NO20035791L - Nye derivater av oksazolidinoner som antibakterielle midler - Google Patents

Nye derivater av oksazolidinoner som antibakterielle midler

Info

Publication number
NO20035791L
NO20035791L NO20035791A NO20035791A NO20035791L NO 20035791 L NO20035791 L NO 20035791L NO 20035791 A NO20035791 A NO 20035791A NO 20035791 A NO20035791 A NO 20035791A NO 20035791 L NO20035791 L NO 20035791L
Authority
NO
Norway
Prior art keywords
oxazolidinones
antibacterial agents
new derivatives
derivatives
medicament
Prior art date
Application number
NO20035791A
Other languages
English (en)
Norwegian (no)
Inventor
Juan Huguet Clotet
Marisabel Mourelle Mancini
Jose Hidalgo Rodriguez
Juan Carlos Castillo
Original Assignee
Vita Lab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Vita Lab filed Critical Vita Lab
Publication of NO20035791L publication Critical patent/NO20035791L/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D498/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
NO20035791A 2001-06-27 2003-12-22 Nye derivater av oksazolidinoner som antibakterielle midler NO20035791L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
ES200101559A ES2186550B2 (es) 2001-06-27 2001-06-27 Nuevos derivados de oxazolidinonas como antibacterianos.
PCT/IB2002/002408 WO2003002560A1 (en) 2001-06-27 2002-06-24 New derivatives of oxazolidinones as antibacterial agents

Publications (1)

Publication Number Publication Date
NO20035791L true NO20035791L (no) 2004-02-19

Family

ID=8498288

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20035791A NO20035791L (no) 2001-06-27 2003-12-22 Nye derivater av oksazolidinoner som antibakterielle midler

Country Status (29)

Country Link
US (1) US20040147545A1 (is)
EP (1) EP1401834A1 (is)
JP (1) JP2004521147A (is)
KR (1) KR20040030712A (is)
CN (1) CN1520412A (is)
AP (1) AP2003002942A0 (is)
AR (1) AR035254A1 (is)
BG (1) BG108498A (is)
BR (1) BR0210667A (is)
CA (1) CA2450982A1 (is)
CO (1) CO5540387A2 (is)
CR (1) CR7195A (is)
CZ (1) CZ2004101A3 (is)
EA (1) EA200400086A1 (is)
EE (1) EE200400004A (is)
ES (1) ES2186550B2 (is)
HR (1) HRP20031063A2 (is)
HU (1) HUP0400370A2 (is)
IL (1) IL159434A0 (is)
IS (1) IS7088A (is)
MA (1) MA27046A1 (is)
MX (1) MXPA04000185A (is)
NO (1) NO20035791L (is)
NZ (1) NZ530206A (is)
OA (1) OA12639A (is)
PE (1) PE20030134A1 (is)
PL (1) PL365476A1 (is)
SK (1) SK572004A3 (is)
WO (1) WO2003002560A1 (is)

