OA12295A - Combinations of depeptidyl peptidase IV inhibitorsand other antidabetic agents for the treatment of diabetes mellitus. - Google Patents

Combinations of depeptidyl peptidase IV inhibitorsand other antidabetic agents for the treatment of diabetes mellitus. Download PDF

Info

Publication number: OA12295A
Authority: OA; OAPI
Prior art keywords: inhibitor; use according; diabètes; dipeptidyl peptidase; insulin
Prior art date: 2000-06-19

Application number

OA1200200388A

Other languages

English (en)

Inventor

Jonathan Robert Sanders Arch

James Martin Lenhard

Original Assignee

Smithkline Beecham Plc

Smithkline Beecham Corp

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2000-06-19

Filing date

2001-06-19

Publication date

2003-11-10

2001-06-19 Application filed by Smithkline Beecham Plc, Smithkline Beecham Corp filed Critical Smithkline Beecham Plc

2003-11-10 Publication of OA12295A publication Critical patent/OA12295A/en

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235000019833 protease Nutrition 0.000 title claims description 5
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239000003472 antidiabetic agent Substances 0.000 claims abstract description 25
229940125708 antidiabetic agent Drugs 0.000 claims abstract description 24
238000000034 method Methods 0.000 claims abstract description 18
229940124213 Dipeptidyl peptidase 4 (DPP IV) inhibitor Drugs 0.000 claims abstract description 13
239000003603 dipeptidyl peptidase IV inhibitor Substances 0.000 claims abstract description 13
241000124008 Mammalia Species 0.000 claims abstract description 4
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- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
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- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
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- A61K31/427—Thiazoles not condensed and containing further heterocyclic rings
- A—HUMAN NECESSITIES
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/06—Antihyperlipidemics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics

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Diabetes (AREA)
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OA1200200388A 2000-06-19 2001-06-19 Combinations of depeptidyl peptidase IV inhibitorsand other antidabetic agents for the treatment of diabetes mellitus. OA12295A (en)

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GBGB0014969.0A GB0014969D0 (en)	2000-06-19	2000-06-19	Novel method of treatment

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OA1200200388A OA12295A (en)	2000-06-19	2001-06-19	Combinations of depeptidyl peptidase IV inhibitorsand other antidabetic agents for the treatment of diabetes mellitus.

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US (2)	US7241756B2 (fr)
EP (2)	EP1292300B1 (fr)
JP (1)	JP2003535898A (fr)
KR (1)	KR20030019440A (fr)
CN (1)	CN1443068A (fr)
AP (1)	AP2002002703A0 (fr)
AT (1)	ATE419850T1 (fr)
AU (3)	AU2001264148A1 (fr)
BG (1)	BG107385A (fr)
BR (1)	BR0111800A (fr)
CA (1)	CA2413299A1 (fr)
CZ (1)	CZ20024069A3 (fr)
DE (1)	DE60137329D1 (fr)
DZ (1)	DZ3390A1 (fr)
EA (1)	EA200300036A1 (fr)
EC (1)	ECSP024397A (fr)
GB (1)	GB0014969D0 (fr)
HR (1)	HRP20020994A2 (fr)
HU (1)	HUP0301194A3 (fr)
IL (2)	IL153529A0 (fr)
MA (1)	MA25820A1 (fr)
MX (1)	MXPA02012763A (fr)
NO (1)	NO20026038L (fr)
OA (1)	OA12295A (fr)
PL (1)	PL360493A1 (fr)
SK (1)	SK17832002A3 (fr)
WO (1)	WO2001097808A1 (fr)
YU (1)	YU1703A (fr)
ZA (1)	ZA200300203B (fr)

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2000
- 2000-06-19 GB GBGB0014969.0A patent/GB0014969D0/en not_active Ceased
2001
- 2001-06-19 BR BR0111800-5A patent/BR0111800A/pt not_active Application Discontinuation
- 2001-06-19 PL PL36049301A patent/PL360493A1/xx unknown
- 2001-06-19 AT AT01938472T patent/ATE419850T1/de not_active IP Right Cessation
- 2001-06-19 EA EA200300036A patent/EA200300036A1/ru unknown
- 2001-06-19 DZ DZ013390A patent/DZ3390A1/fr active
- 2001-06-19 CA CA002413299A patent/CA2413299A1/fr not_active Abandoned
- 2001-06-19 KR KR1020027017279A patent/KR20030019440A/ko not_active Ceased
- 2001-06-19 IL IL15352901A patent/IL153529A0/xx unknown
- 2001-06-19 EP EP01938472A patent/EP1292300B1/fr not_active Expired - Lifetime
- 2001-06-19 AP APAP/P/2002/002703A patent/AP2002002703A0/en unknown
- 2001-06-19 YU YU1703A patent/YU1703A/sh unknown
- 2001-06-19 DE DE60137329T patent/DE60137329D1/de not_active Expired - Fee Related
- 2001-06-19 MX MXPA02012763A patent/MXPA02012763A/es active IP Right Grant
- 2001-06-19 OA OA1200200388A patent/OA12295A/en unknown
- 2001-06-19 JP JP2002503292A patent/JP2003535898A/ja not_active Withdrawn
- 2001-06-19 WO PCT/GB2001/002696 patent/WO2001097808A1/fr not_active Ceased
- 2001-06-19 EP EP08168689A patent/EP2036554A1/fr not_active Withdrawn
- 2001-06-19 CN CN01813126A patent/CN1443068A/zh active Pending
- 2001-06-19 HR HR20020994A patent/HRP20020994A2/hr not_active Application Discontinuation
- 2001-06-19 CZ CZ20024069A patent/CZ20024069A3/cs unknown
- 2001-06-19 SK SK17832002A patent/SK17832002A3/sk not_active Application Discontinuation
- 2001-06-19 AU AU2001264148A patent/AU2001264148A1/en not_active Abandoned
- 2001-06-19 HU HU0301194A patent/HUP0301194A3/hu unknown
2002
- 2002-12-12 BG BG107385A patent/BG107385A/bg unknown
- 2002-12-16 NO NO20026038A patent/NO20026038L/no not_active Application Discontinuation
- 2002-12-18 MA MA26965A patent/MA25820A1/fr unknown
- 2002-12-19 EC EC2002004397A patent/ECSP024397A/es unknown
2003
- 2003-01-08 ZA ZA200300203A patent/ZA200300203B/en unknown
2005
- 2005-11-11 AU AU2005232303A patent/AU2005232303A1/en not_active Abandoned
2006
- 2006-06-01 US US11/421,548 patent/US7241756B2/en not_active Expired - Fee Related
2007
- 2007-06-05 US US11/758,259 patent/US20070238756A1/en not_active Abandoned
- 2007-12-27 IL IL188471A patent/IL188471A0/en unknown
2008
- 2008-09-08 AU AU2008212061A patent/AU2008212061A1/en not_active Abandoned

