NO20061978L - Imidazopyridinsubstituerte tropanderivater med CCR5-reseptorantagonist aktivitet for behandling av HIV og inflammasjon - Google Patents

Imidazopyridinsubstituerte tropanderivater med CCR5-reseptorantagonist aktivitet for behandling av HIV og inflammasjon

Info

Publication number: NO20061978L
Authority: NO; Norway
Prior art keywords: treatment; hiv; imidazopyridine; inflammation; receptor antagonist
Prior art date: 2003-10-03

Application number

NO20061978A

Other languages

English (en)

Norwegian (no)

Inventor

Paul Anthony Stupple

Original Assignee

Pfizer

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2003-10-03

Filing date

2006-05-03

Publication date

2006-07-03

2003-10-03 Priority claimed from GBGB0323236.0A external-priority patent/GB0323236D0/en

2003-10-27 Priority claimed from GB0325020A external-priority patent/GB0325020D0/en

2004-08-19 Priority claimed from GB0418566A external-priority patent/GB0418566D0/en

2006-05-03 Application filed by Pfizer filed Critical Pfizer

2006-07-03 Publication of NO20061978L publication Critical patent/NO20061978L/no

Links

230000000694 effects Effects 0.000 title abstract 2
206010061218 Inflammation Diseases 0.000 title 1
239000003067 chemokine receptor CCR5 antagonist Substances 0.000 title 1
230000004054 inflammatory process Effects 0.000 title 1
150000003813 tropane derivatives Chemical class 0.000 title 1
102000004274 CCR5 Receptors Human genes 0.000 abstract 2
108010017088 CCR5 Receptors Proteins 0.000 abstract 2
150000001875 compounds Chemical class 0.000 abstract 2
102000019034 Chemokines Human genes 0.000 abstract 1
108010012236 Chemokines Proteins 0.000 abstract 1
239000005557 antagonist Substances 0.000 abstract 1
208000015181 infectious disease Diseases 0.000 abstract 1
208000027866 inflammatory disease Diseases 0.000 abstract 1
241001430294 unidentified retrovirus Species 0.000 abstract 1

Classifications

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- C07—ORGANIC CHEMISTRY
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
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- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/4164—1,3-Diazoles
- A61K31/4188—1,3-Diazoles condensed with other heterocyclic ring systems, e.g. biotin, sorbinil
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Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Organic Chemistry (AREA)
Veterinary Medicine (AREA)
Medicinal Chemistry (AREA)
Pharmacology & Pharmacy (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
General Chemical & Material Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Chemical Kinetics & Catalysis (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Virology (AREA)
Oncology (AREA)
Communicable Diseases (AREA)
Diabetes (AREA)
Immunology (AREA)
Cardiology (AREA)
Hematology (AREA)
Epidemiology (AREA)
Molecular Biology (AREA)
Heart & Thoracic Surgery (AREA)
Obesity (AREA)
Endocrinology (AREA)
Rheumatology (AREA)
Tropical Medicine & Parasitology (AREA)
Dermatology (AREA)
Urology & Nephrology (AREA)
Pulmonology (AREA)
Child & Adolescent Psychology (AREA)
Vascular Medicine (AREA)
Hospice & Palliative Care (AREA)
Biotechnology (AREA)
Biomedical Technology (AREA)
Neurology (AREA)
Neurosurgery (AREA)
Pain & Pain Management (AREA)

NO20061978A 2003-10-03 2006-05-03 Imidazopyridinsubstituerte tropanderivater med CCR5-reseptorantagonist aktivitet for behandling av HIV og inflammasjon NO20061978L (no)

Applications Claiming Priority (4)

Application Number	Priority Date	Filing Date	Title
GBGB0323236.0A GB0323236D0 (en)	2003-10-03	2003-10-03	Chemical compounds
GB0325020A GB0325020D0 (en)	2003-10-27	2003-10-27	Chemical compounds
GB0418566A GB0418566D0 (en)	2004-08-19	2004-08-19	Tropane derivatives
PCT/IB2004/003153 WO2005033107A1 (en)	2003-10-03	2004-09-28	Imidazopyridine substituted tropane derivatives with ccr5 receptor antagonist activity for the treatment of hiv and inflammation

