MA55142A - Amino-triazolopyrimidine et amino-triazolopyrazine substitués antagoniste du récepteur de l'adénosine, compositions pharmaceutiques et leur utilisation - Google Patents
Amino-triazolopyrimidine et amino-triazolopyrazine substitués antagoniste du récepteur de l'adénosine, compositions pharmaceutiques et leur utilisationInfo
- Publication number
- MA55142A MA55142A MA055142A MA55142A MA55142A MA 55142 A MA55142 A MA 55142A MA 055142 A MA055142 A MA 055142A MA 55142 A MA55142 A MA 55142A MA 55142 A MA55142 A MA 55142A
- Authority
- MA
- Morocco
- Prior art keywords
- amino
- triazolopyrazine
- triazolopyrimidine
- pharmaceutical compositions
- receptor antagonist
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/4985—Pyrazines or piperazines ortho- or peri-condensed with heterocyclic ring systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K16/00—Immunoglobulins [IG], e.g. monoclonal or polyclonal antibodies
- C07K16/18—Immunoglobulins [IG], e.g. monoclonal or polyclonal antibodies against material from animals or humans
- C07K16/28—Immunoglobulins [IG], e.g. monoclonal or polyclonal antibodies against material from animals or humans against receptors, cell surface antigens or cell surface determinants
- C07K16/2803—Immunoglobulins [IG], e.g. monoclonal or polyclonal antibodies against material from animals or humans against receptors, cell surface antigens or cell surface determinants against the immunoglobulin superfamily
- C07K16/2818—Immunoglobulins [IG], e.g. monoclonal or polyclonal antibodies against material from animals or humans against receptors, cell surface antigens or cell surface determinants against the immunoglobulin superfamily against CD28 or CD152
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K39/00—Medicinal preparations containing antigens or antibodies
- A61K2039/505—Medicinal preparations containing antigens or antibodies comprising antibodies
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K2300/00—Mixtures or combinations of active ingredients, wherein at least one active ingredient is fully defined in groups A61K31/00 - A61K41/00
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Animal Behavior & Ethology (AREA)
- Epidemiology (AREA)
- Immunology (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Molecular Biology (AREA)
- Genetics & Genomics (AREA)
- Biophysics (AREA)
- Biochemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201862769843P | 2018-11-20 | 2018-11-20 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| MA55142A true MA55142A (fr) | 2022-02-23 |
Family
ID=70774154
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MA055142A MA55142A (fr) | 2018-11-20 | 2019-11-15 | Amino-triazolopyrimidine et amino-triazolopyrazine substitués antagoniste du récepteur de l'adénosine, compositions pharmaceutiques et leur utilisation |
Country Status (11)
| Country | Link |
|---|---|
| US (2) | US12466831B2 (fr) |
| EP (1) | EP3883575B1 (fr) |
| JP (1) | JP2022507734A (fr) |
| KR (1) | KR20210093964A (fr) |
| CN (1) | CN113015530A (fr) |
| AU (1) | AU2019383948A1 (fr) |
| BR (1) | BR112021009078A8 (fr) |
| CA (1) | CA3119774A1 (fr) |
| MA (1) | MA55142A (fr) |
| MX (1) | MX2021005839A (fr) |
| WO (1) | WO2020106558A1 (fr) |
