NO20081617L - Metoder for fremstilling av Glutaminsyrederivater - Google Patents

Metoder for fremstilling av Glutaminsyrederivater

Info

Publication number
NO20081617L
NO20081617L NO20081617A NO20081617A NO20081617L NO 20081617 L NO20081617 L NO 20081617L NO 20081617 A NO20081617 A NO 20081617A NO 20081617 A NO20081617 A NO 20081617A NO 20081617 L NO20081617 L NO 20081617L
Authority
NO
Norway
Prior art keywords
preparation
glutamic acid
acid derivatives
methods
novel methods
Prior art date
Application number
NO20081617A
Other languages
English (en)
Inventor
Joseph Zeldis
David Michael Blum
Ronald Stanley Michalak
Mel Jennings
Timothy Doyle
Original Assignee
Wyeth Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Wyeth Corp filed Critical Wyeth Corp
Publication of NO20081617L publication Critical patent/NO20081617L/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C269/00—Preparation of derivatives of carbamic acid, i.e. compounds containing any of the groups, the nitrogen atom not being part of nitro or nitroso groups
    • C07C269/06—Preparation of derivatives of carbamic acid, i.e. compounds containing any of the groups, the nitrogen atom not being part of nitro or nitroso groups by reactions not involving the formation of carbamate groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C237/00—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups
    • C07C237/02—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups having the carbon atoms of the carboxamide groups bound to acyclic carbon atoms of the carbon skeleton
    • C07C237/04—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups having the carbon atoms of the carboxamide groups bound to acyclic carbon atoms of the carbon skeleton the carbon skeleton being acyclic and saturated
    • C07C237/06—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups having the carbon atoms of the carboxamide groups bound to acyclic carbon atoms of the carbon skeleton the carbon skeleton being acyclic and saturated having the nitrogen atoms of the carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C231/00—Preparation of carboxylic acid amides
    • C07C231/12—Preparation of carboxylic acid amides by reactions not involving the formation of carboxamide groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C237/00—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups
    • C07C237/02—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups having the carbon atoms of the carboxamide groups bound to acyclic carbon atoms of the carbon skeleton
    • C07C237/04—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups having the carbon atoms of the carboxamide groups bound to acyclic carbon atoms of the carbon skeleton the carbon skeleton being acyclic and saturated
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C237/00—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups
    • C07C237/02—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups having the carbon atoms of the carboxamide groups bound to acyclic carbon atoms of the carbon skeleton
    • C07C237/22—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups having the carbon atoms of the carboxamide groups bound to acyclic carbon atoms of the carbon skeleton having nitrogen atoms of amino groups bound to the carbon skeleton of the acid part, further acylated
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C271/00—Derivatives of carbamic acids, i.e. compounds containing any of the groups, the nitrogen atom not being part of nitro or nitroso groups
    • C07C271/06—Esters of carbamic acids
    • C07C271/08—Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms
    • C07C271/10—Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms with the nitrogen atoms of the carbamate groups bound to hydrogen atoms or to acyclic carbon atoms
    • C07C271/22—Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms with the nitrogen atoms of the carbamate groups bound to hydrogen atoms or to acyclic carbon atoms to carbon atoms of hydrocarbon radicals substituted by carboxyl groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2603/00—Systems containing at least three condensed rings
    • C07C2603/02—Ortho- or ortho- and peri-condensed systems
    • C07C2603/04—Ortho- or ortho- and peri-condensed systems containing three rings
    • C07C2603/06—Ortho- or ortho- and peri-condensed systems containing three rings containing at least one ring with less than six ring members
    • C07C2603/10—Ortho- or ortho- and peri-condensed systems containing three rings containing at least one ring with less than six ring members containing five-membered rings
    • C07C2603/12—Ortho- or ortho- and peri-condensed systems containing three rings containing at least one ring with less than six ring members containing five-membered rings only one five-membered ring
    • C07C2603/18—Fluorenes; Hydrogenated fluorenes

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)

