NO923580L - Substituerte imidazolylpropensyrederivater - Google Patents

Substituerte imidazolylpropensyrederivater

Info

Publication number
NO923580L
NO923580L NO92923580A NO923580A NO923580L NO 923580 L NO923580 L NO 923580L NO 92923580 A NO92923580 A NO 92923580A NO 923580 A NO923580 A NO 923580A NO 923580 L NO923580 L NO 923580L
Authority
NO
Norway
Prior art keywords
imidazolylpropenic
substituted
acid derivatives
derivatives
acid
Prior art date
Application number
NO92923580A
Other languages
English (en)
Norwegian (no)
Other versions
NO923580D0 (no
Inventor
Thomas Kraemer
Juergen Dressel
Rudolf Hanko
Walter Huebsch
Ulrich Mueller
Matthias Mueller-Gliemann
Martin Beuck
Stanislav Kazda
Johannes-Peter Stasch
Andreas Knorr
Stefan Wohlfeil
Original Assignee
Bayer Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Ag filed Critical Bayer Ag
Publication of NO923580D0 publication Critical patent/NO923580D0/no
Publication of NO923580L publication Critical patent/NO923580L/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/10—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing aromatic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
NO92923580A 1991-10-01 1992-09-15 Substituerte imidazolylpropensyrederivater NO923580L (no)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE4132632A DE4132632A1 (de) 1991-10-01 1991-10-01 Substituierte imidazolyl-propensaeurederivate

Publications (2)

Publication Number Publication Date
NO923580D0 NO923580D0 (no) 1992-09-15
NO923580L true NO923580L (no) 1993-04-02

Family

ID=6441874

Family Applications (1)

Application Number Title Priority Date Filing Date
NO92923580A NO923580L (no) 1991-10-01 1992-09-15 Substituerte imidazolylpropensyrederivater

Country Status (15)

Country Link
EP (1) EP0539713A1 (cs)
JP (1) JPH05213939A (cs)
KR (1) KR930007937A (cs)
AU (1) AU646596B2 (cs)
CA (1) CA2079268A1 (cs)
CZ (1) CZ297692A3 (cs)
DE (1) DE4132632A1 (cs)
FI (1) FI924355A7 (cs)
HU (1) HUT62576A (cs)
IL (1) IL103293A0 (cs)
MX (1) MX9205435A (cs)
NO (1) NO923580L (cs)
SK (1) SK297692A3 (cs)
TW (1) TW206223B (cs)
ZA (1) ZA927500B (cs)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE4132631A1 (de) * 1991-10-01 1993-04-08 Bayer Ag Imidazolyl-propensaeurederivate
DE4132633A1 (de) * 1991-10-01 1993-04-08 Bayer Ag Cyclisch substituierte imidazolyl-propensaeurederivate
AT398202B (de) * 1991-10-04 1994-10-25 Chem Pharm Forsch Gmbh Neue imidazolderivate, verfahren zu ihrer herstellung und ihre verwendung
GB9218449D0 (en) 1992-08-29 1992-10-14 Boots Co Plc Therapeutic agents
DK0668272T3 (da) * 1994-01-28 2000-09-18 Takeda Chemical Industries Ltd Fremgangsmåde til fremstilling af tetrazolylforbindelser
EP0754042A4 (en) * 1994-03-29 2004-06-23 Merck & Co Inc TREATING ATHEROSCLEROSIS WITH IMIDAZOLES BLOCKING THE ANGIOTENSIN II RECEPTOR
EP1013273A1 (en) * 1998-12-23 2000-06-28 Novartis AG Use of AT-1 receptor antagonist or AT-2 receptor modulator for treating diseases associated with an increase of AT-1 or AT-2 receptors
NZ511938A (en) * 1998-12-23 2004-02-27 Novartis Ag Use of AT-1 receptor antagonist or treating diseases associated with an increase of AT-1 receptor
US6465502B1 (en) * 1998-12-23 2002-10-15 Novartis Ag Additional therapeutic use
US8969514B2 (en) 2007-06-04 2015-03-03 Synergy Pharmaceuticals, Inc. Agonists of guanylate cyclase useful for the treatment of hypercholesterolemia, atherosclerosis, coronary heart disease, gallstone, obesity and other cardiovascular diseases
WO2008151257A2 (en) 2007-06-04 2008-12-11 Synergy Pharmaceuticals Inc. Agonists of guanylate cyclase useful for the treatment of gastrointestinal disorders, inflammation, cancer and other disorders
ES2627848T3 (es) 2008-06-04 2017-07-31 Synergy Pharmaceuticals Inc. Agonistas de la guanilato ciclasa útiles para el tratamiento de trastornos gastrointestinales, inflamación, cáncer y otros trastornos
ES2624828T3 (es) 2008-07-16 2017-07-17 Synergy Pharmaceuticals Inc. Agonistas de la guanilato ciclasa útiles para el tratamiento de trastornos gastrointestinales, inflamación, cáncer y otros
US9616097B2 (en) 2010-09-15 2017-04-11 Synergy Pharmaceuticals, Inc. Formulations of guanylate cyclase C agonists and methods of use
EP2968439A2 (en) 2013-03-15 2016-01-20 Synergy Pharmaceuticals Inc. Compositions useful for the treatment of gastrointestinal disorders
US9708367B2 (en) 2013-03-15 2017-07-18 Synergy Pharmaceuticals, Inc. Agonists of guanylate cyclase and their uses
PL3004138T3 (pl) 2013-06-05 2024-07-29 Bausch Health Ireland Limited Ultra-oczyszczeni agoniści peptydowi cyklazy guanylanowej C, sposób ich uzyskiwania i ich zastosowanie

