NO20002214L - FremgangsmÕte for syntese av pyrrolaminer - Google Patents

FremgangsmÕte for syntese av pyrrolaminer

Info

Publication number: NO20002214L
Authority: NO; Norway
Prior art keywords: reaction; pyrrolamines; synthesis; followed; cycloakane
Prior art date: 1997-11-13

Application number

NO20002214A

Other languages

English (en)

Norwegian (no)

Other versions

NO20002214D0 (no

Inventor

John Anthony Ragan

Teresa Woodall Makowski

David Jon Am Ende

Pamela Jane Clifford

Gregory Randall Young

Alyson Kay Conrad

Shane Allen Eisenbeis

Douglas John Meldrum Allen

George Joseph Quallich

Original Assignee

Pfizer Prod Inc

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1997-11-13

Filing date

2000-04-28

Publication date

2000-05-12

2000-04-28 Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc

2000-04-28 Publication of NO20002214D0 publication Critical patent/NO20002214D0/no

2000-05-12 Publication of NO20002214L publication Critical patent/NO20002214L/no

Links

238000000034 method Methods 0.000 title abstract 2
QLSWIGRIBOSFMV-UHFFFAOYSA-N 1h-pyrrol-2-amine Chemical class NC1=CC=CN1 QLSWIGRIBOSFMV-UHFFFAOYSA-N 0.000 title 1
230000015572 biosynthetic process Effects 0.000 title 1
238000003786 synthesis reaction Methods 0.000 title 1
NHNHWBFFDARHFO-UHFFFAOYSA-N 2-(1h-pyrrol-2-yl)acetamide Chemical class NC(=O)CC1=CC=CN1 NHNHWBFFDARHFO-UHFFFAOYSA-N 0.000 abstract 1
RGHQKFQZGLKBCF-UHFFFAOYSA-N 2-bromoethyl acetate Chemical compound CC(=O)OCCBr RGHQKFQZGLKBCF-UHFFFAOYSA-N 0.000 abstract 1
102000027484 GABAA receptors Human genes 0.000 abstract 1
108091008681 GABAA receptors Proteins 0.000 abstract 1
239000002253 acid Substances 0.000 abstract 1
150000004982 aromatic amines Chemical class 0.000 abstract 1
150000004820 halides Chemical class 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/04—Indoles; Hydrogenated indoles
- C07D209/30—Indoles; Hydrogenated indoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to carbon atoms of the hetero ring
- C07D209/42—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
- C07D307/77—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
- C07D307/78—Benzo [b] furans; Hydrogenated benzo [b] furans
- C07D307/82—Benzo [b] furans; Hydrogenated benzo [b] furans with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the hetero ring
- C07D307/83—Oxygen atoms
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
- C07D307/77—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
- C07D307/78—Benzo [b] furans; Hydrogenated benzo [b] furans
- C07D307/82—Benzo [b] furans; Hydrogenated benzo [b] furans with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the hetero ring
- C07D307/84—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Public Health (AREA)
Pharmacology & Pharmacy (AREA)
Neurosurgery (AREA)
Biomedical Technology (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Bioinformatics & Cheminformatics (AREA)
Veterinary Medicine (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Engineering & Computer Science (AREA)
Neurology (AREA)
Psychiatry (AREA)
Pain & Pain Management (AREA)
Plural Heterocyclic Compounds (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Pyrrole Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Indole Compounds (AREA)
Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Furan Compounds (AREA)
Tea And Coffee (AREA)
Fats And Perfumes (AREA)
Treatment Of Liquids With Adsorbents In General (AREA)

NO20002214A 1997-11-13 2000-04-28 FremgangsmÕte for syntese av pyrrolaminer NO20002214L (no)

Applications Claiming Priority (3)

Application Number	Priority Date	Filing Date	Title
US6542297P	1997-11-13	1997-11-13
US7426698P	1998-02-10	1998-02-10
PCT/IB1998/001672 WO1999025684A1 (en)	1997-11-13	1998-10-21	Method of synthesis of pyrrole amides

