PE20141002A1 - Derivados de heteroarilpiperidina y -piperazina como fungicidas - Google Patents

Derivados de heteroarilpiperidina y -piperazina como fungicidas

Info

Publication number
PE20141002A1
PE20141002A1 PE2013000891A PE2013000891A PE20141002A1 PE 20141002 A1 PE20141002 A1 PE 20141002A1 PE 2013000891 A PE2013000891 A PE 2013000891A PE 2013000891 A PE2013000891 A PE 2013000891A PE 20141002 A1 PE20141002 A1 PE 20141002A1
Authority
PE
Peru
Prior art keywords
alkyl
heteroaryl
heteroarylpiperidine
piperazine
fungicides
Prior art date
Application number
PE2013000891A
Other languages
English (en)
Inventor
Stefan Hillebrand
Pierre Cristau
Sebastian Hoffmann
Joachim Kluth
Thomas Seitz
Pierre Wasnaire
Tomoki Tsuchiya
Jurgen Benting
Ulrike Wachendorff-Neumann
Original Assignee
Bayer Ip Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Ip Gmbh filed Critical Bayer Ip Gmbh
Publication of PE20141002A1 publication Critical patent/PE20141002A1/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/72Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms
    • A01N43/74Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms five-membered rings with one nitrogen atom and either one oxygen atom or one sulfur atom in positions 1,3
    • A01N43/781,3-Thiazoles; Hydrogenated 1,3-thiazoles
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/72Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms
    • A01N43/80Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms five-membered rings with one nitrogen atom and either one oxygen atom or one sulfur atom in positions 1,2

Landscapes

  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Environmental Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Plant Pathology (AREA)
  • Pest Control & Pesticides (AREA)
  • Agronomy & Crop Science (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Hydrogenated Pyridines (AREA)

Abstract

SE REFIERE A COMPUESTOS DERIVADOS HETEROARILPIPERIDINA Y -PIPERAZINA DE LA FORMULA (I) , DONDE A ES FENILO, ES UN HETEROARILO, ENTRE OTROS; L1 ES NRL12, C(RL11)2; RL11 ES H, HALOGENO, HIDROXILO, ALCOXI, ENTRE OTROS; RL12 ES H, ALQUILO, ALQUENILO, ENTRE OTROS; Y ES AZUFRE, OXIGENO; X ES CARBONO, NITROGENO; R2 ES H, ALQUILO, HALOALQUILO, HALOGENO, ENTRE OTROS; R10 ES OXO, ALQUILO, ALQUENILO, ALCOXI, ENTRE OTROS; p ES 0,1,2; G ES HETEROARILO DE 5 MIEMBROS QUE ESTA SUSTITUIDO CON Q; Q ES HETEROARILO DE 5 MIEMBROS SATURADO O PARCIAL; ; L2 ES UN ENLACE DIRECTO, O, C(=O), S(O)m CHR20, m ES 0-2; R20 ES HIDROGENO, ALQUILO O HALOALQUILO; R1 ES NAFTILO, DIHIDRONAFTALENILO, TETRAHIDRONAFTALENILO, ENTRE OTROS. SE REFIERE TAMBIEN A UNA COMPOSICION PARA COMBATIR HONGOS FITOPATOGENOS.
PE2013000891A 2010-10-27 2011-10-25 Derivados de heteroarilpiperidina y -piperazina como fungicidas PE20141002A1 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US40720010P 2010-10-27 2010-10-27
EP10189067 2010-10-27

Publications (1)

Publication Number Publication Date
PE20141002A1 true PE20141002A1 (es) 2014-08-17

Family

ID=43640234

Family Applications (1)

Application Number Title Priority Date Filing Date
PE2013000891A PE20141002A1 (es) 2010-10-27 2011-10-25 Derivados de heteroarilpiperidina y -piperazina como fungicidas

Country Status (13)

Country Link
US (4) US20140005224A1 (es)
EP (1) EP2632922B1 (es)
JP (2) JP5918773B2 (es)
KR (1) KR101797074B1 (es)
CN (2) CN103492379B (es)
BR (1) BR112013010497B1 (es)
CA (1) CA2815716C (es)
CO (1) CO6731072A2 (es)
IL (1) IL225766A (es)
MX (1) MX352731B (es)
PE (1) PE20141002A1 (es)
UA (1) UA112534C2 (es)
WO (1) WO2012055837A1 (es)

