MA27080A1 - Forme polymorphe du rimonabant, son procede de preparation et les compositions pharmaceutiques en contenant - Google Patents

Forme polymorphe du rimonabant, son procede de preparation et les compositions pharmaceutiques en contenant

Info

Publication number
MA27080A1
MA27080A1 MA27659A MA27659A MA27080A1 MA 27080 A1 MA27080 A1 MA 27080A1 MA 27659 A MA27659 A MA 27659A MA 27659 A MA27659 A MA 27659A MA 27080 A1 MA27080 A1 MA 27080A1
Authority
MA
Morocco
Prior art keywords
same
rimonabant
preparing
pharmaceutical compositions
compositions containing
Prior art date
Application number
MA27659A
Other languages
English (en)
Inventor
Alain Alcade
Corinne Gavory
Gilles Anne-Archard
Olivier Monnier
Original Assignee
Sanofi Aventis
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sanofi Aventis filed Critical Sanofi Aventis
Publication of MA27080A1 publication Critical patent/MA27080A1/fr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/10—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing aromatic rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Child & Adolescent Psychology (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Steroid Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
MA27659A 2001-11-08 2004-04-28 Forme polymorphe du rimonabant, son procede de preparation et les compositions pharmaceutiques en contenant MA27080A1 (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR0114579A FR2831883B1 (fr) 2001-11-08 2001-11-08 Forme polymorphe du rimonabant, son procede de preparation et les compositions pharmaceutiques en contenant

Publications (1)

Publication Number Publication Date
MA27080A1 true MA27080A1 (fr) 2004-12-20

Family

ID=8869285

Family Applications (1)

Application Number Title Priority Date Filing Date
MA27659A MA27080A1 (fr) 2001-11-08 2004-04-28 Forme polymorphe du rimonabant, son procede de preparation et les compositions pharmaceutiques en contenant

Country Status (33)

Country Link
US (2) US20050043356A1 (fr)
EP (1) EP1446384A1 (fr)
JP (2) JP4181994B2 (fr)
KR (2) KR20050043774A (fr)
CN (1) CN100412063C (fr)
AP (1) AP1830A (fr)
AR (1) AR037253A1 (fr)
AU (1) AU2002350869B2 (fr)
BR (1) BR0213931A (fr)
CA (1) CA2464145A1 (fr)
CO (1) CO5580827A2 (fr)
CR (1) CR7333A (fr)
EA (1) EA006771B1 (fr)
EC (1) ECSP045088A (fr)
FR (1) FR2831883B1 (fr)
GE (1) GEP20063894B (fr)
HR (1) HRP20040403A2 (fr)
HU (1) HUP0402043A3 (fr)
IL (2) IL161533A0 (fr)
IS (1) IS7226A (fr)
MA (1) MA27080A1 (fr)
ME (1) MEP21908A (fr)
MX (1) MXPA04004394A (fr)
NO (1) NO326648B1 (fr)
NZ (1) NZ532369A (fr)
OA (1) OA12721A (fr)
PL (1) PL369372A1 (fr)
RS (1) RS36904A (fr)
TN (1) TNSN04079A1 (fr)
TW (1) TW200302824A (fr)
UA (1) UA76776C2 (fr)
WO (1) WO2003040105A1 (fr)
ZA (1) ZA200402999B (fr)