Publications (2)

Publication Number	Publication Date
NO20002214D0 NO20002214D0 (no)	2000-04-28
NO20002214L true NO20002214L (no)	2000-05-12

Family

ID=26745584

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
NO20002214A NO20002214L (no)	1997-11-13	2000-04-28	FremgangsmÕte for syntese av pyrrolaminer

Country Status (35)

Country	Link
US (1)	US6262272B1 (id)
EP (1)	EP1030838B1 (id)
JP (1)	JP3497469B2 (id)
KR (1)	KR100386722B1 (id)
CN (2)	CN1508129A (id)
AT (1)	ATE231492T1 (id)
AU (1)	AU745788B2 (id)
BG (1)	BG64530B1 (id)
BR (1)	BR9814161A (id)
CA (1)	CA2310095A1 (id)
CZ (1)	CZ20001769A3 (id)
DE (1)	DE69810959T2 (id)
DK (1)	DK1030838T3 (id)
DZ (1)	DZ2651A1 (id)
EA (1)	EA002243B1 (id)
ES (1)	ES2186232T3 (id)
HR (1)	HRP20000298A2 (id)
HU (1)	HUP0100235A3 (id)
ID (1)	ID24135A (id)
IL (1)	IL135710A0 (id)
IS (1)	IS5469A (id)
MA (1)	MA24697A1 (id)
NO (1)	NO20002214L (id)
NZ (1)	NZ503916A (id)
OA (1)	OA11378A (id)
PA (1)	PA8462901A1 (id)
PL (1)	PL340554A1 (id)
PT (1)	PT1030838E (id)
SK (1)	SK6872000A3 (id)
TN (1)	TNSN98204A1 (id)
TR (1)	TR200001343T2 (id)
TW (1)	TW509675B (id)
UY (1)	UY25249A1 (id)
WO (1)	WO1999025684A1 (id)
YU (1)	YU27300A (id)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
HUP0202534A3 (en) *	1999-08-31	2002-12-28	Neurogen Corp Branford	Fused pyrrolecarboxamides: gaba brain receptor ligands and pharmaceutical compositions containing them
WO2002020492A1 (en) *	2000-09-06	2002-03-14	Neurogen Corporation	Aryl substituted tetrahydroindazoles and their use as ligands for the gaba-a receptor
BR0115874A (pt) *	2000-12-04	2003-10-28	Pfizer Prod Inc	Sìntese de pirrole-amidas
AU2003212979A1 (en)	2002-02-07	2003-09-02	Neurogen Corporation	Substituted fused pyrazolecarboxylic acid arylamides and related compounds
US20080153629A1 (en) *	2004-05-07	2008-06-26	Sullivan Michael J	Thick Outer Cover Layer Golf Ball
CN102786458B (zh) *	2012-06-04	2014-02-12	天津渤海职业技术学院	吡咯甲酰胺衍生物、其制备方法和用途
EP3097095A1 (en) *	2014-01-24	2016-11-30	AbbVie Inc.	Furo-3-carboxamide derivatives and methods of use

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US5750702A (en)	1993-10-27	1998-05-12	Neurogen Corporation	Certain pyrrolo pyridine-3-carboxamides; a new class of GABA brain receptor ligands
US5484944A (en) *	1993-10-27	1996-01-16	Neurogen Corporation	Certain fused pyrrolecarboxanilides and their use as GABA brain receptor ligands
US5804686A (en)	1996-01-19	1998-09-08	Neurogen Corporation	fused pyrrolecarboxamides; a new class of GABA brain receptor ligands
WO1997034870A1 (en)	1996-03-22	1997-09-25	Neurogen Corporation	Certain fused pyrrolecarboxamides as gaba brain receptor ligands

