NO830011L - Fremgangsmaate for fremstilling av farmakologisk aktive n-acyl-peptider. - Google Patents

Fremgangsmaate for fremstilling av farmakologisk aktive n-acyl-peptider.

Info

Publication number
NO830011L
NO830011L NO830011A NO830011A NO830011L NO 830011 L NO830011 L NO 830011L NO 830011 A NO830011 A NO 830011A NO 830011 A NO830011 A NO 830011A NO 830011 L NO830011 L NO 830011L
Authority
NO
Norway
Prior art keywords
lower alkyl
carboxy
hexadecanoyloxyoctadecanoyl
valyl
compound
Prior art date
Application number
NO830011A
Other languages
English (en)
Norwegian (no)
Inventor
Kazuyoshi Umehara
Keizo Yoshida
Hirokazu Tanaka
Itsuo Uchida
Masanobu Kohsaka
Hiroshi Imanaka
Original Assignee
Fujisawa Pharmaceutical Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Fujisawa Pharmaceutical Co filed Critical Fujisawa Pharmaceutical Co
Publication of NO830011L publication Critical patent/NO830011L/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C231/00—Preparation of carboxylic acid amides
    • C07C231/12—Preparation of carboxylic acid amides by reactions not involving the formation of carboxamide groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06—Dipeptides
    • C07K5/06104—Dipeptides with the first amino acid being acidic
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06—Dipeptides
    • C07K5/06008—Dipeptides with the first amino acid being neutral
    • C07K5/06017—Dipeptides with the first amino acid being neutral and aliphatic
    • C07K5/06034—Dipeptides with the first amino acid being neutral and aliphatic the side chain containing 2 to 4 carbon atoms
    • C07K5/06052—Val-amino acid
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06—Dipeptides
    • C07K5/06008—Dipeptides with the first amino acid being neutral
    • C07K5/06078—Dipeptides with the first amino acid being neutral and aromatic or cycloaliphatic
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06—Dipeptides
    • C07K5/06086—Dipeptides with the first amino acid being basic
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Biophysics (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Medicinal Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Biochemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
NO830011A 1982-01-05 1983-01-04 Fremgangsmaate for fremstilling av farmakologisk aktive n-acyl-peptider. NO830011L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB8200212 1982-01-05
GB8215910 1982-06-01

Publications (1)

Publication Number Publication Date
NO830011L true NO830011L (no) 1983-07-06

Family

ID=26281659

Family Applications (1)

Application Number Title Priority Date Filing Date
NO830011A NO830011L (no) 1982-01-05 1983-01-04 Fremgangsmaate for fremstilling av farmakologisk aktive n-acyl-peptider.

Country Status (11)

Country Link
US (1) US4643990A (fr)
EP (1) EP0085255B1 (fr)
KR (1) KR840003235A (fr)
AT (1) ATE22087T1 (fr)
AU (1) AU9173582A (fr)
DE (1) DE3273256D1 (fr)
DK (1) DK579682A (fr)
ES (1) ES8500892A1 (fr)
FI (1) FI824453L (fr)
GR (1) GR77060B (fr)
NO (1) NO830011L (fr)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0099709A3 (fr) * 1982-07-19 1985-11-13 Imperial Chemical Industries Plc Dérivés d'amide
EP0136879A3 (fr) * 1983-09-30 1987-01-07 Yamanouchi Pharmaceutical Co., Ltd. Dérivés d'acides gras et procédés de leur préparation
DE3423582A1 (de) * 1984-06-27 1986-01-09 Bayer Ag, 5090 Leverkusen Substituierte 5-acylamino-1-phenylpyrazole
DE3700173A1 (de) * 1987-01-05 1988-07-14 Hoechst Ag Verfahren zur herstellung von lipophilen aminosaeurederivaten sowie lipophile aminosaeurederivate
FR2611205B1 (fr) * 1987-02-20 1990-03-02 Serbio Dipeptides, procede de preparation et utilisation dans le dosage de proteases
US5464825A (en) * 1991-03-14 1995-11-07 Cornell Research Foundation, Inc. Raising glutathione equivalent levels using N-acyl glutathione monoesters
GB9110298D0 (en) * 1991-05-13 1991-07-03 Fujisawa Pharmaceutical Co New peptide compound and a process for the preparation thereof
JPH08509737A (ja) * 1993-05-03 1996-10-15 コーネル・リサーチ・ファウンデーション・インコーポレイテッド グルタチオンジエステルの使用
US5627210A (en) * 1995-02-06 1997-05-06 Chiron Corporation Branched combinatorial libraries
AU1180200A (en) * 1999-11-12 2001-05-30 Fujimoto Brothers Co., Ltd. Antiinflammatory medicinal compositions
WO2005053727A2 (fr) * 2003-11-29 2005-06-16 Sangstat Medical Corporation Compositions pharmaceutiques pour agents peptidiques bioactifs

