NO20003083D0 - Karboksylsubstituerte kromanderivater som er nyttige som beta- 3-adrenoreseptorantagonister - Google Patents

Karboksylsubstituerte kromanderivater som er nyttige som beta- 3-adrenoreseptorantagonister

Info

Publication number
NO20003083D0
NO20003083D0 NO20003083A NO20003083A NO20003083D0 NO 20003083 D0 NO20003083 D0 NO 20003083D0 NO 20003083 A NO20003083 A NO 20003083A NO 20003083 A NO20003083 A NO 20003083A NO 20003083 D0 NO20003083 D0 NO 20003083D0
Authority
NO
Norway
Prior art keywords
beta
carboxyl
derivatives useful
adrenoceptor antagonists
chromane derivatives
Prior art date
Application number
NO20003083A
Other languages
English (en)
Other versions
NO20003083L (no
Inventor
Richard D Connell
Timothy G Lease
Jeremy Baryza
Original Assignee
Bayer Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Ag filed Critical Bayer Ag
Publication of NO20003083D0 publication Critical patent/NO20003083D0/no
Publication of NO20003083L publication Critical patent/NO20003083L/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D311/00—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings
    • C07D311/02—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D311/04—Benzo[b]pyrans, not hydrogenated in the carbocyclic ring
    • C07D311/58—Benzo[b]pyrans, not hydrogenated in the carbocyclic ring other than with oxygen or sulphur atoms in position 2 or 4
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Diabetes (AREA)
  • Veterinary Medicine (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Neurosurgery (AREA)
  • Emergency Medicine (AREA)
  • Endocrinology (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Child & Adolescent Psychology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pyrane Compounds (AREA)
  • Peptides Or Proteins (AREA)
  • Pyrrole Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Solid-Sorbent Or Filter-Aiding Compositions (AREA)
  • Detergent Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
NO20003083A 1997-12-19 2000-06-15 Karboksylsubstituerte kromanderivater som er nyttige som <beta>-3-adrenoreseptorantagonister NO20003083L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US99462097A 1997-12-19 1997-12-19
PCT/US1998/026735 WO1999032476A1 (en) 1997-12-19 1998-12-16 Carboxyl substituted chroman derivatives useful as beta 3 adrenoreceptor agonists

Publications (2)

Publication Number Publication Date
NO20003083D0 true NO20003083D0 (no) 2000-06-15
NO20003083L NO20003083L (no) 2000-08-15

Family

ID=25540853

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20003083A NO20003083L (no) 1997-12-19 2000-06-15 Karboksylsubstituerte kromanderivater som er nyttige som <beta>-3-adrenoreseptorantagonister

Country Status (24)

Country Link
EP (1) EP1040106B1 (no)
JP (1) JP2001526282A (no)
KR (1) KR20010033188A (no)
CN (1) CN1284952A (no)
AT (1) ATE222901T1 (no)
AU (1) AU749097B2 (no)
BG (1) BG104593A (no)
BR (1) BR9814302A (no)
CA (1) CA2316971A1 (no)
DE (1) DE69807523T2 (no)
DK (1) DK1040106T3 (no)
ES (1) ES2183434T3 (no)
HU (1) HUP0004565A3 (no)
ID (1) ID26524A (no)
IL (1) IL136689A0 (no)
NO (1) NO20003083L (no)
NZ (1) NZ505200A (no)
PL (1) PL341229A1 (no)
PT (1) PT1040106E (no)
RU (1) RU2223269C2 (no)
SK (1) SK9362000A3 (no)
TR (1) TR200001927T2 (no)
UA (1) UA62993C2 (no)
WO (1) WO1999032476A1 (no)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AR035605A1 (es) 2000-12-11 2004-06-16 Bayer Corp Derivados de aminometil cromano di-sustituidos, un metodo para su preparacion, composiciones farmaceuticas y el uso de dichos derivados para la manufactura de medicamentos utiles como agonistas beta-3-adreno-receptores
AR035858A1 (es) * 2001-04-23 2004-07-21 Bayer Corp Derivados de cromano 2,6-sustituidos,composiciones farmaceuticas,uso de dichos derivados para la manufactura de medicamentos utiles como agonistas adrenorreceptores beta-3
US20040265991A1 (en) * 2001-10-17 2004-12-30 Naoaki Taoka Process for preparation of (s)-alpha-halomethylpyridine-methanol derivatives
MY147767A (en) * 2004-06-16 2013-01-31 Janssen Pharmaceutica Nv Novel sulfamate and sulfamide derivatives useful for the treatment of epilepsy and related disorders
JP2008530229A (ja) 2005-02-17 2008-08-07 ワイス シクロアルキル縮合インドール、ベンゾチオフェン、ベンゾフランおよびインデン誘導体
EP1803716B1 (en) * 2005-12-28 2012-07-25 Acino Pharma AG A process for preparation of racemic nebivolol
US7560575B2 (en) 2005-12-28 2009-07-14 Acino Pharma Ag Process for preparation of racemic Nebivolol
RU2392277C2 (ru) * 2005-12-28 2010-06-20 Асино Фарма Аг Способ получения рацемического небиволола
ES2534336B1 (es) * 2013-10-18 2016-01-28 Artax Biopharma Inc. Derivados de cromeno como inhibidores de la interacción TCR-Nck
ES2534318B1 (es) * 2013-10-18 2016-01-28 Artax Biopharma Inc. Derivados de cromeno sustituidos por alcóxido como inhibidores de la interacción TCR-Nck

