NO20090854L - Serin-treonin protein kinase og parp modulatorer - Google Patents

Serin-treonin protein kinase og parp modulatorer

Info

Publication number
NO20090854L
NO20090854L NO20090854A NO20090854A NO20090854L NO 20090854 L NO20090854 L NO 20090854L NO 20090854 A NO20090854 A NO 20090854A NO 20090854 A NO20090854 A NO 20090854A NO 20090854 L NO20090854 L NO 20090854L
Authority
NO
Norway
Prior art keywords
protein kinase
serine
activity
threonine protein
molecules
Prior art date
Application number
NO20090854A
Other languages
English (en)
Norwegian (no)
Inventor
Jeffrey P Whitten
Fabrice Pierre
Peter C Chua
Original Assignee
Cylene Pharmaceuticals Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Cylene Pharmaceuticals Inc filed Critical Cylene Pharmaceuticals Inc
Publication of NO20090854L publication Critical patent/NO20090854L/no

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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47—Quinolines; Isoquinolines
    • A61K31/4738—Quinolines; Isoquinolines ortho- or peri-condensed with heterocyclic ring systems
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    • C07D221/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00
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    • C07D221/04—Ortho- or peri-condensed ring systems
    • C07D221/18—Ring systems of four or more rings
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    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
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    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04—Ortho-condensed systems

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
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  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Neurology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Biomedical Technology (AREA)
  • Rheumatology (AREA)
  • Neurosurgery (AREA)
  • Pulmonology (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Dermatology (AREA)
  • Urology & Nephrology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Obesity (AREA)
  • Endocrinology (AREA)
  • Oncology (AREA)
  • Immunology (AREA)
  • Pain & Pain Management (AREA)
  • Reproductive Health (AREA)
  • Ophthalmology & Optometry (AREA)
  • Psychology (AREA)
  • Communicable Diseases (AREA)
  • Psychiatry (AREA)
  • Hospice & Palliative Care (AREA)
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NO20090854A 2006-09-01 2009-02-25 Serin-treonin protein kinase og parp modulatorer NO20090854L (no)

Applications Claiming Priority (6)

Application Number Priority Date Filing Date Title
US84206106P 2006-09-01 2006-09-01
US84454206P 2006-09-13 2006-09-13
US84668306P 2006-09-22 2006-09-22
US87393606P 2006-12-07 2006-12-07
US89571607P 2007-03-19 2007-03-19
PCT/US2007/077464 WO2008028168A2 (en) 2006-09-01 2007-08-31 Serine-threonine protein kinase and parp modulators

Publications (1)

Publication Number Publication Date
NO20090854L true NO20090854L (no) 2009-04-29

Family

ID=39136972

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20090854A NO20090854L (no) 2006-09-01 2009-02-25 Serin-treonin protein kinase og parp modulatorer

Country Status (16)

Country Link
US (2) US7956064B2 (pt)
EP (1) EP2061765B1 (pt)
JP (1) JP5399905B2 (pt)
KR (1) KR20090050094A (pt)
AU (1) AU2007289065B2 (pt)
BR (1) BRPI0719123A2 (pt)
CA (2) CA2974246C (pt)
DK (1) DK2061765T3 (pt)
ES (1) ES2528316T3 (pt)
IL (1) IL197088A0 (pt)
MX (1) MX2009002298A (pt)
NO (1) NO20090854L (pt)
PL (1) PL2061765T3 (pt)
PT (1) PT2061765E (pt)
RU (1) RU2681209C2 (pt)
WO (1) WO2008028168A2 (pt)

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KR20150038395A (ko) * 2006-04-04 2015-04-08 더 리젠트스 오브 더 유니이버시티 오브 캘리포니아 키나제 길항물질
DK2061765T3 (en) 2006-09-01 2015-01-26 Senhwa Biosciences Inc Serine-threonine protein kinase AND PARP-MODULATOR
US20110160232A1 (en) * 2007-10-04 2011-06-30 Pingda Ren Certain chemical entities and therapeutic uses thereof
BRPI0906473A8 (pt) 2008-01-04 2016-02-10 Intellikine Inc Certas entidades químicas, composições e métodos
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MX2011000216A (es) * 2008-07-08 2011-03-29 Intellikine Inc Inhibidores de cinasa y metodos para su uso.
US20110224223A1 (en) * 2008-07-08 2011-09-15 The Regents Of The University Of California, A California Corporation MTOR Modulators and Uses Thereof
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WO2010036380A1 (en) 2008-09-26 2010-04-01 Intellikine, Inc. Heterocyclic kinase inhibitors
AU2009305669A1 (en) 2008-10-16 2010-04-22 The Regents Of The University Of California Fused ring heteroaryl kinase inhibitors
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PL2364983T3 (pl) * 2008-11-11 2014-04-30 Jeil Pharmaceutical Co Ltd Nowa pochodna tricykliczna lub jej farmaceutycznie dopuszczalne sole, sposób jej wytwarzania, oraz zawierająca ją kompozycja farmaceutyczna
ES2550101T3 (es) 2008-12-17 2015-11-04 Merck Patent Gmbh Inhibidores de proteína quinasa de benzonaftiridinona tricíclica modificada con anillo C y su uso
CN102341107A (zh) * 2009-01-08 2012-02-01 赛林药物股份有限公司 用于肿瘤疾病的联合治疗
US20100173013A1 (en) * 2009-01-08 2010-07-08 Denis Drygin Treatment of neoplastic disorders using combination therapies
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