NO20006323L - Glykopeptid-derivater og farmasöytiske sammensetninger som inneholder disse - Google Patents

Glykopeptid-derivater og farmasöytiske sammensetninger som inneholder disse

Info

Publication number: NO20006323L
Authority: NO; Norway
Prior art keywords: pharmaceutical compositions; compositions containing; derivatives; glycopeptide; glycopeptide derivatives
Prior art date: 1998-12-23

Application number

NO20006323A

Other languages

English (en)

Other versions

NO326066B1 (no

NO20006323D0 (no

Inventor

J Kevin Judice

Paul Ross Fatheree

Bernice M T Lam

Michael R Leadbetter

Martin Sheringham Linsell

Yongqi Mu

Sean Gary Trapp

Guang Yang

Yan Zhu

Original Assignee

Advanced Medicine Inc

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1998-12-23

Filing date

2000-12-12

Publication date

2001-02-12

2000-12-12 Application filed by Advanced Medicine Inc filed Critical Advanced Medicine Inc

2000-12-12 Publication of NO20006323D0 publication Critical patent/NO20006323D0/no

2001-02-12 Publication of NO20006323L publication Critical patent/NO20006323L/no

2008-09-08 Publication of NO326066B1 publication Critical patent/NO326066B1/no

Links

DQJCDTNMLBYVAY-ZXXIYAEKSA-N (2S,5R,10R,13R)-16-{[(2R,3S,4R,5R)-3-{[(2S,3R,4R,5S,6R)-3-acetamido-4,5-dihydroxy-6-(hydroxymethyl)oxan-2-yl]oxy}-5-(ethylamino)-6-hydroxy-2-(hydroxymethyl)oxan-4-yl]oxy}-5-(4-aminobutyl)-10-carbamoyl-2,13-dimethyl-4,7,12,15-tetraoxo-3,6,11,14-tetraazaheptadecan-1-oic acid Chemical class NCCCC[C@H](C(=O)N[C@@H](C)C(O)=O)NC(=O)CC[C@H](C(N)=O)NC(=O)[C@@H](C)NC(=O)C(C)O[C@@H]1[C@@H](NCC)C(O)O[C@H](CO)[C@H]1O[C@H]1[C@H](NC(C)=O)[C@@H](O)[C@H](O)[C@@H](CO)O1 DQJCDTNMLBYVAY-ZXXIYAEKSA-N 0.000 title abstract 4
239000008194 pharmaceutical composition Substances 0.000 title abstract 2
239000003242 anti bacterial agent Substances 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K9/00—Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K9/00—Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof
- C07K9/006—Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof the peptide sequence being part of a ring structure
- C07K9/008—Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof the peptide sequence being part of a ring structure directly attached to a hetero atom of the saccharide radical, e.g. actaplanin, avoparcin, ristomycin, vancomycin
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
- C07K7/04—Linear peptides containing only normal peptide links
- C07K7/06—Linear peptides containing only normal peptide links having 5 to 11 amino acids
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Medicinal Chemistry (AREA)
General Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Biochemistry (AREA)
Biophysics (AREA)
Proteomics, Peptides & Aminoacids (AREA)
Molecular Biology (AREA)
Genetics & Genomics (AREA)
Animal Behavior & Ethology (AREA)
Oncology (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Communicable Diseases (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Chemical Kinetics & Catalysis (AREA)
Pharmacology & Pharmacy (AREA)
General Chemical & Material Sciences (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Peptides Or Proteins (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

NO20006323A 1998-12-23 2000-12-12 Glykopeptid-derivater, farmasøytiske sammensetninger samt anvendelser derav. NO326066B1 (no)

Applications Claiming Priority (5)

Application Number	Priority Date	Filing Date	Title
US11372898P	1998-12-23	1998-12-23
US12931399P	1999-04-14	1999-04-14
US16402499P	1999-11-04	1999-11-04
US16997899P	1999-12-10	1999-12-10
PCT/US1999/030543 WO2000039156A1 (en)	1998-12-23	1999-12-22	Glycopeptide derivatives and pharmaceutical compositions containing the same

Publications (3)

Publication Number	Publication Date
NO20006323D0 NO20006323D0 (no)	2000-12-12
NO20006323L true NO20006323L (no)	2001-02-12
NO326066B1 NO326066B1 (no)	2008-09-08

Family

ID=27493926

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
NO20006323A NO326066B1 (no)	1998-12-23	2000-12-12	Glykopeptid-derivater, farmasøytiske sammensetninger samt anvendelser derav.