Families Citing this family (21)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2003031443A1 (en) 2001-10-04 2003-04-17 Morphochem Aktiengesellschaft für kombinatorische Chemie Dual actions antibiotics comprising a oxazoldinone and a quinolone or naphthyridinone moiety
NZ543757A (en) * 2003-04-30 2009-02-28 Morphochem Ag Komb Chemie Use of oxazolidinone-quinoline hybrid antibiotics for the treatment of anthrax and other infections
DE10340485B4 (de) 2003-09-03 2015-05-13 Morphochem AG Aktiengesellschaft für kombinatorische Chemie Verfahren zur Herstellung von Oxazolidinon-Chinolon Hybriden
US7304050B2 (en) * 2003-09-16 2007-12-04 Pfizer Inc. Antibacterial agents
WO2005051933A1 (en) * 2003-11-28 2005-06-09 Ranbaxy Laboratories Limited An improved process for the synthesis of 4-(4-benzyloxy-carbonylamino-2-fluorophenyl)-piperazine-1-carboxylic acid tert-butyl ester, a key intermediate for oxazolidinone antimicrobials and compounds prepared thereby
AU2004299278C9 (en) * 2003-12-18 2013-10-24 Morphochem Aktiengesellschaft Fuer Kombinatorische Chemie Oxazolidinone-quinolone hybrid antibiotics
EP1557416A1 (en) * 2004-01-23 2005-07-27 Morphochem Aktiengesellschaft Für Kombinatorische Chemie Oxazolidinone-quinolone hybrid antibiotics
US8158797B2 (en) 2003-12-18 2012-04-17 Morphochem Aktiengesellschaft Fur Kombinatorische Chemie Oxazolidinone-quinolone hybrid antibiotics
US20060105941A1 (en) * 2004-11-12 2006-05-18 Allergan, Inc. Mixed antibiotic codrugs
KR20080110877A (ko) 2006-03-31 2008-12-19 재단법인 이쯔우 연구소 헤테로환을 갖는 신규 화합물
WO2009044777A1 (ja) 2007-10-02 2009-04-09 Research Foundation Itsuu Laboratory ７員ヘテロ環を有するオキサゾリジノン誘導体
CA2723232C (en) * 2008-05-09 2016-08-02 Actelion Pharmaceuticals Ltd 5-hydroxymethyl-oxazolidin-2-one derivatives for treating bacterial intestinal diseases
ES2726828T3 (es) 2013-05-28 2019-10-09 Morphochem Gmbh Administración de antibacterianos híbridos de oxazolidinona-quinolona
RU2675847C2 (ru) 2013-05-28 2018-12-25 Морфохем Акциенгезельшафт Фюр Комбинаторише Хеми Комбинированные терапевтические средства, содержащие оксазолидинон-хинолоны, предназначенные для лечения бактериальных инфекций
CN107286111B (zh) * 2016-03-30 2020-06-19 广东赛法洛药业有限公司 一种噁唑烷酮化合物的制备方法
CN107286182A (zh) * 2016-04-12 2017-10-24 李靖 新型噁唑烷酮‑氟喹诺酮衍生物及用途
US10087171B2 (en) 2016-12-19 2018-10-02 Actelion Pharmaceuticals Ltd Crystalline forms of cadazolid
GB201708606D0 (en) 2017-05-30 2017-07-12 King S College London Antibiotic resistance breakers
WO2019106693A1 (en) * 2017-11-29 2019-06-06 Bugworks Research India Pvt Ltd Anti-bacterial heterocyclic compounds and their synthesis
CN111087409B (zh) * 2018-10-24 2021-06-08 江阴安博生物医药有限公司 一种喹诺酮类化合物及其制备方法和应用
CN117567455A (zh) * 2019-12-11 2024-02-20 华创合成制药股份有限公司 一种新型噁唑烷酮类化合物及其合成方法和应用

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SE444566B (sv) * 1977-09-20 1986-04-21 Bellon Labor Sa Roger 7-dialkylamin-6-halogen-4-oxo-1,4-dihydrokinolin-3-karboxylsyra, forfarande for framstellning derav och farmaceutiskt preparat derav
DE69019859T2 (de) * 1989-03-30 1995-10-05 Wakunaga Seiyaku Kk Chinolon-Derivate und deren Salze, Verfahren zu deren Herstellung und diese enthaltende antibakterielle Wirkstoffe.
SK283420B6 (sk) * 1992-05-08 2003-07-01 Pharmacia & Upjohn Company Antimikrobiálne oxazolidinóny obsahujúce substituované diazínové skupiny
MY115155A (en) 1993-09-09 2003-04-30 Upjohn Co Substituted oxazine and thiazine oxazolidinone antimicrobials.
JP3933198B2 (ja) * 1994-10-26 2007-06-20 ファルマシア・アンド・アップジョン・カンパニー フェニルオキサゾリジノン抗菌剤
CA2245179A1 (en) * 1996-01-31 1997-08-07 Ube Industries Limited Remedies or preventives for aids
ES2166073T3 (es) * 1996-04-11 2002-04-01 Upjohn Co Procedimiento para preparar oxazolidinonas.
GB9614236D0 (en) * 1996-07-06 1996-09-04 Zeneca Ltd Chemical compounds

Also Published As

Publication number Publication date
NZ530206A (en) 2005-07-29
CO5540387A2 (es) 2005-07-29
HRP20031063A2 (en) 2004-04-30
SK572004A3 (en) 2004-08-03
MA27046A1 (fr) 2004-12-20
IS7088A (is) 2003-12-22
PL365476A1 (en) 2005-01-10
US20040147545A1 (en) 2004-07-29
PE20030134A1 (es) 2003-04-04
OA12639A (en) 2006-06-15
ES2186550B2 (es) 2003-11-16
CZ2004101A3 (cs) 2004-07-14
JP2004521147A (ja) 2004-07-15
AP2003002942A0 (en) 2003-12-24
MXPA04000185A (es) 2004-03-18
BG108498A (en) 2005-03-31
HUP0400370A2 (hu) 2004-08-30
CR7195A (es) 2004-03-05
WO2003002560A1 (en) 2003-01-09
EA200400086A1 (ru) 2004-06-24
CA2450982A1 (en) 2003-01-09
ES2186550A1 (es) 2003-05-01
CN1520412A (zh) 2004-08-11
EP1401834A1 (en) 2004-03-31
IL159434A0 (en) 2004-06-01
EE200400004A (et) 2004-02-16
BR0210667A (pt) 2004-10-05
KR20040030712A (ko) 2004-04-09
AR035254A1 (es) 2004-05-05

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