NO20071871L - Fosfoindoler som HIV-inhibitorer. - Google Patents

Fosfoindoler som HIV-inhibitorer.

Info

Publication number
NO20071871L
NO20071871L NO20071871A NO20071871A NO20071871L NO 20071871 L NO20071871 L NO 20071871L NO 20071871 A NO20071871 A NO 20071871A NO 20071871 A NO20071871 A NO 20071871A NO 20071871 L NO20071871 L NO 20071871L
Authority
NO
Norway
Prior art keywords
phosphoindoles
hiv inhibitors
compounds
hiv
retroviral
Prior art date
Application number
NO20071871A
Other languages
English (en)
Inventor
Richard Storer
Cyril Dousson
Francois-Rene Alexandre
Arlene Roland
Original Assignee
Idenix Cayman Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=36407947&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=NO20071871(L) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Idenix Cayman Ltd filed Critical Idenix Cayman Ltd
Publication of NO20071871L publication Critical patent/NO20071871L/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/6561—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing systems of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring or ring system, with or without other non-condensed hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/6558—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing at least two different or differently substituted hetero rings neither condensed among themselves nor condensed with a common carbocyclic ring or ring system
    • C07F9/65586—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing at least two different or differently substituted hetero rings neither condensed among themselves nor condensed with a common carbocyclic ring or ring system at least one of the hetero rings does not contain nitrogen as ring hetero atom
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • A61P31/18—Antivirals for RNA viruses for HIV
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/553—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having one nitrogen atom as the only ring hetero atom
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/553—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having one nitrogen atom as the only ring hetero atom
    • C07F9/572—Five-membered rings
    • C07F9/5728—Five-membered rings condensed with carbocyclic rings or carbocyclic ring systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/6558—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing at least two different or differently substituted hetero rings neither condensed among themselves nor condensed with a common carbocyclic ring or ring system
    • C07F9/65583—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing at least two different or differently substituted hetero rings neither condensed among themselves nor condensed with a common carbocyclic ring or ring system each of the hetero rings containing nitrogen as ring hetero atom

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Molecular Biology (AREA)
  • Biochemistry (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Virology (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • AIDS & HIV (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Indole Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

Abstract

3-fosfoindolforbindelser for behandling av retrovirale infeksjoner og særlig for HTV, er beskrevet.Også inkludert er sammensetninger som innbefatter 3-fosfoindolderivatene, alene eller i kombinasjon med ett eller flere andre antiretrovirale midler, fremgangsmåter for deres fremstilling og fremgangsmåter for fremstilling av et medikament som inkorporerer disse forbindelsene.
NO20071871A 2004-09-17 2007-04-12 Fosfoindoler som HIV-inhibitorer. NO20071871L (no)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US61106104P 2004-09-17 2004-09-17
US71144505P 2005-08-25 2005-08-25
US71156505P 2005-08-26 2005-08-26
PCT/IB2005/004063 WO2006054182A2 (en) 2004-09-16 2005-09-16 Phosphoindoles as hiv inhibitors

Publications (1)

Publication Number Publication Date
NO20071871L true NO20071871L (no) 2007-05-15

Family

ID=36407947

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20071871A NO20071871L (no) 2004-09-17 2007-04-12 Fosfoindoler som HIV-inhibitorer.

Country Status (24)

Country Link
US (2) US7534809B2 (no)
EP (3) EP1961757B1 (no)
JP (1) JP5031569B2 (no)
KR (1) KR101242962B1 (no)
CN (1) CN102304150B (no)
AT (2) ATE479693T1 (no)
AU (1) AU2005305609B2 (no)
BR (1) BRPI0515344A (no)
CA (1) CA2583409C (no)
CY (1) CY1109440T1 (no)
DE (2) DE602005011031D1 (no)
DK (1) DK1799696T3 (no)
ES (1) ES2320252T3 (no)
HR (1) HRP20090086T3 (no)
IL (1) IL181909A0 (no)
MX (1) MX2007003040A (no)
NO (1) NO20071871L (no)
NZ (1) NZ554232A (no)
PL (1) PL1799696T3 (no)
PT (1) PT1799696E (no)
RS (1) RS50981B (no)
SG (1) SG155939A1 (no)
SI (1) SI1799696T1 (no)
WO (1) WO2006054182A2 (no)