Country Status (23)

Country	Link
US (9)	US6392012B1 (no)
EP (1)	EP1140993B1 (no)
JP (1)	JP4362017B2 (no)
KR (1)	KR100665204B1 (no)
CN (1)	CN1249081C (no)
AT (1)	ATE242783T1 (no)
AU (1)	AU768204B2 (no)
BR (1)	BRPI9914221B8 (no)
CA (1)	CA2336445C (no)
CZ (1)	CZ301184B6 (no)
DE (1)	DE69908819T2 (no)
DK (1)	DK1140993T3 (no)
ES (1)	ES2201825T3 (no)
HK (1)	HK1040721B (no)
HU (1)	HU230190B1 (no)
IL (2)	IL140093A0 (no)
NO (1)	NO326066B1 (no)
NZ (1)	NZ508594A (no)
PL (1)	PL198311B1 (no)
PT (1)	PT1140993E (no)
SI (1)	SI1140993T1 (no)
WO (1)	WO2000039156A1 (no)
ZA (1)	ZA200007222B (no)

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US6392012B1 (en) *	1998-12-23	2002-05-21	Advanced Medicine, Inc.	Glycopeptide derivatives and pharmaceutical compositions containing the same
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WO2001057071A2 (en) *	2000-02-04	2001-08-09	Advanced Medicine, Inc.	Glycopeptide derivatives having antibiotic activity
EP1278549B1 (en) *	2000-05-02	2008-12-10	Theravance, Inc.	Composition containing a cyclodextrin and a glycopeptide antibiotic
SI1276759T1 (sl)	2000-05-02	2008-12-31	Theravance Inc	Postopek reduktivnega alkiliranja na glikopeptidih
WO2001083520A2 (en)	2000-05-02	2001-11-08	Theravance,Inc	Polyacid glycopeptide derivatives
UA75083C2 (uk)	2000-06-22	2006-03-15	Тераванс, Інк.	Похідні глікопептидфосфонатів
US6872804B2 (en)	2000-06-22	2005-03-29	Theravance, Inc.	Glycopeptide disulfide and thioester derivatives
AU2001259816A1 (en)	2000-06-22	2002-01-02	Advanced Medecine, Inc.	Polyhydroxy glycopeptide derivatives
WO2001098327A2 (en) *	2000-06-22	2001-12-27	Theravance, Inc.	Glycopeptide carboxy-saccharide derivatives
US6905669B2 (en) *	2001-04-24	2005-06-14	Supergen, Inc.	Compositions and methods for reestablishing gene transcription through inhibition of DNA methylation and histone deacetylase
TWI312785B (en) *	2001-08-24	2009-08-01	Theravance Inc	Process for preparing vancomycin derivatives
TWI275594B (en)	2001-08-24	2007-03-11	Theravance Inc	Process for preparing vancomycin phosphonate derivatives
EP1295711B1 (en)	2001-09-19	2006-04-12	The Procter & Gamble Company	A color printed laminated structure, absorbent article comprising the same and process for manufacturing the same
TWI335332B (en) *	2001-10-12	2011-01-01	Theravance Inc	Cross-linked vancomycin-cephalosporin antibiotics
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US7067481B2 (en) *	2003-05-23	2006-06-27	Theravance, Inc.	Cross-linked glycopeptide-cephalosporin antibiotics
ATE388153T1 (de) *	2003-07-11	2008-03-15	Theravance Inc	Quervernetzte glycopeptid-cephalosporin- antibiotika
DE102004055582A1 (de) *	2004-11-18	2006-05-24	Bayer Cropscience Ag	N-Heterocyclyl-phthalsäurediamide
