NO20076317L - Sammensetning av en tienopyridinblodplateaggregeringsinhibitor - Google Patents

Sammensetning av en tienopyridinblodplateaggregeringsinhibitor

Info

Publication number
NO20076317L
NO20076317L NO20076317A NO20076317A NO20076317L NO 20076317 L NO20076317 L NO 20076317L NO 20076317 A NO20076317 A NO 20076317A NO 20076317 A NO20076317 A NO 20076317A NO 20076317 L NO20076317 L NO 20076317L
Authority
NO
Norway
Prior art keywords
composition
platelet aggregation
aggregation inhibitor
thienopyridine
thienopyridine platelet
Prior art date
Application number
NO20076317A
Other languages
English (en)
Norwegian (no)
Inventor
David Brian Dziennik
Tamara Beth Edelman
Peter Lloyd Oren
Robert Louis Ternik
Original Assignee
Lilly Co Eli
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=37198935&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=NO20076317(L) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Lilly Co Eli filed Critical Lilly Co Eli
Publication of NO20076317L publication Critical patent/NO20076317L/no

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/4365—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system having sulfur as a ring hetero atom, e.g. ticlopidine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/06—Antiarrhythmics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Landscapes

  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Epidemiology (AREA)
  • Diabetes (AREA)
  • Vascular Medicine (AREA)
  • Urology & Nephrology (AREA)
  • Hematology (AREA)
  • Pulmonology (AREA)
  • Hospice & Palliative Care (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Medical Preparation Storing Or Oral Administration Devices (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
NO20076317A 2005-06-10 2007-12-07 Sammensetning av en tienopyridinblodplateaggregeringsinhibitor NO20076317L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US68918305P 2005-06-10 2005-06-10
PCT/US2006/021860 WO2006135605A2 (fr) 2005-06-10 2006-06-06 Formulation d'une thienopyridine, comme inhibiteur de l'agregation plaquettaire

Publications (1)

Publication Number Publication Date
NO20076317L true NO20076317L (no) 2008-02-29

Family

ID=37198935

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20076317A NO20076317L (no) 2005-06-10 2007-12-07 Sammensetning av en tienopyridinblodplateaggregeringsinhibitor

Country Status (34)

Country Link
US (1) US20080176893A1 (fr)
EP (1) EP1896019B1 (fr)
JP (1) JP2008543755A (fr)
KR (2) KR20100076050A (fr)
CN (1) CN101193633B (fr)
AR (1) AR054283A1 (fr)
AT (1) ATE441413T1 (fr)
AU (1) AU2006258102B2 (fr)
BR (1) BRPI0611350B8 (fr)
CA (1) CA2611668C (fr)
CY (1) CY1109502T1 (fr)
DE (1) DE602006008942D1 (fr)
DK (1) DK1896019T3 (fr)
DO (1) DOP2006000126A (fr)
EA (1) EA011693B1 (fr)
EC (1) ECSP077984A (fr)
ES (1) ES2330373T3 (fr)
HR (1) HRP20090516T1 (fr)
IL (1) IL187830A0 (fr)
MA (1) MA29688B1 (fr)
MX (1) MX2007015431A (fr)
MY (1) MY151038A (fr)
NO (1) NO20076317L (fr)
NZ (1) NZ564003A (fr)
PE (1) PE20070320A1 (fr)
PL (1) PL1896019T3 (fr)
PT (1) PT1896019E (fr)
RS (1) RS51194B (fr)
SI (1) SI1896019T1 (fr)
TN (1) TNSN07466A1 (fr)
TW (1) TWI318571B (fr)
UA (1) UA91051C2 (fr)
WO (1) WO2006135605A2 (fr)
ZA (1) ZA200710697B (fr)

