NO20090138L - Substituted phenyl acetic acids as DP-2 antagonists - Google Patents
Substituted phenyl acetic acids as DP-2 antagonistsInfo
- Publication number
- NO20090138L NO20090138L NO20090138A NO20090138A NO20090138L NO 20090138 L NO20090138 L NO 20090138L NO 20090138 A NO20090138 A NO 20090138A NO 20090138 A NO20090138 A NO 20090138A NO 20090138 L NO20090138 L NO 20090138L
- Authority
- NO
- Norway
- Prior art keywords
- antagonists
- substituted phenyl
- acetic acids
- phenyl acetic
- processes
- Prior art date
Links
- WLJVXDMOQOGPHL-UHFFFAOYSA-N phenylacetic acid Chemical class OC(=O)CC1=CC=CC=C1 WLJVXDMOQOGPHL-UHFFFAOYSA-N 0.000 title abstract 2
- 239000005557 antagonist Substances 0.000 title 1
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 abstract 2
- 238000000034 method Methods 0.000 abstract 2
- 206010012438 Dermatitis atopic Diseases 0.000 abstract 1
- 101150034985 Ptgdr2 gene Proteins 0.000 abstract 1
- 206010039085 Rhinitis allergic Diseases 0.000 abstract 1
- 201000010105 allergic rhinitis Diseases 0.000 abstract 1
- 201000008937 atopic dermatitis Diseases 0.000 abstract 1
- 230000002757 inflammatory effect Effects 0.000 abstract 1
- 239000008194 pharmaceutical composition Substances 0.000 abstract 1
- 230000002265 prevention Effects 0.000 abstract 1
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- C07D295/20—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms by radicals derived from carbonic acid, or sulfur or nitrogen analogues thereof
- C07D295/205—Radicals derived from carbonic acid
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Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US81239806P | 2006-06-09 | 2006-06-09 | |
| PCT/US2007/070803 WO2007143745A2 (en) | 2006-06-09 | 2007-06-08 | Substituted phenyl acetic acids as dp-2 antagonists |
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| NO20090138L true NO20090138L (no) | 2009-03-05 |
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| NO20090138A NO20090138L (no) | 2006-06-09 | 2009-01-09 | Substituted phenyl acetic acids as DP-2 antagonists |
Country Status (10)
| Country | Link |
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| EP (1) | EP2044044A2 (pt) |
| JP (1) | JP2009539880A (pt) |
| CN (1) | CN101490024A (pt) |
| AU (1) | AU2007256597A1 (pt) |
| BR (1) | BRPI0712301A2 (pt) |
| CA (1) | CA2654784A1 (pt) |
| EA (1) | EA200802415A1 (pt) |
| MX (1) | MX2008015696A (pt) |
| NO (1) | NO20090138L (pt) |
| WO (1) | WO2007143745A2 (pt) |
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| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AU2007286829B2 (en) | 2006-08-21 | 2013-05-02 | Array Biopharma, Inc. | 4-substituted phenoxyphenylacetic acid derivatives |
| CN101903335A (zh) * | 2007-10-19 | 2010-12-01 | 詹森药业有限公司 | 连接有胺的γ-分泌酶调节剂 |
| KR101618068B1 (ko) * | 2007-10-19 | 2016-05-04 | 얀센 파마슈티카 엔.브이. | γ-세크레타아제의 탄소 결합된 조절제 |
| KR20100090265A (ko) * | 2007-10-19 | 2010-08-13 | 얀센 파마슈티카 엔.브이. | γ-세크레타아제의 아미드 결합된 조절제 |
| WO2011153359A1 (en) | 2010-06-04 | 2011-12-08 | Albany Molecular Research, Inc. | Glycine transporter-1 inhibitors, methods of making them, and uses thereof |
