PE20120320A1 - Pirazinilpirazoles - Google Patents

Pirazinilpirazoles

Info

Publication number
PE20120320A1
PE20120320A1 PE2011002013A PE2011002013A PE20120320A1 PE 20120320 A1 PE20120320 A1 PE 20120320A1 PE 2011002013 A PE2011002013 A PE 2011002013A PE 2011002013 A PE2011002013 A PE 2011002013A PE 20120320 A1 PE20120320 A1 PE 20120320A1
Authority
PE
Peru
Prior art keywords
halogen
haloalkyl
phenyl
alkyl
refers
Prior art date
Application number
PE2011002013A
Other languages
English (en)
Inventor
Hans-Georg Schwarz
Jens Frackenpohl
Achim Hense
Simon Maechling
Stefan Schnatterer
Robert Velten
Stefan Werner
Angela Becker
Olga Malsam
Eva-Maria Franken
Arnd Voerste
Ulrich Gorgens
Peter Lummen
Original Assignee
Bayer Cropscience Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Cropscience Ag filed Critical Bayer Cropscience Ag
Publication of PE20120320A1 publication Critical patent/PE20120320A1/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/14Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Pyridine Compounds (AREA)

Abstract

SE REFIERE A COMPUESTOS DERIVADOS DE PIRAZIN-2-ILPIRAZOLES DE FORMULA (I) DONDE X ES FENILO, 2-PIRIDILO O 3-PIRIDILO OPCIONALMENTE SUSTITUIDOS CON HALOGENO, CN, NITRO, ENTRE OTROS; R1 ES H, ALQUILO, HALOALQUILO, FENILO, ENTRE OTROS; R2 ES AMINO, ALQUINILO, ALCOXICARBONILO, HETEROARILO, ENTRE OTROS; R3 Y R4 SON CADA UNO H, HALOGENO, ALQUILO, CICLOALQUILO, ENTRE OTROS; R5 ES HALOGENO, HALOALQUILO, ALCOXI, CN, ENTRE OTROS. TAMBIEN SE REFIERE A UN PROCEDIMIENTO DE PREPARACION Y A UNA COMPOSICION. DICHOS COMPUESTOS SON UTILES COMO INSECTICIDAS Y PARASITICIDAS
PE2011002013A 2009-05-29 2010-05-19 Pirazinilpirazoles PE20120320A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP09161568A EP2266973A1 (de) 2009-05-29 2009-05-29 Pyrazinylpyrazole

Publications (1)

Publication Number Publication Date
PE20120320A1 true PE20120320A1 (es) 2012-03-30

Family

ID=40897591

Family Applications (1)

Application Number Title Priority Date Filing Date
PE2011002013A PE20120320A1 (es) 2009-05-29 2010-05-19 Pirazinilpirazoles

Country Status (21)

Country Link
US (2) US20120190687A1 (es)
EP (2) EP2266973A1 (es)
KR (1) KR101758935B1 (es)
CN (1) CN102459235B (es)
AR (1) AR076798A1 (es)
AU (1) AU2010252346B2 (es)
BR (1) BRPI1012771A2 (es)
CA (1) CA2763498A1 (es)
CO (1) CO6470821A2 (es)
DO (1) DOP2011000366A (es)
EC (1) ECSP11011487A (es)
ES (1) ES2409891T3 (es)
IL (1) IL216337A (es)
MX (1) MX2011012504A (es)
NI (1) NI201100208A (es)
NZ (1) NZ596681A (es)
PE (1) PE20120320A1 (es)
TW (1) TW201107310A (es)
UY (1) UY32659A (es)
WO (1) WO2010136145A1 (es)
ZA (1) ZA201108637B (es)

Families Citing this family (21)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2488510B1 (de) * 2009-10-12 2017-03-29 Bayer Intellectual Property GmbH Amide und Thioamide als Schädlingsbekämpfungsmittel
BR112012006956A2 (pt) * 2009-10-12 2015-09-15 Bayer Cropscience Ag 1- (pirida-3-il) -pirazóisol e 1- (pirimida-5-il) - pirazóisol como pesticidas
EP2499130A1 (de) 2009-11-11 2012-09-19 Bayer CropScience AG Neue diazinyl-pyrazolylverbindungen
CA2803695A1 (en) 2010-06-28 2012-01-05 Bayer Intellectual Property Gmbh Heteroaryl-substituted pyridine compounds for use as pesticides
DE102010063691A1 (de) * 2010-12-21 2012-06-21 Bayer Animal Health Gmbh Ektoparasitizide Wirkstoffkombinationen
ES2565821T3 (es) 2011-11-21 2016-04-07 Basf Se Proceso para preparar compuestos 1H-pirazol-5-carboxilato N-sustituidos y derivados de los mismos
CA2868385A1 (en) 2012-05-04 2013-11-07 Basf Se Substituted pyrazole-containing compounds and their use as pesticides
DK2903440T3 (en) * 2012-10-02 2017-12-11 Bayer Cropscience Ag THETEROCYCLIC COMPOUNDS AS PESTICIDES
JP2016503395A (ja) * 2012-10-31 2016-02-04 バイエル・クロップサイエンス・アクチェンゲゼルシャフト 病害生物防除剤としての複素環化合物
WO2016174049A1 (en) 2015-04-30 2016-11-03 Bayer Animal Health Gmbh Anti-parasitic combinations including halogen-substituted compounds
EP3805213A3 (en) 2015-06-18 2021-06-09 Nippon Soda Co., Ltd. 1-(2-(ethylsulfonyl)-phenyl)-4-(phenyl)-1h-1,2,3-triazole and 4-(2-(ethylsulfonyl)-phenyl)-1-(phenyl)-1h-1,2,3-triazole and related compounds derivatives as pesticides
JP6802805B2 (ja) 2015-11-30 2020-12-23 北興化学工業株式会社 1,2,3−トリアゾール誘導体および当該誘導体を有効成分とする殺虫・殺ダニ剤
WO2017104741A1 (ja) 2015-12-16 2017-06-22 日本曹達株式会社 アリールアゾール化合物および有害生物防除剤
TWI766916B (zh) 2016-12-19 2022-06-11 日商日本曹達股份有限公司 二芳基吡唑化合物及有害生物防治劑
CN110305115A (zh) * 2019-08-19 2019-10-08 南通大学 一种含1-(6-氯吡嗪-2-基)-3-甲氧基吡唑单元的吡唑肟衍生物的制备和应用
WO2021219527A1 (de) * 2020-04-29 2021-11-04 Bayer Aktiengesellschaft 1-pyrazinylpyrazolyl-3-oxyalkylsäuren sowie deren derivate und deren verwendung zur bekämpfung unerwünschten pflanzenwachstums
WO2024121262A1 (en) 2022-12-09 2024-06-13 Syngenta Crop Protection Ag Insecticidal compound based on pyrazole derivatives
WO2024121263A1 (en) 2022-12-09 2024-06-13 Syngenta Crop Protection Ag Insecticidal compound based on pyrazole derivatives
WO2024121261A1 (en) 2022-12-09 2024-06-13 Syngenta Crop Protection Ag Insecticidal compound based on pyrazole derivatives
WO2024121264A1 (en) 2022-12-09 2024-06-13 Syngenta Crop Protection Ag Insecticidal compound based on pyrazole derivatives
CN120136787A (zh) * 2023-12-13 2025-06-13 青岛清原化合物有限公司 一种吡唑取代的芳基硫化物类化合物及其应用

