NO20071095L - Hittil ukjente tiofenderivater - Google Patents

Hittil ukjente tiofenderivater

Info

Publication number
NO20071095L
NO20071095L NO20071095A NO20071095A NO20071095L NO 20071095 L NO20071095 L NO 20071095L NO 20071095 A NO20071095 A NO 20071095A NO 20071095 A NO20071095 A NO 20071095A NO 20071095 L NO20071095 L NO 20071095L
Authority
NO
Norway
Prior art keywords
thiophene derivatives
hitherto unknown
derivatives
hitherto
unknown
Prior art date
Application number
NO20071095A
Other languages
English (en)
Inventor
Martin Bolli
Thomas Weller
Walter Fischli
Martine Clozel
Oliver Nayler
Daniel Bur
Claus Mueller
Michael Scherz
David Lehmann
Boris Mathys
Original Assignee
Actelion Pharmaceuticals Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Actelion Pharmaceuticals Ltd filed Critical Actelion Pharmaceuticals Ltd
Publication of NO20071095L publication Critical patent/NO20071095L/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/50—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
    • C07D333/78—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems condensed with rings other than six-membered or with ring systems containing such rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/06—Antipsoriatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/14—Drugs for disorders of the endocrine system of the thyroid hormones, e.g. T3, T4
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Immunology (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Transplantation (AREA)
  • Diabetes (AREA)
  • Endocrinology (AREA)
  • Dermatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Transition And Organic Metals Composition Catalysts For Addition Polymerization (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)

Abstract

Oppfinnelsen angår hittil ukjente tiofenderivater, deres fremstilling og deres anvendelse som farmasøytisk aktive forbindelser. Forbindelsene fungerer især som immunsuppressive 5 midler.
NO20071095A 2004-07-29 2007-02-27 Hittil ukjente tiofenderivater NO20071095L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
PCT/EP2004/008501 WO2006010379A1 (en) 2004-07-29 2004-07-29 Novel thiophene derivatives as immunosuppressive agents
PCT/EP2005/007892 WO2006010544A2 (en) 2004-07-29 2005-07-20 1, 1a, 5, 5a-tetrahydro-3-thia-cyclopropa’a! pentalenes: tricyclic thiophene derivatives as s1p1/edg1 receptor agonists

Publications (1)

Publication Number Publication Date
NO20071095L true NO20071095L (no) 2007-02-27

Family

ID=34958296

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20071095A NO20071095L (no) 2004-07-29 2007-02-27 Hittil ukjente tiofenderivater

Country Status (23)

Country Link
US (1) US7750040B2 (no)
EP (1) EP1805163B1 (no)
JP (1) JP4807884B2 (no)
KR (1) KR20070046849A (no)
CN (1) CN1993346B (no)
AR (1) AR050273A1 (no)
AT (1) ATE409697T1 (no)
AU (1) AU2005266529A1 (no)
BR (1) BRPI0513841A (no)
CA (1) CA2574305A1 (no)
DE (1) DE602005010109D1 (no)
DK (1) DK1805163T3 (no)
ES (1) ES2313391T3 (no)
IL (1) IL180962A0 (no)
MX (1) MX2007000972A (no)
NO (1) NO20071095L (no)
PL (1) PL1805163T3 (no)
PT (1) PT1805163E (no)
RU (1) RU2386626C2 (no)
SI (1) SI1805163T1 (no)
TW (1) TW200616994A (no)
WO (2) WO2006010379A1 (no)
ZA (1) ZA200700535B (no)

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Also Published As

Publication number Publication date
ES2313391T3 (es) 2009-03-01
KR20070046849A (ko) 2007-05-03
AU2005266529A1 (en) 2006-02-02
CN1993346B (zh) 2011-04-27
JP2008508210A (ja) 2008-03-21
EP1805163A2 (en) 2007-07-11
RU2386626C2 (ru) 2010-04-20
DK1805163T3 (da) 2008-12-15
PT1805163E (pt) 2008-12-05
AR050273A1 (es) 2006-10-11
TW200616994A (en) 2006-06-01
WO2006010544A2 (en) 2006-02-02
RU2007107164A (ru) 2008-09-10
ATE409697T1 (de) 2008-10-15
US7750040B2 (en) 2010-07-06
EP1805163B1 (en) 2008-10-01
US20080064740A1 (en) 2008-03-13
IL180962A0 (en) 2007-07-04
CN1993346A (zh) 2007-07-04
MX2007000972A (es) 2007-04-10
WO2006010379A1 (en) 2006-02-02
SI1805163T1 (sl) 2009-02-28
BRPI0513841A (pt) 2008-05-20
ZA200700535B (en) 2008-10-29
DE602005010109D1 (de) 2008-11-13
PL1805163T3 (pl) 2009-04-30
WO2006010544A3 (en) 2006-03-30
CA2574305A1 (en) 2006-02-02
JP4807884B2 (ja) 2011-11-02

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