| CN102958914B (zh) | 2010-07-05 | 2015-05-27 | 埃科特莱茵药品有限公司 | 1-苯基取代的杂环衍生物及其作为前列腺素d2受体调节剂的用途 |
| EP2457900A1 (en) | 2010-11-25 | 2012-05-30 | Almirall, S.A. | New pyrazole derivatives having CRTh2 antagonistic behaviour |
| JP2014525932A (ja) | 2011-08-15 | 2014-10-02 | インターミューン, インコーポレイテッド | リゾホスファチド酸レセプターアンタゴニスト |
| TW201331179A (zh) | 2011-12-21 | 2013-08-01 | Actelion Pharmaceuticals Ltd | 雜環衍生物及其作為前列腺素d2受體調節劑之用途 |
| CA2876808A1 (en) | 2012-07-05 | 2014-01-09 | Actelion Pharmaceuticals Ltd | 1-phenyl-substituted heterocyclyl derivatives and their use as prostaglandin d2 receptor modulators |
| CN102757339A (zh) * | 2012-08-01 | 2012-10-31 | 北京联本医药化学技术有限公司 | 一种改进的4-(2-羧基苄氧基)苯乙酸制备方法 |
| KR20160005356A (ko) | 2013-05-07 | 2016-01-14 | 더 리젠츠 오브 더 유니버시티 오브 캘리포니아 | 방사선완화 약제학적 제형 |
| CN112300120B (zh) * | 2019-07-31 | 2023-04-14 | 北京四环制药有限公司 | 一种用于制备巴罗萨韦或其衍生物的化合物及其制备方法和其应用 |
| EP4065112A4 (en) * | 2019-11-22 | 2023-12-27 | The Regents of the University of California | Taspase1 inhibitors and uses thereof |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| PL377314A1 (pl) * | 2002-12-20 | 2006-01-23 | Amgen Inc. | Modulatory astmy i zapaleń na tle alergicznym |
| PT1471057E (pt) * | 2003-04-25 | 2006-05-31 | Actimis Pharmaceuticals Inc | Derivados de acido pirimidinilacetico uteis para o tratamento de doencas mediadas por crth2 |
| SE0302811D0 (sv) * | 2003-10-23 | 2003-10-23 | Astrazeneca Ab | Novel compounds |
| AR048523A1 (es) * | 2004-04-07 | 2006-05-03 | Kalypsys Inc | Compuestos con estructura de aril sulfonamida y sulfonilo como moduladores de ppar y metodos para tratar trastornos metabolicos |
| JP2008534678A (ja) * | 2005-04-04 | 2008-08-28 | アストラゼネカ・アクチエボラーグ | 新規ジアザスピロアルカン類およびccr8介在疾患の処置のためのそれらの使用 |
| US8097610B2 (en) * | 2005-08-26 | 2012-01-17 | Shionogi & Co., Ltd. | Derivative having PPAR agonistic activity |
| JPWO2007034882A1 (ja) * | 2005-09-22 | 2009-03-26 | 大日本住友製薬株式会社 | 新規アデニン化合物 |
-
2007
- 2007-06-08 AU AU2007256597A patent/AU2007256597A1/en not_active Abandoned
- 2007-06-08 JP JP2009514556A patent/JP2009539880A/ja not_active Withdrawn
- 2007-06-08 EA EA200802415A patent/EA200802415A1/ru unknown
- 2007-06-08 CN CNA2007800263804A patent/CN101490024A/zh active Pending
- 2007-06-08 MX MX2008015696A patent/MX2008015696A/es not_active Application Discontinuation
- 2007-06-08 EP EP07812086A patent/EP2044044A2/en not_active Withdrawn
- 2007-06-08 WO PCT/US2007/070803 patent/WO2007143745A2/en not_active Ceased
- 2007-06-08 BR BRPI0712301-9A patent/BRPI0712301A2/pt not_active IP Right Cessation
- 2007-06-08 CA CA002654784A patent/CA2654784A1/en not_active Abandoned
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2009
- 2009-01-09 NO NO20090138A patent/NO20090138L/no not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| AU2007256597A1 (en) | 2007-12-13 |
| CA2654784A1 (en) | 2007-12-13 |
| CN101490024A (zh) | 2009-07-22 |
| WO2007143745A2 (en) | 2007-12-13 |
| EA200802415A1 (ru) | 2009-06-30 |
| JP2009539880A (ja) | 2009-11-19 |
| BRPI0712301A2 (pt) | 2012-01-17 |
| MX2008015696A (es) | 2009-02-10 |
| WO2007143745A3 (en) | 2008-04-17 |
| EP2044044A2 (en) | 2009-04-08 |
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