MA27195A1 - Derives d'acyl-3 -carboxyphenyluree, procedes pour les preparer et leur utilisation. - Google Patents
Derives d'acyl-3 -carboxyphenyluree, procedes pour les preparer et leur utilisation.Info
- Publication number
- MA27195A1 MA27195A1 MA27903A MA27903A MA27195A1 MA 27195 A1 MA27195 A1 MA 27195A1 MA 27903 A MA27903 A MA 27903A MA 27903 A MA27903 A MA 27903A MA 27195 A1 MA27195 A1 MA 27195A1
- Authority
- MA
- Morocco
- Prior art keywords
- acyl
- preparation
- processes
- derivatives
- carboxyphenylurea
- Prior art date
Links
- 238000000034 method Methods 0.000 title abstract 3
- 150000001875 compounds Chemical class 0.000 abstract 2
- 150000003839 salts Chemical class 0.000 abstract 2
- 230000003178 anti-diabetic effect Effects 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C275/00—Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups
- C07C275/46—Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups containing any of the groups, X being a hetero atom, Y being any atom, e.g. acylureas
- C07C275/48—Y being a hydrogen or a carbon atom
- C07C275/54—Y being a carbon atom of a six-membered aromatic ring, e.g. benzoylureas
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/54—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
Landscapes
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Diabetes (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Obesity (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Endocrinology (AREA)
- Hematology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Emergency Medicine (AREA)
- Engineering & Computer Science (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Abstract
Dérivés d'acyl-3-carboxyphénylurée, procédés pour les préparer et leur utilisation. L'invention concerne des dérivés d'acyl-3-carboxyphénylurée ainsi que leurs sels tolérés physiologiquement et dérivés physiologiquement fonctionnels. L'invention concerne les composés de formule (I) dans laquelle les restes ont les significations indiquées, ainsi que leurs sels tolérés physiologiquement et procédé pour leur préparation. Les composés conviennent, par exemple, en tant qu'antidiabétiques.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE10215908A DE10215908B4 (de) | 2002-04-11 | 2002-04-11 | Acyl-3-carboxyphenyl-harnstoffderivate und deren Verwendung als Arzneimittel |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| MA27195A1 true MA27195A1 (fr) | 2005-01-03 |
Family
ID=28684936
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MA27903A MA27195A1 (fr) | 2002-04-11 | 2004-10-08 | Derives d'acyl-3 -carboxyphenyluree, procedes pour les preparer et leur utilisation. |
Country Status (23)
| Country | Link |
|---|---|
| EP (1) | EP1497263B1 (fr) |
| JP (1) | JP4328212B2 (fr) |
| KR (1) | KR20040097332A (fr) |
| CN (1) | CN1263734C (fr) |
| AR (1) | AR039402A1 (fr) |
| AT (1) | ATE404532T1 (fr) |
| AU (1) | AU2003232192A1 (fr) |
| BR (1) | BR0309130A (fr) |
| CA (1) | CA2481819A1 (fr) |
| DE (2) | DE10215908B4 (fr) |
| HR (1) | HRP20040931A2 (fr) |
| HU (1) | HUP0500203A2 (fr) |
| IL (1) | IL164248A0 (fr) |
| MA (1) | MA27195A1 (fr) |
| MX (1) | MXPA04009239A (fr) |
