NO314685B1 - Anvendelse av cGMP-fosfodiesteraseinhibitorer for fremstilling av et medikament for behandling av erektil dysfunksjon eller seksuelldysfunksjon forbundetmed klitorisforstyrrelser hos en kvinne - Google Patents

Anvendelse av cGMP-fosfodiesteraseinhibitorer for fremstilling av et medikament for behandling av erektil dysfunksjon eller seksuelldysfunksjon forbundetmed klitorisforstyrrelser hos en kvinne Download PDF

Info

Publication number: NO314685B1
Authority: NO; Norway
Prior art keywords: 3alkyl; alkyl; optionally; hydrogen; compound
Prior art date: 1995-07-14

Application number

NO19980153A

Other languages

English (en)

Norwegian (no)

Other versions

NO980153D0 (no

NO980153L (no

Inventor

Alain Claude-Marie Daugan

Original Assignee

Icos Corp

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1995-07-14

Filing date

1998-01-13

Publication date

2003-05-05

Family has litigation

First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=10777695&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=NO314685(B1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.

1998-01-13 Application filed by Icos Corp filed Critical Icos Corp

1998-01-13 Publication of NO980153D0 publication Critical patent/NO980153D0/no

1998-03-10 Publication of NO980153L publication Critical patent/NO980153L/no

2003-05-05 Publication of NO314685B1 publication Critical patent/NO314685B1/no

Links

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IIRDTKBZINWQAW-UHFFFAOYSA-N hexaethylene glycol Chemical class OCCOCCOCCOCCOCCOCCO IIRDTKBZINWQAW-UHFFFAOYSA-N 0.000 description 1
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JUKHNCNDFOAFLT-UHFFFAOYSA-N methyl 1-(1,3-benzodioxol-5-yl)-2-(2-chloroacetyl)-1,3,4,9-tetrahydropyrido[3,4-b]indole-3-carboxylate Chemical compound C1=C2OCOC2=CC(C2C3=C(C4=CC=CC=C4N3)CC(N2C(=O)CCl)C(=O)OC)=C1 JUKHNCNDFOAFLT-UHFFFAOYSA-N 0.000 description 1
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239000008194 pharmaceutical composition Substances 0.000 description 1
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QEVHRUUCFGRFIF-MDEJGZGSSA-N reserpine Chemical compound O([C@H]1[C@@H]([C@H]([C@H]2C[C@@H]3C4=C(C5=CC=C(OC)C=C5N4)CCN3C[C@H]2C1)C(=O)OC)OC)C(=O)C1=CC(OC)=C(OC)C(OC)=C1 QEVHRUUCFGRFIF-MDEJGZGSSA-N 0.000 description 1
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Classifications

- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/4985—Pyrazines or piperazines ortho- or peri-condensed with heterocyclic ring systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/08—Drugs for genital or sexual disorders; Contraceptives for gonadal disorders or for enhancing fertility, e.g. inducers of ovulation or of spermatogenesis
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/10—Drugs for genital or sexual disorders; Contraceptives for impotence
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

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Health & Medical Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Veterinary Medicine (AREA)
Chemical & Material Sciences (AREA)
Public Health (AREA)
General Health & Medical Sciences (AREA)
Medicinal Chemistry (AREA)
Animal Behavior & Ethology (AREA)
Life Sciences & Earth Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Engineering & Computer Science (AREA)
General Chemical & Material Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
Bioinformatics & Cheminformatics (AREA)
Organic Chemistry (AREA)
Reproductive Health (AREA)
Endocrinology (AREA)
Epidemiology (AREA)
Gynecology & Obstetrics (AREA)
Pregnancy & Childbirth (AREA)
Urology & Nephrology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Credit Cards Or The Like (AREA)
Networks Using Active Elements (AREA)
Ultra Sonic Daignosis Equipment (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

NO19980153A 1995-07-14 1998-01-13 Anvendelse av cGMP-fosfodiesteraseinhibitorer for fremstilling av et medikament for behandling av erektil dysfunksjon eller seksuelldysfunksjon forbundetmed klitorisforstyrrelser hos en kvinne NO314685B1 (no)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
GBGB9514464.8A GB9514464D0 (en)	1995-07-14	1995-07-14	Medicaments
PCT/EP1996/003024 WO1997003675A1 (en)	1995-07-14	1996-07-11	Use of cgmp-phosphodiesterase inhibitors to treat impotence