Families Citing this family (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2020106560A1 (fr) | 2018-11-20 | 2020-05-28 | Merck Sharp & Dohme Corp. | Composés amino-triazolopyrimidine et amino-triazolopyrazine substitués utilisés en tant qu'antagonistes de récepteur de l'adénosine, compositions pharmaceutiques et leur utilisation |
| WO2020106558A1 (fr) | 2018-11-20 | 2020-05-28 | Merck Sharp & Dohme Corp. | Amino-triazolopyrimidine et amino-triazolopyrazine substitués antagoniste du récepteur de l'adénosine, compositions pharmaceutiques et leur utilisation |
| CR20210271A (es) | 2018-11-30 | 2021-07-14 | Merck Sharp & Dohme | Derivados de amino triazolo quinazolina 9-sustituidos como antagonistas del receptor de adenosina, composiciones farmacéuticas y su uso |
| JP2022511778A (ja) | 2018-11-30 | 2022-02-01 | メルク・シャープ・アンド・ドーム・コーポレーション | アデノシン受容体拮抗薬としての7-、8-及び10-置換されたアミノトリアゾロキナゾリン誘導体、医薬組成物及びそれらの使用 |
| MX2022002219A (es) * | 2019-08-26 | 2022-06-14 | Incyte Corp | Triazolopirimidinas como inhibidores de a2a/a2b. |
| KR102863028B1 (ko) * | 2021-04-23 | 2025-09-22 | 주식회사 종근당 | 아데노신 A2a 수용체 길항제로서의 화합물 및 이를 포함하는 약학적 조성물 |
| KR20250004779A (ko) | 2022-04-13 | 2025-01-08 | 길리애드 사이언시즈, 인코포레이티드 | Trop-2 발현 암을 치료하기 위한 병용 요법 |
| WO2025137640A1 (fr) | 2023-12-22 | 2025-06-26 | Gilead Sciences, Inc. | Inhibiteurs azaspiro de wrn |
Family Cites Families (52)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB9524395D0 (en) | 1995-11-29 | 1996-01-31 | Nickerson Biocem Ltd | Promoters |
| CA2284737C (fr) | 1997-03-24 | 2007-03-13 | Kyowa Hakko Kogyo Co., Ltd. | Derives [1,2,4]triazolo[1,5-c]pyrimidiniques |
| US6759759B2 (en) | 2000-08-29 | 2004-07-06 | Tamagawa Seiki Kabushiki Kaisha | Rotary contactless connector and non-rotary contactless connector |
| US20040110826A1 (en) * | 2001-09-28 | 2004-06-10 | Noriaki Uesaka | Receptor Antagonists |
| AR037243A1 (es) | 2001-10-15 | 2004-11-03 | Schering Corp | Antagonistas del receptor de adenosina a2a,a5-amino-imidazolo-[4,3-e]-1,2,4-triazolo-[1,5-c]pirimidina, composiciones farmaceuticas y el uso de dichos compuestos para la preparacion de un medicamento |
| US6916811B2 (en) | 2001-11-30 | 2005-07-12 | Schering Corporation | Adenosine A2a receptor antagonists |
| TW200300686A (en) | 2001-11-30 | 2003-06-16 | Schering Corp | Adenosine A2a receptor antagonists |
| JPWO2003068776A1 (ja) | 2002-02-15 | 2005-06-02 | 協和醗酵工業株式会社 | [1,2,4]トリアゾロ[1,5−c]ピリミジン誘導体 |
| PT1537878E (pt) | 2002-07-03 | 2010-11-18 | Ono Pharmaceutical Co | Composições de imunopotenciação |
| AU2003272886A1 (en) | 2002-09-24 | 2004-04-19 | Kyowa Hakko Kogyo Co., Ltd. | (1,2,4)-TRIAZOLO(1,5-c)PYRIMIDINE DERIVATIVE |
| WO2004056875A1 (fr) | 2002-12-23 | 2004-07-08 | Wyeth | Anticorps anti pd-1 et utilisations |
| WO2004072286A1 (fr) | 2003-01-23 | 2004-08-26 | Ono Pharmaceutical Co., Ltd. | Substance specifique a pd-1 humain |
| WO2004092177A1 (fr) * | 2003-04-09 | 2004-10-28 | Biogen Idec Ma Inc. | Triazolopyrazines et procedes de preparation et d'utilisation ce celles-ci |
| PT1678182E (pt) | 2003-10-28 | 2007-04-30 | Schering Corp | Processo para preparar 5-amino-pirazolo-[4,3-e]-1,2,4-triazolo[1,5-c]pirimidinas |
| KR20060135901A (ko) | 2004-04-21 | 2006-12-29 | 쉐링 코포레이션 | 피라졸로-[4,3-e]-1,2,4-트리아졸로-[1,5-c]피리미딘아데노신 A2a 수용체 길항제 |
| US7472383B2 (en) | 2004-08-13 | 2008-12-30 | Sun Microsystems, Inc. | System and method for providing exceptional flow control in protected code through memory layers |
