NO975150L - Fremgangsmåte for fremstilling av enantiomere former av aminoalkylaminofenylpropansyre - Google Patents
Fremgangsmåte for fremstilling av enantiomere former av aminoalkylaminofenylpropansyreInfo
- Publication number
- NO975150L NO975150L NO975150A NO975150A NO975150L NO 975150 L NO975150 L NO 975150L NO 975150 A NO975150 A NO 975150A NO 975150 A NO975150 A NO 975150A NO 975150 L NO975150 L NO 975150L
- Authority
- NO
- Norway
- Prior art keywords
- preparation
- acid
- aminoalkylaminophenylpropanoic
- phenylalanine
- enantiomeric forms
- Prior art date
Links
- 239000002253 acid Substances 0.000 title abstract 2
- 238000000034 method Methods 0.000 title abstract 2
- COLNVLDHVKWLRT-QMMMGPOBSA-N L-phenylalanine Chemical compound OC(=O)[C@@H](N)CC1=CC=CC=C1 COLNVLDHVKWLRT-QMMMGPOBSA-N 0.000 abstract 2
- ATUOYWHBWRKTHZ-UHFFFAOYSA-N Propane Chemical compound CCC ATUOYWHBWRKTHZ-UHFFFAOYSA-N 0.000 abstract 2
- GOJUJUVQIVIZAV-UHFFFAOYSA-N 2-amino-4,6-dichloropyrimidine-5-carbaldehyde Chemical group NC1=NC(Cl)=C(C=O)C(Cl)=N1 GOJUJUVQIVIZAV-UHFFFAOYSA-N 0.000 abstract 1
- COLNVLDHVKWLRT-MRVPVSSYSA-N D-phenylalanine Chemical compound OC(=O)[C@H](N)CC1=CC=CC=C1 COLNVLDHVKWLRT-MRVPVSSYSA-N 0.000 abstract 1
- 125000003282 alkyl amino group Chemical group 0.000 abstract 1
- 150000001412 amines Chemical group 0.000 abstract 1
- 238000006243 chemical reaction Methods 0.000 abstract 1
- 239000001257 hydrogen Chemical group 0.000 abstract 1
- 229910052739 hydrogen Chemical group 0.000 abstract 1
- 125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 1
- 125000000636 p-nitrophenyl group Chemical group [H]C1=C([H])C(=C([H])C([H])=C1*)[N+]([O-])=O 0.000 abstract 1
- COLNVLDHVKWLRT-UHFFFAOYSA-N phenylalanine Natural products OC(=O)C(N)CC1=CC=CC=C1 COLNVLDHVKWLRT-UHFFFAOYSA-N 0.000 abstract 1
- 239000001294 propane Substances 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C227/00—Preparation of compounds containing amino and carboxyl groups bound to the same carbon skeleton
- C07C227/14—Preparation of compounds containing amino and carboxyl groups bound to the same carbon skeleton from compounds containing already amino and carboxyl groups or derivatives thereof
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C229/00—Compounds containing amino and carboxyl groups bound to the same carbon skeleton
- C07C229/02—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton
- C07C229/04—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and saturated
- C07C229/06—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and saturated having only one amino and one carboxyl group bound to the carbon skeleton
- C07C229/10—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and saturated having only one amino and one carboxyl group bound to the carbon skeleton the nitrogen atom of the amino group being further bound to acyclic carbon atoms or to carbon atoms of rings other than six-membered aromatic rings
- C07C229/12—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and saturated having only one amino and one carboxyl group bound to the carbon skeleton the nitrogen atom of the amino group being further bound to acyclic carbon atoms or to carbon atoms of rings other than six-membered aromatic rings to carbon atoms of acyclic carbon skeletons
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Peptides Or Proteins (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Abstract
Fremgangsmåte for fremstilling av enantiomere former av aminoalkylaminofcnylpropansyre En fremgangsmåte for fremstilling av en enantiomcr form av 2-amino 3-(4-alkylamino- fenyl)propans>TC med den generelle formel (1) CO^H m-, der Alk betyr en Ci.j-alkylrcst, i S- cllcr R-form, samt sallcr derav, fra rcspckliw (L)- fcnylalanin cllcr (D)-fcnylalanin, ved nilrcring med cftcrfolgcndc omdanning av nilrorcslcn av det oppnådde 4-nitrofcnylalanin med den generelle formel (II) «0- :02H NH-R der R er et hydrogenatom eller en bcsk>'tlcndc gnippe, til en alkylaminorcst, cfler eventuell besk'yttelse av aminfunksjoncn av fenylalanin.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR9506890A FR2735126B1 (fr) | 1995-06-12 | 1995-06-12 | Procede de preparation des formes enantiomeres de l'acide amino alkylaminophenylpropanoique |
