NL8005346A - 2-amino-3-benzoyl-fenylaceetamiden en cyclische homologen. - Google Patents

2-amino-3-benzoyl-fenylaceetamiden en cyclische homologen. Download PDF

Info

Publication number
NL8005346A
NL8005346A NL8005346A NL8005346A NL8005346A NL 8005346 A NL8005346 A NL 8005346A NL 8005346 A NL8005346 A NL 8005346A NL 8005346 A NL8005346 A NL 8005346A NL 8005346 A NL8005346 A NL 8005346A
Authority
NL
Netherlands
Prior art keywords
amino
compound
benzoyl
phenylacetamide
administered
Prior art date
Application number
NL8005346A
Other languages
English (en)
Dutch (nl)
Inventor
J R Shanklin
D A Shamblee
D A Walsh
Original Assignee
Robins Co Inc A H
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Robins Co Inc A H filed Critical Robins Co Inc A H
Publication of NL8005346A publication Critical patent/NL8005346A/nl

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
    • C07D295/16—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms
    • C07D295/18—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms by radicals derived from carboxylic acids, or sulfur or nitrogen analogues thereof
    • C07D295/182—Radicals derived from carboxylic acids
    • C07D295/185—Radicals derived from carboxylic acids from aliphatic carboxylic acids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pain & Pain Management (AREA)
  • Hematology (AREA)
  • Diabetes (AREA)
  • Rheumatology (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
NL8005346A 1979-09-26 1980-09-25 2-amino-3-benzoyl-fenylaceetamiden en cyclische homologen. NL8005346A (nl)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US7886079A 1979-09-26 1979-09-26
US7886079 1979-09-26

Publications (1)

Publication Number Publication Date
NL8005346A true NL8005346A (nl) 1981-03-30

Family

ID=22146633

Family Applications (1)

Application Number Title Priority Date Filing Date
NL8005346A NL8005346A (nl) 1979-09-26 1980-09-25 2-amino-3-benzoyl-fenylaceetamiden en cyclische homologen.

Country Status (36)

Country Link
JP (1) JPS5657751A (fr)
KR (1) KR840000763B1 (fr)
AT (1) AT374170B (fr)
AU (1) AU532359B2 (fr)
BE (1) BE885393A (fr)
BR (1) BR8006042A (fr)
CA (1) CA1128512A (fr)
CH (1) CH646138A5 (fr)
CS (1) CS227012B2 (fr)
DE (1) DE3035688A1 (fr)
DK (1) DK154136C (fr)
EG (1) EG15020A (fr)
ES (2) ES495329A0 (fr)
FI (1) FI72967C (fr)
FR (1) FR2465710A1 (fr)
GB (1) GB2059963B (fr)
GR (1) GR70049B (fr)
HK (1) HK59383A (fr)
HU (1) HU183215B (fr)
IE (1) IE50268B1 (fr)
IL (1) IL60999A (fr)
IN (3) IN151313B (fr)
IT (1) IT1133823B (fr)
KE (1) KE3307A (fr)
LU (1) LU82797A1 (fr)
MX (1) MX7159E (fr)
NL (1) NL8005346A (fr)
NO (1) NO152128C (fr)
NZ (1) NZ195061A (fr)
PH (1) PH22628A (fr)
PL (1) PL128998B1 (fr)
PT (1) PT71839B (fr)
SE (1) SE448626B (fr)
SG (1) SG42983G (fr)
YU (3) YU41734B (fr)
ZA (1) ZA805476B (fr)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL61945A (en) * 1980-02-19 1984-09-30 Robins Co Inc A H 2-amino-3-(hydroxy(phenyl)methyl)phenylacetic acids,esters and amides and pharmaceutical compositions containing them
US6646001B2 (en) 1997-12-19 2003-11-11 Alcon Manufacturing, Ltd. Use of non-steroidal anti-inflammatory agents in combination with prostaglandin FP receptor agonists to treat glaucoma and ocular hypertension
US6066671A (en) * 1997-12-19 2000-05-23 Alcon Laboratories, Inc. Treatment of GLC1A glaucoma with 3-benzoyl-phenylacetic acids, esters, or amides
GB9727523D0 (en) 1997-12-31 1998-02-25 Pharmacia & Upjohn Spa Alpha-aminoamide derivatives useful as analgesic agents
AR030345A1 (es) * 2000-08-14 2003-08-20 Alcon Inc Metodo de tratamiento de desordenes relacionados con angiogenesis
SI1423168T1 (sl) 2001-09-03 2006-06-30 Newron Pharm Spa Farmacevtski sestavek, ki vsebuje gabapentin ali njegov analog in alfa-aminoamid, in njegova analgetska uporaba
EP1438956A1 (fr) 2003-01-16 2004-07-21 Newron Pharmaceuticals S.p.A. Dérivés alpha-aminoamides en tant qu'agents antimigraine
CZ301776B6 (cs) * 2009-06-08 2010-06-16 Farmak, A.S. Postup prípravy 2-amino-3-benzoylfenylacetamidu (nepafenacu) s minimem vedlejších produktu
CN112794809B (zh) * 2019-11-14 2023-12-29 南京济群医药科技股份有限公司 一种高纯度奈帕芬胺中间体的制备方法

