OA11051A - Fused bicyclic pyrimidine derivatives - Google Patents

Fused bicyclic pyrimidine derivatives Download PDF

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Publication number
OA11051A
OA11051A OA9900107A OA9900107A OA11051A OA 11051 A OA11051 A OA 11051A OA 9900107 A OA9900107 A OA 9900107A OA 9900107 A OA9900107 A OA 9900107A OA 11051 A OA11051 A OA 11051A
Authority
OA
OAPI
Prior art keywords
phenyl
alkyl
compound
pyrrolo
cancer
Prior art date
Application number
OA9900107A
Other languages
English (en)
Inventor
Daniel Arnold Lee
Mikel Paul Moyer
Susan Beth Sobolov-Jaynes
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of OA11051A publication Critical patent/OA11051A/en

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/08—Drugs for disorders of the urinary system of the prostate
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Diabetes (AREA)
  • Urology & Nephrology (AREA)
  • Emergency Medicine (AREA)
  • Endocrinology (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Dermatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
OA9900107A 1996-11-27 1999-05-24 Fused bicyclic pyrimidine derivatives OA11051A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US3186296P 1996-11-27 1996-11-27
US4184697P 1997-04-09 1997-04-09

Publications (1)

Publication Number Publication Date
OA11051A true OA11051A (en) 2003-03-07

Family

ID=26707706

Family Applications (1)

Application Number Title Priority Date Filing Date
OA9900107A OA11051A (en) 1996-11-27 1999-05-24 Fused bicyclic pyrimidine derivatives

Country Status (24)

Country Link
US (1) US6413971B1 (fr)
EP (1) EP0946554A1 (fr)
JP (1) JP2000505109A (fr)
KR (1) KR20000057228A (fr)
CN (1) CN1237177A (fr)
AP (1) AP9701146A0 (fr)
AR (1) AR010740A1 (fr)
AU (1) AU4718997A (fr)
BG (1) BG103417A (fr)
BR (1) BR9713552A (fr)
CA (1) CA2272705C (fr)
CO (1) CO4650037A1 (fr)
HN (1) HN1997000146A (fr)
HR (1) HRP970641A2 (fr)
ID (1) ID18958A (fr)
IL (1) IL129825A0 (fr)
IS (1) IS5041A (fr)
MA (1) MA26452A1 (fr)
NO (1) NO992524D0 (fr)
OA (1) OA11051A (fr)
PA (1) PA8442001A1 (fr)
PE (1) PE17299A1 (fr)
TN (1) TNSN97192A1 (fr)
WO (1) WO1998023613A1 (fr)

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Also Published As

Publication number Publication date
EP0946554A1 (fr) 1999-10-06
BR9713552A (pt) 2000-01-25
WO1998023613A1 (fr) 1998-06-04
AU4718997A (en) 1998-06-22
TNSN97192A1 (fr) 2005-03-15
MA26452A1 (fr) 2004-12-20
NO992524L (no) 1999-05-26
HN1997000146A (es) 1998-02-26
CN1237177A (zh) 1999-12-01
PA8442001A1 (es) 2000-05-24
BG103417A (en) 2000-06-30
CA2272705A1 (fr) 1998-06-04
PE17299A1 (es) 1999-02-19
AP9701146A0 (en) 1998-01-31
HRP970641A2 (en) 1998-10-31
US6413971B1 (en) 2002-07-02
NO992524D0 (no) 1999-05-26
ID18958A (id) 1998-05-28
US20020045630A1 (en) 2002-04-18
CA2272705C (fr) 2003-03-18
JP2000505109A (ja) 2000-04-25
KR20000057228A (ko) 2000-09-15
IS5041A (is) 1999-04-30
CO4650037A1 (es) 1998-09-03
IL129825A0 (en) 2000-02-29
AR010740A1 (es) 2000-07-12

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