| EP1836205B1 (fr) | 2004-12-21 | 2009-06-10 | Schering Corporation | ANTAGONISTES DE RECEPTEUR A2a DE PYRAZOLO [1,5-A]PYRIMIDINE ADENOSINE |
| PL2161336T5 (pl) | 2005-05-09 | 2017-10-31 | Ono Pharmaceutical Co | Ludzkie przeciwciała monoklonalne przeciwko białku Programmed Death 1 (PD-1) oraz sposoby leczenia raka z zastosowaniem samych przeciwciał anty-PD-1 lub w połączeniu z innymi środkami immunoterapeutycznymi |
| CA2612241C (fr) | 2005-07-01 | 2018-11-06 | Medarex, Inc. | Anticorps monoclonaux humains diriges contre un ligand de mort programmee de type 1(pd-l1) |
| CA2622741A1 (fr) | 2005-09-19 | 2007-03-29 | Schering Corporation | 2-heteroaryl-pyrazolo-[4, 3-e]-1, 2, 4-triazolo-[1,5-c]-pyrimidine en tant qu'antagonistes du recepteur a2a d'adenosine |
| ATE457988T1 (de) | 2006-06-26 | 2010-03-15 | Schering Corp | A2a-adenosin-rezeptor-antagonisten |
| KR101586617B1 (ko) | 2007-06-18 | 2016-01-20 | 머크 샤프 앤 도메 비.브이. | 사람 프로그램된 사멸 수용체 pd-1에 대한 항체 |
| PE20091101A1 (es) | 2007-12-18 | 2009-07-26 | Pharminox Ltd | AMIDAS DE ACIDO 3-SUBSTITUIDO-4-OXO-3,4-DIHIDRO-IMIDAZO[5,1-d] [1,2,3,5-TETRACINA-8-CARBOXILICO Y SU EMPLEO |
| US8415353B2 (en) | 2008-03-04 | 2013-04-09 | Merck Sharp & Dohme Corp. | Amino-quinoxaline and amino-quinoline compounds for use as adenosine A2a receptor antagonists |
| US8168757B2 (en) | 2008-03-12 | 2012-05-01 | Merck Sharp & Dohme Corp. | PD-1 binding proteins |
| DE102008023801A1 (de) | 2008-05-15 | 2009-11-19 | Bayer Schering Pharma Aktiengesellschaft | Substituierte Imidazo- und Triazolopyrimidine, Imidazo- und Pyrazolopyrazine und Imidazotriazine |
| GB0906579D0 (en) * | 2009-04-16 | 2009-05-20 | Vernalis R&D Ltd | Pharmaceuticals, compositions and methods of making and using the same |
| JP2012500652A (ja) | 2008-08-25 | 2012-01-12 | アンプリミューン、インコーポレーテッド | 標的化共刺激ポリペプチドおよび癌を処置するための使用方法 |
| PL2342226T3 (pl) | 2008-09-26 | 2017-01-31 | Dana-Farber Cancer Institute, Inc. | Ludzkie przeciwciała anty-PD-1, PD-L1 i PD-L2 oraz ich zastosowania |
| EP4209510B1 (fr) | 2008-12-09 | 2024-01-31 | F. Hoffmann-La Roche AG | Anticorps anti-pd-l1 et leur utilisation pour améliorer la fonction des lymphocytes t |
| EP2509983B1 (fr) | 2009-11-16 | 2014-09-17 | Merck Sharp & Dohme Corp. | Composés tricycliques condensés possédant une activité antagoniste des récepteurs a2a de l'adénosine |
| US20130017199A1 (en) | 2009-11-24 | 2013-01-17 | AMPLIMMUNE ,Inc. a corporation | Simultaneous inhibition of pd-l1/pd-l2 |
| EP2739358B1 (fr) | 2011-08-01 | 2018-11-28 | F.Hoffmann-La Roche Ag | Procédés de traitement du cancer à l'aide d'antagonistes se liant à l'axe pd-1 et inhibiteurs de mek |
| WO2014101113A1 (fr) | 2012-12-28 | 2014-07-03 | Merck Sharp & Dohme Corp. | Composés de 7-méthoxy-[1,2,4]triazolo[1,5-c]quinazoline-5-amine à substitution pipérazine présentant des propriétés d'antagoniste d'a2a |
| WO2014101120A1 (fr) | 2012-12-28 | 2014-07-03 | Merck Sharp & Dohme Corp. | Composés de 7-méthoxy-[1,2,4]triazolo[1,5-c]quinazoline-5-amine à substitution hétérobicyclo présentant des propriétés d'antagoniste d'a2a |
| WO2015027431A1 (fr) | 2013-08-29 | 2015-03-05 | Merck Sharp & Dohme Corp. | Antagonistes 2,2-difluorodioxolo du récepteur a2a |
| JP6779204B2 (ja) | 2014-11-18 | 2020-11-04 | メルク・シャープ・アンド・ドーム・コーポレーションMerck Sharp & Dohme Corp. | A2a拮抗薬特性を有するアミノピラジン化合物 |
