MA23452A1 - Procede de preparation d'agents antiparasitaires consistant en derives d'avermectines et de milbemycines. - Google Patents

Procede de preparation d'agents antiparasitaires consistant en derives d'avermectines et de milbemycines.

Info

Publication number
MA23452A1
MA23452A1 MA23780A MA23780A MA23452A1 MA 23452 A1 MA23452 A1 MA 23452A1 MA 23780 A MA23780 A MA 23780A MA 23780 A MA23780 A MA 23780A MA 23452 A1 MA23452 A1 MA 23452A1
Authority
MA
Morocco
Prior art keywords
avmectins
milbemycins
derivatives
antiparasitic agents
agents consisting
Prior art date
Application number
MA23780A
Other languages
English (en)
Inventor
Nigel Derek Arthur Walshe
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of MA23452A1 publication Critical patent/MA23452A1/fr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/01—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing oxygen
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/10—Anthelmintics

Landscapes

  • Life Sciences & Earth Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Agronomy & Crop Science (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Dentistry (AREA)
  • Plant Pathology (AREA)
  • Pest Control & Pesticides (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Wood Science & Technology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Saccharide Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
MA23780A 1994-02-16 1995-02-15 Procede de preparation d'agents antiparasitaires consistant en derives d'avermectines et de milbemycines. MA23452A1 (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB9402916A GB9402916D0 (en) 1994-02-16 1994-02-16 Antiparasitic agents

Publications (1)

Publication Number Publication Date
MA23452A1 true MA23452A1 (fr) 1995-10-01

Family

ID=10750420

Family Applications (1)

Application Number Title Priority Date Filing Date
MA23780A MA23452A1 (fr) 1994-02-16 1995-02-15 Procede de preparation d'agents antiparasitaires consistant en derives d'avermectines et de milbemycines.

Country Status (30)

Country Link
US (1) US5723488A (fr)
EP (1) EP0745089B1 (fr)
JP (2) JP3194959B2 (fr)
KR (1) KR100196751B1 (fr)
CN (1) CN1043996C (fr)
AP (1) AP547A (fr)
AT (1) ATE174340T1 (fr)
AU (1) AU686326B2 (fr)
CA (1) CA2183453C (fr)
CZ (1) CZ241496A3 (fr)
DE (1) DE69506525T2 (fr)
DK (1) DK0745089T3 (fr)
EG (1) EG20774A (fr)
ES (1) ES2124529T3 (fr)
FI (1) FI963201A7 (fr)
GB (1) GB9402916D0 (fr)
HU (1) HUT76521A (fr)
IL (1) IL112596A0 (fr)
MA (1) MA23452A1 (fr)
MX (1) MX9603486A (fr)
NO (1) NO963389L (fr)
NZ (1) NZ279494A (fr)
OA (1) OA10309A (fr)
PL (1) PL315902A1 (fr)
RU (1) RU2134272C1 (fr)
SI (1) SI9520021A (fr)
SK (1) SK106096A3 (fr)
WO (1) WO1995022552A1 (fr)
YU (1) YU8795A (fr)
ZA (1) ZA951218B (fr)

Families Citing this family (191)