Families Citing this family (23)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP5785560B2 (ja) * 2009-12-21 2015-09-30 バイエル・クロップサイエンス・アクチェンゲゼルシャフト 殺真菌剤としてのビス(ジフルオロメチル)ピラゾール
PE20141002A1 (es) * 2010-10-27 2014-08-17 Bayer Ip Gmbh Derivados de heteroarilpiperidina y -piperazina como fungicidas
KR101848116B1 (ko) 2011-02-01 2018-04-11 바이엘 인텔렉쳐 프로퍼티 게엠베하 살진균제로서의 헤테로아릴 피페리딘 및 헤테로아릴 피페라진 유도체
ES2661849T3 (es) * 2011-09-15 2018-04-04 Bayer Intellectual Property Gmbh Piperidinpirazoles como fungicidas
DK2921493T3 (da) 2011-12-27 2017-11-27 Bayer Ip Gmbh Heteroarylpiperidin og ¿piperazinderivater
AU2013216354B2 (en) 2012-02-02 2017-08-31 Idorsia Pharmaceuticals Ltd 4-(benzoimidazol-2-yl)-thiazole compounds and related aza derivatives
EP2801575A1 (en) 2013-05-07 2014-11-12 Bayer CropScience AG Heteroaryldihydropyridine derivatives as fungicides
JP6430494B2 (ja) 2013-06-24 2018-11-28 バイエル・クロップサイエンス・アクチェンゲゼルシャフト 殺真菌剤としてのピペリジンカルボン酸誘導体
JP6330040B2 (ja) 2013-07-22 2018-05-23 イドーシア ファーマシューティカルズ リミテッドIdorsia Pharmaceuticals Ltd 1−(ピペラジン−1−イル)−2−([1,2,4]トリアゾール−1−イル)−エタノン誘導体
US9924721B2 (en) 2013-08-28 2018-03-27 Bayer Cropscience Aktiengesellschaft Malonic ester derivatives of heteroarylpiperidines and -piperazines as fungicides
AR099789A1 (es) 2014-03-24 2016-08-17 Actelion Pharmaceuticals Ltd Derivados de 8-(piperazin-1-il)-1,2,3,4-tetrahidro-isoquinolina
PE20161176A1 (es) * 2014-03-24 2016-11-19 Bayer Cropscience Ag Derivados de fenilpiperidincarboxamida como fungicidas
WO2016024350A1 (ja) 2014-08-13 2016-02-18 株式会社エス・ディー・エス バイオテック 縮合11員環化合物及びそれらを含有する農園芸用殺菌剤
AR103399A1 (es) 2015-01-15 2017-05-10 Actelion Pharmaceuticals Ltd Derivados de (r)-2-metil-piperazina como moduladores del receptor cxcr3
PL3245203T3 (pl) 2015-01-15 2019-05-31 Idorsia Pharmaceuticals Ltd Pochodne hydroksyalkilopiperazyny jako modulatory receptora cxcr3
AU2016236669B2 (en) 2015-03-24 2018-11-08 Shanghai Yingli Pharmaceutical Co., Ltd Condensed ring derivative, and preparation method, intermediate, pharmaceutical composition and use thereof
WO2016202761A1 (en) 2015-06-17 2016-12-22 Bayer Cropscience Aktiengesellschaft Active compound combinations
JP6407457B2 (ja) 2016-02-08 2018-10-17 株式会社エス・ディー・エス バイオテック 1,2−ベンゼンジメタノール化合物の製造方法
WO2017138069A1 (ja) 2016-02-08 2017-08-17 株式会社エス・ディー・エス バイオテック 殺菌性組成物
TW201838974A (zh) 2017-04-19 2018-11-01 印度商Pi工業公司 具殺菌性質之雜環化合物
US20200281202A1 (en) 2017-09-08 2020-09-10 Pi Industries Ltd. Novel fungicidal heterocyclic compounds
WO2019048988A1 (en) 2017-09-08 2019-03-14 Pi Industries Ltd. Novel fungidal heterocyclic compounds
UY39763A (es) * 2021-05-15 2022-11-30 Pi Industries Ltd Composición agroquímica novedosa que comprende compuestos de piperidin-tiazol