Publications (3)

Publication Number	Publication Date
NO980153D0 NO980153D0 (no)	1998-01-13
NO980153L NO980153L (no)	1998-03-10
NO314685B1 true NO314685B1 (no)	2003-05-05

Family

ID=10777695

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
NO19980153A NO314685B1 (no)	1995-07-14	1998-01-13	Anvendelse av cGMP-fosfodiesteraseinhibitorer for fremstilling av et medikament for behandling av erektil dysfunksjon eller seksuelldysfunksjon forbundetmed klitorisforstyrrelser hos en kvinne

Country Status (24)

Country	Link
US (2)	US6140329A (pl)
EP (1)	EP0839040B1 (pl)
JP (1)	JP4169365B2 (pl)
CN (2)	CN1311828C (pl)
AT (1)	ATE327756T1 (pl)
AU (1)	AU704955B2 (pl)
BR (1)	BR9609758A (pl)
CA (1)	CA2226784C (pl)
CY (2)	CY2563B1 (pl)
CZ (1)	CZ289686B6 (pl)
DE (1)	DE69636193T2 (pl)
DK (1)	DK0839040T3 (pl)
ES (1)	ES2267111T3 (pl)
GB (1)	GB9514464D0 (pl)
HU (1)	HU228369B1 (pl)
IL (1)	IL122870A (pl)
MX (2)	MXPA02009987A (pl)
NO (1)	NO314685B1 (pl)
PL (2)	PL185737B1 (pl)
PT (1)	PT839040E (pl)
RU (1)	RU2181288C2 (pl)
SI (1)	SI0839040T1 (pl)
SK (2)	SK284494B6 (pl)
WO (1)	WO1997003675A1 (pl)

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1995
- 1995-07-14 GB GBGB9514464.8A patent/GB9514464D0/en active Pending
1996
- 1996-07-11 EP EP96923985A patent/EP0839040B1/en not_active Expired - Lifetime
- 1996-07-11 SI SI9630740T patent/SI0839040T1/sl unknown
- 1996-07-11 WO PCT/EP1996/003024 patent/WO1997003675A1/en not_active Ceased
- 1996-07-11 SK SK1259-2003A patent/SK284494B6/sk not_active IP Right Cessation
- 1996-07-11 PL PL96324495A patent/PL185737B1/pl unknown
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- 1996-07-11 PT PT96923985T patent/PT839040E/pt unknown
- 1996-07-11 CN CNB021557918A patent/CN1311828C/zh not_active Expired - Lifetime
- 1996-07-11 AT AT96923985T patent/ATE327756T1/de active
- 1996-07-11 CZ CZ199833A patent/CZ289686B6/cs not_active IP Right Cessation
- 1996-07-11 MX MXPA02009987A patent/MXPA02009987A/es active IP Right Grant
- 1996-07-11 CA CA002226784A patent/CA2226784C/en not_active Expired - Lifetime
- 1996-07-11 US US08/981,989 patent/US6140329A/en not_active Expired - Lifetime
- 1996-07-11 RU RU98102398/14A patent/RU2181288C2/ru active
- 1996-07-11 HU HU9900065A patent/HU228369B1/hu unknown
- 1996-07-11 DK DK96923985T patent/DK0839040T3/da active
- 1996-07-11 PL PL96357665A patent/PL185999B1/pl unknown
- 1996-07-11 AU AU64191/96A patent/AU704955B2/en not_active Expired
- 1996-07-11 BR BR9609758A patent/BR9609758A/pt unknown
- 1996-07-11 JP JP50624897A patent/JP4169365B2/ja not_active Expired - Lifetime
- 1996-07-11 SK SK39-98A patent/SK284141B6/sk not_active IP Right Cessation
- 1996-07-11 ES ES96923985T patent/ES2267111T3/es not_active Expired - Lifetime
- 1996-07-11 DE DE69636193T patent/DE69636193T2/de not_active Expired - Lifetime
- 1996-07-11 CN CN96196723A patent/CN1112928C/zh not_active Expired - Lifetime
1998
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- 1998-01-13 NO NO19980153A patent/NO314685B1/no not_active IP Right Cessation
2000
- 2000-05-18 US US09/573,905 patent/US6608065B1/en not_active Expired - Lifetime
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Also Published As