| PCT/FR1996/000872 WO1996041794A1 (fr) | 1995-06-12 | 1996-06-10 | Procede de preparation des formes enantiomeres de l'acide amino alkylaminophenyl propanoique |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| NO975150L true NO975150L (no) | 1997-11-10 |
| NO975150D0 NO975150D0 (no) | 1997-11-10 |
Family
ID=9479840
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NO975150A NO975150D0 (no) | 1995-06-12 | 1997-11-10 | Fremgangsmåte for fremstilling av enantiomere former av aminoalkylaminofenylpropansyre |
Country Status (23)
| Country | Link |
|---|---|
| US (1) | US5969179A (no) |
| EP (1) | EP0837843B1 (no) |
| JP (1) | JPH11509182A (no) |
| KR (1) | KR19990022841A (no) |
| AR (1) | AR002468A1 (no) |
| AT (1) | ATE205471T1 (no) |
| AU (1) | AU6308396A (no) |
| BR (1) | BR9608974A (no) |
| CA (1) | CA2220403A1 (no) |
| CZ (1) | CZ399497A3 (no) |
| DE (1) | DE69615195T2 (no) |
| DK (1) | DK0837843T3 (no) |
| ES (1) | ES2164252T3 (no) |
| FR (1) | FR2735126B1 (no) |
| GR (1) | GR3036612T3 (no) |
| HU (1) | HUP9900051A3 (no) |
| IL (1) | IL122531A0 (no) |
| NO (1) | NO975150D0 (no) |
| PT (1) | PT837843E (no) |
| SK (1) | SK170197A3 (no) |
| TW (1) | TW415930B (no) |
| WO (1) | WO1996041794A1 (no) |
| ZA (1) | ZA964931B (no) |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| HU204026B (en) * | 1984-03-12 | 1991-11-28 | Alkaloida Vegyeszeti Gyar | Process for producing di-beta-substituted phenylamino acids |
-
1995
- 1995-06-12 FR FR9506890A patent/FR2735126B1/fr not_active Expired - Fee Related
-
1996
- 1996-06-10 IL IL12253196A patent/IL122531A0/xx unknown
- 1996-06-10 ES ES96922085T patent/ES2164252T3/es not_active Expired - Lifetime
- 1996-06-10 JP JP9502697A patent/JPH11509182A/ja not_active Ceased
- 1996-06-10 PT PT96922085T patent/PT837843E/pt unknown
- 1996-06-10 AT AT96922085T patent/ATE205471T1/de not_active IP Right Cessation
- 1996-06-10 KR KR1019970709310A patent/KR19990022841A/ko not_active Withdrawn
- 1996-06-10 US US08/981,038 patent/US5969179A/en not_active Expired - Fee Related
- 1996-06-10 DK DK96922085T patent/DK0837843T3/da active
- 1996-06-10 AU AU63083/96A patent/AU6308396A/en not_active Abandoned
- 1996-06-10 EP EP96922085A patent/EP0837843B1/fr not_active Expired - Lifetime
- 1996-06-10 BR BR9608974A patent/BR9608974A/pt not_active Application Discontinuation
- 1996-06-10 WO PCT/FR1996/000872 patent/WO1996041794A1/fr not_active Ceased
- 1996-06-10 TW TW085106958A patent/TW415930B/zh active
- 1996-06-10 SK SK1701-97A patent/SK170197A3/sk unknown
- 1996-06-10 ZA ZA964931A patent/ZA964931B/xx unknown
- 1996-06-10 CZ CZ973994A patent/CZ399497A3/cs unknown
- 1996-06-10 DE DE69615195T patent/DE69615195T2/de not_active Expired - Fee Related
- 1996-06-10 HU HU9900051A patent/HUP9900051A3/hu unknown
- 1996-06-10 CA CA002220403A patent/CA2220403A1/fr not_active Abandoned
- 1996-06-12 AR ARP960103117A patent/AR002468A1/es unknown
-
1997
- 1997-11-10 NO NO975150A patent/NO975150D0/no not_active Application Discontinuation
-
2001
- 2001-09-13 GR GR20010400340T patent/GR3036612T3/el not_active IP Right Cessation
Also Published As
| Publication number | Publication date |
|---|---|
| ZA964931B (en) | 1997-01-08 |
| HUP9900051A3 (en) | 2000-07-28 |
| FR2735126B1 (fr) | 1997-07-18 |
| FR2735126A1 (fr) | 1996-12-13 |
| WO1996041794A1 (fr) | 1996-12-27 |
| DE69615195D1 (de) | 2001-10-18 |
| EP0837843A1 (fr) | 1998-04-29 |
| PT837843E (pt) | 2001-12-28 |
| ATE205471T1 (de) | 2001-09-15 |
| GR3036612T3 (en) | 2001-12-31 |
| DE69615195T2 (de) | 2002-07-04 |
| KR19990022841A (ko) | 1999-03-25 |
| CA2220403A1 (fr) | 1996-12-27 |
| JPH11509182A (ja) | 1999-08-17 |
| BR9608974A (pt) | 1999-02-02 |
| CZ399497A3 (cs) | 1998-07-15 |
| NO975150D0 (no) | 1997-11-10 |
| MX9708753A (es) | 1998-03-31 |
| SK170197A3 (en) | 1998-05-06 |
| EP0837843B1 (fr) | 2001-09-12 |
| AR002468A1 (es) | 1998-03-25 |
| DK0837843T3 (da) | 2001-11-19 |
| HUP9900051A2 (hu) | 1999-04-28 |
| AU6308396A (en) | 1997-01-09 |
| ES2164252T3 (es) | 2002-02-16 |
| US5969179A (en) | 1999-10-19 |
| TW415930B (en) | 2000-12-21 |
| IL122531A0 (en) | 1998-06-15 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FC2A | Withdrawal, rejection or dismissal of laid open patent application |