* Cited by examiner, † Cited by third party
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NZ601638A (en) 2010-02-22 2014-07-25 Syngenta Participations Ag Dihydrofuran derivatives as insecticidal compounds
US20140206633A1 (en) 2010-02-25 2014-07-24 Syngenta Crop Protection Llc Process for the preparation of isoxazoline derivatives
WO2012045700A1 (fr) 2010-10-05 2012-04-12 Syngenta Participations Ag Pyrolidin-yl-aryl-carboxamides insecticides
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BR112013023798A2 (pt) 2011-03-22 2016-09-20 Syngenta Participations Ag compostos inseticidas
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RU2453553C1 (ru) * 2011-05-11 2012-06-20 Игорь Викторович Заварзин 5-о-сукциноилавермектин, способ его получения и антипаразитарное средство на его основе
MX2013013211A (es) 2011-05-18 2014-02-20 Syngenta Participations Ag Compuestos insecticidas a base de derivados de ariltioacetamida.
WO2012163948A1 (fr) 2011-05-31 2012-12-06 Syngenta Participations Ag Mélanges pesticides comprenant des dérivés d'isoxazoline
UY34104A (es) 2011-05-31 2013-01-03 Syngenta Participations Ag ?compuestos derivados benzamídicos heterocíclicos, procesos e intermedios para su preparación, composiciones y métodos para su uso?.
WO2012175474A1 (fr) 2011-06-20 2012-12-27 Syngenta Participations Ag Pesticides à base de 1,2,3-triazole
CN103732567A (zh) 2011-08-22 2014-04-16 先正达参股股份有限公司 作为杀虫化合物的二氢呋喃衍生物
WO2013026724A1 (fr) 2011-08-22 2013-02-28 Syngenta Participations Ag Dérivés de dihydrofurane en tant que composés insecticides
JP6061934B2 (ja) 2011-08-25 2017-01-18 シンジェンタ パーティシペーションズ アーゲー 殺虫化合物としてのイソオキサゾリン誘導体
BR112014003730A2 (pt) 2011-08-25 2017-03-14 Syngenta Participations Ag processo para a preparação de derivados de tietano
BR112014004275A2 (pt) 2011-08-25 2017-03-21 Syngenta Participations Ag derivados de isoxazolina como compostos inseticidas
WO2013026695A1 (fr) 2011-08-25 2013-02-28 Syngenta Participations Ag Dérivés d'isoxazoline en tant que composés insecticides
WO2013026929A1 (fr) 2011-08-25 2013-02-28 Syngenta Participations Ag Dérivés de dihydropyrrole en tant que composés insecticides
US9078444B2 (en) 2011-09-13 2015-07-14 Syngenta Participations Ag Isothiazoline derivatives as insecticidal compounds
JP2014528957A (ja) 2011-10-03 2014-10-30 シンジェンタ パーティシペーションズ アクチェンゲゼルシャフト 殺虫性化合物
JP2014534182A (ja) 2011-10-03 2014-12-18 シンジェンタ パーティシペーションズ アクチェンゲゼルシャフト 殺虫化合物としてのイソオキサゾリン誘導体
WO2013135674A1 (fr) 2012-03-12 2013-09-19 Syngenta Participations Ag Composés de 2-aryl-acétamide insecticides
WO2014001121A1 (fr) 2012-06-25 2014-01-03 Syngenta Participations Ag Dérivés d'isothiazole en tant que composés insecticides
WO2014001120A1 (fr) 2012-06-25 2014-01-03 Syngenta Participations Ag Dérivés d'isothiazole en tant que composés insecticides
JP6494516B2 (ja) 2012-10-31 2019-04-03 シンジェンタ パーティシペーションズ アーゲー 殺虫性化合物
WO2014079935A1 (fr) 2012-11-21 2014-05-30 Syngenta Participations Ag Composés insecticides à base de dérivés d'arylthioacétamide
JP6488278B2 (ja) 2013-04-02 2019-03-20 シンジェンタ パーティシペーションズ アーゲー 殺虫性化合物
CN105189457A (zh) 2013-04-02 2015-12-23 先正达参股股份有限公司 杀虫化合物
CN104231022B (zh) * 2013-06-14 2018-10-09 南开大学 一种大环内酯类化合物的制备及应用
CN103421065B (zh) * 2013-07-03 2016-05-18 大庆志飞生物化工有限公司 一类新型阿维菌素衍生物及其制备方法
WO2015007451A1 (fr) 2013-07-15 2015-01-22 Syngenta Participations Ag Dérivés hétérobicycliques microbiocides
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CN103896961A (zh) * 2014-03-25 2014-07-02 武汉大学 一种米尔贝肟类化合物及其制备方法
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UA120960C2 (uk) 2015-03-27 2020-03-10 Сінгента Партісіпейшнс Аг Мікробіоцидні гетеробіциклічні похідні
WO2016155831A1 (fr) 2015-04-02 2016-10-06 Syngenta Participations Ag Dérivés d'isoxazoline-styrène utilisés comme composés insecticides
PL3356358T3 (pl) 2015-10-02 2020-11-02 Syngenta Participations Ag Mikrobiocydowe pochodne oksadiazolowe
