NO20041792L - Peptider som virker bade som GLP-1-reseptoragonister og glukagonreseptorantagonister og deres farmakologiske fremgangsmater for anvendelse - Google Patents

Peptider som virker bade som GLP-1-reseptoragonister og glukagonreseptorantagonister og deres farmakologiske fremgangsmater for anvendelse

Info

Publication number
NO20041792L
NO20041792L NO20041792A NO20041792A NO20041792L NO 20041792 L NO20041792 L NO 20041792L NO 20041792 A NO20041792 A NO 20041792A NO 20041792 A NO20041792 A NO 20041792A NO 20041792 L NO20041792 L NO 20041792L
Authority
NO
Norway
Prior art keywords
glp
pharmacological methods
receptor antagonists
peptides acting
receptor agonists
Prior art date
Application number
NO20041792A
Other languages
English (en)
Inventor
Clark Pan
James Whelan
Kevin Clairmont
Original Assignee
Bayer Pharmaceuticals Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Pharmaceuticals Corp filed Critical Bayer Pharmaceuticals Corp
Publication of NO20041792L publication Critical patent/NO20041792L/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K16/00—Immunoglobulins [IG], e.g. monoclonal or polyclonal antibodies
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • C07K14/575—Hormones
    • C07K14/605—Glucagons
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/48—Drugs for disorders of the endocrine system of the pancreatic hormones
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Diabetes (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Endocrinology (AREA)
  • Genetics & Genomics (AREA)
  • Biochemistry (AREA)
  • Hematology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Molecular Biology (AREA)
  • Obesity (AREA)
  • Biophysics (AREA)
  • Zoology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Toxicology (AREA)
  • Emergency Medicine (AREA)
  • Child & Adolescent Psychology (AREA)
  • Immunology (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Micro-Organisms Or Cultivation Processes Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
NO20041792A 2001-10-05 2004-05-03 Peptider som virker bade som GLP-1-reseptoragonister og glukagonreseptorantagonister og deres farmakologiske fremgangsmater for anvendelse NO20041792L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US32773001P 2001-10-05 2001-10-05
PCT/US2002/031693 WO2003040309A2 (en) 2001-10-05 2002-10-04 Peptides acting as both glp-1 receptor agonists and glucagon receptor antagonists and their pharmacological methods of use

Publications (1)

Publication Number Publication Date
NO20041792L true NO20041792L (no) 2004-07-02

Family

ID=23277790

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20041792A NO20041792L (no) 2001-10-05 2004-05-03 Peptider som virker bade som GLP-1-reseptoragonister og glukagonreseptorantagonister og deres farmakologiske fremgangsmater for anvendelse

Country Status (27)

Country Link
US (6) US7399745B2 (no)
EP (1) EP1436330A4 (no)
JP (1) JP2005508639A (no)
KR (1) KR20050034580A (no)
CN (1) CN1326876C (no)
AR (1) AR036711A1 (no)
BR (1) BR0213132A (no)
CA (1) CA2462462A1 (no)
CO (1) CO5570710A2 (no)
DO (1) DOP2002000475A (no)
EC (2) ECSP024346A (no)
HN (1) HN2002000282A (no)
HR (1) HRP20040327A2 (no)
HU (1) HUP0401797A2 (no)
IL (1) IL160706A0 (no)
MA (1) MA26228A1 (no)
MX (1) MXPA04002140A (no)
MY (1) MY138267A (no)
NO (1) NO20041792L (no)
NZ (1) NZ532685A (no)
PE (1) PE20030850A1 (no)
PL (1) PL368760A1 (no)
RU (1) RU2334761C2 (no)
SG (2) SG149693A1 (no)
UY (1) UY27469A1 (no)
WO (1) WO2003040309A2 (no)
ZA (1) ZA200403322B (no)

