OA11569A - Therapeutic combinations of (selective) estrogen receptor modulators (serm) and growth hormone secretagogues(GHS) for treating musculoskeletal frailty. - Google Patents

Therapeutic combinations of (selective) estrogen receptor modulators (serm) and growth hormone secretagogues(GHS) for treating musculoskeletal frailty. Download PDF

Info

Publication number: OA11569A
Authority: OA; OAPI
Prior art keywords: oxo; pyridin; ethyl; phenyl; compound
Prior art date: 1998-06-16

Application number

OA1200000346A

Other languages

English (en)

Inventor

Hua Zhu Ke

Mei Li

Lydia Codetta Pan

David Duane Thompson

Original Assignee

Pfizer Prod Inc

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1998-06-16

Filing date

1999-05-03

Publication date

2004-07-01

1999-05-03 Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc

2004-07-01 Publication of OA11569A publication Critical patent/OA11569A/en

Links

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Classifications

- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/02—Stomatological preparations, e.g. drugs for caries, aphtae, periodontitis
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
- A61P19/10—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease for osteoporosis
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

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Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Chemical & Material Sciences (AREA)
Veterinary Medicine (AREA)
Public Health (AREA)
Medicinal Chemistry (AREA)
General Health & Medical Sciences (AREA)
Animal Behavior & Ethology (AREA)
Pharmacology & Pharmacy (AREA)
Physical Education & Sports Medicine (AREA)
General Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Engineering & Computer Science (AREA)
Chemical Kinetics & Catalysis (AREA)
Bioinformatics & Cheminformatics (AREA)
Orthopedic Medicine & Surgery (AREA)
Rheumatology (AREA)
Epidemiology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)

OA1200000346A 1998-06-16 1999-05-03 Therapeutic combinations of (selective) estrogen receptor modulators (serm) and growth hormone secretagogues(GHS) for treating musculoskeletal frailty. OA11569A (en)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
US8942498P	1998-06-16	1998-06-16

Publications (1)

Publication Number	Publication Date
OA11569A true OA11569A (en)	2004-07-01

Family

ID=22217565

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
OA1200000346A OA11569A (en)	1998-06-16	1999-05-03	Therapeutic combinations of (selective) estrogen receptor modulators (serm) and growth hormone secretagogues(GHS) for treating musculoskeletal frailty.

Country Status (29)

Country	Link
EP (1)	EP1085867A1 (id)
JP (1)	JP2002518328A (id)
KR (1)	KR20010052817A (id)
CN (1)	CN1305378A (id)
AP (1)	AP9901581A0 (id)
AR (1)	AR018868A1 (id)
AU (1)	AU3342099A (id)
BG (1)	BG105128A (id)
BR (1)	BR9911357A (id)
CA (1)	CA2335112A1 (id)
CO (1)	CO5070586A1 (id)
EA (1)	EA200001189A1 (id)
GT (1)	GT199900083A (id)
HR (1)	HRP20000857A2 (id)
HU (1)	HUP0102395A2 (id)
ID (1)	ID26726A (id)
IL (1)	IL139587A0 (id)
IS (1)	IS5727A (id)
MA (1)	MA26648A1 (id)
NO (1)	NO20006381L (id)
OA (1)	OA11569A (id)
PA (1)	PA8472101A1 (id)
PE (1)	PE20000633A1 (id)
PL (1)	PL345064A1 (id)
SK (1)	SK18902000A3 (id)
TN (1)	TNSN99118A1 (id)
UY (1)	UY25557A1 (id)
WO (1)	WO1999065488A1 (id)
ZA (1)	ZA993973B (id)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
EP1004306A3 (en) *	1998-08-06	2000-06-07	Pfizer Products Inc.	Estrogen agonists/antagonists
CA2420535A1 (en) *	2000-08-30	2002-03-07	Mary Tanya Am Ende	Sustained release formulations for growth hormone secretagogues
IL145106A0 (en) *	2000-08-30	2002-06-30	Pfizer Prod Inc	Intermittent administration of a geowth hormone secretagogue
MXPA04005112A (es) *	2001-11-29	2005-04-29	Gtx Inc	Prevencion y tratamiento de osteoporosis inducida por privacion de androgeno.
US7524866B2 (en)	2001-11-29	2009-04-28	Gtx, Inc.	Prevention and treatment of androgen—deprivation induced osteoporosis
US7476653B2 (en)	2003-06-18	2009-01-13	Tranzyme Pharma, Inc.	Macrocyclic modulators of the ghrelin receptor
CU23558A1 (es)	2006-02-28	2010-07-20	Ct Ingenieria Genetica Biotech	Compuestos análogos a los secretagogos peptidicos de la hormona de crecimiento
ES2602789T3 (es)	2007-02-09	2017-02-22	Ocera Therapeutics, Inc.	Productos intermedios conectores para la síntesis de moduladores macrocíclicos del receptor de la grelina