JP4330169B2 (ja)	2004-11-29	2009-09-16	国立大学法人名古屋大学	グリコペプチド抗生物質モノマー誘導体
US8304597B2 (en)	2004-12-15	2012-11-06	The Procter And Gamble Company	Method of using an absorbent article having a functional enhancement indicator
US20070185015A1 (en) *	2005-02-28	2007-08-09	Chiron Corporation and North China Pharmaceutical Corporation	Semi-synthetic desmethyl-vancomycin-based glycopeptides with antibiotic activity
US7632918B2 (en) *	2005-02-28	2009-12-15	Novartis Vaccines And Diagnostics, Inc.	Semi-synthetic glycopeptides with antibiotic activity
US7368422B2 (en) *	2005-02-28	2008-05-06	Novartis Vaccines And Diagnostics Inc.	Semi-synthetic rearranged vancomycin/desmethyl-vancomycin-based glycopeptides with antibiotic activity
JP5192384B2 (ja)	2005-09-22	2013-05-08	メディバスエルエルシー	ビス−（α−アミノ）−ジオール−ジエステル含有ポリ（エステルアミド）およびポリ（エステルウレタン）組成物および使用の方法
JP5178520B2 (ja)	2005-09-22	2013-04-10	メディバスエルエルシー	固体ポリマー送達組成物およびその使用法
US20070173438A1 (en) *	2006-01-13	2007-07-26	The Scripps Research Institute	[PSI[CH2NH]PG4] glycopeptide antibiotic analogs
TW200808818A (en) *	2006-05-26	2008-02-16	Shionogi & Co	Glycopeptide antibiotic derivatives
CN101959849A (zh) *	2007-12-26	2011-01-26	利德治疗公司	作为抗菌剂的新型半合成糖肽
KR20100109934A (ko)	2007-12-26	2010-10-11	시오노기세야쿠 가부시키가이샤	글리코펩티드 항생 물질 배당화 유도체
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GB2465863A (en) *	2008-12-05	2010-06-09	Lead Therapeutics Inc	Semi-synthetic heptapeptidic glycopeptides for the treatment of bacterial infections
CN101928330B (zh) *	2009-06-26	2013-10-16	上海来益生物药物研究开发中心有限责任公司	一种新的化合物及其应用
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CA2904387C (en)	2013-03-15	2021-12-07	Melinta Therapeutics, Inc.	Methods of treating infections in overweight and obese patients using antibiotics
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US20170342110A1 (en) *	2014-12-25	2017-11-30	Jawaharlal Nehru Centre for Advanced Scientific Research (JNCASR)	Glycopeptides and uses thereof
US20190203240A1 (en) *	2016-01-15	2019-07-04	Universitaet Hamburg	Methods for the production of rhamnosylated flavonoids
CA3012176A1 (en) *	2016-01-28	2017-08-03	ACatechol, Inc.	Photo-cleavable primer compositions and methods of use
CN107325159A (zh) *	2016-04-29	2017-11-07	中国科学院上海药物研究所	一类万古霉素衍生物、其制备方法、药物组合物和用途
GB2577420B (en)	2017-05-22	2022-07-06	Insmed Inc	Glycopeptide derivative compounds and uses thereof
CN107987131B (zh) *	2017-11-16	2021-03-09	上海来益生物药物研究开发中心有限责任公司	一组具有抗耐药性细菌活性的化合物、其制备方法和应用
CN108409837B (zh)	2018-03-06	2021-09-24	上海来益生物药物研究开发中心有限责任公司	一组具有抗耐药性细菌活性的糖肽类化合物、其制备方法和应用
NL2023883B1 (en) *	2019-09-24	2021-04-26	Univ Leiden	Antibiotic compounds
CN111620931B (zh) *	2020-06-12	2021-12-17	苏州博源医疗科技有限公司	万古霉素衍生物及其制备方法和应用
