NO20092293L - Sulfonyl-fenyl-2H-[1,2,4]oksodiazol-5-onderivater, fremgangsmate for fremstilling derav og deres anvendelse som farmasoytiske midler - Google Patents

Sulfonyl-fenyl-2H-[1,2,4]oksodiazol-5-onderivater, fremgangsmate for fremstilling derav og deres anvendelse som farmasoytiske midler

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Publication number
NO20092293L
NO20092293L NO20092293A NO20092293A NO20092293L NO 20092293 L NO20092293 L NO 20092293L NO 20092293 A NO20092293 A NO 20092293A NO 20092293 A NO20092293 A NO 20092293A NO 20092293 L NO20092293 L NO 20092293L
Authority
NO
Norway
Prior art keywords
disorders
preparation
derivatives
oxodiazole
sulfonyl
Prior art date
Application number
NO20092293A
Other languages
English (en)
Inventor
Karl Schoenafinger
Hans-Ludwig Schaefer
Stefanie Keil
Matthias Urmann
Wolfgang Wendler
Maike Glien
Eugen Falk
Original Assignee
Sanofi Aventis
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First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=37998695&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=NO20092293(L) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Sanofi Aventis filed Critical Sanofi Aventis
Publication of NO20092293L publication Critical patent/NO20092293L/no

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4245—Oxadiazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47—Quinolines; Isoquinolines
    • A61K31/472—Non-condensed isoquinolines, e.g. papaverine
    • A61K31/4725—Non-condensed isoquinolines, e.g. papaverine containing further heterocyclic rings
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Abstract

Det er beskrevet sulfonylfenyl-2H-[l,2,4]oksadiazoloner og deres fysiologisk akseptable salter og fysiologisk funksjonelle derivater som viser PPARdelta- eller PPARdelta- og PPARgamma-agonistaktivitet. Det er beskrevet forbindelser av formel I, hvori restene er som definert, og deres fysiologisk akseptable salter og fremgangsmåter for deres fremstilling. Forbindelsene er egnede for behandling og/eller forebyggelse av lidelser ved fettsyremetabolisme og glukose utnyttelsesforstyrrelser, så vel som lidelser hvori insulinresistens er involvert og demyelinerende og andre neurodegenerative lidelser i det sentrale og perifere nervesystem.
NO20092293A 2006-12-14 2009-06-15 Sulfonyl-fenyl-2H-[1,2,4]oksodiazol-5-onderivater, fremgangsmate for fremstilling derav og deres anvendelse som farmasoytiske midler NO20092293L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP06025880A EP1932843A1 (en) 2006-12-14 2006-12-14 Sulfonyl-phenyl-2H-(1,2,4) oxadiazole-5-one derivatives, processes for their preparation and their use as pharmaceuticals
PCT/EP2007/010390 WO2008071311A1 (en) 2006-12-14 2007-11-30 Sulfonyl-phenyl-2h-[1,2,4]oxodiazol-5-one derivatives, processes for their preparation and their use as pharmaceuticals

Publications (1)

Publication Number Publication Date
NO20092293L true NO20092293L (no) 2009-09-08

Family

ID=37998695

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20092293A NO20092293L (no) 2006-12-14 2009-06-15 Sulfonyl-fenyl-2H-[1,2,4]oksodiazol-5-onderivater, fremgangsmate for fremstilling derav og deres anvendelse som farmasoytiske midler

Country Status (24)

Country Link
US (1) US8173674B2 (no)
EP (2) EP1932843A1 (no)
JP (1) JP2010512352A (no)
KR (1) KR20090087922A (no)
CN (1) CN101558064A (no)
AR (1) AR064299A1 (no)
AU (1) AU2007331805A1 (no)
BR (1) BRPI0720416A2 (no)
CA (1) CA2672347A1 (no)
CL (1) CL2007003614A1 (no)
CO (1) CO6210729A2 (no)
CR (1) CR10778A (no)
EC (1) ECSP099409A (no)
MA (1) MA30981B1 (no)
MX (1) MX2009005535A (no)
NO (1) NO20092293L (no)
PE (1) PE20081404A1 (no)
RU (1) RU2009126745A (no)
SV (1) SV2009003293A (no)
TN (1) TN2009000242A1 (no)
TW (1) TW200843749A (no)
UY (1) UY30783A1 (no)
WO (1) WO2008071311A1 (no)
ZA (1) ZA200903160B (no)

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