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
UA51676C2 (uk) *	1995-11-02	2002-12-16	Пфайзер Інк.	(-)цис-6(s)-феніл-5(r)[4-(2-піролідин-1-ілетокси)феніл]-5,6,7,8-тетрагідронафталін-2-ол d-тартрат, спосіб його одержання, спосіб лікування захворювань, що піддаються лікуванню агоністами естрогену, та фармацевтична композиція
TW432073B (en) *	1995-12-28	2001-05-01	Pfizer	Pyrazolopyridine compounds
HN1996000101A (es) *	1996-02-28	1997-06-26	Inc Pfizer	Terapia combinada para la osteoporosis

1999
- 1999-05-03 AU AU33420/99A patent/AU3342099A/en not_active Abandoned
- 1999-05-03 WO PCT/IB1999/000796 patent/WO1999065488A1/en not_active Ceased
- 1999-05-03 IL IL13958799A patent/IL139587A0/xx unknown
- 1999-05-03 EA EA200001189A patent/EA200001189A1/ru unknown
- 1999-05-03 OA OA1200000346A patent/OA11569A/en unknown
- 1999-05-03 CN CN99807381A patent/CN1305378A/zh active Pending
- 1999-05-03 KR KR1020007014140A patent/KR20010052817A/ko not_active Ceased
- 1999-05-03 EP EP99914723A patent/EP1085867A1/en not_active Withdrawn
- 1999-05-03 JP JP2000554368A patent/JP2002518328A/ja active Pending
- 1999-05-03 PL PL99345064A patent/PL345064A1/xx unknown
- 1999-05-03 HU HU0102395A patent/HUP0102395A2/hu unknown
- 1999-05-03 HR HR20000857A patent/HRP20000857A2/hr not_active Application Discontinuation
- 1999-05-03 CA CA002335112A patent/CA2335112A1/en not_active Abandoned
- 1999-05-03 SK SK1890-2000A patent/SK18902000A3/sk unknown
- 1999-05-03 BR BR9911357-0A patent/BR9911357A/pt not_active Application Discontinuation
- 1999-05-03 ID IDW20002604A patent/ID26726A/id unknown
- 1999-05-07 PA PA19998472101A patent/PA8472101A1/es unknown
- 1999-06-10 AP APAP/P/1999/001581A patent/AP9901581A0/en unknown
- 1999-06-11 UY UY25557A patent/UY25557A1/es not_active Application Discontinuation
- 1999-06-11 PE PE1999000522A patent/PE20000633A1/es not_active Application Discontinuation
- 1999-06-14 GT GT199900083A patent/GT199900083A/es unknown
- 1999-06-15 ZA ZA9903973A patent/ZA993973B/xx unknown
- 1999-06-15 AR ARP990102847A patent/AR018868A1/es not_active Application Discontinuation
- 1999-06-15 MA MA25622A patent/MA26648A1/fr unknown
- 1999-06-15 TN TNTNSN99118A patent/TNSN99118A1/fr unknown
- 1999-06-16 CO CO99037624A patent/CO5070586A1/es unknown
2000
- 2000-11-24 IS IS5727A patent/IS5727A/is unknown
- 2000-12-14 NO NO20006381A patent/NO20006381L/no not_active Application Discontinuation
2001
- 2001-01-08 BG BG105128A patent/BG105128A/xx unknown