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DE602005011031D1 (en) 2004-09-17 2008-12-24 Idenix Pharmaceuticals Inc Phosphoindole als hiv-inhibitoren
ES2488922T3 (es) 2006-09-29 2014-09-01 Idenix Pharmaceuticals, Inc. Fosfoindoles enantiómeramente puros como inhibidores del HIV
WO2008054605A2 (en) * 2006-10-06 2008-05-08 Merck & Co., Inc. Non-nucleoside reverse transcriptase inhibitors
CA2687747C (en) 2007-05-30 2015-11-17 F. Hoffmann-La Roche Ag Non-nucleoside reverse transcriptase inhibitors
TW200946541A (en) 2008-03-27 2009-11-16 Idenix Pharmaceuticals Inc Solid forms of an anti-HIV phosphoindole compound
TW200944537A (en) * 2008-04-03 2009-11-01 Idenix Pharmaceuticals Inc Formulations comprising a phosphoindole compound and one or more second active agents
WO2010090976A1 (en) * 2009-02-03 2010-08-12 Idenix Pharmaceuticals, Inc. Phosphinate ruthenium complexes
JP5690286B2 (ja) * 2009-03-04 2015-03-25 イデニク プハルマセウティカルス，インコーポレイテッド ホスホチオフェン及びホスホチアゾールｈｃｖポリメラーゼ阻害剤
UA105556C2 (uk) 2010-01-27 2014-05-26 Віів Гелскер Компані Комбінація сполук, що містить інгібітори віл інтегрази з іншими терапевтичними агентами
CN103275126B (zh) * 2013-05-28 2016-03-23 兰州大学 一种立体选择性合成3-位膦酰化吲哚的方法
ITMI20131218A1 (it) * 2013-07-19 2015-01-20 Need Pharma Srl Nuovi ureido derivati di acidi naftalensolfonici
EP3695225A4 (en) * 2017-10-13 2021-06-30 Ursure, Inc. PRODUCTS AND METHODS FOR MONITORING ADHERENCE IN NUCLEOSIDE REVERSE TRANSCRIPTASE INHIBITOR THERAPY

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Also Published As

Publication number Publication date
BRPI0515344A (pt) 2008-07-15
US7534809B2 (en) 2009-05-19
NZ554232A (en) 2010-09-30
JP5031569B2 (ja) 2012-09-19
ATE414092T1 (de) 2008-11-15
MX2007003040A (es) 2007-08-02
DE602005011031D1 (en) 2008-12-24
WO2006054182A2 (en) 2006-05-26
JP2008515782A (ja) 2008-05-15
DE602005023360D1 (de) 2010-10-14
RS50981B (sr) 2010-10-31
KR20070063545A (ko) 2007-06-19
WO2006054182A3 (en) 2007-03-01
EP1799696A2 (en) 2007-06-27
PL1799696T3 (pl) 2009-04-30
AU2005305609A1 (en) 2006-05-26
EP1799696B1 (en) 2008-11-12
PT1799696E (pt) 2009-02-16
AU2005305609B2 (en) 2011-10-06
CY1109440T1 (el) 2014-08-13
US20090163444A1 (en) 2009-06-25
ATE479693T1 (de) 2010-09-15
ES2320252T3 (es) 2009-05-20
CA2583409A1 (en) 2006-05-26
CN102304150B (zh) 2014-06-18
SG155939A1 (en) 2009-10-29
DK1799696T3 (da) 2009-03-09
US8044091B2 (en) 2011-10-25
HRP20090086T3 (en) 2009-03-31
SI1799696T1 (sl) 2009-04-30
IL181909A0 (en) 2007-07-04
CA2583409C (en) 2014-06-17
EP1961757A1 (en) 2008-08-27
WO2006054182A9 (en) 2006-08-17
CN102304150A (zh) 2012-01-04
HK1100142A1 (en) 2007-09-07
EP1961757B1 (en) 2010-09-01
EP2256124A1 (en) 2010-12-01
US20060074054A1 (en) 2006-04-06
KR101242962B1 (ko) 2013-03-13

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