| NO (1) | NO20044881L (fr) |
| NZ (1) | NZ535833A (fr) |
| PL (1) | PL371317A1 (fr) |
| RS (1) | RS88704A (fr) |
| RU (1) | RU2004133046A (fr) |
| TW (1) | TW200401765A (fr) |
| WO (1) | WO2003084923A1 (fr) |
| ZA (1) | ZA200407361B (fr) |
Families Citing this family (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE10215907A1 (de) * | 2002-04-11 | 2003-11-06 | Aventis Pharma Gmbh | Acyl-4-carboxyphenyl-harnstoffderivate, Verfahren zu deren Herstellung und deren Verwendung |
| DE10306502B4 (de) * | 2003-02-17 | 2005-03-17 | Aventis Pharma Deutschland Gmbh | Substituierte 3-(Benzoylureido)-thiophenderivate und sie enthaltende Arzneimittel |
| DE10308352A1 (de) | 2003-02-27 | 2004-09-09 | Aventis Pharma Deutschland Gmbh | Arylcycloalkylderivate mit verzweigten Seitenketten, Verfahren zu ihrer Herstellung und ihre Anwendung als Arzneimittel |
| US7148246B2 (en) | 2003-02-27 | 2006-12-12 | Sanofi-Aventis Deutschland Gmbh | Cycloalkyl derivatives having bioisosteric carboxylic acid groups, processes for their preparation and their use as pharmaceuticals |
| DE10308355A1 (de) | 2003-02-27 | 2004-12-23 | Aventis Pharma Deutschland Gmbh | Aryl-cycloalkyl substituierte Alkansäurederivate, Verfahren zu ihrer Herstellung und ihre Anwendung als Arzneimittel |
| DE10308353A1 (de) | 2003-02-27 | 2004-12-02 | Aventis Pharma Deutschland Gmbh | Diarylcycloalkylderivate, Verfahren zu ihrer Herstellung und ihre Verwendung als Arzneimittel |
| DE10308351A1 (de) | 2003-02-27 | 2004-11-25 | Aventis Pharma Deutschland Gmbh | 1,3-substituierte Cycloalkylderivate mit sauren, meist heterocyclischen Gruppen, Verfahren zu ihrer Herstellung und ihre Verwendung als Arzneimittel |
| US7241787B2 (en) | 2004-01-25 | 2007-07-10 | Sanofi-Aventis Deutschland Gmbh | Substituted N-cycloexylimidazolinones, process for their preparation and their use as medicaments |
| EP1586573B1 (fr) | 2004-04-01 | 2007-02-07 | Sanofi-Aventis Deutschland GmbH | Oxadiazolones, procédé pour leur préparation, usage comme agents pharmaceutiques |
| DE102005026762A1 (de) | 2005-06-09 | 2006-12-21 | Sanofi-Aventis Deutschland Gmbh | Azolopyridin-2-on-derivate als Inhibitoren von Lipasen und Phospholipasen |
| PE20110235A1 (es) | 2006-05-04 | 2011-04-14 | Boehringer Ingelheim Int | Combinaciones farmaceuticas que comprenden linagliptina y metmorfina |
Family Cites Families (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| ZA867420B (en) * | 1985-09-30 | 1987-05-27 | Union Carbide Corp | Pesticidal 1-(4-aryloxyphenyl)-3-benzoyl urea compounds and process for preparation |
| GB9313268D0 (en) * | 1993-06-28 | 1993-08-11 | Zeneca Ltd | Chemical compounds |
| FI974437A7 (fi) * | 1995-06-06 | 1997-12-05 | Pfizer | Substituoituja N-(indoli-2-karbonyyli)amideja ja johdannaisia glykogee nifosforylaasi-inhibiittoreina |
| WO2000056707A1 (fr) * | 1999-03-24 | 2000-09-28 | Sepracor, Inc. | Thioethers de diaryle, compositions et utilisations de ces dernieres |
| US20010053791A1 (en) * | 2000-03-16 | 2001-12-20 | Babcock Walter C. | Glycogen phosphorylase inhibitor |
| TR200401029T4 (tr) * | 2000-06-09 | 2004-06-21 | Aventis Pharma Deutschland Gmbh | Asilfenil-üre türevleri, imalat yöntemleri ve ilaç maddesi olarak kullanımları |
