MA26818A1 - Formulations contenant des inhibiteurs de lipase - Google Patents

Formulations contenant des inhibiteurs de lipase

Info

Publication number
MA26818A1
MA26818A1 MA26545A MA26545A MA26818A1 MA 26818 A1 MA26818 A1 MA 26818A1 MA 26545 A MA26545 A MA 26545A MA 26545 A MA26545 A MA 26545A MA 26818 A1 MA26818 A1 MA 26818A1
Authority
MA
Morocco
Prior art keywords
formulations containing
lipase inhibitors
containing lipase
inhibitors
formulations
Prior art date
Application number
MA26545A
Other languages
English (en)
Inventor
Smidt Passchier Christiaan De
Hans Lengsfeld
Hans Steffen
Joseph Tardio
Paul Hadvary
Thomas Rades
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=8238990&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=MA26818(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of MA26818A1 publication Critical patent/MA26818A1/fr

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/10—Dispersions; Emulsions
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/10—Dispersions; Emulsions
    • A61K9/107—Emulsions ; Emulsion preconcentrates; Micelles
    • A61K9/1075—Microemulsions or submicron emulsions; Preconcentrates or solids thereof; Micelles, e.g. made of phospholipids or block copolymers
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/365—Lactones
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/4841—Filling excipients; Inactive ingredients
    • A61K9/485—Inorganic compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/4841—Filling excipients; Inactive ingredients
    • A61K9/4858—Organic compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/06—Antihyperlipidemics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0002—Galenical forms characterised by the drug release technique; Application systems commanded by energy
    • A61K9/0007—Effervescent

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Dispersion Chemistry (AREA)
  • Hematology (AREA)
  • Diabetes (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • Obesity (AREA)
  • Inorganic Chemistry (AREA)
  • Child & Adolescent Psychology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Medicines Containing Plant Substances (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
MA26545A 1999-09-13 2002-03-11 Formulations contenant des inhibiteurs de lipase MA26818A1 (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP99118180 1999-09-13

Publications (1)

Publication Number Publication Date
MA26818A1 true MA26818A1 (fr) 2004-12-20

Family

ID=8238990

Family Applications (1)

Application Number Title Priority Date Filing Date
MA26545A MA26818A1 (fr) 1999-09-13 2002-03-11 Formulations contenant des inhibiteurs de lipase

Country Status (38)

Country Link
US (3) US20030181512A1 (fr)
EP (1) EP1216025B1 (fr)
JP (1) JP4217016B2 (fr)
KR (1) KR100572434B1 (fr)
CN (1) CN1197551C (fr)
AR (1) AR025587A1 (fr)
AT (1) ATE333866T1 (fr)
AU (1) AU769415B2 (fr)
BR (2) BRPI0013939B1 (fr)
CA (1) CA2383916C (fr)
CO (1) CO5180587A1 (fr)
CY (1) CY1106180T1 (fr)
CZ (1) CZ301901B6 (fr)
DE (1) DE60029602T2 (fr)
DK (1) DK1216025T3 (fr)
EG (1) EG24117A (fr)
ES (1) ES2267563T3 (fr)
HR (1) HRP20020205B1 (fr)
HU (1) HU228858B1 (fr)
IL (1) IL148494A0 (fr)
JO (1) JO2386B1 (fr)
MA (1) MA26818A1 (fr)
ME (1) ME00674B (fr)
MX (1) MXPA02002034A (fr)
MY (1) MY130200A (fr)
NO (1) NO331906B1 (fr)
NZ (1) NZ517545A (fr)
PE (1) PE20010595A1 (fr)
PL (1) PL199870B1 (fr)
PT (1) PT1216025E (fr)
RS (1) RS50422B (fr)
RU (1) RU2239428C2 (fr)
SI (1) SI1216025T1 (fr)
TR (1) TR200200606T2 (fr)
TW (1) TWI243060B (fr)
UY (1) UY26338A1 (fr)
WO (1) WO2001019340A1 (fr)
ZA (1) ZA200201518B (fr)

