NO781053L - Kinazolinderivater. - Google Patents

Kinazolinderivater.

Info

Publication number
NO781053L
NO781053L NO781053A NO781053A NO781053L NO 781053 L NO781053 L NO 781053L NO 781053 A NO781053 A NO 781053A NO 781053 A NO781053 A NO 781053A NO 781053 L NO781053 L NO 781053L
Authority
NO
Norway
Prior art keywords
formula
pyrido
quinazoline
oxo
stated
Prior art date
Application number
NO781053A
Other languages
English (en)
Norwegian (no)
Inventor
Richard Wightman Kierstead
Jefferson Wright Tilley
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of NO781053L publication Critical patent/NO781053L/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/78—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C07D213/81—Amides; Imides
    • C07D213/82—Amides; Imides in position 3
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C205/00—Compounds containing nitro groups bound to a carbon skeleton
    • C07C205/49—Compounds containing nitro groups bound to a carbon skeleton the carbon skeleton being further substituted by carboxyl groups
    • C07C205/57—Compounds containing nitro groups bound to a carbon skeleton the carbon skeleton being further substituted by carboxyl groups having nitro groups and carboxyl groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton
    • C07C205/59—Compounds containing nitro groups bound to a carbon skeleton the carbon skeleton being further substituted by carboxyl groups having nitro groups and carboxyl groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton the carbon skeleton being further substituted by singly-bound oxygen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C323/00—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/61—Halogen atoms or nitro radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/89—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members with hetero atoms directly attached to the ring nitrogen atom
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pulmonology (AREA)
  • Engineering & Computer Science (AREA)
  • Immunology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Plural Heterocyclic Compounds (AREA)
NO781053A 1977-03-24 1978-03-22 Kinazolinderivater. NO781053L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US78093977A 1977-03-24 1977-03-24
US87156478A 1978-01-23 1978-01-23

Publications (1)

Publication Number Publication Date
NO781053L true NO781053L (no) 1978-09-26

Family

ID=27119777

Family Applications (2)

Application Number Title Priority Date Filing Date
NO781053A NO781053L (no) 1977-03-24 1978-03-22 Kinazolinderivater.
NO781051A NO781051L (no) 1977-03-24 1978-03-22 Kinazolinderivater.

Family Applications After (1)

Application Number Title Priority Date Filing Date
NO781051A NO781051L (no) 1977-03-24 1978-03-22 Kinazolinderivater.

Country Status (23)

Country Link
JP (2) JPS53119896A (de)
AR (3) AR218060A1 (de)
AT (2) AT367051B (de)
AU (2) AU521352B2 (de)
DE (2) DE2812585A1 (de)
DK (2) DK128878A (de)
ES (13) ES468126A1 (de)
FI (2) FI780918A7 (de)
FR (2) FR2384771A1 (de)
GB (2) GB1601371A (de)
GR (2) GR72948B (de)
HU (1) HU180782B (de)
IE (1) IE46505B1 (de)
IL (2) IL54328A (de)
IT (2) IT1093710B (de)
LU (2) LU79293A1 (de)
MC (2) MC1185A1 (de)
NL (2) NL7803122A (de)
NO (2) NO781053L (de)
NZ (2) NZ186759A (de)
PH (2) PH14130A (de)
PT (2) PT67821B (de)
SE (2) SE7803418L (de)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2557425C2 (de) * 1975-12-19 1987-03-19 C.H. Boehringer Sohn, 6507 Ingelheim 11-Oxo-11-H-pyrido[2,1-b]-chinazolin-2-carbonsäure und ihre Salze, Verfahren zu ihrer Herstellung und Arzneimittel
DE2845766A1 (de) * 1978-10-18 1980-04-30 Schering Ag Pyrido eckige klammer auf 2,1-b eckige klammer zu -chinazolinon-derivate, ihre herstellung und verwendung
US4395549A (en) 1981-10-02 1983-07-26 Chinoin Gyogyszer Es Vegyeszeti Termekek Gyara Rt. 6-Hydrazono-pyrido[2,1-b] quinazoline-11 ones
ES8306729A1 (es) * 1982-04-30 1983-06-01 Lafarquim "procedimiento de obtencion de 2-isopropil pirido (2-1-b) quinazolinas y sus sales no toxicas con actividad antianafilactica".
US4551460A (en) * 1982-05-10 1985-11-05 Hoffmann-La Roche Inc. Pyrido[2,1-b]quinazoline derivatives useful as agents for treatment of allergic conditions and vascular disorders involving thrombosis
DE3300477A1 (de) * 1983-01-08 1984-07-12 Boehringer Ingelheim KG, 6507 Ingelheim Neue heterocyclische verbindungen, ihre herstellung und verwendung
JPS62238264A (ja) * 1986-04-04 1987-10-19 Nippon Tokushu Noyaku Seizo Kk ２−ハロ−５−アセチルピリジン

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4012387A (en) * 1975-09-18 1977-03-15 Warner-Lambert Company Benzo-[g]pyrido[2,1-b]quinazolinones
US4033961A (en) * 1975-10-07 1977-07-05 Warner-Lambert Company Pyrido[2-1-b]quinazolin-ones and their methods of preparation