| GB0021831D0 (en) * | 2000-09-06 | 2000-10-18 | Astrazeneca Ab | Chemical compounds |
| PE20021091A1 (es) * | 2001-05-25 | 2003-02-04 | Aventis Pharma Gmbh | Derivados de fenilurea sustituidos con carbonamida y procedimiento para su preparacion |
-
2002
- 2002-04-11 DE DE10215908A patent/DE10215908B4/de not_active Expired - Fee Related
-
2003
- 2003-03-28 BR BR0309130-9A patent/BR0309130A/pt not_active IP Right Cessation
- 2003-03-28 MX MXPA04009239A patent/MXPA04009239A/es active IP Right Grant
- 2003-03-28 IL IL16424803A patent/IL164248A0/xx unknown
- 2003-03-28 CA CA002481819A patent/CA2481819A1/fr not_active Abandoned
- 2003-03-28 WO PCT/EP2003/003254 patent/WO2003084923A1/fr not_active Ceased
- 2003-03-28 HR HR20040931A patent/HRP20040931A2/hr not_active Application Discontinuation
- 2003-03-28 PL PL03371317A patent/PL371317A1/xx not_active Application Discontinuation
- 2003-03-28 HU HU0500203A patent/HUP0500203A2/hu unknown
- 2003-03-28 JP JP2003582122A patent/JP4328212B2/ja not_active Expired - Fee Related
- 2003-03-28 CN CNB038082241A patent/CN1263734C/zh not_active Expired - Fee Related
- 2003-03-28 KR KR10-2004-7016149A patent/KR20040097332A/ko not_active Withdrawn
- 2003-03-28 RU RU2004133046/04A patent/RU2004133046A/ru not_active Application Discontinuation
- 2003-03-28 RS YUP-887/04A patent/RS88704A/sr unknown
- 2003-03-28 DE DE50310320T patent/DE50310320D1/de not_active Expired - Lifetime
- 2003-03-28 AT AT03745772T patent/ATE404532T1/de not_active IP Right Cessation
- 2003-03-28 AU AU2003232192A patent/AU2003232192A1/en not_active Abandoned
- 2003-03-28 NZ NZ535833A patent/NZ535833A/xx unknown
- 2003-03-28 EP EP03745772A patent/EP1497263B1/fr not_active Expired - Lifetime
- 2003-04-09 AR ARP030101246A patent/AR039402A1/es unknown
- 2003-04-09 TW TW092108055A patent/TW200401765A/zh unknown
-
2004
- 2004-09-14 ZA ZA200407361A patent/ZA200407361B/xx unknown
- 2004-10-08 MA MA27903A patent/MA27195A1/fr unknown
- 2004-11-09 NO NO20044881A patent/NO20044881L/no unknown
Also Published As
| Publication number | Publication date |
|---|---|
| HK1075650A1 (en) | 2005-12-23 |
| CN1263734C (zh) | 2006-07-12 |
| PL371317A1 (en) | 2005-06-13 |
| IL164248A0 (en) | 2005-12-18 |
| EP1497263B1 (fr) | 2008-08-13 |
| TW200401765A (en) | 2004-02-01 |
| NZ535833A (en) | 2006-03-31 |
| DE10215908B4 (de) | 2005-08-18 |
| WO2003084923A1 (fr) | 2003-10-16 |
| AR039402A1 (es) | 2005-02-16 |
| HRP20040931A2 (en) | 2005-02-28 |
| ATE404532T1 (de) | 2008-08-15 |
| BR0309130A (pt) | 2005-02-01 |
| JP2005522481A (ja) | 2005-07-28 |
| CN1646486A (zh) | 2005-07-27 |
| MXPA04009239A (es) | 2005-01-25 |
| AU2003232192A1 (en) | 2003-10-20 |
| ZA200407361B (en) | 2006-02-22 |
| DE50310320D1 (de) | 2008-09-25 |
| RS88704A (sr) | 2007-02-05 |
| DE10215908A1 (de) | 2003-11-06 |
| CA2481819A1 (fr) | 2003-10-16 |
| NO20044881L (no) | 2005-01-07 |
| KR20040097332A (ko) | 2004-11-17 |
| RU2004133046A (ru) | 2005-04-20 |
| EP1497263A1 (fr) | 2005-01-19 |
| JP4328212B2 (ja) | 2009-09-09 |
| HUP0500203A2 (hu) | 2005-06-28 |
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