EP3367798A1 (fr) 2015-10-28 2018-09-05 Syngenta Participations AG Dérivés d'oxadiazole microbiocides
WO2017076982A1 (fr) 2015-11-04 2017-05-11 Syngenta Participations Ag Dérivés d'anilides microbiocides
CN108289448B (zh) 2015-12-02 2021-10-22 先正达参股股份有限公司 杀微生物的噁二唑衍生物
EP3390399A1 (fr) 2015-12-17 2018-10-24 Syngenta Participations AG Dérivés d'oxadiazole microbiocides
CN108779109B (zh) 2016-03-15 2022-03-11 先正达参股股份有限公司 杀微生物的噁二唑衍生物
WO2017162868A1 (fr) 2016-03-24 2017-09-28 Syngenta Participations Ag Dérivés d'oxadiazole microbiocides
PL3439477T3 (pl) 2016-04-08 2020-11-16 Syngenta Participations Ag Mikrobiocydowe pochodne oksadiazolowe
BR112018070785B1 (pt) 2016-04-12 2023-01-10 Syngenta Participations Ag Compostos derivados de oxadiazol microbiocidas, composição agroquímica, método de controle ou prevenção de infestação de plantas úteis por microrganismos fitopatogênicos e uso dos referidos compostos
WO2017178408A1 (fr) 2016-04-15 2017-10-19 Syngenta Participations Ag Silicium microbiocide contenant des dérivés d'aryle
MX2018014441A (es) 2016-05-30 2019-04-01 Syngenta Participations Ag Derivados de tiazol microbiocidas.
WO2017207757A1 (fr) 2016-06-03 2017-12-07 Syngenta Participations Ag Dérivés d'oxadiazole microbiocides
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JP2019526535A (ja) 2016-07-22 2019-09-19 シンジェンタ パーティシペーションズ アーゲー 殺微生物オキサジアゾール誘導体
WO2018015447A1 (fr) 2016-07-22 2018-01-25 Syngenta Participations Ag Dérivés d'oxadiazole microbiocides
US20190284148A1 (en) 2016-07-22 2019-09-19 Syngenta Participations Ag Microbiocidal oxadiazole derivatives
WO2018029242A1 (fr) 2016-08-11 2018-02-15 Syngenta Participations Ag Dérivés d'oxadiazole microbicides
WO2018055133A1 (fr) 2016-09-23 2018-03-29 Syngenta Participations Ag Dérivés de tétrazolone microbiocides
CN109923112A (zh) 2016-09-23 2019-06-21 先正达参股股份有限公司 杀微生物的噁二唑衍生物
PL3522715T3 (pl) 2016-10-06 2021-06-28 Syngenta Participations Ag Mikrobiocydowe pochodne oksadiazolowe
UY37623A (es) 2017-03-03 2018-09-28 Syngenta Participations Ag Derivados de oxadiazol tiofeno fungicidas
US20200187502A1 (en) 2017-03-10 2020-06-18 Syngenta Participations Ag Microbiocidal oxadiazole derivatives
WO2018185013A1 (fr) 2017-04-03 2018-10-11 Syngenta Participations Ag Dérivés d'oxadiazole microbiocides
BR112019021019B1 (pt) 2017-04-05 2023-12-05 Syngenta Participations Ag Compostos derivados de oxadiazol microbiocidas, composição agrícola, método para controlar ou prevenir a infestação de plantas úteis por microrganismos fitopatogênicos e uso de um composto derivado de oxadiazol
BR112019020734B1 (pt) 2017-04-05 2023-12-05 Syngenta Participations Ag Compostos derivados de oxadiazol, composição agroquímica, método para controlar ou prevenir a infestação de plantas úteis por microrganismos fitopatogênicos e uso dos referidos compostos
WO2018184984A1 (fr) 2017-04-05 2018-10-11 Syngenta Participations Ag Dérivés d'oxadiazole microbiocides
WO2018184982A1 (fr) 2017-04-05 2018-10-11 Syngenta Participations Ag Dérivés d'oxadiazole microbiocides
BR112019020819B1 (pt) 2017-04-05 2023-12-05 Syngenta Participations Ag Composto de fórmula (i), composição agroquímica, método para controlar ou prevenir a infestação de plantas úteis por micro-organismos fitopatogênicos e uso de um composto de fórmula (i)
BR112019020739B1 (pt) 2017-04-05 2023-12-19 Syngenta Participations Ag Compostos derivados de oxadiazol microbiocidas e seu uso, composição agroquímica, método para controlar ou prevenir a infestação de plantas úteis por microrganismos fitopatogênicos
WO2018185211A1 (fr) 2017-04-06 2018-10-11 Syngenta Participations Ag Dérivés d'oxadiazole microbiocides
WO2018206419A1 (fr) 2017-05-12 2018-11-15 Syngenta Participations Ag Dérivés hétérobicycliques microbiocides
CN110709395A (zh) 2017-06-02 2020-01-17 先正达参股股份有限公司 杀微生物的噁二唑衍生物
CN107118247B (zh) * 2017-06-14 2019-07-26 博瑞生物医药(苏州)股份有限公司 塞拉菌素的制备方法
CN107021990B (zh) * 2017-06-14 2019-07-12 博瑞生物医药(苏州)股份有限公司 高纯度塞拉菌素的制备方法
