NO940250L - Fluorerte kinoloner, fremgangsmaate for fremstilling og farmasoeytiske preparater inneholdende slike - Google Patents

Fluorerte kinoloner, fremgangsmaate for fremstilling og farmasoeytiske preparater inneholdende slike

Info

Publication number
NO940250L
NO940250L NO940250A NO940250A NO940250L NO 940250 L NO940250 L NO 940250L NO 940250 A NO940250 A NO 940250A NO 940250 A NO940250 A NO 940250A NO 940250 L NO940250 L NO 940250L
Authority
NO
Norway
Prior art keywords
preparation
methods
pharmaceutical preparations
preparations containing
formula
Prior art date
Application number
NO940250A
Other languages
English (en)
Other versions
NO940250D0 (no
Inventor
Claude Perrin
Original Assignee
Bouchara Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bouchara Sa filed Critical Bouchara Sa
Publication of NO940250D0 publication Critical patent/NO940250D0/no
Publication of NO940250L publication Critical patent/NO940250L/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

Nye 6-fluor-7-piperidin-kinolon- 3-karboksylsyrer med generell formel (I), hvori Z er et aminoradikal, Rj er hydrogen, et (eventuelt hydroksylert) lavere alkylradikal, et acylradikal avledet fra en organisk karboksylsyre, en alkylkarbonsyre, eller en aryl- sulfonsyre eller et arylaminokarbonyl- radikal med formel (a): hvori Ar er et mono- eller bisyklisk aromatisk radikal eventuelt substituert med l, 2 eller 3 substituenter utvalgt fra lavere alkyl, halogen og trifluormetyl, T er oksygen eller svovel, og R, R2, R3, m og n er definert som angitt i beskrivelsen. Forbindelsene med formel (I) utgjør aktive bestanddeler i antibakterielle legemidler.
NO940250A 1992-05-26 1994-01-25 Fluorerte kinoloner, fremgangsmaate for fremstilling og farmasoeytiske preparater inneholdende slike NO940250L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR9206404A FR2692577B1 (fr) 1992-05-26 1992-05-26 Nouvelles quinolones fluorees, leur procede de preparation et les compositions pharmaceutiques en renfermant.
PCT/FR1993/000505 WO1993024479A1 (fr) 1992-05-26 1993-05-25 Nouvelles quinolones fluorees, leur procede de preparation et les compositions pharmaceutiques en renfermant

Publications (2)

Publication Number Publication Date
NO940250D0 NO940250D0 (no) 1994-01-25
NO940250L true NO940250L (no) 1994-01-25

Family

ID=9430170

Family Applications (1)

Application Number Title Priority Date Filing Date
NO940250A NO940250L (no) 1992-05-26 1994-01-25 Fluorerte kinoloner, fremgangsmaate for fremstilling og farmasoeytiske preparater inneholdende slike

Country Status (10)

Country Link
US (1) US5478841A (no)
EP (1) EP0598089A1 (no)
JP (1) JPH06509589A (no)
CA (1) CA2114132A1 (no)
FI (1) FI940357L (no)
FR (1) FR2692577B1 (no)
HU (1) HUT67679A (no)
NO (1) NO940250L (no)
OA (1) OA09881A (no)
WO (1) WO1993024479A1 (no)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2005033108A1 (en) * 2003-09-22 2005-04-14 Janssen Pharmaceutica, N.V. 7-amino alkylidenyl-heterocyclic quinolones and naphthyridones
US7732612B2 (en) * 2004-09-09 2010-06-08 Janssen Pharmaceutica, N.V. 7-amino alkylidenyl-heterocyclic quinolones and naphthyridones
US20090156577A1 (en) * 2004-09-09 2009-06-18 Benjamin Davis 7-amino alkylidenyl-heterocyclic quinolones and naphthyridones

