NL2000291A1 - 1- (1- (2-ethoxyethyl)-3-ethyl-7- (4-methylpyridin-2-ylamino)-1H- pyrazool[4,3-d]pyrimidine-5-yl)piperidine-4-carbonzuur en zouten daarvan. - Google Patents

1- (1- (2-ethoxyethyl)-3-ethyl-7- (4-methylpyridin-2-ylamino)-1H- pyrazool[4,3-d]pyrimidine-5-yl)piperidine-4-carbonzuur en zouten daarvan.

Info

Publication number: NL2000291A1
Authority: NL; Netherlands
Prior art keywords: methylpyridin; ylamino; ethoxyethyl; pyrimidin; pyrazole
Prior art date: 2005-11-10

Application number

NL2000291A

Other languages

English (en)

Other versions

NL2000291C2 (nl

Inventor

Michael Brent Tollefson

Original Assignee

Pfizer Prod Inc

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2005-11-10

Filing date

2006-10-27

Publication date

2007-05-11

2006-10-27 Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc

2007-05-11 Publication of NL2000291A1 publication Critical patent/NL2000291A1/nl

2009-02-17 Application granted granted Critical

2009-02-17 Publication of NL2000291C2 publication Critical patent/NL2000291C2/nl

Links

-1 2-ethoxyethyl Chemical group 0.000 title 1
SRJOCJYGOFTFLH-UHFFFAOYSA-N isonipecotic acid Chemical compound OC(=O)C1CCNCC1 SRJOCJYGOFTFLH-UHFFFAOYSA-N 0.000 title 1
125000004528 pyrimidin-5-yl group Chemical group N1=CN=CC(=C1)* 0.000 title 1
150000003839 salts Chemical class 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
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- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
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NL2000291A 2005-11-10 2006-10-27 1-(1-(2-ethoxyethyl)-3-ethyl-7-(4-methylpyridin-2-ylamino)-1H- pyrazool(4,3-d)pyrimidine-5-yl)piperidine-4-carbonzuur en zouten daarvan. NL2000291C2 (nl)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US73532005P	2005-11-10	2005-11-10
US73532005		2005-11-10

Publications (2)

Publication Number	Publication Date
NL2000291A1 true NL2000291A1 (nl)	2007-05-11
NL2000291C2 NL2000291C2 (nl)	2009-02-17

Family

ID=37685872

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
NL2000291A NL2000291C2 (nl)	2005-11-10	2006-10-27	1-(1-(2-ethoxyethyl)-3-ethyl-7-(4-methylpyridin-2-ylamino)-1H- pyrazool(4,3-d)pyrimidine-5-yl)piperidine-4-carbonzuur en zouten daarvan.

Country Status (29)

Country	Link
US (2)	US20090156618A1 (nl)
EP (1)	EP1948661B1 (nl)
JP (1)	JP4208959B1 (nl)
KR (1)	KR101012592B1 (nl)
CN (1)	CN101305007B (nl)
AP (1)	AP2008004437A0 (nl)
AR (1)	AR057885A1 (nl)
AT (1)	ATE435865T1 (nl)
AU (1)	AU2006313486B2 (nl)
BR (1)	BRPI0618284A2 (nl)
CA (1)	CA2629339C (nl)
CR (1)	CR9966A (nl)
DE (1)	DE602006007728D1 (nl)
DK (1)	DK1948661T3 (nl)
DO (1)	DOP2006000248A (nl)
EA (1)	EA200800920A1 (nl)
EC (1)	ECSP088441A (nl)
ES (1)	ES2326919T3 (nl)
IL (1)	IL190456A (nl)
MA (1)	MA29943B1 (nl)
NL (1)	NL2000291C2 (nl)
NO (1)	NO20082593L (nl)
PE (1)	PE20070764A1 (nl)
RS (1)	RS20080197A (nl)
TN (1)	TNSN08209A1 (nl)
TW (1)	TW200738723A (nl)
UY (1)	UY29909A1 (nl)
WO (1)	WO2007054778A1 (nl)
ZA (1)	ZA200803173B (nl)

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EP2324020A2 (en) *	2008-08-01	2011-05-25	Biocryst Pharmaceuticals, Inc.	Piperidine derivatives as jak3 inhibitors
WO2010043633A1 (en) *	2008-10-15	2010-04-22	Palau Pharma, S. A.	2h-pyrazolo [4,3-d]pyrimidin-5-amine derivatives as h4 histamine receptor antagonists for the treatment of allergic, immunological and inflammatory diseases
JP2013523809A (ja) *	2010-04-05	2013-06-17	エスケーケミカルズカンパニーリミテッド	Ｐｄｅ５抑制剤を含む皮膚しわ改善用組成物
WO2012118042A1 (ja) *	2011-02-28	2012-09-07	独立行政法人国立循環器病研究センター	悪性腫瘍転移抑制用医薬
AU2012244550C1 (en)	2011-04-21	2017-06-22	Origenis Gmbh	Pyrazolo [4, 3-d] pyrimidines useful as kinase inhibitors
US9637491B2 (en)	2012-10-19	2017-05-02	Origenis Gmbh	Pyrazolo[4,3-D]pyrimidines as kinase inhibitors
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Publication number	Publication date
NL2000291C2 (nl)	2009-02-17
MA29943B1 (fr)	2008-11-03
AU2006313486A1 (en)	2007-05-18
KR20080063830A (ko)	2008-07-07
RS20080197A (sr)	2009-05-06
ES2326919T3 (es)	2009-10-21
JP2009519215A (ja)	2009-05-14
IL190456A0 (en)	2008-11-03
WO2007054778A1 (en)	2007-05-18
DE602006007728D1 (de)	2009-08-20
EP1948661B1 (en)	2009-07-08
CN101305007B (zh)	2011-07-20
US8518956B2 (en)	2013-08-27
CR9966A (es)	2008-06-16
NO20082593L (no)	2008-07-22
CA2629339A1 (en)	2007-05-18
US20090156618A1 (en)	2009-06-18
AP2008004437A0 (en)	2008-04-30
BRPI0618284A2 (pt)	2011-08-23
KR101012592B1 (ko)	2011-02-07
ATE435865T1 (de)	2009-07-15
US20110059993A1 (en)	2011-03-10
ECSP088441A (es)	2008-06-30
HK1120803A1 (en)	2009-04-09
EA200800920A1 (ru)	2008-10-30
ZA200803173B (en)	2009-01-28
TNSN08209A1 (fr)	2009-10-30
TW200738723A (en)	2007-10-16
DOP2006000248A (es)	2007-10-15
AU2006313486B2 (en)	2011-10-27
JP4208959B1 (ja)	2009-01-14
EP1948661A1 (en)	2008-07-30
IL190456A (en)	2012-10-31
DK1948661T3 (da)	2009-09-07
AR057885A1 (es)	2007-12-26
UY29909A1 (es)	2007-06-29
CN101305007A (zh)	2008-11-12
PE20070764A1 (es)	2007-08-13
CA2629339C (en)	2010-07-27

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