WO2019011926A1 (fr) 2017-07-11 2019-01-17 Syngenta Participations Ag Dérivés d'oxadiazole microbiocides
WO2019011928A1 (fr) 2017-07-11 2019-01-17 Syngenta Participations Ag Dérivés d'oxadiazole microbiocides
WO2019011929A1 (fr) 2017-07-11 2019-01-17 Syngenta Participations Ag Dérivés d'oxadiazole microbiocides
BR112020000465B1 (pt) 2017-07-11 2024-02-20 Syngenta Participations Ag Derivados oxadiazol microbiocidas
WO2019012001A1 (fr) 2017-07-12 2019-01-17 Syngenta Participations Ag Dérivés d'oxadiazole microbiocides
BR112020000371A2 (pt) 2017-07-12 2020-07-14 Syngenta Participations Ag derivados de oxadiazol microbiocidas
BR112020000463A2 (pt) 2017-07-13 2020-07-21 Syngenta Participations Ag derivados oxadiazol microbiocidas
CN107266511B (zh) * 2017-07-25 2019-08-20 中国农业大学 一类新颖的5-肟酯B2a结构的化合物及其制备方法与应用
US11584740B2 (en) 2017-09-13 2023-02-21 Syngenta Participations Ag Microbiocidal quinoline (thio)carboxamide derivatives
ES2904910T3 (es) 2017-09-13 2022-04-06 Syngenta Participations Ag Derivados de quinolina (tio)carboxamida microbiocidas
EP3681867B1 (fr) 2017-09-13 2021-08-11 Syngenta Participations AG Dérivés de (thio)carboxamide de quinoline microbiocide
CN111164076A (zh) 2017-09-13 2020-05-15 先正达参股股份有限公司 杀微生物的喹啉(硫代)甲酰胺衍生物
ES2894763T3 (es) 2017-09-13 2022-02-15 Syngenta Participations Ag Derivados de quinolina (tio)carboxamida microbiocidas
CN111051286A (zh) 2017-09-13 2020-04-21 先正达参股股份有限公司 杀微生物的喹啉(硫代)甲酰胺衍生物
EP3681870B1 (fr) 2017-09-13 2021-08-04 Syngenta Participations AG Dérivés de (thio)carboxamide de quinoline microbiocide
UY37913A (es) 2017-10-05 2019-05-31 Syngenta Participations Ag Derivados de picolinamida fungicidas que portan un grupo terminal cuaternario
UY37912A (es) 2017-10-05 2019-05-31 Syngenta Participations Ag Derivados de picolinamida fungicidas que portan grupos terminales heteroarilo o heteroariloxi
BR112020009659A2 (pt) 2017-11-15 2020-11-10 Syngenta Participations Ag derivados picolinamida microbiocidas
CN111356679A (zh) 2017-11-20 2020-06-30 先正达参股股份有限公司 杀微生物的噁二唑衍生物
KR102697953B1 (ko) 2017-11-29 2024-08-21 신젠타 파티서페이션즈 아게 살미생물 티아졸 유도체
GB201721235D0 (en) 2017-12-19 2018-01-31 Syngenta Participations Ag Polymorphs
EP3728191B1 (fr) 2017-12-19 2022-07-13 Syngenta Participations Ag Dérivés de picolinamide microbicides
CN112020503A (zh) 2018-04-26 2020-12-01 先正达参股股份有限公司 杀微生物的噁二唑衍生物
BR112020023915A2 (pt) 2018-05-25 2021-02-09 Syngenta Participations Ag derivados de picolinamida microbiocidas
CN112351981A (zh) 2018-06-29 2021-02-09 先正达农作物保护股份公司 杀微生物的噁二唑衍生物
EP3818058A1 (fr) 2018-07-02 2021-05-12 Syngenta Crop Protection AG Dérivés de 3-(2-thiényl)-5-(trifluorométhyl) -1,2,4-oxadiazole en tant que fongicides agrochimiques
CN112689631A (zh) 2018-07-16 2021-04-20 先正达农作物保护股份公司 杀微生物的噁二唑衍生物
GB201812692D0 (en) 2018-08-03 2018-09-19 Syngenta Participations Ag Microbiocidal compounds
US11440888B2 (en) 2018-09-19 2022-09-13 Syngenta Crop Protection Ag Microbiocidal quinoline carboxamide derivatives
WO2020070132A1 (fr) 2018-10-06 2020-04-09 Syngenta Participations Ag Dérivés de quinoléine dihydro-(thiazine) oxazine microbiocides
JP2022504304A (ja) 2018-10-06 2022-01-13 シンジェンタ パーティシペーションズ アーゲー 殺微生物性キノリンジヒドロ-(チアジン)オキサジン誘導体
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FI963201A0 (fi) 1996-08-15
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AP9500714A0 (en) 1995-01-31
SI9520021A (en) 1997-04-30
EP0745089B1 (fr) 1998-12-09
ES2124529T3 (es) 1999-02-01
WO1995022552A1 (fr) 1995-08-24
OA10309A (en) 1997-10-07
US5723488A (en) 1998-03-03
ATE174340T1 (de) 1998-12-15
GB9402916D0 (en) 1994-04-06
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JPH11263791A (ja) 1999-09-28
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IL112596A0 (en) 1995-05-26
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DE69506525T2 (de) 1999-05-06
AU686326B2 (en) 1998-02-05
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YU8795A (sh) 1997-12-05
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