Also Published As

Publication number Publication date
NL7803122A (nl) 1978-09-26
DK128878A (da) 1978-09-25
AU521352B2 (en) 1982-04-01
PH14130A (en) 1981-02-26
IL54328A0 (en) 1978-06-15
IL54326A0 (en) 1978-06-15
FI780918A7 (fi) 1978-09-25
ES478326A1 (es) 1979-11-01
DE2812585A1 (de) 1978-09-28
IT1093710B (it) 1985-07-26
FR2384770A1 (fr) 1978-10-20
ES478330A1 (es) 1979-11-01
ES478328A1 (es) 1979-11-01
MC1185A1 (fr) 1978-12-22
AR218480A1 (es) 1980-06-13
FR2384770B1 (de) 1980-10-24
ES478324A1 (es) 1979-11-01
GR73170B (de) 1983-02-14
JPS53119896A (en) 1978-10-19
FR2384771A1 (fr) 1978-10-20
ES468126A1 (es) 1979-09-01
FR2384771B1 (de) 1980-04-04
PT67820A (en) 1978-04-01
ES478325A1 (es) 1979-11-01
AR225415A1 (es) 1982-03-31
DK132778A (da) 1978-09-25
PT67821A (en) 1978-04-01
ES478333A1 (es) 1979-11-16
ES478332A1 (es) 1979-11-16
IT7821655A0 (it) 1978-03-24
LU79293A1 (de) 1979-05-25
AU3447578A (en) 1979-09-27
DE2812586A1 (de) 1978-09-28
IE780582L (en) 1978-09-24
ATA210278A (de) 1981-10-15
AU521096B2 (en) 1982-03-18
LU79290A1 (de) 1979-05-25
AU3447478A (en) 1979-09-27
GR72948B (de) 1984-01-17
IL54328A (en) 1982-03-31
SE7803418L (sv) 1978-09-25
GB1601371A (en) 1981-10-28
ES478323A1 (es) 1979-11-01
NZ186760A (en) 1981-03-16
HU180782B (en) 1983-04-29
PT67821B (en) 1980-03-04
IE46505B1 (en) 1983-06-29
ATA210478A (de) 1981-10-15
NO781051L (no) 1978-09-26
NL7803112A (nl) 1978-09-26
PH13915A (en) 1980-11-04
ES478327A1 (es) 1979-11-01
AR218060A1 (es) 1980-05-15
MC1186A1 (fr) 1978-12-22
GB1601991A (en) 1981-11-04
FI780917A7 (fi) 1978-09-25
IL54326A (en) 1982-04-30
JPS53119897A (en) 1978-10-19
ES478331A1 (es) 1979-11-16
ES468127A1 (es) 1979-09-16
NZ186759A (en) 1981-03-16
SE7803419L (sv) 1978-09-25
IT7821578A0 (it) 1978-03-23
ES478329A1 (es) 1979-11-01
AT367050B (de) 1982-05-25
IT1095493B (it) 1985-08-10
AT367051B (de) 1982-05-25

Similar Documents

Publication Publication Date Title
KR900007780B1 (ko) 축합된 피롤리논 유도체의 제조방법
JP4790703B2 (ja) 環式化合物
AU749224B2 (en) Novel camptothecin tetracyclic analogues, preparation, methods, applications as medicines and pharmaceutical compositions containing them
EP0481429B1 (de) Quinolin-Derivate
JP2008528496A (ja) エストロゲン受容体のモジュレーターとして有用な新規な複素環式ベンゾ［ｃ］クロメン誘導体
CA2173876C (en) Alkoxy alkyl carbamates from imidazo(1,2-a)pyridines
EP0222576A2 (de) Heterocyclische Oxophthalazinylessigsäure
NO161373B (no) Analogifremgangsmaate for fremstilling av terapeutisk aktive pteridin-derivater.
EP0181136B1 (de) Oxindol-Derivate als antiinflammatorische Mittel
CA2717013A1 (en) Tricyclic pyridine derivatives, medicaments containing such compounds, their use and process for their preparation
MXPA06014337A (es) Derivados de cromona utiles como antagonistas vanilloides.
NO781053L (no) Kinazolinderivater.
JP3860618B2 (ja) 置換キノリン誘導体、それらの製造方法およびそれらの使用
UA63891C2 (en) Camptothecine analogues, method for preparing thereof, intermediate compounds and a pharmaceutical composition containing said camptothecine analogues
WO2004002484A1 (ja) ホスホジエステラーゼ阻害剤
JP2000508299A (ja) 抗ウイルス作用を有する置換キノリン誘導体
CS207619B2 (en) Method of making the new derivatives of 5,11-dihydro-6h-pyrido 2,3-b 1,4 benzodiazepin-6-on
US5034531A (en) Fused polycyclic pyranyl compounds as antiviral agents
US4348396A (en) Substituted 11-oxo-11H-pyrido[2,1-b]quinazolines and method of inhibiting allergic reactions with them
WO1994017075A1 (en) Diazepin derivatives and antiviral compositions
US5990106A (en) Bicyclic amino group-substituted pyridonecarboxylic acid derivatives, esters thereof and salts thereof, and bicyclic amines useful as intermediates thereof
NO312463B1 (no) Pyrimid [4,5-b] indoler og forbindelser
EP0481243A1 (de) Tricyclische heterocyclische Verbindungen, ihre Herstellung und Anwendung
JPS61137885A (ja) １，８−ナフチリジン誘導体、そのエステルおよびその塩
CA2196076A1 (en) Acyl imidazopyridines