MA47504A - Composés et méthodes de traitement de l'angiocholite biliaire primitive - Google Patents

Composés et méthodes de traitement de l'angiocholite biliaire primitive

Info

Publication number
MA47504A
MA47504A MA047504A MA47504A MA47504A MA 47504 A MA47504 A MA 47504A MA 047504 A MA047504 A MA 047504A MA 47504 A MA47504 A MA 47504A MA 47504 A MA47504 A MA 47504A
Authority
MA
Morocco
Prior art keywords
angiocholitis
compounds
treatment methods
biliary
primitive
Prior art date
Application number
MA047504A
Other languages
English (en)
Inventor
Ronald J Christopher
Robert Mark Jones
Cheryl Geraldine Lassen
Que Liu
Original Assignee
Arena Pharm Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Arena Pharm Inc filed Critical Arena Pharm Inc
Publication of MA47504A publication Critical patent/MA47504A/fr

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/403—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
    • A61K31/404—Indoles, e.g. pindolol
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K2300/00—Mixtures or combinations of active ingredients, wherein at least one active ingredient is fully defined in groups A61K31/00 - A61K41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/575—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of three or more carbon atoms, e.g. cholane, cholestane, ergosterol, sitosterol

Landscapes

  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Organic Chemistry (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
MA047504A 2017-02-16 2018-02-16 Composés et méthodes de traitement de l'angiocholite biliaire primitive MA47504A (fr)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201762459916P 2017-02-16 2017-02-16
US201762502129P 2017-05-05 2017-05-05
US201762506906P 2017-05-16 2017-05-16

Publications (1)

Publication Number Publication Date
MA47504A true MA47504A (fr) 2019-12-25

Family

ID=61873875

Family Applications (1)

Application Number Title Priority Date Filing Date
MA047504A MA47504A (fr) 2017-02-16 2018-02-16 Composés et méthodes de traitement de l'angiocholite biliaire primitive

Country Status (10)

Country Link
US (2) US11534424B2 (fr)
EP (1) EP3582772A1 (fr)
JP (1) JP2020507611A (fr)
KR (1) KR20190116416A (fr)
CN (1) CN110520124A (fr)
AU (1) AU2018220521A1 (fr)
CA (1) CA3053418A1 (fr)
MA (1) MA47504A (fr)
MX (1) MX2019009841A (fr)
WO (1) WO2018151873A1 (fr)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN108558740B (zh) 2010-01-27 2021-10-19 艾尼纳制药公司 S1p1受体调节剂及其盐的制备方法
PL3242666T3 (pl) 2015-01-06 2025-02-17 Arena Pharmaceuticals, Inc. Związek do zastosowania w leczeniu dolegliwości związanych z receptorem s1p1
HUE060476T2 (hu) * 2015-06-22 2023-03-28 Arena Pharm Inc (R)-2-(7-(4-ciklopentil-3-(trifluormetil)benziloxi)-1,2,3,4- tetrahidrociklopenta[B]indol-3-il)ecetsav kristályos L-arginin-sója S1P1 receptorral kapcsolatos rendellenességek esetén való alkalmazásra
WO2018151873A1 (fr) 2017-02-16 2018-08-23 Arena Pharmaceuticals, Inc. Composés et méthodes de traitement de l'angiocholite biliaire primitive
CN110545848A (zh) 2017-02-16 2019-12-06 艾尼纳制药公司 用于治疗具有肠外表现的炎症性肠病的化合物和方法
US12156866B2 (en) * 2018-06-06 2024-12-03 Arena Pharmaceuticals, Inc. Methods of treating conditions related to the S1P1 receptor
WO2020072824A1 (fr) * 2018-10-03 2020-04-09 Arena Pharmaceuticals, Inc. Méthodes pour le traitement des troubles de la sclérodermie
CA3120706A1 (fr) * 2018-11-30 2020-06-04 Arena Pharmaceuticals, Inc. Methodes de traitement d'etats lies au recepteur s1p1
AU2021205465A1 (en) * 2020-01-06 2022-07-14 Arena Pharmaceuticals, Inc. Methods of treating conditions related to the S1P1 receptor
JP2023513670A (ja) * 2020-02-10 2023-04-03 ジェンフィット エラフィブラノールを用いた原発性胆汁性胆管炎の治療
WO2025177319A2 (fr) * 2024-02-22 2025-08-28 Msn Laboratories Private Limited, R&D Center Formes à l'état solide de l-arginine, (3r)-7-[[4-cyclopentyl-3-(trifluorométhyl)phényl]méthoxy]-1,2,3,4-tétrahydrocyclopent[b]indole-3-acétate et leurs procédés de préparation

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US11534424B2 (en) 2022-12-27
WO2018151873A1 (fr) 2018-08-23
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MX2019009841A (es) 2020-01-30
CA3053418A1 (fr) 2018-08-23
US20200000770A1 (en) 2020-01-02
JP2020507611A (ja) 2020-03-12
KR20190116416A (ko) 2019-10-14
US20230149353A1 (en) 2023-05-18
CN110520124A (zh) 2019-11-29

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