NO308772B1 - Sublingual eller buckal farmasoytisk blanding inneholdende trans-5-klor-2-metyl-2,3,3a,12b-tetrahydro-1H-dibenz[2,3:6,7]oksepino[4,5-c]pyrrol, samt anvendelse av forbindelsen for fremstilling av farmasoytisk blanding - Google Patents

Sublingual eller buckal farmasoytisk blanding inneholdende trans-5-klor-2-metyl-2,3,3a,12b-tetrahydro-1H-dibenz[2,3:6,7]oksepino[4,5-c]pyrrol, samt anvendelse av forbindelsen for fremstilling av farmasoytisk blanding

Info

Publication number
NO308772B1
NO308772B1 NO19963639A NO963639A NO308772B1 NO 308772 B1 NO308772 B1 NO 308772B1 NO 19963639 A NO19963639 A NO 19963639A NO 963639 A NO963639 A NO 963639A NO 308772 B1 NO308772 B1 NO 308772B1
Authority
NO
Norway
Prior art keywords
pharmaceutical composition
sublingual
buccal
oxepino
dibenz
Prior art date
Application number
NO19963639A
Other languages
English (en)
Norwegian (no)
Other versions
NO963639D0 (no
NO963639L (no
Inventor
Leonardus Petrus Carla Delbressine
Johannes Hubertus Wieringa
Original Assignee
Akzo Nobel Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=8216678&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=NO308772(B1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Akzo Nobel Nv filed Critical Akzo Nobel Nv
Publication of NO963639D0 publication Critical patent/NO963639D0/no
Publication of NO963639L publication Critical patent/NO963639L/no
Publication of NO308772B1 publication Critical patent/NO308772B1/no

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/407Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with other heterocyclic ring systems, e.g. ketorolac, physostigmine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0053Mouth and digestive tract, i.e. intraoral and peroral administration
    • A61K9/006Oral mucosa, e.g. mucoadhesive forms, sublingual droplets; Buccal patches or films; Buccal sprays
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2095Tabletting processes
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/18Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/22Anxiolytics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0053Mouth and digestive tract, i.e. intraoral and peroral administration
    • A61K9/0056Mouth soluble or dispersible forms; Suckable, eatable, chewable coherent forms; Forms rapidly disintegrating in the mouth; Lozenges; Lollipops; Bite capsules; Baked products; Baits or other oral forms for animals

Landscapes

  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Biomedical Technology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Organic Chemistry (AREA)
  • Nutrition Science (AREA)
  • Physiology (AREA)
  • Psychiatry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
NO19963639A 1994-03-02 1996-08-30 Sublingual eller buckal farmasoytisk blanding inneholdende trans-5-klor-2-metyl-2,3,3a,12b-tetrahydro-1H-dibenz[2,3:6,7]oksepino[4,5-c]pyrrol, samt anvendelse av forbindelsen for fremstilling av farmasoytisk blanding NO308772B1 (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP94200521 1994-03-02
PCT/EP1995/000765 WO1995023600A1 (en) 1994-03-02 1995-03-01 Sublingual or buccal pharmaceutical composition

Publications (3)

Publication Number Publication Date
NO963639D0 NO963639D0 (no) 1996-08-30
NO963639L NO963639L (no) 1996-10-30
NO308772B1 true NO308772B1 (no) 2000-10-30

Family

ID=8216678

Family Applications (2)

Application Number Title Priority Date Filing Date
NO19963639A NO308772B1 (no) 1994-03-02 1996-08-30 Sublingual eller buckal farmasoytisk blanding inneholdende trans-5-klor-2-metyl-2,3,3a,12b-tetrahydro-1H-dibenz[2,3:6,7]oksepino[4,5-c]pyrrol, samt anvendelse av forbindelsen for fremstilling av farmasoytisk blanding
NO2010024C NO2010024I2 (no) 1994-03-02 2010-12-13 Trans-5-klor-2-metyl-2,3,3a,12b-tetrahydro-1H-dibenz[2,3:6,7]oksepino[4,5-c]pyrrol eller et salt derav

Family Applications After (1)

Application Number Title Priority Date Filing Date
NO2010024C NO2010024I2 (no) 1994-03-02 2010-12-13 Trans-5-klor-2-metyl-2,3,3a,12b-tetrahydro-1H-dibenz[2,3:6,7]oksepino[4,5-c]pyrrol eller et salt derav

Country Status (22)

Country Link
US (1) US5763476A (pl)
EP (1) EP0746317B1 (pl)
JP (2) JP4099224B2 (pl)
KR (1) KR100330942B1 (pl)
CN (1) CN1079670C (pl)
AT (1) ATE167057T1 (pl)
AU (1) AU692530B2 (pl)
BR (2) BR9506924A (pl)
CA (1) CA2182981C (pl)
CZ (1) CZ284633B6 (pl)
DE (2) DE69502939T2 (pl)
DK (1) DK0746317T3 (pl)
ES (1) ES2118584T3 (pl)
FI (1) FI117923B (pl)
FR (1) FR10C0056I2 (pl)
HU (1) HU225051B1 (pl)
LU (1) LU91751I2 (pl)
NO (2) NO308772B1 (pl)
NZ (1) NZ282394A (pl)
PL (1) PL180465B1 (pl)
RU (1) RU2139051C1 (pl)
WO (1) WO1995023600A1 (pl)

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Also Published As

Publication number Publication date
FR10C0056I2 (pl) 2011-11-25
DK0746317T3 (da) 1999-03-22
NZ282394A (en) 1997-12-19
BR1100625A (pt) 1999-12-28
DE122010000050I2 (de) 2011-07-21
RU2139051C1 (ru) 1999-10-10
KR100330942B1 (ko) 2002-11-16
US5763476A (en) 1998-06-09
EP0746317A1 (en) 1996-12-11
CN1143320A (zh) 1997-02-19
NO963639D0 (no) 1996-08-30
JPH09509674A (ja) 1997-09-30
NO2010024I2 (no) 2012-04-10
NO2010024I1 (no) 2011-01-03
FI963398A0 (fi) 1996-08-30
EP0746317B1 (en) 1998-06-10
PL316080A1 (en) 1996-12-23
NO963639L (no) 1996-10-30
CA2182981C (en) 2006-10-17
AU692530B2 (en) 1998-06-11
CA2182981A1 (en) 1995-09-08
MX9603713A (es) 1997-12-31
ES2118584T3 (es) 1998-09-16
WO1995023600A1 (en) 1995-09-08
HK1008417A1 (en) 1999-05-07
LU91751I2 (fr) 2011-01-04
DE69502939D1 (de) 1998-07-16
CZ284633B6 (cs) 1999-01-13
DE122010000050I1 (de) 2011-05-05
JP4616810B2 (ja) 2011-01-19
FI963398L (fi) 1996-08-30
AU1947895A (en) 1995-09-18
DE69502939T2 (de) 1998-10-22
BR9506924A (pt) 1997-09-30
FR10C0056I1 (pl) 2011-01-28
CN1079670C (zh) 2002-02-27
PL180465B1 (pl) 2001-02-28
ATE167057T1 (de) 1998-06-15
CZ254196A3 (en) 1997-10-15
JP4099224B2 (ja) 2008-06-11
HU9602383D0 (en) 1996-10-28
JP2006342178A (ja) 2006-12-21
HU225051B1 (en) 2006-05-29
HUT76319A (en) 1997-08-28
FI117923B (fi) 2007-04-30

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