MA30209B1 - Derives de l'acide benzo(f)isoindol-2-ylphenyl acetique comme agonistes du recepteur ep 4 - Google Patents

Derives de l'acide benzo(f)isoindol-2-ylphenyl acetique comme agonistes du recepteur ep 4

Info

Publication number
MA30209B1
MA30209B1 MA31159A MA31159A MA30209B1 MA 30209 B1 MA30209 B1 MA 30209B1 MA 31159 A MA31159 A MA 31159A MA 31159 A MA31159 A MA 31159A MA 30209 B1 MA30209 B1 MA 30209B1
Authority
MA
Morocco
Prior art keywords
ylphenyl
isoindol
benzo
acetic acid
acid derivatives
Prior art date
Application number
MA31159A
Other languages
English (en)
Inventor
Andrew Billinton
Nicholas Maughan Clayton
Gerard Martin Paul Giblin
Mark Patrick Healy
Original Assignee
Glaxo Group Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=37944208&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=MA30209(B1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Priority claimed from GB0602237A external-priority patent/GB0602237D0/en
Priority claimed from GB0608976A external-priority patent/GB0608976D0/en
Application filed by Glaxo Group Ltd filed Critical Glaxo Group Ltd
Publication of MA30209B1 publication Critical patent/MA30209B1/fr

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
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    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/56—Ring systems containing three or more rings
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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/403—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
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  • Communicable Diseases (AREA)
  • Gynecology & Obstetrics (AREA)

Abstract

UN COMPOSÉ DE FORMULE (I) OU UN DE SES DÉRIVÉS PHARMACEUTIQUEMENT ACCEPTABLES FORMULE DANS LAQUELLE R1, R2, R3, R4, R5, R6, X ET Y SONT TELS QUE DÉFINIS DANS LA DESCRIPTION ; UN PROCÉDÉ POUR LA PRÉPARATION DE TELS COMPOSÉS ; UNE COMPOSITION PHARMACEUTIQUE COMPRENANT DE TELS COMPOSÉS ; ET L'UTILISATION DE CES COMPOSÉS EN MÉDECINE.
MA31159A 2006-02-03 2008-08-06 Derives de l'acide benzo(f)isoindol-2-ylphenyl acetique comme agonistes du recepteur ep 4 MA30209B1 (fr)

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GB0602237A GB0602237D0 (en) 2006-02-03 2006-02-03 Novel compounds
GB0608976A GB0608976D0 (en) 2006-05-05 2006-05-05 Novel compounds

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GB0620619D0 (en) * 2006-10-17 2006-11-29 Glaxo Group Ltd Novel compounds
GB0623203D0 (en) * 2006-11-21 2007-01-03 Glaxo Group Ltd Novel compounds
AU2008246579A1 (en) 2007-05-08 2008-11-13 National University Corporation, Hamamatsu University School Of Medicine Cytotoxic T cell activator comprising EP4 agonist
GB0721611D0 (en) 2007-11-02 2007-12-12 Glaxo Group Ltd Novel compounds
CN103012111B (zh) * 2012-09-12 2016-01-13 衢州学院 一种2,4,5-三氟苯乙酸的制备方法
CN110003129B (zh) * 2019-04-18 2021-04-06 济南立德医药技术有限公司 一种佐米曲普坦中间体的制备方法
WO2021082705A1 (fr) 2019-10-29 2021-05-06 宁波舜宇光电信息有限公司 Module de caméra et lentille optique associée, feuille de lentille optique, procédé de fabrication associé et procédé d'assemblage de module de caméra grand angle

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EA200870224A1 (ru) 2009-02-27
JP5250427B2 (ja) 2013-07-31
WO2007088190A1 (fr) 2007-08-09
AR059282A1 (es) 2008-03-19
JP2009525309A (ja) 2009-07-09
CA2640277A1 (fr) 2007-08-09
EP2457897A1 (fr) 2012-05-30
EP1979316A1 (fr) 2008-10-15
CR10207A (es) 2008-09-22
AU2007211484A1 (en) 2007-08-09
TW200808722A (en) 2008-02-16
JP2013082734A (ja) 2013-05-09
US20110201663A1 (en) 2011-08-18
BRPI0708024A2 (pt) 2011-05-17
US8252833B2 (en) 2012-08-28
EP1979316B1 (fr) 2012-07-11
IL192934A0 (en) 2009-02-11
UY30121A1 (es) 2007-08-31
ES2390491T3 (es) 2012-11-13
NO20083448L (no) 2008-10-23
KR20080097417A (ko) 2008-11-05
PE20070949A1 (es) 2007-11-22
SG169380A1 (en) 2011-03-30

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