NO981241L - Heteroarylsubstituerte akryloylguanidinderivater og farmas÷ytiske preparater inneholdende disse - Google Patents
Heteroarylsubstituerte akryloylguanidinderivater og farmas÷ytiske preparater inneholdende disseInfo
- Publication number
- NO981241L NO981241L NO981241A NO981241A NO981241L NO 981241 L NO981241 L NO 981241L NO 981241 A NO981241 A NO 981241A NO 981241 A NO981241 A NO 981241A NO 981241 L NO981241 L NO 981241L
- Authority
- NO
- Norway
- Prior art keywords
- optionally substituted
- derivatives
- pharmaceutical preparations
- preparations containing
- heteroaryl substituted
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/78—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
- C07D213/81—Amides; Imides
- C07D213/82—Amides; Imides in position 3
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D207/30—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members
- C07D207/32—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
- C07D207/325—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms with substituted hydrocarbon radicals directly attached to the ring nitrogen atom
- C07D207/327—Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
- A61K31/357—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having two or more oxygen atoms in the same ring, e.g. crown ethers, guanadrel
- A61K31/36—Compounds containing methylenedioxyphenyl groups, e.g. sesamin
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Epidemiology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP24171695 | 1995-09-20 | ||
| PCT/JP1996/002696 WO1997011055A1 (en) | 1995-09-20 | 1996-09-19 | Heteroaryl-substituted acryloylguanidine derivatives and medicinal composition thereof |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| NO981241D0 NO981241D0 (no) | 1998-03-19 |
| NO981241L true NO981241L (no) | 1998-05-20 |
Family
ID=17078479
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NO981241A NO981241L (no) | 1995-09-20 | 1998-03-19 | Heteroarylsubstituerte akryloylguanidinderivater og farmas÷ytiske preparater inneholdende disse |
Country Status (13)
| Country | Link |
|---|---|
| EP (1) | EP0861831A4 (de) |
| KR (1) | KR19990063589A (de) |
| CN (1) | CN1196721A (de) |
| AU (1) | AU702092B2 (de) |
| BR (1) | BR9610530A (de) |
| CA (1) | CA2232497A1 (de) |
| CZ (1) | CZ84098A3 (de) |
| HU (1) | HUP9901336A3 (de) |
| NO (1) | NO981241L (de) |
| PL (1) | PL326033A1 (de) |
| SK (1) | SK35198A3 (de) |
| WO (1) | WO1997011055A1 (de) |
| ZA (1) | ZA967800B (de) |
Families Citing this family (17)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5942516A (en) * | 1995-08-02 | 1999-08-24 | Elliott; John Duncan | Endothelin receptor antagonists |
| CA2283404A1 (en) * | 1997-03-06 | 1998-09-11 | Jun Sasamori | Cycloalka¬b|pyridine-3-carbonylguanidine derivatives, process for producing the same, and drugs containing the same |
| JP2003507468A (ja) * | 1999-08-23 | 2003-02-25 | スミスクライン・ビーチャム・コーポレイション | 脂肪酸シンターゼ阻害剤 |
| EP1695716A2 (de) * | 2000-12-26 | 2006-08-30 | Sankyo Company, Limited | Medizinische Zusammensetzungen enthaltend ein Diuretikum und einen Insulin-Sensibilisator |
| ES2332659T3 (es) | 2004-06-16 | 2010-02-10 | Wyeth | Derivados de amino-5,5-difenilimidazolona para la inhibicion de beta-secretasa. |
| BRPI0512220A (pt) | 2004-06-16 | 2008-02-19 | Wyeth Corp | método para tratamento, prevenção ou melhora de uma doença ou distúrbio; composição farmacêutica; processo para a preparação de um composto; e uso de um composto |
| EP1836208A2 (de) | 2005-01-14 | 2007-09-26 | Wyeth Incoporated | Amino-imidazolone als beta-sekretase-hemmer |
| RU2007124935A (ru) | 2005-02-01 | 2009-03-10 | Вайет (Us) | АМИНОПИРИДИНЫ В КАЧЕСТВЕ ИНГИБИТОРОВ β-СЕКТРЕТАЗЫ |
| WO2006088694A1 (en) | 2005-02-14 | 2006-08-24 | Wyeth | SUBSTITUTED THIENYL AND FURYL ACYLGUANIDINES AS β-SECRETASE MODULATORS |