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1226344A (fr) * 1967-07-31 1971-03-24
CH577461A5 (fr) * 1975-08-13 1976-07-15 Robins Co Inc A H
IL61945A (en) * 1980-02-19 1984-09-30 Robins Co Inc A H 2-amino-3-(hydroxy(phenyl)methyl)phenylacetic acids,esters and amides and pharmaceutical compositions containing them

Also Published As

Publication number Publication date
FI72967C (fi) 1987-08-10
KR830004210A (ko) 1983-07-06
BE885393A (fr) 1981-01-16
IN151313B (fr) 1983-03-26
FR2465710A1 (fr) 1981-03-27
PL128998B1 (en) 1984-03-31
YU73083A (en) 1983-12-31
IE50268B1 (en) 1986-03-19
KE3307A (en) 1983-08-19
IT1133823B (it) 1986-07-24
SE8006668L (sv) 1981-03-27
CA1128512A (fr) 1982-07-27
ATA474580A (de) 1983-08-15
DE3035688C2 (fr) 1990-05-17
JPS5657751A (en) 1981-05-20
YU41734B (en) 1987-12-31
EG15020A (en) 1985-03-31
ES8204715A1 (es) 1982-05-01
PL226919A1 (fr) 1982-02-01
NO802834L (no) 1981-03-27
DK154136B (da) 1988-10-17
YU43305B (en) 1989-06-30
IN156255B (fr) 1985-06-08
CS227012B2 (en) 1984-04-16
DE3035688A1 (de) 1981-04-16
ZA805476B (en) 1981-11-25
SE448626B (sv) 1987-03-09
AU6211680A (en) 1981-04-02
AT374170B (de) 1984-03-26
ES8200329A1 (es) 1981-10-16
AU532359B2 (en) 1983-09-29
NO152128C (no) 1985-08-07
NZ195061A (en) 1984-04-27
PT71839B (en) 1981-06-25
YU73183A (en) 1983-12-31
MX7159E (es) 1987-12-02
FR2465710B1 (fr) 1984-10-12
YU245080A (en) 1983-09-30
HU183215B (en) 1984-04-28
IT8024948A0 (it) 1980-09-26
JPH0141616B2 (fr) 1989-09-06
PH22628A (en) 1988-10-28
BR8006042A (pt) 1981-04-07
IL60999A (en) 1984-05-31
LU82797A1 (fr) 1982-05-10
CH646138A5 (fr) 1984-11-15
YU43306B (en) 1989-06-30
IN156254B (fr) 1985-06-08
HK59383A (en) 1983-12-02
IL60999A0 (en) 1980-11-30
NO152128B (no) 1985-04-29
IE801946L (en) 1981-03-26
ES503019A0 (es) 1982-05-01
DK405780A (da) 1981-03-27
SG42983G (en) 1985-01-11
FI72967B (fi) 1987-04-30
GB2059963A (en) 1981-04-29
ES495329A0 (es) 1981-10-16
DK154136C (da) 1989-03-06
GR70049B (fr) 1982-07-26
FI803002A7 (fi) 1981-03-27
KR840000763B1 (ko) 1984-06-08
PT71839A (en) 1980-10-01
GB2059963B (en) 1983-04-20

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Legal Events

Date Code Title Description
A85 Still pending on 85-01-01
BA A request for search or an international-type search has been filed
BB A search report has been drawn up
BC A request for examination has been filed
BV The patent application has lapsed