Family Cites Families (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NL109134C (fr) * 1900-01-01
NL279057A (fr) * 1900-01-01
FR2907E (fr) * 1903-03-09 1904-07-12 Brunet Loiseau Freres Soc Interrupteur-vibreur pour bobine d'induction, en vue de l'allumage des moteurs
FR4629E (fr) * 1904-04-21 1905-09-02 Jean Victorin Poplawski Générateur de vapeur à mèche
FR7648E (fr) * 1906-02-26 1907-09-17 Georges Clesse Dispositif de changement de vitesse et de renversement de marche pour voitures automobiles
NL299197A (fr) * 1957-07-11
JPS4211925Y1 (fr) * 1966-02-09 1967-07-05
DE1593858A1 (de) * 1967-03-02 1970-10-29 Hoechst Ag Verfahren zur Herstellung tyrosinhaltiger Peptide und deren Derivaten
JPS468685Y1 (fr) * 1967-08-02 1971-03-27
JPS46164Y1 (fr) * 1967-09-05 1971-01-07
US3893992A (en) * 1970-11-19 1975-07-08 Rohm & Haas N-acylated peptides of amino aromatic sulfonic acids and their derivatives
FR2340983A1 (fr) * 1976-02-10 1977-09-09 Ugine Kuhlmann Activateurs pour percomposes
LU78804A1 (de) * 1977-12-30 1979-07-20 Byk Gulden Lomberg Chem Fab N-substituierte w-aminoalkanoyl-w-aminoalkansaeuren,ihre verwendung und verfahren zu ihrer herstellung sowie diese verbindungen enthaltende arzneimittel
US4205069A (en) * 1978-09-29 1980-05-27 American Home Products Corporation Dipeptide narcotic antagonists
US4311640A (en) * 1978-11-14 1982-01-19 Fujisawa Pharmaceutical Co., Ltd. Peptide, process for preparation thereof and use thereof
EP0011283B1 (fr) * 1978-11-14 1982-07-28 Fujisawa Pharmaceutical Co., Ltd. Lactyl-tétrapeptide, procédé pour sa préparation et compositions pharmaceutiques le contenant
FR2460288A1 (fr) * 1979-06-29 1981-01-23 Rhone Poulenc Ind Nouveaux dipeptides, leur preparation et les medicaments qui les contiennent
US4436726A (en) * 1980-12-15 1984-03-13 Fujisawa Pharmaceutical Co., Ltd. N-Acylpeptide compound, processes for the preparation thereof and the pharmaceutical compositions

Also Published As

Publication number Publication date
FI824453A7 (fi) 1983-07-06
DK579682A (da) 1983-07-06
EP0085255A2 (fr) 1983-08-10
EP0085255A3 (en) 1984-08-01
GR77060B (fr) 1984-09-05
DE3273256D1 (en) 1986-10-16
AU9173582A (en) 1983-07-14
KR840003235A (ko) 1984-08-20
EP0085255B1 (fr) 1986-09-10
ATE22087T1 (de) 1986-09-15
FI824453L (fi) 1983-07-06
ES518771A0 (es) 1984-03-01
FI824453A0 (fi) 1982-12-27
ES8500892A1 (es) 1984-03-01
US4643990A (en) 1987-02-17

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