Family Cites Families (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NL253320A (es) 1959-07-03
FR2326421A1 (fr) 1975-09-30 1977-04-29 Ugine Kuhlmann Nouveaux trifluoromethyl-3-aryl-4 amino-5 pyrazoles et leur application comme bases diazotables pour la synthese de matieres colorantes
US4101540A (en) 1975-09-30 1978-07-18 Produits Chimiques Ugine Kuhlmann 3-Trifluoromethyl-4-phenyl-pyrazolium azo dyestuffs
JPH08208620A (ja) 1995-02-03 1996-08-13 Takeda Chem Ind Ltd アミノピラゾール誘導体、その製造法および用途
DE19544799A1 (de) * 1995-12-01 1997-06-05 Bayer Ag Substituierte 5-Aminopyrazole
US6169086B1 (en) 1997-01-27 2001-01-02 Daiichi Pharmaceutical Co., Ltd. Pyrazole derivatives
CA2278677A1 (en) 1997-01-27 1998-07-30 Daiichi Pharmaceutical Co., Ltd. Pyrazole derivatives
CA2297780A1 (en) 1998-06-10 1999-12-16 Boulder Scientific Company Synthesis of aryl boronic acids
WO2001007413A1 (en) * 1999-07-22 2001-02-01 3-Dimensional Pharmaceuticals, Inc. 1-aryl-3-thioalkyl pyrazoles, the synthesis thereof and the use thereof as insecticides
US7514464B2 (en) 2003-12-18 2009-04-07 Pfizer Limited Substituted arylpyrazoles
CA2620425A1 (en) 2005-08-31 2007-03-08 Bayer Healthcare Llc Anilinopyrazole derivatives useful for the treatment of diabetes
WO2007048733A1 (de) 2005-10-28 2007-05-03 Basf Se Verwendung von 5-amino-pyrazolen zur bekämpfung pflanzenpathogener schadpilze, neue 5-amino-pyrazole, verfahren zu ihrer herstellung und sie enthaltende mittel
DE102007003036A1 (de) 2006-12-20 2008-06-26 Bayer Cropscience Ag Pyrimidinylpyrazole
WO2009156090A2 (de) * 2008-06-26 2009-12-30 Bayer Cropscience Aktiengesellschaft Insektizide schwefel-derivatisierte 1-azinylpyrazole
EP2499130A1 (de) * 2009-11-11 2012-09-19 Bayer CropScience AG Neue diazinyl-pyrazolylverbindungen

Also Published As

Publication number Publication date
CA2763498A1 (en) 2010-12-02
CO6470821A2 (es) 2012-06-29
KR101758935B1 (ko) 2017-07-17
MX2011012504A (es) 2011-12-12
AR076798A1 (es) 2011-07-06
IL216337A0 (en) 2012-01-31
EP2435420B1 (de) 2013-04-03
WO2010136145A1 (de) 2010-12-02
US8513260B2 (en) 2013-08-20
BRPI1012771A2 (pt) 2016-03-29
DOP2011000366A (es) 2011-12-15
NI201100208A (es) 2012-08-17
US20110021539A1 (en) 2011-01-27
ZA201108637B (en) 2013-01-30
CN102459235A (zh) 2012-05-16
AU2010252346A1 (en) 2011-12-22
IL216337A (en) 2015-09-24
NZ596681A (en) 2015-09-25
UY32659A (es) 2010-12-31
ES2409891T3 (es) 2013-06-28
EP2266973A1 (de) 2010-12-29
CN102459235B (zh) 2015-03-11
TW201107310A (en) 2011-03-01
KR20120061779A (ko) 2012-06-13
US20120190687A1 (en) 2012-07-26
ECSP11011487A (es) 2011-12-30
AU2010252346B2 (en) 2015-11-19
EP2435420A1 (de) 2012-04-04

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