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US8450270B2 (en) * 2008-06-17 2013-05-28 Indiana University Research And Technology Corporation Glucagon analogs exhibiting enhanced solubility and stability in physiological pH buffers
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PT2373681T (pt) 2008-12-10 2017-04-11 Glaxosmithkline Llc Composições farmacêuticas de albiglutida
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US8691763B2 (en) 2010-05-04 2014-04-08 Glaxosmithkline Llc Methods for treating or preventing cardiovascular disorders and providing cardiovascular protection
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MX2012013001A (es) 2010-05-13 2013-02-26 Univ Indiana Res & Tech Corp Peptidos de la superfamilia de glucagon que presentan actividad del receptor nuclear de hormonas.
EP2588126A4 (en) 2010-06-24 2015-07-08 Univ Indiana Res & Tech Corp AMID-BASED GLUCAGON SUPERFAMILY PEPTIDE PRODRUGS
US8507428B2 (en) 2010-12-22 2013-08-13 Indiana University Research And Technology Corporation Glucagon analogs exhibiting GIP receptor activity
CA2828761C (en) * 2011-03-04 2017-04-04 Becton, Dickinson And Company Blood collection device containing lysophospholipase inhibitor
RS56173B1 (sr) 2011-06-22 2017-11-30 Univ Indiana Res & Tech Corp Koagonisti receptora za glukagon/glp-1 receptora
KR20140043793A (ko) 2011-06-22 2014-04-10 인디애나 유니버시티 리서치 앤드 테크놀로지 코퍼레이션 글루카곤/glp-1 수용체 공동-작용물질
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CN104583232B (zh) 2012-06-21 2018-04-13 印第安纳大学研究及科技有限公司 展现gip受体活性的胰高血糖素类似物
JP6538645B2 (ja) 2013-03-14 2019-07-03 インディアナ ユニバーシティー リサーチ アンド テクノロジー コーポレーションＩｎｄｉａｎａ Ｕｎｉｖｅｒｓｉｔｙ Ｒｅｓｅａｒｃｈ Ａｎｄ Ｔｅｃｈｎｏｌｏｇｙ Ｃｏｒｐｏｒａｔｉｏｎ インスリン‐インクレチン複合物
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Also Published As

Publication number Publication date
HN2002000282A (es) 2002-12-12
US7488714B2 (en) 2009-02-10
US20060003418A1 (en) 2006-01-05
IL160706A0 (en) 2004-08-31
SG158736A1 (en) 2010-02-26
US20060003934A1 (en) 2006-01-05
US7494978B2 (en) 2009-02-24
CN1564828A (zh) 2005-01-12
WO2003040309A2 (en) 2003-05-15
ECSP045094A (es) 2004-06-28
MA26228A1 (fr) 2004-07-01
CN1326876C (zh) 2007-07-18
US7399745B2 (en) 2008-07-15
AR036711A1 (es) 2004-09-29
DOP2002000475A (es) 2003-06-30
CA2462462A1 (en) 2003-05-15
PE20030850A1 (es) 2003-10-31
SG149693A1 (en) 2009-02-27
WO2003040309A3 (en) 2003-12-18
UY27469A1 (es) 2003-04-30
US20050288248A1 (en) 2005-12-29
MXPA04002140A (es) 2005-03-07
US20060003417A1 (en) 2006-01-05
US7488715B2 (en) 2009-02-10
CO5570710A2 (es) 2005-10-31
HUP0401797A2 (en) 2006-08-28
JP2005508639A (ja) 2005-04-07
MY138267A (en) 2009-05-29
ZA200403322B (en) 2005-05-03
EP1436330A2 (en) 2004-07-14
HK1073117A1 (zh) 2005-09-23
EP1436330A4 (en) 2006-01-18
KR20050034580A (ko) 2005-04-14
NZ532685A (en) 2006-02-24
RU2334761C2 (ru) 2008-09-27
BR0213132A (pt) 2004-10-19
US20050153890A1 (en) 2005-07-14
US7488716B2 (en) 2009-02-10
RU2004114243A (ru) 2005-05-10
ECSP024346A (es) 2003-05-26
HRP20040327A2 (en) 2007-11-30
PL368760A1 (en) 2005-04-04
US20060003419A1 (en) 2006-01-05

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