PE20141002A1 - Derivados de heteroarilpiperidina y -piperazina como fungicidas - Google Patents

Derivados de heteroarilpiperidina y -piperazina como fungicidas

Info

Publication number
PE20141002A1
PE20141002A1 PE2013000891A PE2013000891A PE20141002A1 PE 20141002 A1 PE20141002 A1 PE 20141002A1 PE 2013000891 A PE2013000891 A PE 2013000891A PE 2013000891 A PE2013000891 A PE 2013000891A PE 20141002 A1 PE20141002 A1 PE 20141002A1
Authority
PE
Peru
Prior art keywords
alkyl
heteroaryl
heteroarylpiperidine
piperazine
fungicides
Prior art date
Application number
PE2013000891A
Other languages
English (en)
Inventor
Stefan Hillebrand
Pierre Cristau
Sebastian Hoffmann
Joachim Kluth
Thomas Seitz
Pierre Wasnaire
Tomoki Tsuchiya
Jurgen Benting
Ulrike Wachendorff-Neumann
Original Assignee
Bayer Ip Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Ip Gmbh filed Critical Bayer Ip Gmbh
Publication of PE20141002A1 publication Critical patent/PE20141002A1/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/72—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms
    • A01N43/74—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms five-membered rings with one nitrogen atom and either one oxygen atom or one sulfur atom in positions 1,3
    • A01N43/78—1,3-Thiazoles; Hydrogenated 1,3-thiazoles
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/72—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms
    • A01N43/80—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms five-membered rings with one nitrogen atom and either one oxygen atom or one sulfur atom in positions 1,2

Landscapes

  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Environmental Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Plant Pathology (AREA)
  • Pest Control & Pesticides (AREA)
  • Agronomy & Crop Science (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Hydrogenated Pyridines (AREA)

Abstract

SE REFIERE A COMPUESTOS DERIVADOS HETEROARILPIPERIDINA Y -PIPERAZINA DE LA FORMULA (I) , DONDE A ES FENILO, ES UN HETEROARILO, ENTRE OTROS; L1 ES NRL12, C(RL11)2; RL11 ES H, HALOGENO, HIDROXILO, ALCOXI, ENTRE OTROS; RL12 ES H, ALQUILO, ALQUENILO, ENTRE OTROS; Y ES AZUFRE, OXIGENO; X ES CARBONO, NITROGENO; R2 ES H, ALQUILO, HALOALQUILO, HALOGENO, ENTRE OTROS; R10 ES OXO, ALQUILO, ALQUENILO, ALCOXI, ENTRE OTROS; p ES 0,1,2; G ES HETEROARILO DE 5 MIEMBROS QUE ESTA SUSTITUIDO CON Q; Q ES HETEROARILO DE 5 MIEMBROS SATURADO O PARCIAL; ; L2 ES UN ENLACE DIRECTO, O, C(=O), S(O)m CHR20, m ES 0-2; R20 ES HIDROGENO, ALQUILO O HALOALQUILO; R1 ES NAFTILO, DIHIDRONAFTALENILO, TETRAHIDRONAFTALENILO, ENTRE OTROS. SE REFIERE TAMBIEN A UNA COMPOSICION PARA COMBATIR HONGOS FITOPATOGENOS.
PE2013000891A 2010-10-27 2011-10-25 Derivados de heteroarilpiperidina y -piperazina como fungicidas PE20141002A1 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US40720010P 2010-10-27 2010-10-27
EP10189067 2010-10-27

Publications (1)

Publication Number Publication Date
PE20141002A1 true PE20141002A1 (es) 2014-08-17

Family

ID=43640234

Family Applications (1)

Application Number Title Priority Date Filing Date
PE2013000891A PE20141002A1 (es) 2010-10-27 2011-10-25 Derivados de heteroarilpiperidina y -piperazina como fungicidas

Country Status (13)