Also Published As

Publication number	Publication date
SK18902000A3 (sk)	2001-12-03
JP2002518328A (ja)	2002-06-25
BG105128A (en)	2001-11-30
PL345064A1 (en)	2001-11-19
IS5727A (is)	2000-11-24
AU3342099A (en)	2000-01-05
BR9911357A (pt)	2001-03-13
HRP20000857A2 (en)	2001-10-31
ZA993973B (en)	2000-12-15
WO1999065488A1 (en)	1999-12-23
CO5070586A1 (es)	2001-08-28
CA2335112A1 (en)	1999-12-23
NO20006381D0 (no)	2000-12-14
UY25557A1 (es)	2001-01-31
PA8472101A1 (es)	2000-09-29
HUP0102395A2 (hu)	2001-11-28
KR20010052817A (ko)	2001-06-25
AR018868A1 (es)	2001-12-12
CN1305378A (zh)	2001-07-25
PE20000633A1 (es)	2000-07-26
ID26726A (id)	2001-02-01
GT199900083A (es)	2000-12-05
AP9901581A0 (en)	1999-06-30
TNSN99118A1 (fr)	2005-11-10
EP1085867A1 (en)	2001-03-28
NO20006381L (no)	2000-12-14
EA200001189A1 (ru)	2001-06-25
IL139587A0 (en)	2002-02-10
MA26648A1 (fr)	2004-12-20

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CN109922812A (zh)	2019-06-21	减少与甲状腺相关的副作用的方法
HRP980356A2 (en)	1999-02-28	Prostaglandin agonists
US20050065133A1 (en)	2005-03-24	Pharmaceutical compositions and methods comprising combinations of 2-alkylidene-19-nor-vitamin D derivatives and an EP2 or EP4 selective agonist
US20050065180A1 (en)	2005-03-24	Pharmaceutical compositions and methods comprising combinations of 2-alkylidene-19-nor-vitamin D derivatives and a growth hormone secretagogue
US7632813B2 (en)	2009-12-15	Bone densifying agent characterized by use of cathepsin K inhibitor with PTH
US6132774A (en)	2000-10-17	Therapeutic combinations comprising a selective estrogen receptor modulator and parathyroid hormone
US20020002137A1 (en)	2002-01-03	Combination of growth hormone secretagogues and antidepressants
WO1999065488A1 (en)	1999-12-23	Therapeutic combinations of (selective) estrogen receptor modulators (serm) and growth hormone secretagogues (ghs) for treating musculoskeletal frailty
OA11505A (en)	2004-05-07	Therapeutic combinations of (selective) estrogen receptor modulators (SERM) and growth hormone secretagogues (GHS) for treating musculoskeletal frailty.
US6284773B1 (en)	2001-09-04	Therapeutic combinations comprising a selective estrogen receptor modulator and prostaglandin E2
CZ20004680A3 (cs)	2001-06-13	Terapeutické kombinace (selektivních) modulátorů estrogenního receptorů (ŠERM) a prostředků podporujících sekreci růstového hormonu (GHS) pro léčbu muskuloskeletární fragility
MXPA00012628A (en)	2001-07-31	Therapeutic combinations of (selective) estrogen receptor modulators (serm) and growth hormone secretagogues (ghs) for treating musculoskeletal frailty
HK1036938A (en)	2002-01-25	Therapeutic combinations of (selective) estrogen receptor modulators (serm) and growth hormone secretagogues (ghs) for treating musculoskeletal frailty
CZ20004679A3 (cs)	2001-05-16	Terapeutické kombinace (selektivních) modulátorů estrogenního receptoru (ŠERM) a prostředků podporujících sekreci růstového hormonu (GHS) pro léčbu muskuloskeletární fragility
MXPA00012727A (en)	2001-07-31	Therapeutic combinations of (selective) estrogen receptor modulators (serm) and growth hormone secretagogues (ghs) for treating musculoskeletal frailty
EA008927B1 (ru)	2007-08-31	Применение производных 2h-[1,3]оксазино[3,2-a]индола для лечения невропатической боли
HK1036414A (en)	2002-01-04	Therapeutic combinations of (selective) estrogen receptor modulators (serm) and growth hormone secretagogues (ghs) for treating musculoskeletal frailty
MXPA00012728A (en)	2001-07-31	Therapeutic combinations comprising a selective estrogen receptor modulator and parathyroid hormone