Publication number	Publication date
CN1112928C (zh)	2003-07-02
HUP9900065A3 (en)	1999-11-29
CA2226784A1 (en)	1997-02-06
MX9800414A (es)	1998-06-30
IL122870A0 (en)	1998-08-16
EP0839040A1 (en)	1998-05-06
NO980153D0 (no)	1998-01-13
MXPA02009987A (es)	2003-02-28
PT839040E (pt)	2006-09-29
CN1513452A (zh)	2004-07-21
DK0839040T3 (da)	2006-09-25
CZ289686B6 (cs)	2002-03-13
US6608065B1 (en)	2003-08-19
SK3998A3 (en)	1998-07-08
DE69636193D1 (de)	2006-07-06
CN1195290A (zh)	1998-10-07
IL122870A (en)	2002-03-10
ATE327756T1 (de)	2006-06-15
SI0839040T1 (sl)	2006-10-31
JPH11509221A (ja)	1999-08-17
CA2226784C (en)	2003-07-08
HK1005363A1 (en)	1999-01-08
ES2267111T3 (es)	2007-03-01
CN1311828C (zh)	2007-04-25
EP0839040B1 (en)	2006-05-31
GB9514464D0 (en)	1995-09-13
SK284494B6 (sk)	2005-05-05
NO980153L (no)	1998-03-10
DE69636193T2 (de)	2007-04-26
HUP9900065A2 (hu)	1999-05-28
WO1997003675A1 (en)	1997-02-06
JP4169365B2 (ja)	2008-10-22
US6140329A (en)	2000-10-31
CY2563B1 (en)	2008-07-02
CY2006007I1 (el)	2009-11-04
SK284141B6 (sk)	2004-10-05
PL185999B1 (pl)	2003-09-30
PL185737B1 (pl)	2003-07-31
BR9609758A (pt)	1999-01-26
CY2006007I2 (el)	2009-11-04
AU6419196A (en)	1997-02-18
AU704955B2 (en)	1999-05-13
CZ3398A3 (cs)	1998-05-13
HU228369B1 (en)	2013-03-28
PL324495A1 (en)	1998-05-25
RU2181288C2 (ru)	2002-04-20

Legal Events

Date	Code	Title	Description
2016-07-18	MK1K	Patent expired

Publication	Publication Date	Title
AU704955B2 (en)	1999-05-13	Use of CGMP-phosphodiesterase inhibitors to treat impotence
JP4150818B2 (ja)	2008-09-17	環状ｇｍｐ特異性ホスフォジエステラーゼインヒビター
US6143757A (en)	2000-11-07	Chemical compounds
US6143746A (en)	2000-11-07	Tetracyclic cyclic GMP-specific phosphodiesterase inhibitors, process of preparation and use
RU2142463C1 (ru)	1999-12-10	Тетрациклические производные, способ их получения (варианты), содержащий их фармацевтический состав, и их использование в терапии
EP1129093A1 (en)	2001-09-05	Pyrazolopyrimidinone derivatives for the treatment of impotence
WO2000002881A2 (fr)	2000-01-20	Utilisation de derives de la cysteine pour preparer un medicament destine a traiter les pathologies qui resultent de la formation de la proteine g heterotrimerique
KR20030005176A (ko)	2003-01-17	4-피리딜- 및 2,4-피리미디닐-치환된 피롤 유도체 및 그의제약학에서의 용도
HK1005363B (en)	2006-12-01	Use of cgmp - phosphodiesterase inhibitors to treat impotence
CZ289832B6 (cs)	2002-04-17	Léčivo pro léčení nebo prevenci samičí sexuální dysfunkce
HK1158519A (en)	2012-07-20	Tetracyclic cyclic gmp-specific phosphodiesterase inhibitors for the treatment of benign prostatic hypertrophy
HK1128423A (en)	2009-10-30	(6r,12ar)-2,3,6,7,12,12a-hexahydro-2-methyl-6-(3,4-methylenedioxyphenyl)-pyrazino[2',1':6,1]pyrido[3,4-b]indole-1,4-dione for the treatment of benign prostatic hypertrophy