NO990793L - 7<alfa>-(<Epsilon>-aminoalkyl)-°stratriener, fremgangsmÕte for fremstilling av disse, farmas°ytiske preparater inneholdende disse, samt deres anvendelse for fremstilling av legemidler - Google Patents

7<alfa>-(<Epsilon>-aminoalkyl)-°stratriener, fremgangsmÕte for fremstilling av disse, farmas°ytiske preparater inneholdende disse, samt deres anvendelse for fremstilling av legemidler

Info

Publication number
NO990793L
NO990793L NO990793A NO990793A NO990793L NO 990793 L NO990793 L NO 990793L NO 990793 A NO990793 A NO 990793A NO 990793 A NO990793 A NO 990793A NO 990793 L NO990793 L NO 990793L
Authority
NO
Norway
Prior art keywords
pharmaceuticals
stratrienes
alfa
epsilon
aminoalkyl
Prior art date
Application number
NO990793A
Other languages
English (en)
Other versions
NO990793D0 (no
NO315655B1 (no
Inventor
Rolf Bohlmann
Dieter Bittler
Josef Heindi
Nikolaus Heinrich
Helmut Hofmeister
Hermann Kuenzer
Gerhard Sauer
Christa Hegele-Hartung
Rosemarie Lichtner
Yukishige Nishino
Karsten Parczyk
Martin Schneider
Original Assignee
Schering Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Schering Ag filed Critical Schering Ag
Publication of NO990793D0 publication Critical patent/NO990793D0/no
Publication of NO990793L publication Critical patent/NO990793L/no
Publication of NO315655B1 publication Critical patent/NO315655B1/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J53/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton has been modified by condensation with a carbocyclic rings or by formation of an additional ring by means of a direct link between two ring carbon atoms, including carboxyclic rings fused to the cyclopenta(a)hydrophenanthrene skeleton are included in this class
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J53/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton has been modified by condensation with a carbocyclic rings or by formation of an additional ring by means of a direct link between two ring carbon atoms, including carboxyclic rings fused to the cyclopenta(a)hydrophenanthrene skeleton are included in this class
    • C07J53/002—Carbocyclic rings fused
    • C07J53/004—3 membered carbocyclic rings
    • C07J53/008—3 membered carbocyclic rings in position 15/16
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
    • A61P5/32—Antioestrogens
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
    • C07J41/0033—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005
    • C07J41/0072—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005 the A ring of the steroid being aromatic
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J43/00—Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton
    • C07J43/006—Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton spiro-condensed
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J53/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton has been modified by condensation with a carbocyclic rings or by formation of an additional ring by means of a direct link between two ring carbon atoms, including carboxyclic rings fused to the cyclopenta(a)hydrophenanthrene skeleton are included in this class
    • C07J53/002—Carbocyclic rings fused

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Diabetes (AREA)
  • Endocrinology (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
NO19990793A 1996-08-20 1999-02-19 7<alfa>-(<Epsilon>-aminoalkyl)-östratriener, farmasöytiske preparater inneholdende disse, samt deres anvendelse for fremstilling avlegemidler NO315655B1 (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE19635525A DE19635525A1 (de) 1996-08-20 1996-08-20 7alpha-(xi-Aminoalkyl)-estratriene, Verfahren zu deren Herstellung, pharmazeutische Präparate, die diese 7alpha(xi-Aminoalkyl-estratriene enthalten sowie deren Verwendung zur Herstellung von Arzneimitteln
PCT/EP1997/004517 WO1998007740A1 (de) 1996-08-20 1997-08-20 7α-(κ-AMINOALKYL)-ESTRATRIENE, VERFAHREN ZU DEREN HERSTELLUNG, PHARMAZEUTISCHE PRÄPARATE, DIE DIESE 7α-(κ-AMINOALKYL)-ESTRATRIENE ENTHALTEN SOWIE DEREN VERWENDUNG ZUR HERSTELLUNG VON ARZNEIMITTELN

Publications (3)

Publication Number Publication Date
NO990793D0 NO990793D0 (no) 1999-02-19
NO990793L true NO990793L (no) 1999-04-20
NO315655B1 NO315655B1 (no) 2003-10-06

Family

ID=7804367

Family Applications (1)

Application Number Title Priority Date Filing Date
NO19990793A NO315655B1 (no) 1996-08-20 1999-02-19 7<alfa>-(<Epsilon>-aminoalkyl)-östratriener, farmasöytiske preparater inneholdende disse, samt deres anvendelse for fremstilling avlegemidler

Country Status (29)