| EP3227299B1 (fr) | 2014-12-04 | 2021-05-26 | Merck Sharp & Dohme Corp. | Formulation inhibant les effets d'un environnement faiblement acide |
| US10138212B2 (en) | 2015-02-06 | 2018-11-27 | Merck Sharp & Dohme Corp. | Aminoquinazoline compounds as A2A antagonist |
| EP3307067B1 (fr) | 2015-06-11 | 2022-11-02 | Merck Sharp & Dohme LLC | Composés d'aminopyrazine ayant des propriétés d'antagoniste a2a |
| US10207002B2 (en) | 2015-06-26 | 2019-02-19 | Merck Sharp & Dohme Corp. | Sustained release formulation and tablets prepared therefrom |
| WO2017008205A1 (fr) | 2015-07-10 | 2017-01-19 | Merck Sharp & Dohme Corp. | Composés d'aminoquinazoline substitués a titre d'antagonistes du récepteur a2a |
| AR108875A1 (es) * | 2016-06-24 | 2018-10-03 | Incyte Corp | COMPUESTOS HETEROCÍCLICOS COMO INHIBIDORES DE PI3K-g |
| JP7065113B2 (ja) | 2017-04-07 | 2022-05-11 | 南京明徳新薬研発有限公司 | A2A受容体阻害剤としての[1,2,4]トリアゾロ[1,5-c]ピリミジン誘導体 |
| CN109535161B (zh) * | 2017-09-22 | 2021-09-03 | 江苏恒瑞医药股份有限公司 | 三唑并嘧啶类衍生物、其制备方法及其在医药上的应用 |
| US11498923B2 (en) | 2017-12-13 | 2022-11-15 | Merck Sharp & Dohme Llc | Substituted imidazo[1,2-c]quinazolines as A2A antagonists |
| BR122023024273A2 (pt) * | 2018-02-27 | 2024-02-20 | Incyte Corporation | Compostos imidazopirimidinas e triazolopirimidinas, seus usos, método para inibir uma atividade de um receptor de adenosina e composição farmacêutica dos mesmos |
| AU2019297361B2 (en) | 2018-07-05 | 2024-06-27 | Incyte Corporation | Fused pyrazine derivatives as A2A / A2B inhibitors |
| WO2020106560A1 (fr) | 2018-11-20 | 2020-05-28 | Merck Sharp & Dohme Corp. | Composés amino-triazolopyrimidine et amino-triazolopyrazine substitués utilisés en tant qu'antagonistes de récepteur de l'adénosine, compositions pharmaceutiques et leur utilisation |
| WO2020106558A1 (fr) | 2018-11-20 | 2020-05-28 | Merck Sharp & Dohme Corp. | Amino-triazolopyrimidine et amino-triazolopyrazine substitués antagoniste du récepteur de l'adénosine, compositions pharmaceutiques et leur utilisation |
| CR20210271A (es) | 2018-11-30 | 2021-07-14 | Merck Sharp & Dohme | Derivados de amino triazolo quinazolina 9-sustituidos como antagonistas del receptor de adenosina, composiciones farmacéuticas y su uso |
| JP2022511778A (ja) | 2018-11-30 | 2022-02-01 | メルク・シャープ・アンド・ドーム・コーポレーション | アデノシン受容体拮抗薬としての7-、8-及び10-置換されたアミノトリアゾロキナゾリン誘導体、医薬組成物及びそれらの使用 |
-
2019
- 2019-11-15 WO PCT/US2019/061622 patent/WO2020106558A1/fr not_active Ceased
- 2019-11-15 AU AU2019383948A patent/AU2019383948A1/en not_active Abandoned
- 2019-11-15 MA MA055142A patent/MA55142A/fr unknown
- 2019-11-15 US US17/292,511 patent/US12466831B2/en active Active
- 2019-11-15 KR KR1020217018498A patent/KR20210093964A/ko not_active Withdrawn
- 2019-11-15 EP EP19886307.8A patent/EP3883575B1/fr active Active
- 2019-11-15 JP JP2021527186A patent/JP2022507734A/ja active Pending
- 2019-11-15 BR BR112021009078A patent/BR112021009078A8/pt not_active Application Discontinuation
- 2019-11-15 CA CA3119774A patent/CA3119774A1/fr active Pending
- 2019-11-15 CN CN201980076511.2A patent/CN113015530A/zh active Pending
- 2019-11-15 MX MX2021005839A patent/MX2021005839A/es unknown
-
2025
- 2025-08-18 US US19/302,594 patent/US20250382300A1/en active Pending
Also Published As
| Publication number | Publication date |
|---|---|
| US20210395255A1 (en) | 2021-12-23 |