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA1337429C (en) * 1983-12-05 1995-10-24 Guy Rosalia Eugene Van Lommen Derivatives of 2,2'-iminobisethanol
GB8801306D0 (en) * 1988-01-21 1988-02-17 Ici Plc Chemical compounds
RU2032684C1 (ru) * 1991-04-08 1995-04-10 Джон Вайс энд Бразер Лимитед Способ получения производных 4-оксохинолина или хромона или их фармацевтически приемлемых солей
US5451677A (en) * 1993-02-09 1995-09-19 Merck & Co., Inc. Substituted phenyl sulfonamides as selective β 3 agonists for the treatment of diabetes and obesity
BR9406823A (pt) * 1993-06-14 1996-03-26 Pfizer Aminas secundárias e agentes anti-diabéticos e antiobesidade
GB9405019D0 (en) * 1994-03-15 1994-04-27 Smithkline Beecham Plc Novel compounds
US5561142A (en) * 1994-04-26 1996-10-01 Merck & Co., Inc. Substituted sulfonamides as selective β3 agonists for the treatment of diabetes and obesity
EP0801060A1 (en) * 1996-04-09 1997-10-15 Pfizer Inc. Heterocyclic Beta-3 Adrenergenic Agonists

Also Published As

Publication number Publication date
UA62993C2 (en) 2004-01-15
ATE222901T1 (de) 2002-09-15
AU1830099A (en) 1999-07-12
PL341229A1 (en) 2001-03-26
PT1040106E (pt) 2002-11-29
EP1040106B1 (en) 2002-08-28
NO20003083L (no) 2000-08-15
IL136689A0 (en) 2001-06-14
EP1040106A1 (en) 2000-10-04
DE69807523T2 (de) 2003-01-09
KR20010033188A (ko) 2001-04-25
DE69807523D1 (de) 2002-10-02
WO1999032476A1 (en) 1999-07-01
BR9814302A (pt) 2000-10-10
ID26524A (id) 2001-01-11
SK9362000A3 (en) 2001-09-11
BG104593A (en) 2001-09-28
JP2001526282A (ja) 2001-12-18
DK1040106T3 (da) 2002-12-02
HUP0004565A2 (hu) 2001-08-28
ES2183434T3 (es) 2003-03-16
AU749097B2 (en) 2002-06-20
RU2223269C2 (ru) 2004-02-10
TR200001927T2 (tr) 2001-06-21
NZ505200A (en) 2002-09-27
CA2316971A1 (en) 1999-07-01
HUP0004565A3 (en) 2002-12-28
CN1284952A (zh) 2001-02-21

Similar Documents

Publication Publication Date Title
EE200100227A (et) Asendatud bensopüraani analoogid põletiku raviks
EE9900506A (et) Asendatud bensopüraani derivaadid põletiku raviks
BG104247A (bg) Производни на резорцинола
ES2186720T3 (es) Composiciones para inhibir la reabsorcion osea mediada por osteoclastos.
ES2184127T3 (es) Derivados de sulfamato anticonvulsivos utiles para el tratamiento de la obesidad.
TR200100267T2 (tr) İkameli anilid bileşimleri ve yöntemler.
NO983431L (no) Anti-klöemidler
NO993634D0 (no) Anvendelse av sentrale cannabinoid-reseptor-antagonister for regulering av appetitt
TR199701146T1 (xx) N�rotensin resept�rleri �zerinde etkili 1-Fenilpirazol-3-Karboksamidler.
DOP2002000385A (es) Derivados de cromano 2,6-sustituidos utiles como agonistas adrenoreceptores beta-3
NO20003083D0 (no) Karboksylsubstituerte kromanderivater som er nyttige som beta- 3-adrenoreseptorantagonister
NO20006293L (no) Nye benzopyran eller tiobenzopyranderivater
EE200000140A (et) Asendatud kromaani derivaadid
HN2001000275A (es) Agonistas beta-3 adreno-receptores de derivados de aminometil cromano d-sustituido
EE200000144A (et) Asendatud kromaani derivaadid
BR9813905A (pt) Instalação para influenciar uma instalação de iluminação
BR9608594B1 (pt) misturas de benzimidazóis substituìdos para o combate de protozoários parasìticos.
IL136688A0 (en) Novel sulfonamide substituted chroman derivatives useful as beta-3 adrenoreceptor agonists
TR200001080T2 (tr) 2 ile ikame edilmiş 1,2-Benisotiyazol türevleri ve bunların serrotonın antagonistleri
ATE265418T1 (de) Neue substituierte 3-phenoxy- und 3- phenylalkyloxy-2-phenyl-propylamine
PT908107E (pt) Composicoes adocantes contendo neohesperidina-dihidrocalcona e pelo menos um outro adocante de elevada intensidade
FR2770126B1 (fr) Vis chirurgicale pour le repositionnement de la tuberosite tibiale
EE200300194A (et) Asendatud bensopüraani derivaatide kasutamine põletiku raviks
ECSP982678A (es) Derivados de resorcinol
SE9802754D0 (sv) Belysning av strömställare, reglerdon eller annat instrument

Legal Events

Date Code Title Description
FC2A Withdrawal, rejection or dismissal of laid open patent application