Country Link
EP (1) EP0920441B1 (no)
JP (1) JP2001503024A (no)
KR (1) KR20000068261A (no)
CN (1) CN1231670A (no)
AR (1) AR009278A1 (no)
AT (1) ATE231882T1 (no)
AU (1) AU728843B2 (no)
BG (1) BG62972B1 (no)
BR (1) BR9711328A (no)
CA (1) CA2263708A1 (no)
CZ (1) CZ57999A3 (no)
DE (2) DE19635525A1 (no)
DK (1) DK0920441T3 (no)
EA (1) EA001577B1 (no)
EE (1) EE04021B1 (no)
ES (1) ES2191857T3 (no)
HU (1) HUP9903106A3 (no)
IL (1) IL128601A (no)
IS (1) IS4976A (no)
NO (1) NO315655B1 (no)
NZ (1) NZ334277A (no)
PL (1) PL186309B1 (no)
PT (1) PT920441E (no)
SK (1) SK18899A3 (no)
TR (1) TR199900432T2 (no)
TW (1) TW552267B (no)
UA (1) UA50792C2 (no)
WO (1) WO1998007740A1 (no)
ZA (1) ZA977482B (no)

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US6548491B2 (en) 1997-12-24 2003-04-15 Sri International Anti-estrogenic steroids, and associated pharmaceutical compositions and methods of use
US6503896B1 (en) 1997-12-24 2003-01-07 Sri International Anti-estrogenic steroids, and associated pharmaceutical compositions and methods of use
DE19807791A1 (de) * 1998-02-19 1999-08-26 Schering Ag Kombinationspräparat aus Östrogen und Antiöstrogen
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DE10019171A1 (de) * 2000-04-07 2001-10-18 Schering Ag Zusammensetzungen zur Verwendung als Penetrationsverstärker in transdermalen Formulierungen für hoch lipophile Wirkstoffe
AU2006202187B2 (en) * 2001-11-27 2008-11-06 Bayer Schering Pharma Aktiengesellschaft 17alpah-alkyl-17beta-oxy-estratrienes and intermediate products for their production, uses thereof and pharmaceutical preparations
DE10159217A1 (de) 2001-11-27 2003-06-05 Schering Ag 17alpha-Alkyl-17ß-oxy-estratriene und Zwischenprodukte zu deren Herstellung, Verwendung der 17alpha-Alkyl-17ß-oxy-estratriene zur Herstellung von Arzneimitteln sowie pharmazeutische Präparate
US20040242551A1 (en) * 2003-05-28 2004-12-02 Schering Ag Composition comprising antiprogestins and pure antiestrogens for prophylaxis and treatment of hormone-dependent diseases
JP2007506805A (ja) 2004-07-27 2007-03-22 シコール インコーポレイティド ７α−アルキル化された１９−ノルステロイドの調製方法
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TW200904329A (en) 2007-05-18 2009-02-01 Sumitomo Chemical Co Organic sulfur compound and its use for controlling harmful arthropod
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DE102007032800A1 (de) 2007-07-10 2009-01-15 Bayer Schering Pharma Aktiengesellschaft Nichtsteroidale Progesteronrezeptor-Modulatoren
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DE102009034362A1 (de) 2009-07-20 2011-01-27 Bayer Schering Pharma Aktiengesellschaft 17-Hydroxy-17-pentafluorethyl-estra-4,9(10)-dien-11-aryl-Derivate, Verfahren zu ihrer Herstellung und ihre Verwendung zur Behandlung von Krankheiten
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Also Published As

Publication number Publication date
BG103185A (en) 1999-11-30
TW552267B (en) 2003-09-11
CZ57999A3 (cs) 1999-08-11
AU728843B2 (en) 2001-01-18
CN1231670A (zh) 1999-10-13
ZA977482B (en) 1998-02-23
DE59709239D1 (de) 2003-03-06
EA001577B1 (ru) 2001-06-25
SK18899A3 (en) 1999-08-06
AU4552097A (en) 1998-03-06
EE04021B1 (et) 2003-04-15
WO1998007740A1 (de) 1998-02-26
AR009278A1 (es) 2000-04-12
TR199900432T2 (xx) 1999-04-21
KR20000068261A (ko) 2000-11-25
UA50792C2 (uk) 2002-11-15
ATE231882T1 (de) 2003-02-15
PL186309B1 (pl) 2003-12-31
EP0920441B1 (de) 2003-01-29
BR9711328A (pt) 1999-08-17
NO990793D0 (no) 1999-02-19
NO315655B1 (no) 2003-10-06
PL331863A1 (en) 1999-08-16
CA2263708A1 (en) 1998-02-26
EA199900210A1 (ru) 1999-08-26
DK0920441T3 (da) 2003-05-26
PT920441E (pt) 2003-06-30
HUP9903106A3 (en) 2000-05-29
DE19635525A1 (de) 1998-02-26
IL128601A (en) 2003-07-31
BG62972B1 (bg) 2000-12-29
EE9900075A (et) 1999-10-15
HUP9903106A2 (hu) 2000-03-28
IS4976A (is) 1999-02-11
JP2001503024A (ja) 2001-03-06
IL128601A0 (en) 2000-01-31
NZ334277A (en) 2000-10-27
ES2191857T3 (es) 2003-09-16
EP0920441A1 (de) 1999-06-09

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