Families Citing this family (33)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2831883B1 (fr) * 2001-11-08 2004-07-23 Sanofi Synthelabo Forme polymorphe du rimonabant, son procede de preparation et les compositions pharmaceutiques en contenant
CA2487849A1 (fr) 2002-07-18 2004-01-29 Cytos Biotechnology Ag Conjugues haptene-porteur et utilisations de ceux-ci
FR2861992B1 (fr) * 2003-11-10 2007-07-20 Sanofi Synthelabo Composition pharmaceutique destinee a l'administration orale d'un derive de pyrazole-3-carboxamide.
MX2007016508A (es) 2005-06-30 2008-03-04 Prosidion Ltd Agonistas del receptor acoplado a la proteina g.
EP1816125A1 (fr) * 2006-02-02 2007-08-08 Ranbaxy Laboratories, Ltd. Formes cristallines d'un antagoniste du récepteur cannabinoïde CB1 et son procédé de préparation
FR2897060B1 (fr) * 2006-02-08 2008-07-25 Sanofi Aventis Sa Le monohydrate de rimonabant, son procede de preparation et les compositions pharmaceutiques en contenant
WO2008038143A2 (fr) * 2006-06-22 2008-04-03 Medichem, S.A. Nouvelles formes solides du rimonabant et procédés de synthèse pour la préparation de celles-ci
WO2008044153A2 (fr) * 2006-08-29 2008-04-17 Medichem, S.A. Procédé de synthèse amélioré de rimonabant
US20100076022A1 (en) * 2006-09-01 2010-03-25 Hetero Drugs Limited Novel polymorphs of rimonabant
EP2061783A2 (fr) * 2006-09-11 2009-05-27 Hetero Drugs Limited Procédé amélioré pour l'obtention de rimonabant
WO2008035023A1 (fr) * 2006-09-19 2008-03-27 Cipla Limited Formes polymorphes de rimonabant
WO2008056377A2 (fr) * 2006-11-06 2008-05-15 Cadila Healthcare Limited Nouvelles formes du rimonabant
WO2008064615A2 (fr) * 2006-12-01 2008-06-05 Zentiva, A.S. Formes cristallines et amorphes du rimonabant et procédés permettant d'obtenir ces formes
CA2673177A1 (fr) * 2006-12-18 2008-06-26 7Tm Pharma A/S Modulateurs de recepteurs cb1
US20100048632A1 (en) 2007-01-04 2010-02-25 Matthew Colin Thor Fyfe Piperidine GPCR Agonists
PE20081849A1 (es) 2007-01-04 2009-01-26 Prosidion Ltd Derivados de piperidin-4-il-propoxi-benzamida como agonistas de gpcr
GB0700122D0 (en) 2007-01-04 2007-02-14 Prosidion Ltd GPCR agonists
US20100048625A1 (en) 2007-01-04 2010-02-25 Matthew Colin Thor Fyfe Piperidine gpcr agonists
PE20081659A1 (es) 2007-01-04 2008-10-24 Prosidion Ltd Agonistas de gpcr
EP1944297A1 (fr) * 2007-01-09 2008-07-16 Miklós Vértessy Rimonabant solide et cristallin et procédés de préparation, ainsi que composition pharmaceutique correspondante
WO2008088900A2 (fr) * 2007-01-18 2008-07-24 Teva Pharmaceutical Industries Ltd. Formes polymorphes d'une base de rimonabant et procédés pour leur préparation
EP1953144A1 (fr) * 2007-01-30 2008-08-06 Sandoz AG Nouvelles formes polymorphes de N-pipéridino-5-(4-chlorophényl)-1-(2, 4-dichlorphényl)-4-méthyl-3-pyrazolecarboxamide
FR2919867A1 (fr) * 2007-08-06 2009-02-13 Sanofi Aventis Sa Le solvate de 2-methoxyethanol de rimonabant et son procede de preparation
FR2919865A1 (fr) * 2007-08-06 2009-02-13 Sanofi Aventis Sa Le solvate de dmso de rimonabant, son procede de preparation et les compositions pharmaceutiques en contenant
FR2919864A1 (fr) * 2007-08-06 2009-02-13 Sanofi Aventis Sa Le solvate de 1,4-dioxane de rimonabant, son procede de preparation et les compositions pharmaceutiques en contenant
FR2919863A1 (fr) * 2007-08-06 2009-02-13 Sanofi Aventis Sa Le solvate de n-methylpyrrolidone de rimonabant, son procede de preparation et les compositions pharmaceutiques en contenant
FR2919862A1 (fr) * 2007-08-06 2009-02-13 Sanofi Aventis Sa Le solvate de 3-methylbutan-1-ol de rimonabant, son procede de preparation et les compositions pharmaceutiques en contenant
GB0720390D0 (en) 2007-10-18 2007-11-28 Prosidion Ltd G-Protein coupled receptor agonists
GB0720389D0 (en) 2007-10-18 2008-11-12 Prosidion Ltd G-Protein Coupled Receptor Agonists
WO2009153804A1 (fr) * 2008-06-16 2009-12-23 Cadila Healthcare Limited Procédé de préparation de la forme 1 du rimonabant
WO2010079241A1 (fr) 2009-01-12 2010-07-15 Fundacion Hospital Nacional De Paraplejicos Para La Investigacion Y La Integracion Utilisation d'antagonistes et/ou d'agonistes inverses des récepteurs cb1 pour la préparation de médicaments qui augmentent l'excitabilité des motoneurones
FR3008620A1 (fr) * 2013-07-22 2015-01-23 Sanofi Sa Formulation de comprime d'un inhibiteur de phosphatidylinositol 3-kinase
CN114555557A (zh) * 2019-10-16 2022-05-27 大塚制药株式会社 森塔纳法啶的制备方法

