NO20053144L - Chk-, Pdk- og Akt-inhibitorpyrimidiner, deres fremstilling og anvendelse som famasoytiske midler. - Google Patents

Chk-, Pdk- og Akt-inhibitorpyrimidiner, deres fremstilling og anvendelse som famasoytiske midler.

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Publication number
NO20053144L
NO20053144L NO20053144A NO20053144A NO20053144L NO 20053144 L NO20053144 L NO 20053144L NO 20053144 A NO20053144 A NO 20053144A NO 20053144 A NO20053144 A NO 20053144A NO 20053144 L NO20053144 L NO 20053144L
Authority
NO
Norway
Prior art keywords
preparation
famasoytic
pdk
chk
pyrimidines
Prior art date
Application number
NO20053144A
Other languages
English (en)
Norwegian (no)
Other versions
NO20053144D0 (no
Inventor
Peter Esperling
Damian O Arnaiz
Monica J Kochanny
Gary B Phillips
Brad O Buckman
Christoph Huwe
Dirk Kosemund
Joachim Kuhnke
Martina Schafer
Judi Bryant
Shendong Yuan
Hans Briem
Ulf Bomer
Seock-Kyu Khim
Lars Wortmann
Emil Eckle
Richard Feldman
Original Assignee
Schering Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Schering Ag filed Critical Schering Ag
Publication of NO20053144L publication Critical patent/NO20053144L/no
Publication of NO20053144D0 publication Critical patent/NO20053144D0/no

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    • C07D239/24Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/47One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine
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NO20053144A 2002-11-28 2005-06-27 Chk-, Pdk- og Akt-inhibitorpyrimidiner, deres fremstilling og anvendelse som famasoytiske midler. NO20053144D0 (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP02026607 2002-11-28
PCT/EP2003/013443 WO2004048343A1 (en) 2002-11-28 2003-11-28 Chk-, pdk- and akt-inhibitory pyrimidines, their production and use as pharmaceutical agents

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NO20053144L true NO20053144L (no) 2005-06-27
NO20053144D0 NO20053144D0 (no) 2005-06-27

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NO20053144A NO20053144D0 (no) 2002-11-28 2005-06-27 Chk-, Pdk- og Akt-inhibitorpyrimidiner, deres fremstilling og anvendelse som famasoytiske midler.

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US (1) US7504410B2 (is)
EP (1) EP1565446A1 (is)
JP (1) JP2006508997A (is)
KR (1) KR20050084027A (is)
CN (1) CN1717396A (is)
AU (1) AU2003288198A1 (is)
BR (1) BR0316680A (is)
CA (1) CA2502970A1 (is)
EA (1) EA200500721A1 (is)
EC (1) ECSP055899A (is)
HR (1) HRP20050601A2 (is)
IL (1) IL168102A0 (is)
IS (1) IS7881A (is)
MX (1) MXPA05005547A (is)
NO (1) NO20053144D0 (is)
NZ (1) NZ539823A (is)
PL (1) PL377795A1 (is)
RS (1) RS20050363A (is)
WO (1) WO2004048343A1 (is)
ZA (1) ZA200505184B (is)

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KR100874791B1 (ko) * 2001-05-29 2008-12-18 바이엘 쉐링 파마 악티엔게젤샤프트 Cdk-억제 피리미딘, 그의 제조방법 및 약제로서의 용도
TWI329105B (en) 2002-02-01 2010-08-21 Rigel Pharmaceuticals Inc 2,4-pyrimidinediamine compounds and their uses
ES2445208T3 (es) 2002-07-29 2014-02-28 Rigel Pharmaceuticals, Inc. Compuestos de 2,4-pirimidindiamina para uso en métodos para tratar o prevenir enfermedades autoinmunitarias
UA80767C2 (en) * 2002-12-20 2007-10-25 Pfizer Prod Inc Pyrimidine derivatives for the treatment of abnormal cell growth
US7157455B2 (en) 2003-02-10 2007-01-02 Hoffmann-La Roche Inc. 4-Aminopyrimidine-5-one derivatives
EP1624873A2 (en) * 2003-04-28 2006-02-15 AB Science Use of tyrosine kinase inhibitors for treating cerebral ischemia
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US7504410B2 (en) 2009-03-17
AU2003288198A1 (en) 2004-06-18
PL377795A1 (pl) 2006-02-20
CA2502970A1 (en) 2004-06-10
EP1565446A1 (en) 2005-08-24
IL168102A0 (en) 2009-02-11
JP2006508997A (ja) 2006-03-16
BR0316680A (pt) 2005-10-18
MXPA05005547A (es) 2005-07-26
WO2004048343A1 (en) 2004-06-10
KR20050084027A (ko) 2005-08-26
NO20053144D0 (no) 2005-06-27
HRP20050601A2 (en) 2005-10-31
EA200500721A1 (ru) 2005-12-29
ECSP055899A (es) 2005-11-22
RS20050363A (sr) 2007-11-15
US20040186118A1 (en) 2004-09-23
ZA200505184B (en) 2006-09-27
NZ539823A (en) 2008-04-30
IS7881A (is) 2005-06-02

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