1998
- 1998-10-21 CN CNA031594727A patent/CN1508129A/zh active Pending
- 1998-10-21 EA EA200000413A patent/EA002243B1/ru not_active IP Right Cessation
- 1998-10-21 WO PCT/IB1998/001672 patent/WO1999025684A1/en not_active Ceased
- 1998-10-21 EP EP98946678A patent/EP1030838B1/en not_active Expired - Lifetime
- 1998-10-21 US US09/403,985 patent/US6262272B1/en not_active Expired - Fee Related
- 1998-10-21 DK DK98946678T patent/DK1030838T3/da active
- 1998-10-21 KR KR10-2000-7005185A patent/KR100386722B1/ko not_active Expired - Fee Related
- 1998-10-21 CA CA002310095A patent/CA2310095A1/en not_active Abandoned
- 1998-10-21 AT AT98946678T patent/ATE231492T1/de not_active IP Right Cessation
- 1998-10-21 ES ES98946678T patent/ES2186232T3/es not_active Expired - Lifetime
- 1998-10-21 JP JP2000521068A patent/JP3497469B2/ja not_active Expired - Fee Related
- 1998-10-21 CZ CZ20001769A patent/CZ20001769A3/cs unknown
- 1998-10-21 TR TR2000/01343T patent/TR200001343T2/xx unknown
- 1998-10-21 ID IDW20000893A patent/ID24135A/id unknown
- 1998-10-21 PT PT98946678T patent/PT1030838E/pt unknown
- 1998-10-21 HR HR20000298A patent/HRP20000298A2/hr not_active Application Discontinuation
- 1998-10-21 CN CN98811119A patent/CN1280566A/zh active Pending
- 1998-10-21 AU AU93639/98A patent/AU745788B2/en not_active Ceased
- 1998-10-21 SK SK687-2000A patent/SK6872000A3/sk unknown
- 1998-10-21 NZ NZ503916A patent/NZ503916A/xx unknown
- 1998-10-21 HU HU0100235A patent/HUP0100235A3/hu unknown
- 1998-10-21 IL IL13571098A patent/IL135710A0/xx unknown
- 1998-10-21 YU YU27300A patent/YU27300A/sh unknown
- 1998-10-21 DE DE69810959T patent/DE69810959T2/de not_active Expired - Fee Related
- 1998-10-21 PL PL98340554A patent/PL340554A1/xx not_active Application Discontinuation
- 1998-10-21 BR BR9814161-9A patent/BR9814161A/pt not_active Application Discontinuation
- 1998-11-10 PA PA19988462901A patent/PA8462901A1/es unknown
- 1998-11-10 TW TW087118708A patent/TW509675B/zh not_active IP Right Cessation
- 1998-11-11 DZ DZ980261A patent/DZ2651A1/xx active
- 1998-11-11 MA MA25342A patent/MA24697A1/fr unknown
- 1998-11-11 TN TNTNSN98204A patent/TNSN98204A1/fr unknown
- 1998-11-13 UY UY25249A patent/UY25249A1/es not_active IP Right Cessation
2000
- 2000-04-26 IS IS5469A patent/IS5469A/is unknown
- 2000-04-28 NO NO20002214A patent/NO20002214L/no unknown
- 2000-05-09 BG BG104413A patent/BG64530B1/bg unknown
- 2000-05-12 OA OA1200000136A patent/OA11378A/en unknown

