NO322011B1 - Aminometylpyrrolidin-derivater som har aromatiske substituenter - Google Patents

Aminometylpyrrolidin-derivater som har aromatiske substituenter Download PDF

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Publication number
NO322011B1
NO322011B1 NO20014374A NO20014374A NO322011B1 NO 322011 B1 NO322011 B1 NO 322011B1 NO 20014374 A NO20014374 A NO 20014374A NO 20014374 A NO20014374 A NO 20014374A NO 322011 B1 NO322011 B1 NO 322011B1
Authority
NO
Norway
Prior art keywords
group
compound
fluoro
salts
hydrates
Prior art date
Application number
NO20014374A
Other languages
English (en)
Norwegian (no)
Other versions
NO20014374L (no
NO20014374D0 (no
Inventor
Katsuhiro Kawakami
Makoto Takemura
Hisashi Takahashi
Rie Miyauchi
Toshiyuki Takeda
Original Assignee
Daiichi Seiyaku Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Daiichi Seiyaku Co filed Critical Daiichi Seiyaku Co
Publication of NO20014374D0 publication Critical patent/NO20014374D0/no
Publication of NO20014374L publication Critical patent/NO20014374L/no
Publication of NO322011B1 publication Critical patent/NO322011B1/no

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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/14Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D498/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/02Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D498/04Ortho-condensed systems
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Pyrrole Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
NO20014374A 1999-03-10 2001-09-07 Aminometylpyrrolidin-derivater som har aromatiske substituenter NO322011B1 (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP6280699 1999-03-10
PCT/JP2000/001439 WO2000053594A1 (en) 1999-03-10 2000-03-09 Aminomethylpyrrolidine derivatives having aromatic substituents

Publications (3)

Publication Number Publication Date
NO20014374D0 NO20014374D0 (no) 2001-09-07
NO20014374L NO20014374L (no) 2001-11-12
NO322011B1 true NO322011B1 (no) 2006-08-07

Family

ID=13210961

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20014374A NO322011B1 (no) 1999-03-10 2001-09-07 Aminometylpyrrolidin-derivater som har aromatiske substituenter

Country Status (10)

Country Link
US (2) US6762181B1 (de)
EP (1) EP1182202B1 (de)
KR (1) KR20010102560A (de)
CN (1) CN1258531C (de)
AT (1) ATE268329T1 (de)
AU (1) AU2940300A (de)
DE (1) DE60011264T2 (de)
NO (1) NO322011B1 (de)
RU (1) RU2255938C2 (de)
WO (1) WO2000053594A1 (de)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2940300A (en) * 1999-03-10 2000-09-28 Daiichi Pharmaceutical Co., Ltd. Aminomethylpyrrolidine derivatives having aromatic substituents
US7384773B1 (en) 2001-05-10 2008-06-10 Pfizer Inc Crystal of HIV protease-cleaved human beta secretase and method for crystallization thereof
US7012144B2 (en) * 2001-12-31 2006-03-14 Korea Research Institute Of Chemical Technology Quinolone carboxylic acid derivatives
US7915418B2 (en) 2003-06-06 2011-03-29 Daiichi Pharmaceutical Co., Ltd. Intermediates and process for the production of optically active quinolonecarboxylic acid derivatives
WO2005111030A1 (en) * 2004-05-12 2005-11-24 Warner-Lambert Company Llc Quinolone antibacterial agents
CN100441580C (zh) * 2006-07-14 2008-12-10 中山大学 喹啉二酮衍生物及其在制备抗菌药物中的应用
FR2928150A1 (fr) 2008-02-29 2009-09-04 Vetoquinol Sa Sa Nouveaux derives 7-substitues de 3-carboxy-oxadiazino-quinolones, leur preparation et leur application comme anti-bacteriens
EP2145891A1 (de) 2008-07-09 2010-01-20 Vetoquinol S.A. 9-substierte 5-Carboxy-Oxadiazin-Chinolon-Derivate, ihre Herstellung und ihre Anwendung als antibakterielle Mittel
US8987242B2 (en) 2008-12-05 2015-03-24 Merck Sharp & Dohme Corp. Morpholinone compounds as factor IXA inhibitors
JP2012511008A (ja) * 2008-12-05 2012-05-17 持田製薬株式会社 IXa因子阻害薬としてのモルホリノン化合物

Family Cites Families (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0207420B1 (de) 1985-06-26 1992-05-06 Daiichi Pharmaceutical Co., Ltd. Pyridoncarbonsäurederivate
JPH0723369B2 (ja) * 1986-12-27 1995-03-15 第一製薬株式会社 ピリドンカルボン酸誘導体
US4920120A (en) * 1988-01-25 1990-04-24 Warner-Lambert Company Antibacterial agents
IL90062A (en) * 1988-04-27 1994-10-07 Daiichi Seiyaku Co Pyridonecarboxylic acid derivatives, their preparation and pharmaceutical compositions containing them
US5157128A (en) * 1990-11-30 1992-10-20 Warner-Lambert Company Certain optically active substituted α,α-dialkyl-pyrrolidine-3-methamines useful as intermediates
DE4230804A1 (de) * 1992-09-15 1994-03-17 Bayer Ag 7-Isoindolinyl-chinolon- und -naphthyridon-Derivate
WO1996023782A1 (en) * 1995-02-02 1996-08-08 Daiichi Pharmaceutical Co., Ltd. Heterocyclic compounds
JP3833738B2 (ja) 1995-11-15 2006-10-18 第一製薬株式会社 置換アミノメチルピロリジン誘導体
JP4323574B2 (ja) * 1995-12-13 2009-09-02 大日本住友製薬株式会社 抗腫瘍剤
WO1997042954A1 (en) * 1996-05-10 1997-11-20 Pharmacia & Upjohn Company Topical administration of antimicrobial agents for the treatment of systemic bacterial diseases
JPH10324686A (ja) 1997-03-27 1998-12-08 Hokuriku Seiyaku Co Ltd 7−(ヒドロキシピロリジニル)キノリンカルボン酸誘導体
JPH10287669A (ja) * 1997-04-10 1998-10-27 Dai Ichi Seiyaku Co Ltd 置換アミノメチルピロリジン誘導体
AU2940300A (en) * 1999-03-10 2000-09-28 Daiichi Pharmaceutical Co., Ltd. Aminomethylpyrrolidine derivatives having aromatic substituents

Also Published As

Publication number Publication date
DE60011264D1 (de) 2004-07-08
CN1350527A (zh) 2002-05-22
NO20014374L (no) 2001-11-12
DE60011264T2 (de) 2005-07-14
US7186843B2 (en) 2007-03-06
KR20010102560A (ko) 2001-11-15
AU2940300A (en) 2000-09-28
ATE268329T1 (de) 2004-06-15
US6762181B1 (en) 2004-07-13
NO20014374D0 (no) 2001-09-07
WO2000053594A1 (en) 2000-09-14
US20040209940A1 (en) 2004-10-21
EP1182202B1 (de) 2004-06-02
CN1258531C (zh) 2006-06-07
RU2255938C2 (ru) 2005-07-10
EP1182202A4 (de) 2002-03-27
EP1182202A1 (de) 2002-02-27

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