NO20050748L - Heterosykliske aromatiske forbindelser anvendelige som veksthormonsekretagoger - Google Patents

Heterosykliske aromatiske forbindelser anvendelige som veksthormonsekretagoger

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Publication number
NO20050748L
NO20050748L NO20050748A NO20050748A NO20050748L NO 20050748 L NO20050748 L NO 20050748L NO 20050748 A NO20050748 A NO 20050748A NO 20050748 A NO20050748 A NO 20050748A NO 20050748 L NO20050748 L NO 20050748L
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Norway
Prior art keywords
growth hormone
aromatic compounds
compounds useful
heterocyclic aromatic
hormone secretagogues
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NO20050748A
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English (en)
Other versions
NO332370B1 (no
Inventor
James J Li
Richard B Sulsky
Joseph A Tino
William R Ewing
Guixue Yu
Jun Li
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Bristol Myers Squibb Co
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First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=31981567&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=NO20050748(L) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Bristol Myers Squibb Co filed Critical Bristol Myers Squibb Co
Publication of NO20050748L publication Critical patent/NO20050748L/no
Publication of NO332370B1 publication Critical patent/NO332370B1/no

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
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    • A61P13/00—Drugs for disorders of the urinary system
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/12—Drugs for disorders of the urinary system of the kidneys
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    • A61P19/00—Drugs for skeletal disorders
    • A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
    • A61P19/10—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease for osteoporosis
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    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/54—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings condensed with carbocyclic rings or ring systems
    • C07D231/56—Benzopyrazoles; Hydrogenated benzopyrazoles
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D261/00—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings
    • C07D261/20—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings condensed with carbocyclic rings or ring systems
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    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
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    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04—Ortho-condensed systems

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  • Health & Medical Sciences (AREA)
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  • Obesity (AREA)
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Abstract

Heterosykliske aromatiske forbindelser anvendelige som veksthormonsekretagoger Det tilveiebringes nye heterocj4[liske aromatiske forbindelser som er anvendelige for å stimulere endogen produksjon eller frigjøring av veksthormon, hvor nevnte forbindelser har den generelle struktur med formel I; hvor Ri, Ri', R2, R3, R4, Xa, Y, Z og n er som beskrevet her. Forbindelsene gitt her er anvendelige for behandling av fedme, osteoporose (forbedrer bentetthet) og forbedre mnskebnasse og muskelstyrke.
NO20050748A 2002-09-04 2005-02-11 Heterocykliske aromatiske forbindelser, farmasoytisk preparat inneholdende slike samt anvendelse av slike for fremstilling av farmasoytisk preparat forbehandling av sykdom NO332370B1 (no)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US40809902P 2002-09-04 2002-09-04
US49164503P 2003-07-31 2003-07-31
PCT/US2003/027513 WO2004021984A2 (en) 2002-09-04 2003-09-02 Heterocyclic aromatic compounds useful as growth hormone secretagogues

Publications (2)

Publication Number Publication Date
NO20050748L true NO20050748L (no) 2005-03-30
NO332370B1 NO332370B1 (no) 2012-09-03

Family

ID=31981567

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20050748A NO332370B1 (no) 2002-09-04 2005-02-11 Heterocykliske aromatiske forbindelser, farmasoytisk preparat inneholdende slike samt anvendelse av slike for fremstilling av farmasoytisk preparat forbehandling av sykdom

Country Status (30)

Country Link
US (8) US7166596B2 (no)
EP (2) EP1551511B1 (no)
JP (1) JP4658600B2 (no)
KR (3) KR20110003592A (no)
CN (2) CN1678372A (no)
AR (1) AR041143A1 (no)
AU (1) AU2003270065B2 (no)
BR (1) BR0314024A (no)
CA (1) CA2496842C (no)
CY (2) CY1120250T1 (no)
DK (2) DK2570414T3 (no)
ES (2) ES2644265T3 (no)
GE (1) GEP20074019B (no)
HR (1) HRP20050188B1 (no)
HU (2) HUE035498T2 (no)
IL (5) IL166802A (no)
IS (1) IS7719A (no)
LT (2) LT1551511T (no)
MX (1) MXPA05002301A (no)
MY (1) MY139563A (no)
NO (1) NO332370B1 (no)
NZ (1) NZ538166A (no)
PE (1) PE20040997A1 (no)
PL (1) PL219563B1 (no)
PT (2) PT2570414T (no)
RS (2) RS55124B1 (no)
RU (1) RU2382042C2 (no)
SI (2) SI1551511T1 (no)
TW (2) TWI362389B (no)
WO (1) WO2004021984A2 (no)

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