NO20083448L - Benzo(f)isoindol-2-ylfenyleddiksyrederivater som EP4 receptoragonister - Google Patents

Benzo(f)isoindol-2-ylfenyleddiksyrederivater som EP4 receptoragonister

Info

Publication number
NO20083448L
NO20083448L NO20083448A NO20083448A NO20083448L NO 20083448 L NO20083448 L NO 20083448L NO 20083448 A NO20083448 A NO 20083448A NO 20083448 A NO20083448 A NO 20083448A NO 20083448 L NO20083448 L NO 20083448L
Authority
NO
Norway
Prior art keywords
isoindol
benzo
acid derivatives
receptor agonists
ylphenylacetic
Prior art date
Application number
NO20083448A
Other languages
English (en)
Inventor
Gerard Martin Paul Giblin
Mark Patrick Healy
Andrew Billinton
Nicholas Maughan Clayton
Original Assignee
Glaxo Group Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=37944208&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=NO20083448(L) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Priority claimed from GB0602237A external-priority patent/GB0602237D0/en
Priority claimed from GB0608976A external-priority patent/GB0608976D0/en
Application filed by Glaxo Group Ltd filed Critical Glaxo Group Ltd
Publication of NO20083448L publication Critical patent/NO20083448L/no

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
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    • C07D209/56—Ring systems containing three or more rings
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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/403—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
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  • Communicable Diseases (AREA)
  • Epidemiology (AREA)
  • Virology (AREA)

Abstract

En forbindelse med formel (I) eller et farmasøytisk akseptabelt derivat derav, hvor R1 R2 R3, R4, R5, R6, X og Y er som definert i spesifikasjonen; en prosess for å lage slike forbindelser; en farmasøytisk sammensetning som omfatter slike forbindelser; og anvendelsen av slike forbindelser i medisin.
NO20083448A 2006-02-03 2008-08-07 Benzo(f)isoindol-2-ylfenyleddiksyrederivater som EP4 receptoragonister NO20083448L (no)

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GB0608976A GB0608976D0 (en) 2006-05-05 2006-05-05 Novel compounds
PCT/EP2007/050992 WO2007088190A1 (en) 2006-02-03 2007-02-01 Benzo (f) isoindol-2-ylphenyl acetic acid derivatives as ep4 receptor agonists

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GB0623203D0 (en) * 2006-11-21 2007-01-03 Glaxo Group Ltd Novel compounds
EP2147672A4 (en) 2007-05-08 2011-11-02 Nat University Corp Hamamatsu University School Of Medicine CYTOTOXIC T CELL ACTIVATOR WITH AN EP4 AGONIST
GB0721611D0 (en) 2007-11-02 2007-12-12 Glaxo Group Ltd Novel compounds
CN103012111B (zh) * 2012-09-12 2016-01-13 衢州学院 一种2,4,5-三氟苯乙酸的制备方法
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EA200870224A1 (ru) 2009-02-27
WO2007088190A1 (en) 2007-08-09
KR20080097417A (ko) 2008-11-05
JP5250427B2 (ja) 2013-07-31
PE20070949A1 (es) 2007-11-22
CR10207A (es) 2008-09-22
EP1979316A1 (en) 2008-10-15
AU2007211484A1 (en) 2007-08-09
EP1979316B1 (en) 2012-07-11
US20110201663A1 (en) 2011-08-18
TW200808722A (en) 2008-02-16
ES2390491T3 (es) 2012-11-13
MA30209B1 (fr) 2009-02-02
JP2013082734A (ja) 2013-05-09
SG169380A1 (en) 2011-03-30
BRPI0708024A2 (pt) 2011-05-17
JP2009525309A (ja) 2009-07-09
UY30121A1 (es) 2007-08-31
CA2640277A1 (en) 2007-08-09
IL192934A0 (en) 2009-02-11
EP2457897A1 (en) 2012-05-30
AR059282A1 (es) 2008-03-19
US8252833B2 (en) 2012-08-28

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