Also Published As

Publication number	Publication date
CA2310095A1 (en)	1999-05-27
OA11378A (en)	2004-01-27
WO1999025684A1 (en)	1999-05-27
CN1508129A (zh)	2004-06-30
AU745788B2 (en)	2002-03-28
CN1280566A (zh)	2001-01-17
NZ503916A (en)	2002-08-28
DZ2651A1 (fr)	2003-03-15
EA200000413A1 (ru)	2000-12-25
HRP20000298A2 (en)	2001-02-28
EP1030838B1 (en)	2003-01-22
IL135710A0 (en)	2001-05-20
JP2001523660A (ja)	2001-11-27
EA002243B1 (ru)	2002-02-28
YU27300A (sh)	2002-10-18
ID24135A (id)	2000-07-06
ES2186232T3 (es)	2003-05-01
BR9814161A (pt)	2000-09-26
PL340554A1 (en)	2001-02-12
TNSN98204A1 (fr)	2005-03-15
US6262272B1 (en)	2001-07-17
BG64530B1 (bg)	2005-06-30
DE69810959T2 (de)	2003-06-05
TW509675B (en)	2002-11-11
DK1030838T3 (da)	2003-02-24
NO20002214D0 (no)	2000-04-28
KR20010032063A (ko)	2001-04-16
UY25249A1 (es)	1999-07-19
PA8462901A1 (es)	2000-05-24
TR200001343T2 (tr)	2001-02-21
JP3497469B2 (ja)	2004-02-16
IS5469A (is)	2000-04-26
CZ20001769A3 (cs)	2001-09-12
HUP0100235A3 (en)	2002-04-29
EP1030838A1 (en)	2000-08-30
MA24697A1 (fr)	1999-07-01
DE69810959D1 (de)	2003-02-27
PT1030838E (pt)	2003-03-31
BG104413A (en)	2001-02-28
ATE231492T1 (de)	2003-02-15
SK6872000A3 (en)	2002-02-05
KR100386722B1 (ko)	2003-06-09
HUP0100235A2 (hu)	2001-12-28
AU9363998A (en)	1999-06-07

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PL326452A1 (en)	1998-09-28	Method of synthesising composunds being affinite to curcumine
TR200000456T2 (tr)	2000-07-21	Glufosinatların ve ara ürünlerinin üretimine dair yöntem.
DE69307699D1 (de)	1997-03-06	Verfahren zur herstellung substituierter aromatischer amine
NO20002214D0 (no)	2000-04-28	FremgangsmÕte for syntese av pyrrolaminer
DK0787124T3 (da)	2000-05-08	Fremgangsmåde til fremstilling af substituerede 3-aminobenzonitriler
DE60102008D1 (de)	2004-03-18	Herstellungsverfahren für ein bekanntes terazolderivat
EP1344772A4 (en)	2005-03-16	ARYLBIS (PERFLUORALKYLSULFONYL) -METHANE, METAL SALT AND METHOD FOR THE PRODUCTION THEREOF
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ATE11401T1 (de)	1985-02-15	Substituierte biphenyl-2-carboxaldehyde und verfahren zu ihrer herstellung.
NO985775L (no)	1999-06-21	FremgangsmÕte til fremstilling av aminocyanacetamid
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DK0971907T3 (da)	2002-06-10	Fremgangsmåde til fremstilling af 1,3-disubstituerede 2-nitroguanidiner
NZ332245A (en)	2000-03-27	Substituted benzo-oxazolol carboxylic acid derivatives, process for their production and medicaments containing them
BR9909570A (pt)	2004-06-01	Processo altamente seletivo, produto preparado pelo mesmo, e, processo para preparar uma quinonaimina a partir de uma hidroxifenilamina correspondente
BR0115874A (pt)	2003-10-28	Sìntese de pirrole-amidas
ATE260883T1 (de)	2004-03-15	Verfahren zur herstellung von atropasäureethylester
IL133719A0 (en)	2001-04-30	Method for the production of n-(5-amino-2-cyano-4- fluorophenyl) - sulphonamides and new intermediate products
HUP9900171A2 (hu)	1999-04-28	Eljárás azo-metinek és alfa-halogén-acetanilidek előállítására
FI915109A0 (fi)	1991-10-30	Foerfarande foer framstaellning av alifatisk amid och salter daerav.
MX9504739A (es)	1997-03-29	Procedimiento para la obtencion de colorantes cationicos del 1,3,4-tiadiazol.
DK1044204T3 (da)	2003-09-29	Fremgangsmåde til fremstiling af alfa-oxolactamer