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US6392012B1 (en) *	1998-12-23	2002-05-21	Advanced Medicine, Inc.	Glycopeptide derivatives and pharmaceutical compositions containing the same
UA75083C2 (uk)	2000-06-22	2006-03-15	Тераванс, Інк.	Похідні глікопептидфосфонатів
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1999
- 1999-12-22 US US09/470,209 patent/US6392012B1/en not_active Expired - Lifetime
- 1999-12-22 DK DK99965331T patent/DK1140993T3/da active
- 1999-12-22 DE DE69908819T patent/DE69908819T2/de not_active Expired - Lifetime
- 1999-12-22 JP JP2000591067A patent/JP4362017B2/ja not_active Expired - Fee Related
- 1999-12-22 CZ CZ20010022A patent/CZ301184B6/cs not_active IP Right Cessation
- 1999-12-22 BR BRPI9914221A patent/BRPI9914221B8/pt not_active IP Right Cessation
- 1999-12-22 AT AT99965331T patent/ATE242783T1/de active
- 1999-12-22 PL PL348451A patent/PL198311B1/pl unknown
- 1999-12-22 IL IL14009399A patent/IL140093A0/xx active IP Right Grant
- 1999-12-22 EP EP99965331A patent/EP1140993B1/en not_active Expired - Lifetime
- 1999-12-22 ES ES99965331T patent/ES2201825T3/es not_active Expired - Lifetime
- 1999-12-22 HU HU0400887A patent/HU230190B1/hu unknown
- 1999-12-22 AU AU31273/00A patent/AU768204B2/en not_active Expired
- 1999-12-22 NZ NZ508594A patent/NZ508594A/en not_active IP Right Cessation
- 1999-12-22 KR KR1020017003918A patent/KR100665204B1/ko not_active Expired - Lifetime
- 1999-12-22 WO PCT/US1999/030543 patent/WO2000039156A1/en not_active Ceased
- 1999-12-22 CA CA2336445A patent/CA2336445C/en not_active Expired - Lifetime
- 1999-12-22 HK HK02102171.5A patent/HK1040721B/en unknown
- 1999-12-22 PT PT99965331T patent/PT1140993E/pt unknown
- 1999-12-22 CN CNB99809434XA patent/CN1249081C/zh not_active Expired - Lifetime
- 1999-12-22 SI SI9930389T patent/SI1140993T1/xx unknown
2000
- 2000-09-06 US US09/656,473 patent/US6444786B1/en not_active Expired - Lifetime
- 2000-11-01 US US09/674,456 patent/US6455669B1/en not_active Expired - Lifetime
- 2000-12-05 IL IL140093A patent/IL140093A/en not_active IP Right Cessation
- 2000-12-06 ZA ZA200007222A patent/ZA200007222B/xx unknown
- 2000-12-12 NO NO20006323A patent/NO326066B1/no not_active IP Right Cessation
2002
- 2002-03-06 US US10/092,088 patent/US6962970B2/en not_active Expired - Lifetime
2004
- 2004-04-15 US US10/825,038 patent/US6949681B2/en not_active Expired - Lifetime
2005
- 2005-05-13 US US11/128,901 patent/US7101964B2/en not_active Expired - Lifetime
2006
- 2006-04-17 US US11/405,234 patent/US7351791B2/en not_active Expired - Fee Related
2007
- 2007-10-24 US US11/977,377 patent/US7723470B2/en not_active Expired - Fee Related
2009
- 2009-05-08 US US12/437,778 patent/US8030445B2/en not_active Expired - Fee Related