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Publication number Priority date Publication date Assignee Title
CA2672134C (fr) * 2006-12-07 2015-02-10 Daiichi Sankyo Company, Limited Preparation medicale sous forme solide contenant un mannitol ou un lactose
KR101665705B1 (ko) * 2006-12-07 2016-10-12 다이이찌 산쿄 가부시키가이샤 안정성이 개선된 필름 코팅 제제
AU2007333302A1 (en) * 2006-12-07 2008-06-19 Eli Lilly And Company An article comprising prasugrel
JPWO2008072532A1 (ja) * 2006-12-07 2010-03-25 第一三共株式会社 貯蔵安定性が改善された医薬組成物
WO2008072533A1 (fr) * 2006-12-07 2008-06-19 Daiichi Sankyo Company, Limited Procédé de production d'une préparation solide
TWI482641B (zh) * 2006-12-07 2015-05-01 Daiichi Sankyo Co Ltd 含有低取代度羥丙基纖維素之醫藥組成物
CN102424686A (zh) * 2007-03-02 2012-04-25 第一三共株式会社 用于制备高纯度普拉格雷盐酸盐的方法
CN101686681B (zh) 2007-04-27 2015-04-01 锡德克斯药物公司 包含氯吡格雷和磺基烷基醚环糊精的制剂和其使用方法
GB2450117A (en) * 2007-06-13 2008-12-17 Reckitt Benckiser Healthcare A water- and oxygen-occlusive blister tablet pack
WO2009098142A1 (fr) * 2008-02-06 2009-08-13 Helm Ag Sels de prasugrel avec des propriétés améliorées
EP2107061A1 (fr) * 2008-04-02 2009-10-07 Krka Tovarna Zdravil, D.D., Novo Mesto Procédé de préparation de clopidogrel enrichi optiquement
DE602008002820D1 (de) 2008-04-25 2010-11-11 Sandoz Ag Hydrogensulfat von 2-Acetoxy-5-(a-cyclopropylcarbonyl-2-fluorbenzyl)-4,5,6,7-tetrahydrothienoÄ3,2-cÜpyridin und dessen Zubereitung
WO2010094471A1 (fr) * 2009-02-17 2010-08-26 Krka, D. D., Novo Mesto Compositions pharmaceutiques comprenant du prasugrel ou ses sels d'addition d'acide pharmaceutiquement acceptables, et leurs procédés de préparation
PL3100728T3 (pl) * 2009-05-13 2020-05-18 Cydex Pharmaceuticals, Inc. Kompozycje farmaceutyczne zawierające prasugrel i pochodne cyklodekstryny oraz sposoby ich wytwarzania i zastosowania
DE102009036646A1 (de) 2009-08-07 2011-02-10 Ratiopharm Gmbh Prasugrel in nicht-kristalliner Form und pharmazeutische Zusammensetzung davon
JP2013032289A (ja) * 2009-10-28 2013-02-14 Daiichi Sankyo Co Ltd ワックス安定製剤
WO2011052499A1 (fr) * 2009-10-28 2011-05-05 第一三共株式会社 Composition pharmaceutique présentant une stabilité au stockage améliorée
WO2011092720A2 (fr) * 2010-02-01 2011-08-04 Msn Laboratories Limited Composition pharmaceutique de prasugrel et ses sels pharmaceutiquement acceptables
EP2409685A3 (fr) 2010-07-19 2012-02-01 Sanovel Ilac Sanayi ve Ticaret A.S. Formulations de prasugrel à désintégration orale
TR201006802A1 (tr) * 2010-08-17 2012-03-21 Sanovel İlaç San. Ve Ti̇c. A.Ş. Prasugrelin oral yolla dağılan formülasyonları.
TR201005900A1 (tr) 2010-07-19 2012-02-21 Sanovel İlaç San. Ve Ti̇c. A.Ş. Geliştirilmiş stabiliteye sahip prasugrel granülleri.
TR201007926A1 (tr) 2010-07-19 2012-02-21 Sanovel İlaç San.Ve Ti̇c.A.Ş. Prasugrel tablet formülasyonları.
CZ2011872A3 (cs) 2011-12-22 2013-07-03 Zentiva, K.S. Farmaceutická formulace prasugrelu hydrobromidu
US8603537B2 (en) 2012-04-02 2013-12-10 Egis Pharmaceuticals Plc Prasugrel containing quickly released stable oral pharmaceutical compositions
WO2014060560A1 (fr) 2012-10-19 2014-04-24 Sanovel Ilac Sanayi Ve Ticaret A.S. Formulations orales solides de prasugrel
EP2722037A1 (fr) 2012-10-19 2014-04-23 Sanovel Ilac Sanayi ve Ticaret A.S. Formulations de prasugrel
CN102993210A (zh) * 2012-12-19 2013-03-27 苏春华 一种吡啶并噻吩的新化合物
EP2979693A1 (fr) 2014-08-01 2016-02-03 Zaklady Farmaceutyczne Polpharma SA Composition pharmaceutique comprenant du prasugrel ou un sel pharmaceutiquement acceptable de celui-ci et son procédé de préparation
WO2016122421A1 (fr) 2015-01-29 2016-08-04 Pharmactive Ilaç Sanayi Ve Ticaret A.Ş. Compositions pharmaceutiques stables contenant une base de prasugrel
EP3158993A1 (fr) 2015-10-22 2017-04-26 Zaklady Farmaceutyczne Polpharma SA Procédé pour préparer un comprimé contenant du prasugrel ou des sels pharmaceutiquement acceptables de celui-ci
CN107304216A (zh) * 2016-04-20 2017-10-31 陕西合成药业股份有限公司 噻吩吡啶类衍生物及其制备方法和用途
HU231079B1 (hu) 2016-06-23 2020-06-29 Richter Gedeon Nyrt. Eljárás nagytisztaságú Prasugrel előállítására bromopentil szennyezés eltávolításával
GR1009230B (el) 2016-10-12 2018-02-22 Φαρματεν Αβεε Φαρμακευτικο σκευασμα που περιλαμβανει βεσυλικη πρασουγρελη

