MA32132B1 - Utilisation de ranolazine pour traiter la douleur - Google Patents
Utilisation de ranolazine pour traiter la douleurInfo
- Publication number
- MA32132B1 MA32132B1 MA33137A MA33137A MA32132B1 MA 32132 B1 MA32132 B1 MA 32132B1 MA 33137 A MA33137 A MA 33137A MA 33137 A MA33137 A MA 33137A MA 32132 B1 MA32132 B1 MA 32132B1
- Authority
- MA
- Morocco
- Prior art keywords
- ranolazine
- pain
- treatment
- patient
- visceral
- Prior art date
Links
- XKLMZUWKNUAPSZ-UHFFFAOYSA-N N-(2,6-dimethylphenyl)-2-{4-[2-hydroxy-3-(2-methoxyphenoxy)propyl]piperazin-1-yl}acetamide Chemical compound COC1=CC=CC=C1OCC(O)CN1CCN(CC(=O)NC=2C(=CC=CC=2C)C)CC1 XKLMZUWKNUAPSZ-UHFFFAOYSA-N 0.000 title abstract 2
- 229960000213 ranolazine Drugs 0.000 title abstract 2
- 208000001294 Nociceptive Pain Diseases 0.000 abstract 1
- 230000002757 inflammatory effect Effects 0.000 abstract 1
- 208000004296 neuralgia Diseases 0.000 abstract 1
- 230000002981 neuropathic effect Effects 0.000 abstract 1
- 208000021722 neuropathic pain Diseases 0.000 abstract 1
- 230000009278 visceral effect Effects 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P23/00—Anaesthetics
- A61P23/02—Local anaesthetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
Landscapes
- Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Chemical & Material Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Anesthesiology (AREA)
- Epidemiology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Pain & Pain Management (AREA)
- Rheumatology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
La présente invention concerne des procédés pour traiter un patient souffrant d'une douleur neuropathique ou nociceptive qui peut être de nature mécanique, viscérale et/ou inflammatoire, comprenant l'administration d'une quantité thérapeutiquement efficace de ranolazine à un patient qui en a besoin.
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US2669908P | 2008-02-06 | 2008-02-06 | |
| US5743708P | 2008-05-30 | 2008-05-30 | |
| PCT/US2009/033464 WO2009100380A1 (fr) | 2008-02-06 | 2009-02-06 | Utilisation de ranolazine pour traiter la douleur |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| MA32132B1 true MA32132B1 (fr) | 2011-03-01 |
Family
ID=40548472
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MA33137A MA32132B1 (fr) | 2008-02-06 | 2010-09-01 | Utilisation de ranolazine pour traiter la douleur |
Country Status (13)
| Country | Link |
|---|---|
| US (1) | US20090203707A1 (fr) |
| EP (1) | EP2252294A1 (fr) |
| KR (1) | KR20110013348A (fr) |
| CN (1) | CN101977605A (fr) |
| AU (1) | AU2009212254A1 (fr) |
| BR (1) | BRPI0908428A2 (fr) |
| CA (1) | CA2713521A1 (fr) |
| CO (1) | CO6290663A2 (fr) |
| EA (1) | EA201070914A1 (fr) |
| EC (1) | ECSP10010446A (fr) |
| IL (1) | IL207292A0 (fr) |
| MA (1) | MA32132B1 (fr) |
| WO (1) | WO2009100380A1 (fr) |
Families Citing this family (26)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US8822473B2 (en) * | 2002-05-21 | 2014-09-02 | Gilead Sciences, Inc. | Method of treating diabetes |
| CN100551370C (zh) * | 2002-05-21 | 2009-10-21 | Cv医药有限公司 | 雷诺嗪在制备治疗糖尿病的药物组合物中的应用 |
| US20090247535A1 (en) * | 2008-03-26 | 2009-10-01 | Duke University | Use of ranolazine for non-cardiovascular disorders |
| CA2761771A1 (fr) * | 2009-05-14 | 2010-11-18 | Gilead Sciences, Inc. | Ranolazine pour le traitement de troubles du snc |