Also Published As

Publication number	Publication date
NO326066B1 (no)	2008-09-08
PT1140993E (pt)	2003-10-31
DE69908819D1 (de)	2003-07-17
IL140093A (en)	2006-06-11
US7351791B2 (en)	2008-04-01
CN1315961A (zh)	2001-10-03
US7723470B2 (en)	2010-05-25
NO20006323D0 (no)	2000-12-12
HU230190B1 (hu)	2015-09-28
EP1140993B1 (en)	2003-06-11
US6949681B2 (en)	2005-09-27
US6392012B1 (en)	2002-05-21
AU768204B2 (en)	2003-12-04
US6455669B1 (en)	2002-09-24
DK1140993T3 (da)	2003-10-06
JP2002533472A (ja)	2002-10-08
HUP0400887A3 (en)	2012-09-28
NZ508594A (en)	2003-05-30
AU3127300A (en)	2000-07-31
US20090215982A1 (en)	2009-08-27
BRPI9914221B8 (pt)	2021-05-25
BR9914221B1 (pt)	2013-12-31
CA2336445A1 (en)	2000-07-06
EP1140993A1 (en)	2001-10-10
US8030445B2 (en)	2011-10-04
KR20010085857A (ko)	2001-09-07
BR9914221A (pt)	2001-06-26
US20030060598A1 (en)	2003-03-27
US6444786B1 (en)	2002-09-03
JP4362017B2 (ja)	2009-11-11
US6962970B2 (en)	2005-11-08
WO2000039156A1 (en)	2000-07-06
PL198311B1 (pl)	2008-06-30
HUP0400887A2 (hu)	2004-08-30
HK1040721A1 (en)	2002-06-21
SI1140993T1 (en)	2003-12-31
KR100665204B1 (ko)	2007-01-04
CN1249081C (zh)	2006-04-05
ES2201825T3 (es)	2004-03-16
IL140093A0 (en)	2002-02-10
PL348451A1 (en)	2002-05-20
ATE242783T1 (de)	2003-06-15
DE69908819T2 (de)	2004-05-06
US20080103292A1 (en)	2008-05-01
US20040204346A1 (en)	2004-10-14
CZ301184B6 (cs)	2009-12-02
HK1040721B (en)	2003-10-17
US20060241024A1 (en)	2006-10-26
US7101964B2 (en)	2006-09-05
ZA200007222B (en)	2002-03-06
US20050239690A1 (en)	2005-10-27
CA2336445C (en)	2011-07-19
CZ200122A3 (en)	2001-06-13

Legal Events

Date	Code	Title	Description
2015-11-09	CHAD	Change of the owner's name or address (par. 44 patent law, par. patentforskriften)	Owner name: THERAVANCE BIOPHARMA R&D IP, US
2015-11-16	CHAD	Change of the owner's name or address (par. 44 patent law, par. patentforskriften)	Owner name: THERAVANCE BIOPHARMA ANTIBIOTICS IP, US
2019-04-15	CHAD	Change of the owner's name or address (par. 44 patent law, par. patentforskriften)	Owner name: CUMBERLAND PHARMACEUTICALS INC., US
2020-01-13	MK1K	Patent expired

Publication	Publication Date	Title
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ATE296826T1 (de)	2005-06-15	Pyrazolo(1,5)pyridinderivate
TR200101126T2 (tr)	2001-09-21	İkameli fenil türevleri, hazırlanma ve kullanımları
EA200300050A1 (ru)	2003-04-24	Гликопептидфосфонатные производные
DK1200418T3 (da)	2004-07-26	Nematodicide trifluorbutener
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DK0920421T3 (da)	2003-03-10	Isoxazolinderivater anvendelige som antimikrobielle midler
NO20012727D0 (no)	2001-06-01	3,4,5-trisubstituerte arylnitronforbindelser og farmasöytiske sammensetninger som inneholder samme
BR9813719A (pt)	2000-10-17	Agentes terapêuticos
AU2002357740A1 (en)	2003-06-23	Pyrazolo-pyridine derivatives as antiherpes agents
AU2002248531A1 (en)	2002-09-24	Pyrazolopyriadine derivatives
DK1073447T3 (da)	2007-09-03	N1-modificerede glycopeptider
SE9904128D0 (sv)	1999-11-15	Novel compounds
ATE282608T1 (de)	2004-12-15	Chinoxalindionen
NO20002321L (no)	2000-05-02	Bifenylderivater som farmasøytiske midler
PT1104419E (pt)	2002-09-30	Derivados de azabicicloheptano substituidos no azoto sua preparacao e utilizacao
MY123217A (en)	2006-05-31	Glycopeptide derivatives and pharmaceutical compositions containing the same
PT1140932E (pt)	2004-08-31	Derivados de 1,8-benzonaftiridina
DK1390056T3 (da)	2010-07-05	Glycopeptid-antibiotika
ECSP993299A (es)	2001-07-27	Derivados glicopeptidicos y composiciones farmaceuticas que los contienen