Family Cites Families (27)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA1092606A (en) * 1976-10-05 1980-12-30 Herbert Berger 1-(n-acylcarbamoyl)-2-cyano-aziridines and the preparation thereof
US4665079A (en) * 1984-02-17 1987-05-12 Warner-Lambert Company Antibacterial agents
DE3318145A1 (de) * 1983-05-18 1984-11-22 Bayer Ag, 5090 Leverkusen 7-amino-1-cyclopropyl-6,8-difluor-1,4-dihydro-4-oxo-3-chinolincarbonsaeuren, verfahren zu ihrer herstellung sowie diese enthaltende antibakterielle mittel
JPS6089480A (ja) * 1983-10-21 1985-05-20 Dainippon Pharmaceut Co Ltd ピリドンカルボン酸誘導体
JPS60228479A (ja) * 1984-04-26 1985-11-13 Toyama Chem Co Ltd １，４−ジヒドロ−４−オキソナフチリジン誘導体およびその塩
US5097032A (en) * 1984-07-20 1992-03-17 Warner-Lambert Company Antibacterial agents - II
US4657913A (en) * 1985-04-18 1987-04-14 Warner-Lambert Company Trifluoro- quinoline -3- carboxylic acids and their use as anti-bacterial agents
JPH0635457B2 (ja) * 1985-06-28 1994-05-11 杏林製薬株式会社 ピリドンカルボン酸誘導体およびその製造方法
JPH089597B2 (ja) * 1986-01-21 1996-01-31 杏林製薬株式会社 選択毒性に優れた８‐アルコキシキノロンカルボン酸およびその塩並びにその製造方法
JPS62215572A (ja) * 1986-03-17 1987-09-22 Kyorin Pharmaceut Co Ltd キノロンカルボン酸誘導体
EP0241206A3 (en) * 1986-03-31 1989-05-10 Sankyo Company Limited Quinoline-3-carboxylic acid derivatives, their preparation and use
JPS63198664A (ja) * 1986-03-31 1988-08-17 Sankyo Co Ltd キノロンカルボン酸誘導体
IL83049A (en) * 1986-07-04 1991-12-12 Chemie Linz Ag 4-quinolinone-3-carboxylic acid derivatives,their manufacture and pharmaceutical compositions containing them
US5563138A (en) * 1987-04-16 1996-10-08 Otsuka Pharmaceutical Company, Limited Benzoheterocyclic compounds
US4851418A (en) * 1987-08-21 1989-07-25 Warner-Lambert Company Naphthyridine antibacterial agents containing an α-amino acid in the side chain of the 7-substituent
FR2634483B2 (fr) * 1987-12-29 1994-03-04 Esteve Labor Dr Derives des acides 7-(1-azetidinyl)-1,4-dihydro-4-oxoquinoleine-3-carboxyliques, leur preparation et leur application en tant que medicaments
US5173484A (en) * 1988-02-05 1992-12-22 Bayer Aktiengesellschaft Quinolone- and naphthyridone carboxylic acid derivatives, process for their production, antibacterial compositions and feed additives containing them
CA1340285C (en) * 1988-05-19 1998-12-22 Hiroyuki Nagano Novel quinolonecarboxylic acid derivatives having at 7-position a piperidin-1-yl substituent
AU618823B2 (en) * 1988-07-20 1992-01-09 Sankyo Company Limited 4-oxoquinoline-3-carboxylic acid derivatives, their preparation and their use
US5328908A (en) * 1988-10-24 1994-07-12 Procter & Gamble Pharmaceuticals, Inc. Antimicrobial quinolone thioureas
DE3918544A1 (de) * 1989-06-07 1990-12-13 Bayer Ag Verfahren zur herstellung von 7-(3-amino- sowie 3-amino-methyl-1-pyrrolidinyl)-3-chinolon- carbonsaeuren sowie -naphthyridoncarbonsaeuren
US5047538A (en) * 1990-04-12 1991-09-10 Warner-Lambert Company Quinolinecarboxylic acid antibacterial agents
US5116834A (en) * 1990-04-12 1992-05-26 Warner-Lambert Company Quinolinecarboxylic acid antibacterial agents
US5342846A (en) * 1990-12-05 1994-08-30 Synphar Laboratories, Inc. 7-substituted-6-fluoro-1,4-dihydro-4-oxo-quinoline-3-carboxylic acid compounds and 7-(substituted triazolyl pyrrolidin-1-yl) 4-oxoquinoline-3-carboxylic acid derivatives useful as antibacterial agents
FR2673426B1 (fr) * 1991-03-01 1993-07-16 Bouchara Sa Nouvelles quinolones, leur procede de preparation et les compositions en refermant.
US5250532A (en) * 1991-04-11 1993-10-05 Dowelanco 3,4,N-trisubstituted-4,5-dihydro-1H-pyrazole-1-carboxamides and their use as insecticides
US5221676A (en) * 1992-02-06 1993-06-22 Warner-Lambert Company 7-substituted quinolones and naphthyridones as antibacterial agents

Also Published As

Publication number Publication date
CA2114132A1 (fr) 1993-12-09
US5478841A (en) 1995-12-26
FR2692577B1 (fr) 1996-02-02
JPH06509589A (ja) 1994-10-27
FI940357A0 (fi) 1994-01-25
FR2692577A1 (fr) 1993-12-24
HUT67679A (en) 1995-04-28
NO940250D0 (no) 1994-01-25
WO1993024479A1 (fr) 1993-12-09
OA09881A (fr) 1994-09-15
EP0598089A1 (fr) 1994-05-25
FI940357A7 (fi) 1994-03-28
FI940357L (fi) 1994-03-28
HU9400211D0 (en) 1994-05-30

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