MC1920A1 - Derives acyles - Google Patents

Derives acyles

Info

Publication number
MC1920A1
MC1920A1 MC881967A MC1967A MC1920A1 MC 1920 A1 MC1920 A1 MC 1920A1 MC 881967 A MC881967 A MC 881967A MC 1967 A MC1967 A MC 1967A MC 1920 A1 MC1920 A1 MC 1920A1
Authority
MC
Monaco
Prior art keywords
methyl
compounds
group
hydrogen
formula
Prior art date
Application number
MC881967A
Other languages
English (en)
French (fr)
Inventor
Furlenmeier Andre
Goetschi Erwin
Hebeisen Paul
Hofheinz Werner
Link Helmut
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of MC1920A1 publication Critical patent/MC1920A1/fr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D501/14—Compounds having a nitrogen atom directly attached in position 7
    • C07D501/16—Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
    • C07D501/20—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids
    • C07D501/24—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids with hydrocarbon radicals, substituted by hetero atoms or hetero rings, attached in position 3
    • C07D501/36—Methylene radicals, substituted by sulfur atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D519/00—Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/00 or C07D455/00
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Saccharide Compounds (AREA)
  • Cephalosporin Compounds (AREA)
MC881967A 1987-04-10 1988-04-07 Derives acyles MC1920A1 (fr)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
CH140787 1987-04-10
CH165787 1987-04-30
CH241487 1987-06-26

Publications (1)

Publication Number Publication Date
MC1920A1 true MC1920A1 (fr) 1989-04-06

Family

ID=27172952

Family Applications (1)

Application Number Title Priority Date Filing Date
MC881967A MC1920A1 (fr) 1987-04-10 1988-04-07 Derives acyles

Country Status (15)

Country Link
US (1) US5055572A (pt)
EP (1) EP0286144A3 (pt)
JP (1) JPH01261392A (pt)
KR (1) KR880012611A (pt)
AU (1) AU611428B2 (pt)
DK (1) DK170088A (pt)
FI (1) FI881641A7 (pt)
HU (1) HU201948B (pt)
IL (1) IL85970A0 (pt)
MC (1) MC1920A1 (pt)
NO (1) NO881530L (pt)
NZ (1) NZ224130A (pt)
PH (1) PH24960A (pt)
PT (1) PT87202B (pt)
YU (1) YU70888A (pt)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FI872879A7 (fi) * 1986-07-21 1988-01-22 Sankei Yakuhin Kk --laktamfoerening, foerfarande foer dess framstaellning, denna innehaollande laekemedelskomposition foer behandling av sjukdom med bakterieinfektion samt mellanprodukter foer dess syntes.
FI883320A7 (fi) * 1987-08-07 1989-02-08 Sankei Pharmaceutical Company Ltd --Laktaami, sen valmistus ja välituotteetsen valmistamiseksi
EP0366189A3 (en) * 1988-10-24 1992-01-02 Norwich Eaton Pharmaceuticals, Inc. Novel antimicrobial lactam-quinolones
DE3939533A1 (de) * 1989-11-30 1991-06-06 Bayer Ag Neue cephalosporine, verfahren zu ihrer herstellung und ihre verwendung als arzneimittel
EP0544166A3 (en) * 1991-11-26 1993-11-03 Hoffmann La Roche Cephalosporinderivatives
GB201111705D0 (en) 2011-07-07 2011-08-24 Takeda Pharmaceutical Compounds and their use
JO3115B1 (ar) 2011-08-22 2017-09-20 Takeda Pharmaceuticals Co مركبات بيريدازينون واستخدامها كمثبطات daao
AU2012337781B2 (en) 2011-11-15 2017-07-06 Takeda Pharmaceutical Company Limited Dihydroxy aromatic heterocyclic compound
GB201222711D0 (en) 2012-12-17 2013-01-30 Takeda Pharmaceutical Novel compounds
CN110655526A (zh) * 2018-06-28 2020-01-07 中国科学院上海药物研究所 头孢菌素-铁载体轭合物及其制备方法和用途

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS60142987A (ja) * 1983-12-29 1985-07-29 Mochida Pharmaceut Co Ltd セフアロスポリン誘導体
EP0150507B1 (en) * 1983-12-29 1992-08-05 Mochida Pharmaceutical Co., Ltd. Cephalosporin derivatives, processes for producing the same and compositions containing them
AU586215B2 (en) * 1985-01-21 1989-07-06 Nippon Pharmaceutical Development Institute Company Limited Novel ```-lactam antibiotics
NZ215527A (en) * 1985-04-01 1989-06-28 Mochida Pharm Co Ltd Cephalosporin derivatives and pharmaceutical compositions
FI872879A7 (fi) * 1986-07-21 1988-01-22 Sankei Yakuhin Kk --laktamfoerening, foerfarande foer dess framstaellning, denna innehaollande laekemedelskomposition foer behandling av sjukdom med bakterieinfektion samt mellanprodukter foer dess syntes.
US4880798A (en) * 1986-11-25 1989-11-14 Mochida Pharmaceutical Co., Ltd. Cephalosporin derivatives

Also Published As

Publication number Publication date
EP0286144A3 (de) 1990-10-03
AU1431088A (en) 1988-10-13
NO881530D0 (no) 1988-04-08
NZ224130A (en) 1991-02-26
AU611428B2 (en) 1991-06-13
FI881641A0 (fi) 1988-04-08
DK170088D0 (da) 1988-03-28
IL85970A0 (en) 1988-09-30
NO881530L (no) 1988-10-11
HUT46920A (en) 1988-12-28
PT87202B (pt) 1992-07-31
HU201948B (en) 1991-01-28
JPH01261392A (ja) 1989-10-18
FI881641A7 (fi) 1988-10-11
US5055572A (en) 1991-10-08
EP0286144A2 (de) 1988-10-12
PT87202A (pt) 1988-05-01
DK170088A (da) 1988-10-11
KR880012611A (ko) 1988-11-28
PH24960A (en) 1990-12-26
YU70888A (en) 1989-12-31

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