MA29841B1 - Comprimes dispersibles contenant du deferasirox - Google Patents

Comprimes dispersibles contenant du deferasirox

Info

Publication number
MA29841B1
MA29841B1 MA30795A MA30795A MA29841B1 MA 29841 B1 MA29841 B1 MA 29841B1 MA 30795 A MA30795 A MA 30795A MA 30795 A MA30795 A MA 30795A MA 29841 B1 MA29841 B1 MA 29841B1
Authority
MA
Morocco
Prior art keywords
dispersible tablets
tablets containing
dispersible
tablet
deferasirox
Prior art date
Application number
MA30795A
Other languages
English (en)
Inventor
Florian Battung
Jean-Pierre Cassiere
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of MA29841B1 publication Critical patent/MA29841B1/fr

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0087Galenical forms not covered by A61K9/02 - A61K9/7023
    • A61K9/0095Drinks; Beverages; Syrups; Compositions for reconstitution thereof, e.g. powders or tablets to be dispersed in a glass of water; Veterinary drenches
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • A61P7/06Antianaemics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2072Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
    • A61K9/2077Tablets comprising drug-containing microparticles in a substantial amount of supporting matrix; Multiparticulate tablets
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2095Tabletting processes

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

La présente invention se rapporte à un comprimé dispersible, qui contient : (a) un composé I représenté par la formule (I) ou un sel pharmaceutiquement acceptable de celui-ci, présent en une quantité comprise entre 42 % et 65 % poids par rapport au poids total du comprimé ; et (b) au moins un excipient pharmaceutiquement acceptable convenant à la préparation de comprimés dispersibles. L'invention a également trait à un procédé de fabrication dudit comprimé dispersible.
MA30795A 2005-10-19 2008-03-31 Comprimes dispersibles contenant du deferasirox MA29841B1 (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR0553182 2005-10-19

Publications (1)

Publication Number Publication Date
MA29841B1 true MA29841B1 (fr) 2008-10-03

Family

ID=36616771

Family Applications (1)

Application Number Title Priority Date Filing Date
MA30795A MA29841B1 (fr) 2005-10-19 2008-03-31 Comprimes dispersibles contenant du deferasirox

Country Status (17)

Country Link
US (1) US20080311194A1 (fr)
EP (1) EP1940360A1 (fr)
JP (1) JP2009512652A (fr)
KR (1) KR20080056225A (fr)
CN (1) CN101291655A (fr)
AU (1) AU2006303514B2 (fr)
BR (1) BRPI0617715A2 (fr)
CA (1) CA2625112A1 (fr)
EC (1) ECSP088379A (fr)
IL (1) IL190397A0 (fr)
MA (1) MA29841B1 (fr)
NO (1) NO20082265L (fr)
NZ (1) NZ567155A (fr)
RU (1) RU2008119410A (fr)
TN (1) TNSN08173A1 (fr)
WO (1) WO2007045445A1 (fr)
ZA (1) ZA200802670B (fr)

Families Citing this family (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2009067557A1 (fr) * 2007-11-19 2009-05-28 Teva Pharmaceutical Industries Ltd. Compositions pharmaceutiques de déférasirox
WO2010035282A1 (fr) * 2008-09-24 2010-04-01 Matrix Laboratories Limited Compositions pharmaceutiques comprenant du deferasirox
ES2543427T3 (es) 2010-07-08 2015-08-19 Ratiopharm Gmbh Forma farmacéutica oral de deferasirox
MX2013003522A (es) * 2010-10-01 2013-05-22 Cipla Ltd Composicion farmaceutica.
MX2015003729A (es) 2012-11-12 2015-06-15 Cipla Ltd Composiciones farmaceuticas de dosis fija que comprende deferasirox y deferiprona.
HRP20190173T1 (hr) 2013-03-08 2019-03-22 Novartis Ag Oralne formulacije deferasiroksa
US20160120847A1 (en) * 2013-05-10 2016-05-05 Cipla Limited Low Dose Pharmaceutical Composition
ES2734675T3 (es) 2014-05-20 2019-12-11 Sanovel Ilac Sanayi Ve Ticaret As Formulación de comprimido dispersable en agua que contiene deferasirox
EP2987482A1 (fr) 2014-08-22 2016-02-24 Santa Farma Ilaç Sanayi A.S. Composition pharmaceutique soluble et dispersible contenant du déférasirox
WO2016167729A1 (fr) 2015-04-16 2016-10-20 Öğün Yusuf Toktamiş Comprimés dispersibles contenant du déférasirox
EP3095443A1 (fr) * 2015-05-21 2016-11-23 Abdi Ibrahim Ilac Sanayi ve Ticaret A.S. Composition pharmaceutique contenant du déférasirox
MA43271A (fr) 2015-06-17 2018-09-26 Dispersol Technologies Llc Formulations améliorées de déférasirox et leurs procédés de fabrication
WO2018007956A1 (fr) * 2016-07-05 2018-01-11 Jubilant Generics Limited Composition pharmaceutique à libération immédiate d'agents chélateurs du fer
EP3518904A1 (fr) 2016-09-30 2019-08-07 Synthon B.V. Composition pharmaceutique comprenant du deferasirox
WO2018208242A1 (fr) * 2017-05-10 2018-11-15 İlko Ilaç Sanayi Ve Ticaret Anonim Şirketi Formulation de comprimé de déférasirox pour composition de suspension orale présentant une capacité de traitement améliorée
WO2019043427A1 (fr) 2017-09-01 2019-03-07 Jordan Sweden Medical And Sterilization Company Formes posologiques à auto-dispersion rapide de déférasirox
WO2019108157A1 (fr) * 2017-11-28 2019-06-06 Biofarma Ilac Sanayi Ve Ticaret A.S. Formulation de comprimé entaillé sous une forme dispersible comprenant du déférasirox
TR201722910A2 (tr) 2017-12-29 2019-07-22 Sanovel Ilac Sanayi Ve Ticaret Anonim Sirketi Deferasi̇roks i̇çeren suda dağilabi̇len tablet formülasyonlari
WO2022240279A1 (fr) * 2021-05-10 2022-11-17 Garcia Perez Miguel Angel Comprimé dispersible contenant du déférasirox sous forme de dispersion solide

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9215908D0 (en) * 1992-07-27 1992-09-09 Wellcome Found Water dispersible tablets
MY129541A (en) * 1996-06-25 2007-04-30 Novartis Ag Substituded 3,5-diphenyl-1,2,4-triazoles and their use as pharmaceutical metal chelators
GB0223978D0 (en) * 2002-10-15 2002-11-20 Novartis Ag Organic compound

Also Published As

Publication number Publication date
NZ567155A (en) 2010-06-25
IL190397A0 (en) 2008-11-03
TNSN08173A1 (en) 2009-10-30
WO2007045445A1 (fr) 2007-04-26
KR20080056225A (ko) 2008-06-20
ECSP088379A (es) 2008-05-30
ZA200802670B (en) 2009-10-28
CA2625112A1 (fr) 2007-04-26
EP1940360A1 (fr) 2008-07-09
BRPI0617715A2 (pt) 2011-08-02
AU2006303514B2 (en) 2010-06-24
JP2009512652A (ja) 2009-03-26
US20080311194A1 (en) 2008-12-18
RU2008119410A (ru) 2009-11-27
NO20082265L (no) 2008-05-16
AU2006303514A1 (en) 2007-04-26
CN101291655A (zh) 2008-10-22

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