MA56032A - Composés, compositions et procédés d'utilisation - Google Patents

Composés, compositions et procédés d'utilisation

Info

Publication number
MA56032A
MA56032A MA056032A MA56032A MA56032A MA 56032 A MA56032 A MA 56032A MA 056032 A MA056032 A MA 056032A MA 56032 A MA56032 A MA 56032A MA 56032 A MA56032 A MA 56032A
Authority
MA
Morocco
Prior art keywords
compositions
compounds
methods
Prior art date
Application number
MA056032A
Other languages
English (en)
Inventor
Allen Taylor Hopper
Daniel La
Steven Mischke
Original Assignee
Sage Therapeutics Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sage Therapeutics Inc filed Critical Sage Therapeutics Inc
Publication of MA56032A publication Critical patent/MA56032A/fr

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/14Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
MA056032A 2019-05-24 2020-05-24 Composés, compositions et procédés d'utilisation MA56032A (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US201962852565P 2019-05-24 2019-05-24

Publications (1)

Publication Number Publication Date
MA56032A true MA56032A (fr) 2022-04-06

Family

ID=71078654

Family Applications (1)

Application Number Title Priority Date Filing Date
MA056032A MA56032A (fr) 2019-05-24 2020-05-24 Composés, compositions et procédés d'utilisation

Country Status (7)

Country Link
US (1) US20220332699A1 (fr)
EP (1) EP3976186A1 (fr)
JP (2) JP7687964B2 (fr)
AR (1) AR119010A1 (fr)
MA (1) MA56032A (fr)
TW (2) TWI855081B (fr)
WO (1) WO2020243027A1 (fr)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FI2753632T3 (fi) 2011-09-08 2023-08-02 Sage Therapeutics Inc Neuroaktiivisia steroideja, koostumuksia ja niiden käyttöjä
SMT202000008T1 (it) 2012-01-23 2020-03-13 Sage Therapeutics Inc Formulazione di steroide neuroattivo comprendente un complesso di allopregnanolone e solfobutil eter beta-ciclodestrina
PL2887944T3 (pl) 2012-08-21 2022-02-21 Sage Therapeutics, Inc. Allopregnanolon do leczenia lekoopornego stanu padaczkowego
CN113527400B (zh) 2013-04-17 2024-06-28 萨奇治疗股份有限公司 19-去甲c3,3-二取代的c21-n-吡唑基类固醇及其使用方法
WO2015195962A1 (fr) 2014-06-18 2015-12-23 Sage Therapeutics, Inc. Stéroïdes neuroactifs, leurs compositions et utilisations
JOP20200195A1 (ar) 2014-09-08 2017-06-16 Sage Therapeutics Inc سترويدات وتركيبات نشطة عصبياً، واستخداماتها
ME03749B (fr) 2014-11-27 2021-04-20 Sage Therapeutics Inc Compositions et procédés pour traiter des troubles du snc
US20190330259A1 (en) 2016-04-01 2019-10-31 Sage Therapeutics, Inc. Oxysterols and methods of use thereof
CN115974956A (zh) 2016-08-23 2023-04-18 萨奇治疗股份有限公司 19-去甲c3,3-二取代的c21-n-吡唑基类固醇的晶体
KR20200096596A (ko) 2017-12-08 2020-08-12 세이지 테라퓨틱스, 인크. Cns 장애의 치료를 위한 중수소화 21 -[4-시아노-피라졸-1 -일]-19-노르-프레간-3. 알파-올-20-온 유도체
AU2022291395A1 (en) 2021-06-11 2024-01-04 Sage Therapeutics, Inc. Neuroactive steroid for the treatment of alzheimer's disease
CN113501787A (zh) * 2021-08-20 2021-10-15 黑龙江省科学院石油化学研究院 一种合成6-三氟甲基-3-甲基吲唑的方法
US20240189312A1 (en) * 2022-12-02 2024-06-13 Morehouse School Of Medicine Composition for treating acute brain injury or neurodegenerative disease, method of making, and use thereof

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5854204A (en) 1995-03-14 1998-12-29 Praecis Pharmaceuticals, Inc. Aβ peptides that modulate β-amyloid aggregation
CA2262453A1 (fr) 1996-08-27 1998-03-05 Praecis Pharmaceuticals Incorporated Modulateurs de l'agregation de peptides beta-amyloides, comprenant des d-aminoacides
AR035016A1 (es) 1999-08-25 2004-04-14 Takeda Chemical Industries Ltd Composicion de azol promotor de produccion/secrecion de neurotrofina, compuesto prodroga del mismo, composicion farmaceutica que lo comprende y uso del mismo para preparar esta ultima.
WO2010068881A1 (fr) * 2008-12-12 2010-06-17 Forest Laboratories Holdings Limited Nouveaux dérivés de benzodioxane et benzoxazine utiles en tant que ligands pour les récepteurs de chimiokine cc
KR101702159B1 (ko) * 2009-09-16 2017-02-02 더 유니버시티 오브 에든버러 (4―페닐―피페리딘―1―일)―[5―(1h―피라졸―4―일)―티오펜―3―일]―메탄온 화합물 및 그의 용도
ES2543692T3 (es) * 2010-04-29 2015-08-21 The University Of Edinburgh (8-aza-biciclo[3.2.1biciclo[oct-8-il)-[5-(1H-pirazol-4-il)-tiofeno-3-il]-metanonas 3,3-disustituidas como inhibidores de 11beta-HSD1
CA2851087C (fr) * 2011-10-07 2019-09-24 Takeda Pharmaceutical Company Limited Composes de 1-arylcarbonyl-4-oxypiperidine utiles pour le traitement de maladies neurodegeneratives
WO2014092100A1 (fr) * 2012-12-11 2014-06-19 武田薬品工業株式会社 Composé hétérocyclique
US9598398B2 (en) * 2013-04-04 2017-03-21 Takeda Pharmaceutical Company Limited Heterocyclic compound
US20230000843A1 (en) * 2019-09-30 2023-01-05 Actinogen Medical Limited Medicinal cognitive treatments

Also Published As

Publication number Publication date
JP2022533436A (ja) 2022-07-22
AR119010A1 (es) 2021-11-17
JP7687964B2 (ja) 2025-06-03
JP2025090698A (ja) 2025-06-17
TW202110824A (zh) 2021-03-16
TW202523658A (zh) 2025-06-16
EP3976186A1 (fr) 2022-04-06
US20220332699A1 (en) 2022-10-20
WO2020243027A1 (fr) 2020-12-03
TWI855081B (zh) 2024-09-11

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