Publications (1)

Publication Number	Publication Date
NO20061978L true NO20061978L (no)	2006-07-03

Family

ID=34426592

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
NO20061978A NO20061978L (no)	2003-10-03	2006-05-03	Imidazopyridinsubstituerte tropanderivater med CCR5-reseptorantagonist aktivitet for behandling av HIV og inflammasjon

Country Status (35)

Country	Link
US (2)	US7309790B2 (es)
EP (1)	EP1682545B1 (es)
JP (1)	JP4874107B2 (es)
KR (1)	KR100777885B1 (es)
AP (1)	AP2174A (es)
AR (1)	AR045856A1 (es)
AT (1)	ATE380813T1 (es)
AU (1)	AU2004278158B2 (es)
BR (1)	BRPI0414862A (es)
CA (1)	CA2540834C (es)
CY (1)	CY1107281T1 (es)
DE (1)	DE602004010708T2 (es)
DK (1)	DK1682545T3 (es)
EA (1)	EA009941B1 (es)
EC (1)	ECSP066475A (es)
ES (1)	ES2295924T3 (es)
GE (1)	GEP20084417B (es)
HN (1)	HN2004000383A (es)
HR (1)	HRP20080052T3 (es)
IL (1)	IL174208A0 (es)
MA (1)	MA28080A1 (es)
MX (1)	MXPA06003749A (es)
MY (1)	MY137609A (es)
NO (1)	NO20061978L (es)
NZ (1)	NZ545837A (es)
OA (1)	OA13266A (es)
PA (1)	PA8614301A1 (es)
PE (1)	PE20050961A1 (es)
PL (1)	PL1682545T3 (es)
PT (1)	PT1682545E (es)
RS (1)	RS20060198A (es)
SI (1)	SI1682545T1 (es)
TW (1)	TWI280244B (es)
UY (1)	UY28546A1 (es)
WO (1)	WO2005033107A1 (es)

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JP2010043063A (ja)	2008-05-09	2010-02-25	Agency For Science Technology & Research	川崎病の診断及び治療
CN102573475B (zh)	2009-08-14	2016-01-20	欧科生医股份有限公司	神经激肽-1拮抗剂的静脉内制剂
US20130023496A1 (en)	2010-04-02	2013-01-24	Randy Tressler	Combination Therapy Comprising A CCR5 Antagonist, A HIV-1 Protease Inhibtior and a Pharmacokinetic Enhancer
WO2012061428A2 (en)	2010-11-01	2012-05-10	Portola Pharmaceuticals, Inc.	Nicotinamides as jak kinase modulators
US20140271680A1 (en)	2011-08-12	2014-09-18	Universite Paris-Est Creteil Val De Marne	Methods and pharmaceutical compositions for treatment of pulmonary hypertension
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JP6224256B2 (ja) *	2013-09-25	2017-11-01	マリンクロッドエルエルシー	放射ヨウ素標識された３−フルオロプロピル−ＮＯＲ−β−ＣＩＴの調製
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2004
- 2004-09-28 HR HR20080052T patent/HRP20080052T3/xx unknown
- 2004-09-28 EA EA200600480A patent/EA009941B1/ru not_active IP Right Cessation
- 2004-09-28 EP EP04769496A patent/EP1682545B1/en not_active Expired - Lifetime
- 2004-09-28 US US10/953,136 patent/US7309790B2/en not_active Expired - Fee Related
- 2004-09-28 MX MXPA06003749A patent/MXPA06003749A/es active IP Right Grant
- 2004-09-28 AU AU2004278158A patent/AU2004278158B2/en not_active Ceased
- 2004-09-28 DE DE602004010708T patent/DE602004010708T2/de not_active Expired - Lifetime
- 2004-09-28 JP JP2006530737A patent/JP4874107B2/ja not_active Expired - Fee Related
- 2004-09-28 OA OA1200600114A patent/OA13266A/en unknown
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- 2004-09-28 KR KR1020067006293A patent/KR100777885B1/ko not_active Expired - Fee Related
- 2004-09-28 WO PCT/IB2004/003153 patent/WO2005033107A1/en not_active Ceased
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- 2004-09-28 PT PT04769496T patent/PT1682545E/pt unknown
- 2004-09-28 DK DK04769496T patent/DK1682545T3/da active
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- 2004-09-28 NZ NZ545837A patent/NZ545837A/en not_active IP Right Cessation
- 2004-09-28 AT AT04769496T patent/ATE380813T1/de active
- 2004-09-29 HN HN2004000383A patent/HN2004000383A/es unknown
- 2004-09-29 TW TW093129475A patent/TWI280244B/zh not_active IP Right Cessation
- 2004-10-01 AR ARP040103581A patent/AR045856A1/es not_active Application Discontinuation
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- 2004-10-01 UY UY28546A patent/UY28546A1/es unknown
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- 2004-10-01 MY MYPI20044043A patent/MY137609A/en unknown
2006
- 2006-03-09 IL IL174208A patent/IL174208A0/en unknown
- 2006-04-03 MA MA28906A patent/MA28080A1/fr unknown
- 2006-04-03 EC EC2006006475A patent/ECSP066475A/es unknown
- 2006-05-03 NO NO20061978A patent/NO20061978L/no not_active Application Discontinuation
2007
- 2007-08-27 US US11/845,500 patent/US7790740B2/en not_active Expired - Fee Related
2008
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Also Published As