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2692575B1 (fr) * 1992-06-23 1995-06-30 Sanofi Elf Nouveaux derives du pyrazole, procede pour leur preparation et compositions pharmaceutiques les contenant.
FR2713225B1 (fr) * 1993-12-02 1996-03-01 Sanofi Sa N-pipéridino-3-pyrazolecarboxamide substitué.
AU2002331595A1 (en) * 2001-08-15 2003-03-03 The Government Of The United States Of America As Represented By The Secretary Of The Department Of Novel vasoconstrictor cannabinoid analogs
FR2831883B1 (fr) * 2001-11-08 2004-07-23 Sanofi Synthelabo Forme polymorphe du rimonabant, son procede de preparation et les compositions pharmaceutiques en contenant

Also Published As

Publication number Publication date
NO20041879D0 (no) 2004-05-07
EP1446384A1 (fr) 2004-08-18
AP1830A (en) 2008-02-22
MEP21908A (en) 2010-06-10
NO326648B1 (no) 2009-01-26
KR20050043774A (ko) 2005-05-11
OA12721A (fr) 2006-06-27
JP2005508383A (ja) 2005-03-31
WO2003040105A1 (fr) 2003-05-15
UA76776C2 (uk) 2006-09-15
KR20090089485A (ko) 2009-08-21
US20100190827A1 (en) 2010-07-29
ZA200402999B (en) 2005-04-20
IL161533A0 (en) 2004-09-27
ECSP045088A (es) 2004-06-28
TW200302824A (en) 2003-08-16
JP2009035547A (ja) 2009-02-19
IL161533A (en) 2010-05-31
EA006771B1 (ru) 2006-04-28
AP2004003024A0 (en) 2004-06-30
GEP20063894B (en) 2006-08-10
NO20041879L (no) 2004-06-08
IS7226A (is) 2004-04-19
NZ532369A (en) 2005-10-28
HRP20040403A2 (en) 2004-08-31
JP4181994B2 (ja) 2008-11-19
BR0213931A (pt) 2004-09-08
CR7333A (es) 2008-09-23
JP4931874B2 (ja) 2012-05-16
FR2831883B1 (fr) 2004-07-23
HUP0402043A3 (en) 2009-07-28
CN1582278A (zh) 2005-02-16
CO5580827A2 (es) 2005-11-30
MXPA04004394A (es) 2004-08-11
RS36904A (sr) 2006-10-27
HUP0402043A2 (hu) 2005-01-28
CA2464145A1 (fr) 2003-05-15
AR037253A1 (es) 2004-11-03
EA200400491A1 (ru) 2004-12-30
FR2831883A1 (fr) 2003-05-09
AU2002350869B2 (en) 2007-07-26
PL369372A1 (en) 2005-04-18
US20050043356A1 (en) 2005-02-24
TNSN04079A1 (fr) 2006-06-01
CN100412063C (zh) 2008-08-20

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