| KR20070102751A (ko) | 2005-02-14 | 2007-10-19 | 와이어쓰 | β-세크레타제 억제제로서의 아졸릴아실구아니딘 |
| TW200738683A (en) | 2005-06-30 | 2007-10-16 | Wyeth Corp | Amino-5-(5-membered)heteroarylimidazolone compounds and the use thereof for β-secretase modulation |
| WO2007005404A1 (en) | 2005-06-30 | 2007-01-11 | Wyeth | AMINO-5-(6-MEMBERED)HETEROARYLIMIDAZOLONE COMPOUNDS AND THE USE THEREOF FOR ß-SECRETASE MODULATION |
| EP2256107A1 (de) | 2005-09-26 | 2010-12-01 | Wyeth LLC | Amino-5-[4-(difluoromethoxy)phenyl]-5-phenylimidazolon-Verbindungen als Beta-Secretase-Hemmer (BACE) |
| WO2007100536A1 (en) | 2006-02-24 | 2007-09-07 | Wyeth | DIHYDROSPIRO[DIBENZO[A,D][7]ANNULENE-5,4'-IMIDAZOL] COMPOUNDS FOR THE INHIBITION OF β-SECRETASE |
| US7700606B2 (en) | 2006-08-17 | 2010-04-20 | Wyeth Llc | Imidazole amines as inhibitors of β-secretase |
| CL2008000791A1 (es) | 2007-03-23 | 2008-05-30 | Wyeth Corp | Compuestos derivados de 2-amino-5-(4-difluorometoxi-fenil)-5-fenil-imidazolidin-4-ona; composicion farmaceutica que comprende a dichos compuestos; y su uso en el tratamiento de una enfermedad asociada con la actividad bace excesiva, tales como enferm |
| WO2018065288A1 (de) | 2016-10-07 | 2018-04-12 | Bayer Cropscience Aktiengesellschaft | 2-[2-phenyl-1-(sulfonylmethyl)vinyl]-imidazo[4,5-b]pyridin-derivate und verwandte verbindungen als schädlingsbekämpfungsmittel im pflanzenschutz |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE3929582A1 (de) | 1989-09-06 | 1991-03-07 | Hoechst Ag | Benzoylguanidine, verfahren zu ihrer herstellung, ihre verwendung als medikament sowie sie enthaltendes medikament |
| DE59302959D1 (de) * | 1992-02-15 | 1996-07-25 | Hoechst Ag | 3,5-Substituierte Benzoylguanidine, mit antiarrythmischer Wirkung und inhibierender Wirkung auf die Proliferationen von Zellen |
| JP3162572B2 (ja) * | 1993-04-28 | 2001-05-08 | 住友製薬株式会社 | インドロイルグアニジン誘導体 |
| US5401758A (en) * | 1993-10-07 | 1995-03-28 | Bristol-Myers Squibb Company | Pyridinyl cyanoguanidine compounds |
| DE4430861A1 (de) * | 1994-08-31 | 1996-03-07 | Merck Patent Gmbh | Heterocyclyl-benzoylguanidine |
| JPH0959245A (ja) * | 1995-08-25 | 1997-03-04 | Yamanouchi Pharmaceut Co Ltd | Ｎ−（２−プロペノイル）グアニジン誘導体 |
-
1996
- 1996-09-16 ZA ZA967800A patent/ZA967800B/xx unknown
- 1996-09-19 CN CN96196999A patent/CN1196721A/zh active Pending
- 1996-09-19 CZ CZ98840A patent/CZ84098A3/cs unknown
- 1996-09-19 HU HU9901336A patent/HUP9901336A3/hu unknown
- 1996-09-19 AU AU70007/96A patent/AU702092B2/en not_active Ceased
- 1996-09-19 WO PCT/JP1996/002696 patent/WO1997011055A1/ja not_active Ceased
- 1996-09-19 SK SK351-98A patent/SK35198A3/sk unknown
- 1996-09-19 PL PL96326033A patent/PL326033A1/xx unknown
- 1996-09-19 BR BR9610530A patent/BR9610530A/pt not_active Application Discontinuation
- 1996-09-19 CA CA002232497A patent/CA2232497A1/en not_active Abandoned
- 1996-09-19 EP EP96931252A patent/EP0861831A4/de not_active Withdrawn
- 1996-09-19 KR KR1019980702028A patent/KR19990063589A/ko not_active Withdrawn
-
1998
- 1998-03-19 NO NO981241A patent/NO981241L/no unknown
Also Published As
| Publication number | Publication date |
|---|---|
| CZ84098A3 (cs) | 1998-09-16 |
| WO1997011055A1 (en) | 1997-03-27 |
| HUP9901336A3 (en) | 2000-02-28 |
| BR9610530A (pt) | 1999-07-06 |
| AU7000796A (en) | 1997-04-09 |
| PL326033A1 (en) | 1998-08-17 |
| CA2232497A1 (en) | 1997-03-27 |
| MX9802238A (es) | 1998-08-30 |
| EP0861831A4 (de) | 1998-11-11 |
| NO981241D0 (no) | 1998-03-19 |
| SK35198A3 (en) | 1999-06-11 |
| ZA967800B (en) | 1997-04-03 |
| HUP9901336A2 (hu) | 1999-08-30 |
| CN1196721A (zh) | 1998-10-21 |
| KR19990063589A (ko) | 1999-07-26 |
| EP0861831A1 (de) | 1998-09-02 |
| AU702092B2 (en) | 1999-02-11 |
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