NO20044135L - Piperazinyl-, piperidinyl- og morfolinylderivater som nye inhibitorer av histon-deacetylase - Google Patents

Piperazinyl-, piperidinyl- og morfolinylderivater som nye inhibitorer av histon-deacetylase

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Publication number
NO20044135L
NO20044135L NO20044135A NO20044135A NO20044135L NO 20044135 L NO20044135 L NO 20044135L NO 20044135 A NO20044135 A NO 20044135A NO 20044135 A NO20044135 A NO 20044135A NO 20044135 L NO20044135 L NO 20044135L
Authority
NO
Norway
Prior art keywords
piperazinyl
piperidinyl
histone deacetylase
novel inhibitors
morpholinyl derivatives
Prior art date
Application number
NO20044135A
Other languages
English (en)
Norwegian (no)
Inventor
Kristof Van Emelen
Original Assignee
Janssen Pharmaceutica Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv
Publication of NO20044135L publication Critical patent/NO20044135L/no

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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
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    • A61K31/402—1-aryl substituted, e.g. piretanide
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NO20044135A 2002-03-13 2004-09-29 Piperazinyl-, piperidinyl- og morfolinylderivater som nye inhibitorer av histon-deacetylase NO20044135L (no)

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