NO20061656L - 2,4 di(hetero)-arylamino-pyrimidin derivaer som ZAP-70 og/aller SYK inhibitorer - Google Patents

2,4 di(hetero)-arylamino-pyrimidin derivaer som ZAP-70 og/aller SYK inhibitorer

Info

Publication number
NO20061656L
NO20061656L NO20061656A NO20061656A NO20061656L NO 20061656 L NO20061656 L NO 20061656L NO 20061656 A NO20061656 A NO 20061656A NO 20061656 A NO20061656 A NO 20061656A NO 20061656 L NO20061656 L NO 20061656L
Authority
NO
Norway
Prior art keywords
zap
arylamino
hetero
pyrimidine derivatives
syk inhibitors
Prior art date
Application number
NO20061656A
Other languages
English (en)
Norwegian (no)
Inventor
Rudolf Duthaler
Gebhard Thoma
Nigel Graham Cooke
Gerhard Zenke
Klaus Hinterding
Anette Von Matt
Rolf Baentell
Marie Claude Bernhard
Peter Buchlmayer
Maurice Van Eis
Louis Walliser
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of NO20061656L publication Critical patent/NO20061656L/no

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    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/48—Two nitrogen atoms
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NO20061656A 2003-09-16 2006-04-11 2,4 di(hetero)-arylamino-pyrimidin derivaer som ZAP-70 og/aller SYK inhibitorer NO20061656L (no)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GBGB0321710.6A GB0321710D0 (en) 2003-09-16 2003-09-16 Organic compounds
GBGB0414440.8A GB0414440D0 (en) 2003-09-16 2004-06-28 Organic compounds
PCT/EP2004/010348 WO2005026158A1 (fr) 2003-09-16 2004-09-15 Derives de 2,4-di(hetero)-arylamino-pyrimidine comme inhibiteurs des kinases zap-70 et/ou syk

Publications (1)

Publication Number Publication Date
NO20061656L true NO20061656L (no) 2006-06-16

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NO20061656A NO20061656L (no) 2003-09-16 2006-04-11 2,4 di(hetero)-arylamino-pyrimidin derivaer som ZAP-70 og/aller SYK inhibitorer

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Country Link
US (2) US7671063B2 (fr)
EP (2) EP2266977B1 (fr)
JP (1) JP4504375B2 (fr)
KR (1) KR100813384B1 (fr)
CN (2) CN102260248A (fr)
AR (1) AR045747A1 (fr)
AT (1) ATE498623T1 (fr)
AU (1) AU2004272283B9 (fr)
BR (1) BRPI0414480A (fr)
CA (1) CA2538909A1 (fr)
DE (1) DE602004031436D1 (fr)
EC (1) ECSP066424A (fr)
ES (2) ES2361412T3 (fr)
GB (2) GB0321710D0 (fr)
IL (1) IL174217A0 (fr)
IS (1) IS8402A (fr)
MA (1) MA28076A1 (fr)
MX (1) MXPA06002966A (fr)
NO (1) NO20061656L (fr)
PE (1) PE20050429A1 (fr)
PL (1) PL1664035T3 (fr)
PT (1) PT1664035E (fr)
RU (1) RU2403251C2 (fr)
SG (1) SG132676A1 (fr)
TN (1) TNSN06083A1 (fr)
TW (1) TW200521118A (fr)
WO (1) WO2005026158A1 (fr)
ZA (1) ZA200601963B (fr)

Families Citing this family (135)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TWI329105B (en) 2002-02-01 2010-08-21 Rigel Pharmaceuticals Inc 2,4-pyrimidinediamine compounds and their uses
GB0206215D0 (en) * 2002-03-15 2002-05-01 Novartis Ag Organic compounds
BR0313059B8 (pt) 2002-07-29 2021-07-27 Rigel Pharmaceuticals composto, e, composição farmacêutica
GB0305929D0 (en) * 2003-03-14 2003-04-23 Novartis Ag Organic compounds
CN102358738A (zh) 2003-07-30 2012-02-22 里格尔药品股份有限公司 2,4-嘧啶二胺化合物及其预防和治疗自体免疫疾病的用途
TWI378923B (en) * 2003-08-15 2012-12-11 Novartis Ag Pyrimidine derivatives
GB0321710D0 (en) * 2003-09-16 2003-10-15 Novartis Ag Organic compounds
JP4801096B2 (ja) 2005-01-19 2011-10-26 ライジェル ファーマシューティカルズ， インコーポレイテッド ２，４−ピリミジンジアミン化合物のプロドラッグおよびそれらの使用
AU2006209216A1 (en) * 2005-01-25 2006-08-03 Galenea Corp Substituted arylamine compounds and their use as 5-HT6 modulators
WO2006129100A1 (fr) * 2005-06-03 2006-12-07 Glaxo Group Limited Nouveaux composes
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