| PT2464645T (pt) * | 2009-07-27 | 2017-10-11 | Gilead Sciences Inc | Compostos heterocíclicos fusionados como moduladores do canal de iões |
| WO2012003392A1 (fr) | 2010-07-02 | 2012-01-05 | Gilead Sciences, Inc. | Composés hétérocycliques condensés en tant que modulateurs des canaux ioniques |
| AU2012253653A1 (en) | 2011-05-10 | 2013-05-02 | Gilead Sciences, Inc. | Fused heterocyclic compounds as sodium channel modulators |
| TWI622583B (zh) | 2011-07-01 | 2018-05-01 | 基利科學股份有限公司 | 作為離子通道調節劑之稠合雜環化合物 |
| NO3175985T3 (fr) | 2011-07-01 | 2018-04-28 | ||
| NZ720651A (en) | 2013-12-19 | 2017-12-22 | Gilead Sciences Inc | Fused heterocyclic compounds as ion channel modulators |
| AU2017228371A1 (en) | 2016-03-04 | 2018-09-13 | Gilead Sciences, Inc. | Compositions and combinations of autotaxin inhibitors |
| WO2018098491A1 (fr) | 2016-11-28 | 2018-05-31 | Praxis Precision Medicines, Inc. | Composés et procédés d'utilisation desdits composés |
| WO2018098499A1 (fr) | 2016-11-28 | 2018-05-31 | Praxis Precision Medicines, Inc. | Composés et procédés d'utilisation desdits composés |
| WO2018148745A1 (fr) | 2017-02-13 | 2018-08-16 | Praxis Precision Medicines , Inc. | Composés et leurs méthodes d'utilisation |
| US11731966B2 (en) | 2017-04-04 | 2023-08-22 | Praxis Precision Medicines, Inc. | Compounds and their methods of use |
| WO2019035951A1 (fr) | 2017-08-15 | 2019-02-21 | Praxis Precision Medicines, Inc. | Composés et leurs méthodes d'utilisation |
| IL309843B2 (en) | 2018-05-30 | 2026-05-01 | Praxis Prec Medicines Inc | History of [4,2,1]triazolo[3,4-a]pyridines and their use as sodium ion channel modulators |
| EA202092908A1 (ru) | 2018-09-28 | 2021-05-14 | Праксис Пресижн Медсинз, Инк. | Модуляторы ионных каналов |
| US11773099B2 (en) | 2019-05-28 | 2023-10-03 | Praxis Precision Medicines, Inc. | Compounds and their methods of use |
| US11505554B2 (en) | 2019-05-31 | 2022-11-22 | Praxis Precision Medicines, Inc. | Substituted pyridines as ion channel modulators |
| US11279700B2 (en) | 2019-05-31 | 2022-03-22 | Praxis Precision Medicines, Inc. | Ion channel modulators |
| AU2020394421A1 (en) | 2019-11-26 | 2022-06-09 | Praxis Precision Medicines, Inc. | Ion channel modulators |
| AU2020392128A1 (en) | 2019-11-27 | 2022-06-09 | Praxis Precision Medicines, Inc. | Formulations of ion channel modulators and methods of preparation and use of ion channel modulators |
| US12533341B2 (en) | 2019-12-11 | 2026-01-27 | Duke University | Small molecule inhibitors of voltage-gated sodium channel 1.7 and methods of using same |
| CA3250706A1 (fr) | 2022-04-26 | 2023-11-02 | Praxis Precision Medicines, Inc. | Traitement de troubles neurologiques |
| WO2025252860A1 (fr) * | 2024-06-04 | 2025-12-11 | Celex Oncology Innovations Limited | Énantiomère de la ranolazine pour utilisation dans le traitement du cancer |
Family Cites Families (17)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4657264A (en) * | 1985-11-01 | 1987-04-14 | Ingersoll-Rand Company | Fluid seal assembly with segmented sub-assembly |
| DK0407780T3 (da) * | 1989-06-23 | 1996-09-30 | Syntex Inc | Ranolazin og beslægtede piperaziner til anvendelse i behandling af væv, der har været udsat for fysisk eller kemisk skade |
| US5455045A (en) * | 1993-05-13 | 1995-10-03 | Syntex (U.S.A.) Inc. | High dose formulations |