Country Link
US (4) US20140005224A1 (es)
EP (1) EP2632922B1 (es)
JP (2) JP5918773B2 (es)
KR (1) KR101797074B1 (es)
CN (2) CN103492379B (es)
BR (1) BR112013010497B1 (es)
CA (1) CA2815716C (es)
CO (1) CO6731072A2 (es)
IL (1) IL225766A (es)
MX (1) MX352731B (es)
PE (1) PE20141002A1 (es)
UA (1) UA112534C2 (es)
WO (1) WO2012055837A1 (es)

Families Citing this family (23)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MX2012007200A (es) 2009-12-21 2012-07-10 Bayer Cropscience Ag Bis(difluorometil)pirazoles como fungicidas.
EP2632922B1 (de) * 2010-10-27 2019-02-27 Bayer CropScience Aktiengesellschaft Heteroarylpiperidin und -piperazinderivate als fungizide
WO2012104273A1 (de) 2011-02-01 2012-08-09 Bayer Cropscience Ag Heteroarylpiperidin und -piperazinderivate als fungizide
US10004232B2 (en) 2011-09-15 2018-06-26 Bayer Intellectual Property Gmbh Piperidine pyrazoles as fungicides
DK2797899T3 (en) * 2011-12-27 2016-04-04 Bayer Ip Gmbh Heteroarylpiperidin and -piperazinderivater as fungicides
US9266876B2 (en) 2012-02-02 2016-02-23 Actelion Pharmaceuticals Ltd. 4-(benzoimidazol-2-yl)-thiazole compounds and related aza derivatives
EP2801575A1 (en) 2013-05-07 2014-11-12 Bayer CropScience AG Heteroaryldihydropyridine derivatives as fungicides
WO2014206896A1 (en) 2013-06-24 2014-12-31 Bayer Cropscience Ag Piperidinecarboxylic acid derivatives as fungicides
EA030067B1 (ru) 2013-07-22 2018-06-29 Идорсиа Фармасьютиклз Лтд Производные 1-(пиперазин-1-ил)-2-([1,2,4]триазол-1-ил)этанона
US9924721B2 (en) 2013-08-28 2018-03-27 Bayer Cropscience Aktiengesellschaft Malonic ester derivatives of heteroarylpiperidines and -piperazines as fungicides
PT3122746T (pt) 2014-03-24 2018-07-27 Bayer Cropscience Ag Derivados de fenilpiperidinacarboxamida como fungicidas
AR099789A1 (es) 2014-03-24 2016-08-17 Actelion Pharmaceuticals Ltd Derivados de 8-(piperazin-1-il)-1,2,3,4-tetrahidro-isoquinolina
WO2016024350A1 (ja) 2014-08-13 2016-02-18 株式会社エス・ディー・エス バイオテック 縮合１１員環化合物及びそれらを含有する農園芸用殺菌剤
JP6337218B2 (ja) 2015-01-15 2018-06-06 イドーシア ファーマシューティカルズ リミテッドＩｄｏｒｓｉａ Ｐｈａｒｍａｃｅｕｔｉｃａｌｓ Ｌｔｄ Ｃｘｃｒ３受容体調節剤としてのヒドロキシアルキル−ピペラジン誘導体
AR103399A1 (es) 2015-01-15 2017-05-10 Actelion Pharmaceuticals Ltd Derivados de (r)-2-metil-piperazina como moduladores del receptor cxcr3
MX383376B (es) 2015-03-24 2025-03-13 Shanghai Yingli Pharm Co Ltd Derivado de un anillo condensado y método de preparación, compuesto intermedio, composición farmacéutica y uso del mismo.
WO2016202761A1 (en) 2015-06-17 2016-12-22 Bayer Cropscience Aktiengesellschaft Active compound combinations
CN108602765B (zh) 2016-02-08 2022-05-03 高文有限公司 1,2-苯二甲醇化合物的制造方法
KR102605762B1 (ko) 2016-02-08 2023-11-27 고완 크롭 프로텍션 리미티드 살균성 조성물
TW201838974A (zh) 2017-04-19 2018-11-01 印度商Ｐｉ工業公司 具殺菌性質之雜環化合物
WO2019048988A1 (en) 2017-09-08 2019-03-14 Pi Industries Ltd. Novel fungidal heterocyclic compounds
CA3073637A1 (en) 2017-09-08 2019-03-14 Pi Industries Ltd Novel fungicidal heterocyclic compounds
AR125834A1 (es) * 2021-05-15 2023-08-16 Pi Industries Ltd Composición agroquímica que comprende compuestos de piperidin-tiazol