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0403158A3 (en) * 1989-06-14 1991-12-18 Smithkline Beecham Corporation Imidazolyl-alkenoic acids
SG52330A1 (en) * 1989-06-14 1998-09-28 Smithkline Beecham Corp Imidazolyl-alkenoic acids
GB9017482D0 (en) * 1990-08-09 1990-09-26 Ici Plc Manufacturing process

Also Published As

Publication number Publication date
ZA927500B (en) 1993-05-03
IL103293A0 (en) 1993-02-21
TW206223B (cs) 1993-05-21
DE4132632A1 (de) 1993-04-08
FI924355A0 (fi) 1992-09-29
NO923580D0 (no) 1992-09-15
CZ297692A3 (en) 1993-04-14
HUT62576A (en) 1993-05-28
SK297692A3 (en) 1995-09-13
CA2079268A1 (en) 1993-04-02
MX9205435A (es) 1993-04-01
KR930007937A (ko) 1993-05-20
AU2602492A (en) 1993-04-08
AU646596B2 (en) 1994-02-24
HU9203123D0 (en) 1992-12-28
EP0539713A1 (de) 1993-05-05
JPH05213939A (ja) 1993-08-24
FI924355L (fi) 1993-04-02
FI924355A7 (fi) 1993-04-02

Similar Documents

Publication Publication Date Title
FI922953A7 (fi) 7-azaisoindolinylkinolon- och naftyridonkarboxylsyraderivat
FI922873A7 (fi) 7-isoindolinyl-kinolon- och -naftyridonkarboxylsyraderivat
FI921163A7 (fi) N-acyl-a-aminosyraderivat
FI933260A7 (fi) Heteroaettiksyraderivat
DE69208877D1 (de) Chinuclidinderivate
FI924160A7 (fi) Benzanilidderivat
FI935726A7 (fi) Atsanorbornaanijohdannaisia
FI924159L (fi) Benzanilidderivat
NO922182D0 (no) Krystallinske oksatiolan-derivater
FI925763L (fi) Fungicida 2-imidazolin-5-on- och 2-imidazolin-5-tionderivat
FI923726L (fi) Sulfaterade glykosaminoglykanoidderivat
FI922095L (fi) Substituerade karboxylsyraderivat
FI924355A7 (fi) Substituoituja imidatsolyylipropeenihappojohdannaisia
FI935243L (fi) Pyridonkarboxylsyraderivat
NO923581D0 (no) Sykliske substituerte imidazolylpropensyrederivater
FI924354A7 (fi) Imidatsolyylipropeenihappojohdannaisia
FI925469A7 (fi) Tiatsolyylillä substituoidut kinolyylimetoksifenyylietikkahappojohdannaiset
FI920394A7 (fi) 3-kinuklidiinijohdannaiset
FI940003L (fi) Aminohappojohdannaiset
FI932953A7 (fi) Imidazolylsubstituerade fenylpropion- och -kanelsyraderivat
FI924145L (fi) 3-cykloalkylprop-2-enamidderivat
DE69202059D1 (de) Propensäurederivate.
FI922125L (fi) Mikrobidogiskt foerfarande foer framstaellning av 5-hydroxipyrazinkarboxylsyra
FI942070A7 (fi) Nitroksialkyyliamidijohdannaiset
FI933346A7 (fi) Aminoalkylpyrrolidinyltiokarbapenemderivat