| CN113015530A (zh) | 2021-06-22 |
| EP3883575A1 (fr) | 2021-09-29 |
| AU2019383948A1 (en) | 2021-05-20 |
| KR20210093964A (ko) | 2021-07-28 |
| WO2020106558A1 (fr) | 2020-05-28 |
| BR112021009078A8 (pt) | 2023-02-07 |
| EP3883575B1 (fr) | 2025-10-08 |
| US12466831B2 (en) | 2025-11-11 |
| EP3883575A4 (fr) | 2022-06-15 |
| BR112021009078A2 (pt) | 2021-08-10 |
| CA3119774A1 (fr) | 2020-05-28 |
| MX2021005839A (es) | 2021-07-15 |
| US20250382300A1 (en) | 2025-12-18 |
| JP2022507734A (ja) | 2022-01-18 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| EP3883575A4 (fr) | Amino-triazolopyrimidine et amino-triazolopyrazine substitués antagoniste du récepteur de l'adénosine, compositions pharmaceutiques et leur utilisation | |
| IL304521A (en) | GPCR receptor agonists, pharmaceutical preparations containing them and methods of using them | |
| MA54298A (fr) | Dérivés amino triazolo quinazoline 9-substitués utiles en tant qu'antagonistes du récepteur de l'adénosine, compositions pharmaceutiques et leur utilisation | |
| MA49753A (fr) | Agents de liaison se liant à pd-l1 et cd137 et leur utilisation | |
| EP3883576A4 (fr) | Composés amino-triazolopyrimidine et amino-triazolopyrazine substitués utilisés en tant qu'antagonistes de récepteur de l'adénosine, compositions pharmaceutiques et leur utilisation | |
| MA52245A (fr) | Promédicaments d'antagonistes de c5ar bicycliques fusionnés | |
| LT3762380T (lt) | Fenilpirolidinono formilpeptido 2 receptoriaus antagonistai | |
| IL283712A (en) | Crf1 receptor antagonist, pharmaceutical formulations and solid forms thereof for the treatment of congenital adrenal hyperplasia | |
| EP4039705A4 (fr) | Anticorps ciblant bcma, anticorps bispécifique et leur utilisation | |
| EP3802500A4 (fr) | Antagonistes du récepteur de la mélanocortine de sous-type 2 (mc2r) et leurs utilisations | |
| EP3450460A4 (fr) | Conjugué de liaison multi-spécifique, compositions pharmaceutiques associées et utilisation | |
| HUE067014T2 (hu) | Szolúbilis 1-es típusú komplementreceptor variánsai és alkalmazásuk | |
| EP3887377A4 (fr) | Dérivés d'amino triazolo quinazoline à substitution en positions 7, 8 et 10 utilisés en tant qu'antagonistes du récepteur de l'adénosine, compositions pharmaceutiques et leur utilisation | |
| EP3860977A4 (fr) | Antagonistes de l'intégrine | |
| EP3770148A4 (fr) | Inhibiteur de récepteur, composition pharmaceutique le comprenant et son utilisation | |
| EP3845528A4 (fr) | Composés de pyrazole, compositions pharmaceutiques correspondantes et utilisation associées | |
| EP3946315A4 (fr) | Compositions de cannabinoïdes et leur utilisation | |
| EP3762386A4 (fr) | Antagonistes du récepteur de l'adénosine et leurs utilisations | |
| EP3790409A4 (fr) | Compositions comprenant du glucose et de l'hémicellulose et leur utilisation | |
| MA42527A (fr) | Agonistes de récepteur 5-ht2c et compositions et procédés d'utilisation | |
| EP3715344A4 (fr) | Dérivés de 1,4-benzodiazépine et leur utilisation | |
| EP3897593A4 (fr) | Formulations de cannabinoïdes et compositions pharmaceutiques | |
| MA53218A (fr) | Antagonistes de l'intégrine | |
| EP3664797A4 (fr) | Ligands de nr4a1, compositions pharmaceutiques et procédés d'utilisation associés | |
| EP3773654C0 (fr) | Compositions médicamenteuses polypharmaceutiques et méthodes associées |