Family Cites Families (47)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4272417A (en) 1979-05-22 1981-06-09 Cargill, Incorporated Stable protective seed coating
US4245432A (en) 1979-07-25 1981-01-20 Eastman Kodak Company Seed coatings
JPS60156601A (ja) 1984-01-26 1985-08-16 Mitsubishi Petrochem Co Ltd 水田用除草剤
US4808430A (en) 1987-02-27 1989-02-28 Yazaki Corporation Method of applying gel coating to plant seeds
GB8810120D0 (en) 1988-04-28 1988-06-02 Plant Genetic Systems Nv Transgenic nuclear male sterile plants
CA2218526C (en) 1995-04-20 2012-06-12 American Cyanamid Company Structure-based designed herbicide resistant products
US5876739A (en) 1996-06-13 1999-03-02 Novartis Ag Insecticidal seed coating
US6503904B2 (en) 1998-11-16 2003-01-07 Syngenta Crop Protection, Inc. Pesticidal composition for seed treatment
US6660690B2 (en) 2000-10-06 2003-12-09 Monsanto Technology, L.L.C. Seed treatment with combinations of insecticides
US20020134012A1 (en) 2001-03-21 2002-09-26 Monsanto Technology, L.L.C. Method of controlling the release of agricultural active ingredients from treated plant seeds
WO2005040159A1 (en) 2003-10-17 2005-05-06 Astrazeneca Ab 4-(pyrazol-3-ylamino) pyrimidine derivatives for use in the treatment of cancer
TW200639163A (en) 2005-02-04 2006-11-16 Genentech Inc RAF inhibitor compounds and methods
WO2006106423A2 (en) 2005-04-07 2006-10-12 Pfizer Inc. Amino sulfonyl derivatives as inhibitors of human 11-.beta.-hydrosysteroid dehydrogenase
GB0508717D0 (en) 2005-04-29 2005-06-08 Astrazeneca Ab Chemical compounds
TW200738701A (en) 2005-07-26 2007-10-16 Du Pont Fungicidal carboxamides
MEP3508A (xx) 2005-08-24 2010-02-10 Pioneer Hi Bred Int Kompozicije koje obezbjeđuju otpornost na više hibricida i njihov postupak upotrebe
MX2008002802A (es) 2005-08-31 2008-04-07 Monsanto Technology Llc Secuencias nucleotidicas que codifican proteinas insecticidas.
MY145633A (en) 2006-03-01 2012-03-15 Theravance Inc 8-azabicyclo[3.2.1]octane compounds as mu opioid receptor antagonists
KR101130380B1 (ko) 2006-06-13 2012-04-23 상하이 인스티튜트 오브 마테리아 메디카 차이니즈 아카데미 오브 싸이언시즈 헤테로시클릭 비뉴클레오시드 화합물, 그의 제조방법, 약학적 조성물 및 항바이러스성 약제로서의 용도
US9090604B2 (en) * 2006-07-27 2015-07-28 E I Du Pont De Nemours And Company Fungicidal azocyclic amides
WO2008013622A2 (en) * 2006-07-27 2008-01-31 E. I. Du Pont De Nemours And Company Fungicidal azocyclic amides
US20080182851A1 (en) 2006-11-20 2008-07-31 Glenmark Pharmaceuticals S.A. Acetylene derivatives as stearoyl coa desaturase inhibitors
WO2008091594A2 (en) 2007-01-24 2008-07-31 E. I. Du Pont De Nemours And Company Fungicidal mixtures