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FI101150B (fi) * 1991-09-09 1998-04-30 Sankyo Co Menetelmä lääkeaineina käyttökelpoisten tetrahydrotienopyridiinin johd annaisten valmistamiseksi
KR20080021152A (ko) * 2000-07-06 2008-03-06 다이이찌 산쿄 가부시키가이샤 히드로피리딘 유도체 산부가염
JP4001199B2 (ja) * 2000-07-06 2007-10-31 第一三共株式会社 ヒドロピリジン誘導体酸付加塩
EP1243524A3 (fr) * 2001-03-16 2004-04-07 Pfizer Products Inc. Trousse pharmaceutique pour médicaments sensibles a l'oxygène
JP4394873B2 (ja) * 2001-12-19 2010-01-06 武田薬品工業株式会社 酸素に不安定な化合物を含有する固形組成物およびその安定化方法
SI21302A (sl) * 2002-10-11 2004-04-30 LEK farmacevtska dru�ba d.d. Stabiliziran farmacevtski izdelek z amorfno aktivno učinkovino
US20050020554A1 (en) * 2003-06-06 2005-01-27 Ahmed Salah U. Stability of hormone formulations
US20080171784A1 (en) * 2003-08-05 2008-07-17 Zentiva, A.S. Methods For the Stabilization of Atorvastatin

Also Published As

Publication number Publication date
CN101193633B (zh) 2011-12-14
AR054283A1 (es) 2007-06-13
WO2006135605A2 (fr) 2006-12-21
JP2008543755A (ja) 2008-12-04
CA2611668C (fr) 2013-10-15
KR20080008413A (ko) 2008-01-23
ATE441413T1 (de) 2009-09-15
RS51194B (sr) 2010-10-31
WO2006135605A3 (fr) 2007-04-12
MX2007015431A (es) 2008-02-21
MY151038A (en) 2014-03-31
DK1896019T3 (da) 2009-10-26
HRP20090516T1 (hr) 2009-10-31
EP1896019A2 (fr) 2008-03-12
CY1109502T1 (el) 2014-08-13
DE602006008942D1 (en) 2009-10-15
PL1896019T3 (pl) 2010-01-29
IL187830A0 (en) 2008-04-13
ZA200710697B (en) 2009-08-26
PE20070320A1 (es) 2007-05-12
PT1896019E (pt) 2009-11-19
SI1896019T1 (sl) 2010-01-29
BRPI0611350B1 (pt) 2020-09-15
EA200702670A1 (ru) 2008-04-28
KR20100076050A (ko) 2010-07-05
CN101193633A (zh) 2008-06-04
BRPI0611350B8 (pt) 2021-05-25
BRPI0611350A2 (pt) 2010-12-07
CA2611668A1 (fr) 2006-12-21
EA011693B1 (ru) 2009-04-28
TNSN07466A1 (en) 2009-03-17
TW200718420A (en) 2007-05-16
HK1116422A1 (en) 2008-12-24
AU2006258102A1 (en) 2006-12-21
DOP2006000126A (es) 2006-12-15
ECSP077984A (es) 2008-01-23
MA29688B1 (fr) 2008-08-01
NZ564003A (en) 2011-07-29
US20080176893A1 (en) 2008-07-24
AU2006258102B2 (en) 2011-09-15
TWI318571B (en) 2009-12-21
EP1896019B1 (fr) 2009-09-02
ES2330373T3 (es) 2009-12-09
UA91051C2 (ru) 2010-06-25

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