| US6303607B1 (en) * | 1998-09-10 | 2001-10-16 | Cv Therapeutics, Inc. | Method for administering a sustained release ranolanolazine formulation |
| US6479496B1 (en) * | 1998-09-10 | 2002-11-12 | Cv Therapeutics, Inc. | Methods for treating angina with ranolazine |
| EP1259230A2 (fr) * | 2000-02-18 | 2002-11-27 | Cv Therapeutics, Inc. | Inhibiteurs partiels de l'oxydation d'acides gras pour le traitement de l'insuffisance cardiaque globale |
| US20030220344A1 (en) * | 2002-04-04 | 2003-11-27 | Luiz Belardinelli | Method of treating arrhythmias |
| US8822473B2 (en) * | 2002-05-21 | 2014-09-02 | Gilead Sciences, Inc. | Method of treating diabetes |
| CN100551370C (zh) * | 2002-05-21 | 2009-10-21 | Cv医药有限公司 | 雷诺嗪在制备治疗糖尿病的药物组合物中的应用 |
| JP2008526879A (ja) * | 2005-01-06 | 2008-07-24 | シーブイ・セラピューティクス・インコーポレイテッド | ラノラジンを含有する徐放性薬学的処方物 |
| AU2006318447A1 (en) * | 2005-11-21 | 2007-05-31 | The Board Of Trustees Of The University Of Alabama For And On Behalf Of The University Of Alabama | Methods of using small molecule compounds for neuroprotection |
| CA2653056A1 (fr) * | 2006-07-27 | 2008-01-31 | Cv Therapeutics, Inc. | Inhibiteurs d'aldh-2 utilises pour le traitement d'une accoutumance |
| CA2678515A1 (fr) * | 2007-02-13 | 2008-08-21 | Cv Therapeutics, Inc. | Utilisation de la ranolazine dans le traitement des maladies cardiovasculaires |
| JP2010518170A (ja) * | 2007-02-13 | 2010-05-27 | ギリアード・パロ・アルト・インコーポレイテッド | 冠微小血管疾患の処置のためのラノラジンの使用 |
| EP2129665A1 (fr) * | 2007-04-05 | 2009-12-09 | CV Therapeutics Inc. | Dérivés de quinazolinone en tant qu'inhibiteurs de l'aldh-2 |
| BRPI0810171A2 (pt) * | 2007-04-12 | 2014-12-30 | Cv Therapeutics Inc | Método para o aumento da secreção de insulina |
| US20090124672A1 (en) * | 2007-11-06 | 2009-05-14 | Ivan Diamond | Aldh-2 inhibitors in the treatment of psychiatric disorders |
-
2009
- 2009-02-06 KR KR1020107019622A patent/KR20110013348A/ko not_active Withdrawn
- 2009-02-06 CA CA2713521A patent/CA2713521A1/fr not_active Abandoned
- 2009-02-06 AU AU2009212254A patent/AU2009212254A1/en not_active Abandoned
- 2009-02-06 EP EP09707821A patent/EP2252294A1/fr not_active Withdrawn
- 2009-02-06 US US12/367,403 patent/US20090203707A1/en not_active Abandoned
- 2009-02-06 CN CN2009801040287A patent/CN101977605A/zh active Pending
- 2009-02-06 EA EA201070914A patent/EA201070914A1/ru unknown
- 2009-02-06 BR BRPI0908428A patent/BRPI0908428A2/pt not_active Application Discontinuation
- 2009-02-06 WO PCT/US2009/033464 patent/WO2009100380A1/fr not_active Ceased
-
2010
- 2010-07-29 IL IL207292A patent/IL207292A0/en unknown
- 2010-08-13 CO CO10099978A patent/CO6290663A2/es not_active Application Discontinuation
- 2010-09-01 MA MA33137A patent/MA32132B1/fr unknown
- 2010-09-03 EC EC2010010446A patent/ECSP10010446A/es unknown
Also Published As
| Publication number | Publication date |
|---|---|
| CN101977605A (zh) | 2011-02-16 |
| BRPI0908428A2 (pt) | 2015-12-08 |
| KR20110013348A (ko) | 2011-02-09 |
| CA2713521A1 (fr) | 2009-08-13 |
| US20090203707A1 (en) | 2009-08-13 |
| AU2009212254A1 (en) | 2009-08-13 |
| EP2252294A1 (fr) | 2010-11-24 |
| ECSP10010446A (es) | 2010-10-30 |
| EA201070914A1 (ru) | 2011-04-29 |
| CO6290663A2 (es) | 2011-06-20 |
| WO2009100380A1 (fr) | 2009-08-13 |
| IL207292A0 (en) | 2010-12-30 |
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