JP5337711B2 (ja) 2007-01-25 2013-11-06 イー・アイ・デュポン・ドウ・ヌムール・アンド・カンパニー 殺菌性アミド
US8338437B2 (en) 2007-02-28 2012-12-25 Methylgene Inc. Amines as small molecule inhibitors
WO2008147831A1 (en) 2007-05-23 2008-12-04 Smithkline Beecham Corporation Anthranilamides
US20090209536A1 (en) 2007-06-17 2009-08-20 Kalypsys, Inc. Aminoquinazoline cannabinoid receptor modulators for treatment of disease
KR101384075B1 (ko) 2007-07-20 2014-04-09 엘지전자 주식회사 플라즈마 디스플레이 패널
TWI428091B (zh) * 2007-10-23 2014-03-01 Du Pont 殺真菌劑混合物
US8349870B2 (en) * 2008-01-25 2013-01-08 E I Du Pont De Nemours And Company Fungicidal hetercyclic compounds
EP2238133A2 (en) * 2008-01-25 2010-10-13 E. I. du Pont de Nemours and Company Fungicidal amides
BRPI0910837B1 (pt) 2008-04-30 2017-03-07 Bayer Cropscience Ag ésteres e tioésteres tiazol-4-carboxílicos, seus usos, e método e composição para controlar fungos fitopatogênicos prejudiciais
EP2334669B1 (de) 2008-10-01 2015-12-23 Bayer Intellectual Property GmbH Heterocyclyl substituierte thiazole als pflanzenschutzmittel
AU2009322486A1 (en) 2008-12-02 2010-06-10 E. I. Du Pont De Nemours And Company Fungicidal heterocyclic compounds
CN102292334A (zh) 2008-12-11 2011-12-21 拜尔农作物科学股份公司 噻唑基肟醚和腙植物保护剂
DE102010000662A1 (de) 2009-03-18 2010-10-21 Bayer Cropscience Ag Aminopropylthiazol-Derivate als Fungizide
EP2272846A1 (de) 2009-06-23 2011-01-12 Bayer CropScience AG Thiazolylpiperidin Derivate als Fungizide
EP2464643A1 (en) 2009-08-12 2012-06-20 Syngenta Participations AG Microbiocidal heterocycles
UA107938C2 (en) 2009-08-12 2015-03-10 Syngenta Participations Ag Heterocycles with microbicidal properties
WO2011051243A1 (en) 2009-10-29 2011-05-05 Bayer Cropscience Ag Active compound combinations
KR20120101019A (ko) 2009-10-30 2012-09-12 바이엘 크롭사이언스 아게 헤테로아릴피페리딘 및 -피페라진 유도체
MX2012007200A (es) * 2009-12-21 2012-07-10 Bayer Cropscience Ag Bis(difluorometil)pirazoles como fungicidas.
US8629286B2 (en) 2009-12-22 2014-01-14 Syngenta Crop Protection, Llc Pyrazole derivatives
BR112012027762B1 (pt) 2010-04-28 2018-06-05 Bayer Intellectual Property Gmbh Derivados de cetoheteroarilpiperidina e - piperazina como fungicidas
US8815775B2 (en) 2010-05-18 2014-08-26 Bayer Cropscience Ag Bis(difluoromethyl)pyrazoles as fungicides
US8759527B2 (en) * 2010-08-25 2014-06-24 Bayer Cropscience Ag Heteroarylpiperidine and -piperazine derivatives as fungicides
EP2632922B1 (de) * 2010-10-27 2019-02-27 Bayer CropScience Aktiengesellschaft Heteroarylpiperidin und -piperazinderivate als fungizide

