MA29080B1 - Derives de la quinuclidine et leur utilisation en tant qu'antagonistes du recepteur m3 muscarinique - Google Patents

Derives de la quinuclidine et leur utilisation en tant qu'antagonistes du recepteur m3 muscarinique

Info

Publication number
MA29080B1
MA29080B1 MA29952A MA29952A MA29080B1 MA 29080 B1 MA29080 B1 MA 29080B1 MA 29952 A MA29952 A MA 29952A MA 29952 A MA29952 A MA 29952A MA 29080 B1 MA29080 B1 MA 29080B1
Authority
MA
Morocco
Prior art keywords
receptor antagonists
muscarinic receptor
quinuclidine derivatives
quinuclidine
derivatives
Prior art date
Application number
MA29952A
Other languages
English (en)
Inventor
Neil John Press
Stephen Paul Collingwood
Urs Baettig
Brian Cox
Sudhakar Devidasrao Garad
Hyungchul Kim
Dimitris Papoutsakis
Simon James Watson
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=33515948&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=MA29080(B1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of MA29080B1 publication Critical patent/MA29080B1/fr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D453/00—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
    • C07D453/02—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids containing not further condensed quinuclidine ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/06—Antiasthmatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/08—Bronchodilators
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/16—Central respiratory analeptics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pulmonology (AREA)
  • Immunology (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Cosmetics (AREA)
  • Hydrogenated Pyridines (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Plural Heterocyclic Compounds (AREA)
MA29952A 2004-11-02 2007-05-30 Derives de la quinuclidine et leur utilisation en tant qu'antagonistes du recepteur m3 muscarinique MA29080B1 (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GBGB0424284.8A GB0424284D0 (en) 2004-11-02 2004-11-02 Organic compounds

Publications (1)

Publication Number Publication Date
MA29080B1 true MA29080B1 (fr) 2007-12-03

Family

ID=33515948

Family Applications (1)

Application Number Title Priority Date Filing Date
MA29952A MA29080B1 (fr) 2004-11-02 2007-05-30 Derives de la quinuclidine et leur utilisation en tant qu'antagonistes du recepteur m3 muscarinique

Country Status (33)

Country Link
US (2) US7723356B2 (fr)
EP (2) EP2206499A1 (fr)
JP (1) JP4950896B2 (fr)
KR (1) KR101252307B1 (fr)
CN (1) CN101056634B (fr)
AR (1) AR054090A1 (fr)
AT (1) ATE481099T1 (fr)
AU (1) AU2005300710B2 (fr)
BR (1) BRPI0517945A (fr)
CA (1) CA2583237C (fr)
CY (1) CY1110952T1 (fr)
DE (1) DE602005023639D1 (fr)
DK (1) DK1811999T3 (fr)
EC (1) ECSP077424A (fr)
ES (1) ES2353142T3 (fr)
GB (1) GB0424284D0 (fr)
HR (1) HRP20100693T1 (fr)
IL (1) IL182695A0 (fr)
JO (1) JO2613B1 (fr)
MA (1) MA29080B1 (fr)
MX (1) MX2007005189A (fr)
MY (1) MY145207A (fr)
NO (1) NO20072371L (fr)
NZ (1) NZ554302A (fr)
PE (1) PE20060609A1 (fr)
PL (1) PL1811999T3 (fr)
PT (1) PT1811999E (fr)
RU (1) RU2399620C2 (fr)
SI (1) SI1811999T1 (fr)
TN (1) TNSN07164A1 (fr)
TW (1) TW200628154A (fr)
WO (1) WO2006048225A1 (fr)
ZA (1) ZA200702772B (fr)

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GB0601951D0 (en) 2006-01-31 2006-03-15 Novartis Ag Organic compounds
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TW200825084A (en) * 2006-11-14 2008-06-16 Astrazeneca Ab New compounds 521
KR20090094460A (ko) * 2006-12-19 2009-09-07 아스트라제네카 아베 무스카린 수용체 길항제로서 퀴누클리디놀 유도체
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US8329729B2 (en) * 2008-05-13 2012-12-11 Astrazeneca Ab Quinuclidine derivatives as muscarinic M3 receptor antagonists
EP2315589A4 (fr) * 2008-05-13 2013-09-11 Astrazeneca Ab PRODUIT PHARMACEUTIQUE COMPRENANT UN ANTAGONISTE DU RÉCEPTEUR MUSCARINIQUE ET UN AGONISTE DES béta2-ADRÉNOCEPTEURS
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KR101290893B1 (ko) 2009-04-09 2013-07-29 노파르티스 아게 피롤리디늄 염의 제조 방법
CA2803418A1 (fr) * 2010-06-22 2011-12-29 Chiesi Farmaceutici S.P.A. Formulation de poudre seche comprenant un medicament antimuscarinique
KR20130111968A (ko) * 2010-06-22 2013-10-11 키에시 파르마슈티시 엣스. 피. 에이. 알칼로이드 아미노에스테르 유도체 및 이의 의약 조성물
WO2012034095A1 (fr) 2010-09-09 2012-03-15 Irm Llc Composés et compositions comme inhibiteurs de trk
UY33597A (es) 2010-09-09 2012-04-30 Irm Llc Compuestos y composiciones como inhibidores de la trk
BR112013021638A2 (pt) 2011-02-25 2016-08-02 Irm Llc "compostos inibidores de trk, seu uso e composições que os compreendem"
JP2011195593A (ja) * 2011-06-30 2011-10-06 Astrazeneca Ab ムスカリンｍ３受容体アンタゴニストとしてのキヌクリジン誘導体
EP2935249B1 (fr) 2012-12-19 2018-12-12 Novartis AG Inhibiteurs d'autotaxine
EP3134398A1 (fr) 2014-04-24 2017-03-01 Novartis Ag Inhibiteurs de l'autotaxine
US20170065589A1 (en) * 2014-05-06 2017-03-09 Anthony G. Visco Methods of treating or preventing preterm labor
CN109851615B (zh) * 2019-04-22 2021-06-08 上海旭东海普药业有限公司 纯化戊乙奎醚的方法

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WO2006048225A1 (fr) 2006-05-11
MX2007005189A (es) 2007-05-11
DE602005023639D1 (de) 2010-10-28
MY145207A (en) 2012-01-13
US8084463B2 (en) 2011-12-27
KR101252307B1 (ko) 2013-04-08
DK1811999T3 (da) 2010-12-13
PT1811999E (pt) 2010-10-29
TNSN07164A1 (en) 2008-11-21
BRPI0517945A (pt) 2008-10-21
US20100168132A1 (en) 2010-07-01
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EP2206499A1 (fr) 2010-07-14
SI1811999T1 (sl) 2011-01-31
AU2005300710A1 (en) 2006-05-11
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