Also Published As

Publication number	Publication date
EA200300036A1 (ru)	2003-04-24
CA2413299A1 (fr)	2001-12-27
BG107385A (bg)	2003-09-30
EP2036554A1 (fr)	2009-03-18
DE60137329D1 (de)	2009-02-26
CN1443068A (zh)	2003-09-17
AP2002002703A0 (en)	2002-12-31
US7241756B2 (en)	2007-07-10
BR0111800A (pt)	2003-05-27
MA25820A1 (fr)	2003-07-01
IL153529A0 (en)	2003-07-06
MXPA02012763A (es)	2003-04-25
ATE419850T1 (de)	2009-01-15
AU2001264148A1 (en)	2002-01-02
CZ20024069A3 (cs)	2004-02-18
HRP20020994A2 (en)	2005-02-28
JP2003535898A (ja)	2003-12-02
IL188471A0 (en)	2008-03-20
PL360493A1 (en)	2004-09-06
HUP0301194A3 (en)	2007-09-28
EP1292300A1 (fr)	2003-03-19
ZA200300203B (en)	2004-03-26
AU2005232303A1 (en)	2005-12-01
GB0014969D0 (en)	2000-08-09
AU2008212061A1 (en)	2008-10-02
SK17832002A3 (en)	2004-10-05
KR20030019440A (ko)	2003-03-06
YU1703A (sh)	2006-03-03
WO2001097808A1 (fr)	2001-12-27
NO20026038L (no)	2003-02-03
US20070238756A1 (en)	2007-10-11
ECSP024397A (es)	2003-02-06
US20060205675A1 (en)	2006-09-14
EP1292300B1 (fr)	2009-01-07
NO20026038D0 (no)	2002-12-16
DZ3390A1 (fr)	2001-12-27
HUP0301194A2 (hu)	2003-08-28

Publication	Publication Date	Title
US7241756B2 (en)	2007-07-10	Combinations of dipeptidyl peptidase IV inhibitors and other antidiabetic agents for the treatment of diabetes mellitus
US7078397B2 (en)	2006-07-18	Combinations of dipeptidyl peptidase IV inhibitors and other antidiabetic agents for the treatment of diabetes mellitus
KR100666591B1 (ko)	2007-01-11	티아졸리딘디온 및 메트포르민을 사용한 당뇨병의 치료
OA11279A (en)	2003-07-31	Treatment of diabetes with thiazolidinedione, insulin secretagogue and diguanide.
US20080058388A1 (en)	2008-03-06	Treatment of diabetes with thiazolidinedione and sulphonylurea
OA11517A (en)	2004-02-04	Treatment of diabetes with rosiglitazone and insulin.
AU743269B2 (en)	2002-01-24	Treatment of diabetes with thiazolidinedione and sulphonylurea
AU766928B2 (en)	2003-10-23	Combinations comprising a beta-agonist and a further antidiabetic agent
OA11510A (en)	2004-02-03	Treatment of diabetes with thiazolidinedione and sulphonylurea.
CN1263467A (zh)	2000-08-16	用噻唑烷二酮、促胰岛素分泌剂和α一葡糖苷酶抑制剂治疗糖尿病
NZ501345A (en)	2001-10-26	Treatment of diabetes mellitus with 5-[4-[2-(N-methyl-N-(2- pyridyl)amino)ethoxy]benzyl]thiazolidine-2,4-dione (2-12 mg) and an alpha-glucosidase inhibitor antihyperglycemic agent
US20030073644A1 (en)	2003-04-17	Combinations comprising a beta-agonist and a further antidiabetic agent
HK1091393A (en)	2007-01-19	Treatment of diabetes with thiazolidinedione and sulphonylurea
AU1540002A (en)	2002-03-21	Treatment of diabetes with thiazolidinedione and sulphonylurea