Also Published As

Publication number Publication date
CA2815716A1 (en) 2012-05-03
CN103492379B (zh) 2018-06-15
MX352731B (es) 2017-12-06
IL225766A (en) 2015-09-24
CN103492379A (zh) 2014-01-01
JP6117387B2 (ja) 2017-04-19
US9914728B2 (en) 2018-03-13
JP5918773B2 (ja) 2016-05-18
US9512117B2 (en) 2016-12-06
CN107033139B (zh) 2019-11-19
BR112013010497A2 (pt) 2016-07-05
BR112013010497B1 (pt) 2018-07-17
IL225766A0 (en) 2013-06-27
WO2012055837A1 (de) 2012-05-03
US20140005224A1 (en) 2014-01-02
US20170044154A1 (en) 2017-02-16
CA2815716C (en) 2019-06-11
US20170044153A1 (en) 2017-02-16
KR101797074B1 (ko) 2017-11-13
KR20130129962A (ko) 2013-11-29
US20150218152A1 (en) 2015-08-06
JP2016128458A (ja) 2016-07-14
JP2013542212A (ja) 2013-11-21
CO6731072A2 (es) 2013-08-15
WO2012055837A9 (de) 2012-09-20
US9975889B2 (en) 2018-05-22
EP2632922A1 (de) 2013-09-04
MX2013004526A (es) 2013-05-30
CN107033139A (zh) 2017-08-11
EP2632922B1 (de) 2019-02-27
UA112534C2 (uk) 2016-09-26

Similar Documents

Publication Publication Date Title
PE20141002A1 (es) Derivados de heteroarilpiperidina y -piperazina como fungicidas
EA201200018A1 (ru) Триазольные соединения, несущие серосодержащий заместитель
PE20181288A1 (es) Derivados de dihidroimidazopirazinona usados en el tratamiento del cancer
UY32313A (es) Composiciones herbicidas que contienen compuestos de benzoilpirazol y otro compuesto herbicida
PH12015500119A1 (en) Composition for controlling plant disease and application therefor
AR079342A1 (es) Derivados de azol y metodos para producirlos, compuestos intermediarios para los derivados y metodos para producirlos, asi como tambien agentes agrohorticolas y agentes protectores de materiales industriales que contienen los derivados
MD4866B1 (ro) Pesticide pe bază de azol biciclic substituit cu heterociclu
UA110657C2 (uk) Сільськогосподарська і садова фунгіцидна композиція
CL2012000310A1 (es) Compuesto derivado de 5-fluoro pirimidinona; composicion fungicida que comprende a dicho compuesto; y un metodo para el control diferencial de ataque fungico en plantas.
MX2010007952A (es) Arilpirrolinas insecticidas.
NI201000054A (es) Compuestos químicos.
AR077722A1 (es) Derivados de pirazol-carboxamidas, composiciones que los contienen e intermediarios usados en la preparacion de dichos compuestos utiles en horticultura para control o prevencion de la infestacion de plantas por hongos patogenos.
AR087119A1 (es) Composiciones plaguicidas y procesos relacionados
UA104203C2 (en) Microbiocidal heterocycles
BRPI0812222A2 (pt) Compostos ciclobutenodiona substituídos anti-inflamatórios.
TN2015000521A1 (en) Processes of making and crystalline forms of a mdm2 inhibitor
PE20121047A1 (es) Derivados de tiazolilpiperidina como fungicidas
UY31750A (es) Compuestos y composiciones como inhibidores de quinasa
MX380421B (es) Compuestos herbicidas de pirimidiniloxi benceno sustituido.
CO6341630A2 (es) Microbiocidas nuevos
PH12015502671A1 (en) Heterocyclic amide compound
EA201270256A1 (ru) Производные т1-замещенного 5-фтор-2-оксопиримидинон-1 (2h) -карбоксамида
PE20141169A1 (es) Derivados de etinilo
AR079316A1 (es) Derivado de azol, compuestos intermedios para obtenerlo, metodos para producirlos y agente agro- horticola o agente de proteccion de material industrial que lo comprende
PE20141168A1 (es) Derivados de pirazolidin-3-ona

Legal Events

Date Code Title Description
FG Grant, registration