MA51611A - Inhibiteurs de pi4kiiibêta - Google Patents

Inhibiteurs de pi4kiiibêta

Info

Publication number
MA51611A
MA51611A MA051611A MA51611A MA51611A MA 51611 A MA51611 A MA 51611A MA 051611 A MA051611 A MA 051611A MA 51611 A MA51611 A MA 51611A MA 51611 A MA51611 A MA 51611A
Authority
MA
Morocco
Prior art keywords
inhibitors
Prior art date
Application number
MA051611A
Other languages
English (en)
Inventor
Nicholas Paul Barton
Sophie Marie Bertrand
Kenneth Down
Matthew Gray
Original Assignee
Glaxosmithkline Ip Dev Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GBGB1800734.4A external-priority patent/GB201800734D0/en
Priority claimed from GBGB1817616.4A external-priority patent/GB201817616D0/en
Application filed by Glaxosmithkline Ip Dev Ltd filed Critical Glaxosmithkline Ip Dev Ltd
Publication of MA51611A publication Critical patent/MA51611A/fr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/02—Nasal agents, e.g. decongestants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/06—Antiasthmatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/16—Otologicals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • A61P31/16—Antivirals for RNA viruses for influenza or rhinoviruses
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
    • Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
    • Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Virology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pulmonology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Molecular Biology (AREA)
  • Cardiology (AREA)
  • Epidemiology (AREA)
  • Hospice & Palliative Care (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Otolaryngology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
MA051611A 2018-01-17 2019-01-15 Inhibiteurs de pi4kiiibêta MA51611A (fr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB1800734.4A GB201800734D0 (en) 2018-01-17 2018-01-17 Novel compounds
GBGB1817616.4A GB201817616D0 (en) 2018-10-29 2018-10-29 Novel compounds

Publications (1)

Publication Number Publication Date
MA51611A true MA51611A (fr) 2021-04-21

Family

ID=65033598

Family Applications (1)

Application Number Title Priority Date Filing Date
MA051611A MA51611A (fr) 2018-01-17 2019-01-15 Inhibiteurs de pi4kiiibêta

Country Status (19)

Country Link
US (3) US11649238B2 (fr)
EP (1) EP3740489A1 (fr)
JP (2) JP7133023B2 (fr)
KR (1) KR102523513B1 (fr)
CN (2) CN111868063B (fr)
AR (1) AR114082A1 (fr)
AU (1) AU2019208416B2 (fr)
BR (1) BR112020014431A2 (fr)
CA (1) CA3088347A1 (fr)
CL (1) CL2020001875A1 (fr)
CO (1) CO2020008887A2 (fr)
IL (1) IL276013B2 (fr)
MA (1) MA51611A (fr)
MX (1) MX2020007521A (fr)
PH (1) PH12020551034A1 (fr)
SG (1) SG11202006453SA (fr)
TW (1) TWI795510B (fr)
UY (1) UY38051A (fr)
WO (1) WO2019141694A1 (fr)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SG11202006453SA (en) * 2018-01-17 2020-08-28 Glaxosmithkline Ip Dev Ltd Pi4kiiibeta inhibitors
AU2020315192A1 (en) 2019-07-17 2022-02-24 2692372 Ontario, Inc. Benzenesulfonamide derivatives and uses thereof
EP4125919A1 (fr) 2020-03-26 2023-02-08 GlaxoSmithKline Intellectual Property Development Limited Inhibiteurs de cathepsine pour la prévention ou le traitement d'infections virales
GB2617477A (en) 2020-11-20 2023-10-11 2692372 Ontario Inc Benzenesulfonamide derivatives and uses thereof
JP2024501118A (ja) 2020-11-20 2024-01-11 ２６９２３７２ オンタリオ，インク． Ｋｒａｓ修飾のための方法および組成物
WO2026013001A1 (fr) 2024-07-10 2026-01-15 Glaxosmithkline Intellectual Property Development Limited Compositions d'inhibiteur de phosphatidylinositol 4-kinase bêta pour le traitement d'une infection par le rhinovirus humain

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Also Published As

Publication number Publication date
BR112020014431A2 (pt) 2020-12-01
CN117069728A (zh) 2023-11-17
CN117069728B (zh) 2025-08-29
AR114082A1 (es) 2020-07-22
KR102523513B1 (ko) 2023-04-18
MX2020007521A (es) 2022-12-05
US20210387988A1 (en) 2021-12-16
CN111868063B (zh) 2023-08-01
US20240336618A1 (en) 2024-10-10
US20230124394A1 (en) 2023-04-20
RU2020123034A (ru) 2022-02-17
JP2022172223A (ja) 2022-11-15
KR20200109343A (ko) 2020-09-22
EP3740489A1 (fr) 2020-11-25
UY38051A (es) 2019-08-30
NZ765884A (en) 2024-10-25
JP7133023B2 (ja) 2022-09-07
AU2019208416A1 (en) 2020-07-23
CA3088347A1 (fr) 2019-07-25
US11649238B2 (en) 2023-05-16
IL276013A (en) 2020-08-31
CO2020008887A2 (es) 2020-07-31
WO2019141694A1 (fr) 2019-07-25
PH12020551034A1 (en) 2021-09-06
SG11202006453SA (en) 2020-08-28
TWI795510B (zh) 2023-03-11
CL2020001875A1 (es) 2021-02-12
IL276013B1 (en) 2023-11-01
CN111868063A (zh) 2020-10-30
TW201940173A (zh) 2019-10-16
AU2019208416B2 (en) 2021-07-29
IL276013B2 (en) 2024-03-01
JP7338017B2 (ja) 2023-09-04
JP2021510711A (ja) 2021-04-30

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