Abstract

Foreliggende oppfinnelse angår nye metoder for fremstilling av glutaminsyrederivater og mellomprodukter derav, og slike forbindelser fremstilt ved de nye metodene. 58
NO20081617A 2005-10-13 2008-04-02 Metoder for fremstilling av Glutaminsyrederivater NO20081617L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US72644105P 2005-10-13 2005-10-13
PCT/US2006/026892 WO2007044100A1 (en) 2005-10-13 2006-07-11 Methods for preparing glutamic acid derivatives

Publications (1)

Publication Number Publication Date
NO20081617L true NO20081617L (no) 2008-05-06

Family

ID=37119907

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20081617A NO20081617L (no) 2005-10-13 2008-04-02 Metoder for fremstilling av Glutaminsyrederivater

Country Status (18)

Country Link
US (1) US7541485B2 (no)
EP (1) EP1934171A1 (no)
JP (1) JP2009511578A (no)
KR (1) KR20080058436A (no)
CN (1) CN101282927A (no)
AR (1) AR057451A1 (no)
AU (1) AU2006299918A1 (no)
BR (1) BRPI0617348A2 (no)
CA (1) CA2624866A1 (no)
CR (1) CR9885A (no)
EC (1) ECSP088360A (no)
GT (1) GT200600305A (no)
IL (1) IL190729A0 (no)
NO (1) NO20081617L (no)
PE (1) PE20070526A1 (no)
RU (1) RU2008113222A (no)
TW (1) TW200740729A (no)
WO (1) WO2007044100A1 (no)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AR061420A1 (es) * 2006-06-02 2008-08-27 Wyeth Corp Metodos para preparar derivados de acido glutamico e intermediarios del mismo
US20100216886A1 (en) * 2006-11-09 2010-08-26 Wyeth Polymorphs of n2-(1,1'-biphenyl-4-ylcarbonyl)-n1-[2-(4-fluorophenyl)-1,1-dimethylethyl]-l-alpha-glutamine
ES2776106T3 (es) * 2011-09-30 2020-07-29 Kemira Oyj Prevención de la degradación de almidón en procesos fabricación de pulpa, papel o cartón
ES2968371T3 (es) 2013-10-10 2024-05-09 Eastern Virginia Medical School Derivados de 4-((2-hidroxi-3-metoxibencil)amino) bencenosulfonamida como inhibidores de la 12-lipoxigenasa
EP3286172B1 (en) 2015-04-23 2019-06-12 Constellation Pharmaceuticals, Inc. Lsd1 inhibitors and uses thereof
LT3532459T (lt) 2016-10-26 2023-11-10 Constellation Pharmaceuticals, Inc. Lsd1 inhibitoriai ir jų medicininis panaudojimas
US12668594B2 (en) 2020-12-23 2026-06-30 Sudo Biosciences Limited TYK2 inhibitors and uses thereof
IL305119A (en) 2021-02-19 2023-10-01 Sudo Biosciences Ltd Tyk2 inhibitors and uses thereof
TW202302583A (zh) 2021-02-19 2023-01-16 英商蘇多生物科學有限公司 Tyk2抑制劑及其用途
KR20230159421A (ko) 2021-02-19 2023-11-21 수도 바이오사이언시즈 리미티드 Tyk2 억제제 및 이의 용도

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Also Published As

Publication number Publication date
ECSP088360A (es) 2008-05-30
CN101282927A (zh) 2008-10-08
WO2007044100A1 (en) 2007-04-19
JP2009511578A (ja) 2009-03-19
RU2008113222A (ru) 2009-11-20
US20070088172A1 (en) 2007-04-19
IL190729A0 (en) 2008-11-03
CA2624866A1 (en) 2007-04-19
PE20070526A1 (es) 2007-06-11
AR057451A1 (es) 2007-12-05
US7541485B2 (en) 2009-06-02
GT200600305A (es) 2007-02-26
CR9885A (es) 2008-06-16
TW200740729A (en) 2007-11-01
AU2006299918A1 (en) 2007-04-19
EP1934171A1 (en) 2008-06-25
BRPI0617348A2 (pt) 2011-07-26
KR20080058436A (ko) 2008-06-25

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