Families Citing this family (27)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR100572785B1 (ko) 2000-07-28 2006-04-19 에프. 호프만-라 로슈 아게 신규한 약학 조성물
US6730319B2 (en) * 2001-06-06 2004-05-04 Hoffmann-La Roche Inc. Pharmaceutical compositions having depressed melting points
US20030027786A1 (en) * 2001-06-06 2003-02-06 Karsten Maeder Lipase inhibiting composition
US8372430B2 (en) 2002-12-17 2013-02-12 The Procter & Gamble Company Compositions, methods, and kits useful for the alleviation of gastrointestinal effects
FI20045076A7 (fi) * 2004-03-15 2005-09-16 Bioferme Oy Funktionaalinen elintarvike
US8241664B2 (en) * 2005-04-15 2012-08-14 Clarus Therapeutics, Inc Pharmaceutical delivery systems for hydrophobic drugs and compositions comprising same
KR100910000B1 (ko) * 2005-05-13 2009-07-29 씨제이제일제당 (주) 리파아제 저해제 함유 약학 조성물
JP5044398B2 (ja) * 2005-06-09 2012-10-10 武田薬品工業株式会社 固形製剤
KR100669497B1 (ko) * 2005-08-17 2007-01-16 보람제약주식회사 안정성과 용출률이 뛰어난 약리학적 조성물 및 그 제조방법
WO2007033522A1 (fr) * 2005-09-21 2007-03-29 Shenzhen Tys R & D Co., Ltd. Formulation de gélule contenant de la moxifloxacine et son procédé de préparation
KR101252635B1 (ko) * 2006-04-20 2013-04-10 (주)아모레퍼시픽 리파아제 저해제 및 친유성 오일흡수제를 포함하는 약학조성물 및 이로부터 제조된 경구 투여용 제제
TR200607613A2 (tr) * 2006-12-29 2008-07-21 NOBEL İLAÇ SAN.ve TiC.A.Ş. Lipaz inhibitörü içeren farmasötik formülasyonlar
EP1970051A1 (fr) * 2007-03-14 2008-09-17 Merz Pharma GmbH & Co.KGaA Utilisation d'une micro-émulsion aqueuse pour la préparation d'une formulation pour le traitement de maladies adipeuses
KR101439470B1 (ko) * 2007-05-22 2014-09-16 한미사이언스 주식회사 오를리스타트 및 대변 연화제를 포함하는 비만의 예방 또는치료용 조성물
ES2350798T3 (es) * 2007-09-12 2011-01-27 Mader S.R.L. Composiciones farmacéuticas para uso oral para tratar a pacientes afectados por la obesidad.
EP2044930A1 (fr) * 2007-10-01 2009-04-08 Nestec S.A. Composition pour le contrôle de réactions catalysées par la lipase
PL216542B1 (pl) 2008-03-20 2014-04-30 Zakłady Farmaceutyczne POLPHARMA Spółka Akcyjna Sposób wytwarzania stabilnej kompozycji orlistatu w postaci kapsułkowanego proszku
US8309107B2 (en) 2008-10-06 2012-11-13 Banner Pharmacaps, Inc. Stable solutions of orlistat for pharmaceutical dosage forms
KR20100075260A (ko) * 2008-12-24 2010-07-02 주식회사종근당 리파아제 저해제의 부작용 개선을 위한 신규한 약제학적 조성물
BRPI0901602B8 (pt) 2009-04-03 2021-05-25 Ems S/A formulação farmacêuticas
RU2441654C2 (ru) * 2010-02-17 2012-02-10 Лабораториос Баго С.А. Фармацевтическая композиция с активностью против ожирения, включающая премикс чистого орлистата, и способ ее изготовления
ITRM20120331A1 (it) 2012-07-12 2014-01-13 Guidotti & C Spa Labor Composizioni pediatriche orali liquide contenenti nepadutant.
WO2016166767A1 (fr) * 2015-04-14 2016-10-20 Zim Laboratories Limited Formulation pharmaceutique comprenant des médicaments à faible point de fusion hautement lipophiles
CN106310287B (zh) * 2015-06-25 2019-03-19 山东省药学科学院 新利司他药用组合物及其制备方法
MY196635A (en) * 2018-06-22 2023-04-25 Sime Darby Plantation Intellectual Property Sdn Bhd Method For Reducing Formation of Free Fatty Acids in Plants
CN115105476B (zh) * 2021-03-23 2023-11-14 山东新时代药业有限公司 一种奥利司他冻干口服制剂及其制备工艺
CN114983938A (zh) * 2022-05-19 2022-09-02 广东嘉博制药有限公司 一种奥利司他口服复合乳液及其制备方法