Publication number	Publication date
AU2004278158B2 (en)	2009-08-13
SI1682545T1 (sl)	2008-04-30
HRP20080052T3 (hr)	2008-02-29
GEP20084417B (en)	2008-07-10
BRPI0414862A (pt)	2006-11-28
KR20060070571A (ko)	2006-06-23
IL174208A0 (en)	2006-08-01
CY1107281T1 (el)	2012-11-21
KR100777885B1 (ko)	2007-11-28
MXPA06003749A (es)	2006-06-14
PL1682545T3 (pl)	2008-04-30
JP4874107B2 (ja)	2012-02-15
WO2005033107A1 (en)	2005-04-14
EA009941B1 (ru)	2008-04-28
TWI280244B (en)	2007-05-01
EP1682545A1 (en)	2006-07-26
UY28546A1 (es)	2005-05-31
US20080045563A1 (en)	2008-02-21
HN2004000383A (es)	2008-10-14
US7309790B2 (en)	2007-12-18
NZ545837A (en)	2009-12-24
PA8614301A1 (es)	2005-05-10
DK1682545T3 (da)	2008-03-17
OA13266A (en)	2007-01-31
MA28080A1 (fr)	2006-08-01
CA2540834C (en)	2010-06-22
MY137609A (en)	2009-02-27
TW200519112A (en)	2005-06-16
PT1682545E (pt)	2008-02-11
AU2004278158A1 (en)	2005-04-14
DE602004010708T2 (de)	2008-12-04
RS20060198A (sr)	2008-09-29
JP2007507483A (ja)	2007-03-29
EA200600480A1 (ru)	2006-08-25
ECSP066475A (es)	2006-10-10
US20050131011A1 (en)	2005-06-16
CA2540834A1 (en)	2005-04-14
ES2295924T3 (es)	2008-04-16
US7790740B2 (en)	2010-09-07
EP1682545B1 (en)	2007-12-12
ATE380813T1 (de)	2007-12-15
AP2174A (en)	2010-11-20
DE602004010708D1 (de)	2008-01-24
AP2006003580A0 (en)	2006-04-30
AR045856A1 (es)	2005-11-16
PE20050961A1 (es)	2005-11-29

Legal Events

Date	Code	Title	Description
2013-04-22	FC2A	Withdrawal, rejection or dismissal of laid open patent application

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