NO20082593L - Pyrazolo[4,3-D]pyrimidin-5-yl)derivater anvendt som PDE5 inhibitorer - Google Patents

Pyrazolo[4,3-D]pyrimidin-5-yl)derivater anvendt som PDE5 inhibitorer

Info

Publication number
NO20082593L
NO20082593L NO20082593A NO20082593A NO20082593L NO 20082593 L NO20082593 L NO 20082593L NO 20082593 A NO20082593 A NO 20082593A NO 20082593 A NO20082593 A NO 20082593A NO 20082593 L NO20082593 L NO 20082593L
Authority
NO
Norway
Prior art keywords
pyrazolo
pyrimidin
derivatives used
pde5 inhibitors
methylpyridin
Prior art date
Application number
NO20082593A
Other languages
English (en)
Inventor
Michael Brent Tollefson
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Publication of NO20082593L publication Critical patent/NO20082593L/no

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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
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Abstract

Foreliggende oppfinnelse omfatter l-(l-(2-etoksyetyI)-3-etyI-7-(4-metyIpyridin-2-ylamino)-1H-pyrazolo[4,3-dlpyrimidin-5-yl)piperidin-4-karboksylsyre og dets salter. Oppfinnelsen innbefatter ytterligere farmasøytiske sammensetninger, behandlingsfremgangsmåter av behandling og syntetiske behandlingsfremgangsmåter relatert til 1-(1-(2-etoksyetyl)-3-etyl-7-(4-metylpyridin-2-ylamino)-1H-pyrazolo[4,3-dlpyrimidin-5-yl)piperidin-4-karboksylsyre og dets salter.
NO20082593A 2005-11-10 2008-06-10 Pyrazolo[4,3-D]pyrimidin-5-yl)derivater anvendt som PDE5 inhibitorer NO20082593L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US73532005P 2005-11-10 2005-11-10
PCT/IB2006/003132 WO2007054778A1 (en) 2005-11-10 2006-10-31 Pyrazolo[4,3-d]pyrimidin-5-yl)derivative used as pde5 inhibitors

Publications (1)

Publication Number Publication Date
NO20082593L true NO20082593L (no) 2008-07-22

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NO20082593A NO20082593L (no) 2005-11-10 2008-06-10 Pyrazolo[4,3-D]pyrimidin-5-yl)derivater anvendt som PDE5 inhibitorer

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US (2) US20090156618A1 (no)
EP (1) EP1948661B1 (no)
JP (1) JP4208959B1 (no)
KR (1) KR101012592B1 (no)
CN (1) CN101305007B (no)
AP (1) AP2008004437A0 (no)
AR (1) AR057885A1 (no)
AT (1) ATE435865T1 (no)
AU (1) AU2006313486B2 (no)
BR (1) BRPI0618284A2 (no)
CA (1) CA2629339C (no)
CR (1) CR9966A (no)
DE (1) DE602006007728D1 (no)
DK (1) DK1948661T3 (no)
DO (1) DOP2006000248A (no)
EA (1) EA200800920A1 (no)
EC (1) ECSP088441A (no)
ES (1) ES2326919T3 (no)
IL (1) IL190456A (no)
MA (1) MA29943B1 (no)
NL (1) NL2000291C2 (no)
NO (1) NO20082593L (no)
PE (1) PE20070764A1 (no)
RS (1) RS20080197A (no)
TN (1) TNSN08209A1 (no)
TW (1) TW200738723A (no)
UY (1) UY29909A1 (no)
WO (1) WO2007054778A1 (no)
ZA (1) ZA200803173B (no)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20110165183A1 (en) * 2008-08-01 2011-07-07 Biocryst Pharmaceuticals, Inc. Piperidine derivatives as jak3 inhibitors
WO2010043633A1 (en) * 2008-10-15 2010-04-22 Palau Pharma, S. A. 2h-pyrazolo [4,3-d]pyrimidin-5-amine derivatives as h4 histamine receptor antagonists for the treatment of allergic, immunological and inflammatory diseases
CN102970965A (zh) * 2010-04-05 2013-03-13 Sk化学公司 含有pde5抑制剂的减少皮肤皱纹的合成物
EP3189835B1 (en) * 2011-02-28 2018-07-25 National Cerebral and Cardiovascular Center Medical agent for suppressing malignant tumor metastasis
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