Family Cites Families (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA1247547A (fr) 1983-06-22 1988-12-28 Paul Hadvary Derives de leucine
ES2061623T3 (es) * 1987-03-02 1994-12-16 Brocades Pharma Bv Procedimiento para la obtencion de una composicion farmaceutica y un granulado farmaceutico.
SU1510148A1 (ru) * 1988-01-26 1995-04-30 Всесоюзный научно-исследовательский институт химии и технологии лекарственных средств Способ получения ингибитора липазы
CA2128044C (fr) 1993-08-05 2007-02-20 Klaus-Dieter Bremer Compositions pharmaceutiques comportant un glucosidase et/ou un inhibiteur d'amylase, et un inhibiteur des lipases
IT1282673B1 (it) 1996-02-23 1998-03-31 Ist Naz Stud Cura Dei Tumori Derivati della camptotecina e loro uso come agenti antitumorali
JP2001523221A (ja) 1996-09-01 2001-11-20 ファーモス コーポレイション 親油性物質の促進された生物学的利用能のための固形共沈物
US5891469A (en) * 1997-04-02 1999-04-06 Pharmos Corporation Solid Coprecipitates for enhanced bioavailability of lipophilic substances
US6004996A (en) * 1997-02-05 1999-12-21 Hoffman-La Roche Inc. Tetrahydrolipstatin containing compositions
PL191222B1 (pl) 1997-02-05 2006-03-31 Hoffmann La Roche Zastosowanie tetrahydrolipstatyny do wytwarzania doustnego farmaceutycznego preparatu do leczenia cukrzycy typu II
US6267952B1 (en) 1998-01-09 2001-07-31 Geltex Pharmaceuticals, Inc. Lipase inhibiting polymers
CA2340056C (fr) 1998-08-14 2007-01-09 F. Hoffmann-La Roche Ag Compositions pharmaceutiques comportant des inhibiteurs de lipase
PT1105123E (pt) 1998-08-14 2004-08-31 Hoffmann La Roche Composicoes farmaceuticas contendo inibidores da lipase e quitosano
US6368622B2 (en) * 1999-01-29 2002-04-09 Abbott Laboratories Process for preparing solid formulations of lipid regulating agents with enhanced dissolution and absorption

Also Published As

Publication number Publication date
HU228858B1 (en) 2013-06-28
NO331906B1 (no) 2012-04-30
CN1197551C (zh) 2005-04-20
CY1106180T1 (el) 2011-06-08
US20030181512A1 (en) 2003-09-25
CO5180587A1 (es) 2002-07-30
HRP20020205B1 (hr) 2011-06-30
PL199870B1 (pl) 2008-11-28
SI1216025T1 (sl) 2006-12-31
NZ517545A (en) 2003-11-28
PE20010595A1 (es) 2001-05-26
DK1216025T3 (da) 2006-10-30
EP1216025B1 (fr) 2006-07-26
DE60029602T2 (de) 2007-07-26
ZA200201518B (en) 2003-07-30
BRPI0013939B1 (pt) 2017-07-18
CZ301901B6 (cs) 2010-07-28
TWI243060B (en) 2005-11-11
US20110275706A1 (en) 2011-11-10
US20040175420A1 (en) 2004-09-09
CA2383916C (fr) 2009-01-20
AU7286300A (en) 2001-04-17
HRP20020205A2 (en) 2004-04-30
UY26338A1 (es) 2000-10-31
MEP90808A (en) 2011-12-20
ME00674B (fr) 2011-12-20
HK1049966A1 (en) 2003-06-06
JP4217016B2 (ja) 2009-01-28
RS50422B (sr) 2009-12-31
EG24117A (en) 2008-07-06
PL356174A1 (en) 2004-06-14
MY130200A (en) 2007-06-29
ATE333866T1 (de) 2006-08-15
YU17202A (sh) 2006-01-16
JO2386B1 (en) 2007-06-17
CN1373656A (zh) 2002-10-09
CA2383916A1 (fr) 2001-03-22
NO20021204L (no) 2002-03-12
HUP0202737A3 (en) 2005-01-28
KR100572434B1 (ko) 2006-04-18
CZ20021276A3 (cs) 2003-04-16
BR0013939A (pt) 2002-05-14
IL148494A0 (en) 2002-09-12
DE60029602D1 (de) 2006-09-07
NO20021204D0 (no) 2002-03-12
RU2239428C2 (ru) 2004-11-10
US8012494B2 (en) 2011-09-06
JP2003509357A (ja) 2003-03-11
MXPA02002034A (es) 2002-08-20
WO2001019340A1 (fr) 2001-03-22
KR20020063852A (ko) 2002-08-05
PT1216025E (pt) 2006-12-29
AR025587A1 (es) 2002-12-04
HUP0202737A2 (hu) 2003-01-28
ES2267563T3 (es) 2007-03-16
AU769415B2 (en) 2004-01-29
TR200200606T2 (tr) 2002-07-22
EP1216025A1 (fr) 2002-06-26

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