DK1948661T3 - Pyrazolo[4,3-D]pyrimidin-5-YL)-derivat anvendt som PDE5-inhibitorer - Google Patents

Pyrazolo[4,3-D]pyrimidin-5-YL)-derivat anvendt som PDE5-inhibitorer

Info

Publication number
DK1948661T3
DK1948661T3 DK06809195T DK06809195T DK1948661T3 DK 1948661 T3 DK1948661 T3 DK 1948661T3 DK 06809195 T DK06809195 T DK 06809195T DK 06809195 T DK06809195 T DK 06809195T DK 1948661 T3 DK1948661 T3 DK 1948661T3
Authority
DK
Denmark
Prior art keywords
pyrazolo
pyrimidin
derivative used
pde5 inhibitors
pde5
Prior art date
Application number
DK06809195T
Other languages
English (en)
Inventor
Michael Brent Tollefson
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Application granted granted Critical
Publication of DK1948661T3 publication Critical patent/DK1948661T3/da

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
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DK06809195T 2005-11-10 2006-10-31 Pyrazolo[4,3-D]pyrimidin-5-YL)-derivat anvendt som PDE5-inhibitorer DK1948661T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US73532005P 2005-11-10 2005-11-10
PCT/IB2006/003132 WO2007054778A1 (en) 2005-11-10 2006-10-31 Pyrazolo[4,3-d]pyrimidin-5-yl)derivative used as pde5 inhibitors

Publications (1)

Publication Number Publication Date
DK1948661T3 true DK1948661T3 (da) 2009-09-07

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DK06809195T DK1948661T3 (da) 2005-11-10 2006-10-31 Pyrazolo[4,3-D]pyrimidin-5-YL)-derivat anvendt som PDE5-inhibitorer

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US (2) US20090156618A1 (da)
EP (1) EP1948661B1 (da)
JP (1) JP4208959B1 (da)
KR (1) KR101012592B1 (da)
CN (1) CN101305007B (da)
AP (1) AP2008004437A0 (da)
AR (1) AR057885A1 (da)
AT (1) ATE435865T1 (da)
AU (1) AU2006313486B2 (da)
BR (1) BRPI0618284A2 (da)
CA (1) CA2629339C (da)
CR (1) CR9966A (da)
DE (1) DE602006007728D1 (da)
DK (1) DK1948661T3 (da)
DO (1) DOP2006000248A (da)
EA (1) EA200800920A1 (da)
EC (1) ECSP088441A (da)
ES (1) ES2326919T3 (da)
IL (1) IL190456A (da)
MA (1) MA29943B1 (da)
NL (1) NL2000291C2 (da)
NO (1) NO20082593L (da)
PE (1) PE20070764A1 (da)
RS (1) RS20080197A (da)
TN (1) TNSN08209A1 (da)
TW (1) TW200738723A (da)
UY (1) UY29909A1 (da)
WO (1) WO2007054778A1 (da)
ZA (1) ZA200803173B (da)

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RU2011105768A (ru) * 2008-08-01 2012-09-10 Биокрист Фармасьютикалз, Инк. (Us) Производные пиперидина в качестве ингибиторов jakз
WO2010043633A1 (en) * 2008-10-15 2010-04-22 Palau Pharma, S. A. 2h-pyrazolo [4,3-d]pyrimidin-5-amine derivatives as h4 histamine receptor antagonists for the treatment of allergic, immunological and inflammatory diseases
EP2556820A4 (en) * 2010-04-05 2015-01-21 Sk Chemicals Co Ltd COMPOSITION CONTAINING PDE5 INHIBITOR FOR MITIGATION OF SKIN WRINKLES
EP3189835B1 (en) * 2011-02-28 2018-07-25 National Cerebral and Cardiovascular Center Medical agent for suppressing malignant tumor metastasis
AU2012244550C1 (en) 2011-04-21 2017-06-22 Origenis Gmbh Pyrazolo [4, 3-d] pyrimidines useful as kinase inhibitors
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