Family Cites Families (47)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4272417A (en) 1979-05-22 1981-06-09 Cargill, Incorporated Stable protective seed coating
US4245432A (en) 1979-07-25 1981-01-20 Eastman Kodak Company Seed coatings
JPS60156601A (ja) 1984-01-26 1985-08-16 Mitsubishi Petrochem Co Ltd 水田用除草剤
US4808430A (en) 1987-02-27 1989-02-28 Yazaki Corporation Method of applying gel coating to plant seeds
GB8810120D0 (en) 1988-04-28 1988-06-02 Plant Genetic Systems Nv Transgenic nuclear male sterile plants
US6576455B1 (en) 1995-04-20 2003-06-10 Basf Corporation Structure-based designed herbicide resistant products
US5876739A (en) 1996-06-13 1999-03-02 Novartis Ag Insecticidal seed coating
US6503904B2 (en) 1998-11-16 2003-01-07 Syngenta Crop Protection, Inc. Pesticidal composition for seed treatment
US6660690B2 (en) 2000-10-06 2003-12-09 Monsanto Technology, L.L.C. Seed treatment with combinations of insecticides
US20020134012A1 (en) 2001-03-21 2002-09-26 Monsanto Technology, L.L.C. Method of controlling the release of agricultural active ingredients from treated plant seeds
CA2542522A1 (en) 2003-10-17 2005-05-06 Astrazeneca Ab 4-(pyrazol-3-ylamino) pyrimidine derivatives for use in the treatment of cancer
TW200639163A (en) 2005-02-04 2006-11-16 Genentech Inc RAF inhibitor compounds and methods
WO2006106423A2 (en) 2005-04-07 2006-10-12 Pfizer Inc. Amino sulfonyl derivatives as inhibitors of human 11-.beta.-hydrosysteroid dehydrogenase
GB0508717D0 (en) 2005-04-29 2005-06-08 Astrazeneca Ab Chemical compounds
TW200738701A (en) 2005-07-26 2007-10-16 Du Pont Fungicidal carboxamides
BRPI0615087A2 (pt) 2005-08-24 2011-05-03 Pioneer Hi Bred Int métodos e composições para a expressão de um polinucleotìdeo de interesse
EA015908B1 (ru) 2005-08-31 2011-12-30 Монсанто Текнолоджи, Ллс Инсектицидный белок в.thuringiensis cry1a.105, кодирующий его полинуклеотид и их применение
MY145633A (en) 2006-03-01 2012-03-15 Theravance Inc 8-azabicyclo[3.2.1]octane compounds as mu opioid receptor antagonists
KR101130380B1 (ko) 2006-06-13 2012-04-23 상하이 인스티튜트 오브 마테리아 메디카 차이니즈 아카데미 오브 싸이언시즈 헤테로시클릭 비뉴클레오시드 화합물, 그의 제조방법, 약학적 조성물 및 항바이러스성 약제로서의 용도
US9090604B2 (en) * 2006-07-27 2015-07-28 E I Du Pont De Nemours And Company Fungicidal azocyclic amides
WO2008013622A2 (en) * 2006-07-27 2008-01-31 E. I. Du Pont De Nemours And Company Fungicidal azocyclic amides
WO2008062276A2 (en) 2006-11-20 2008-05-29 Glenmark Pharmaceuticals S.A. Acetylene derivatives as stearoyl coa desaturase inhibitors
WO2008091594A2 (en) 2007-01-24 2008-07-31 E. I. Du Pont De Nemours And Company Fungicidal mixtures
US8420673B2 (en) 2007-01-25 2013-04-16 E I Du Pont De Nemours And Company Fungicidal amides
EP2137158A4 (en) 2007-02-28 2012-04-18 Methylgene Inc LOW-MOLECULAR INHIBITORS OF PROTEINARGININE METHYLTRANSFERASES (PRMTS)
WO2008147831A1 (en) 2007-05-23 2008-12-04 Smithkline Beecham Corporation Anthranilamides
WO2008157500A1 (en) 2007-06-17 2008-12-24 Kalypsys, Inc. Aminoquinazoline cannabinoid receptor modulators for treatment of disease
KR101384075B1 (ko) 2007-07-20 2014-04-09 엘지전자 주식회사 플라즈마 디스플레이 패널
TWI428091B (zh) * 2007-10-23 2014-03-01 Du Pont 殺真菌劑混合物
CN101925598B (zh) * 2008-01-25 2014-03-05 杜邦公司 杀真菌酰胺
CN101970432B (zh) * 2008-01-25 2014-05-28 杜邦公司 杀真菌杂环化合物
MX2010011879A (es) 2008-04-30 2010-12-06 Bayer Cropscience Ag Esteres y tioesteres del acido tiazol-4-carboxilico como agentes fitoprotectores.
BRPI0920767B1 (pt) 2008-10-01 2018-07-17 Bayer Intellectual Property Gmbh tiazóis substituídos por heterociclila como agentes protetores de cultura, seus usos e seus processos de preparação, composições e seu processo de preparação, e método para combate a fungos nocivos fitopatogênicos
TW201036966A (en) * 2008-12-02 2010-10-16 Du Pont Fungicidal heterocyclic compounds
BRPI0923366A2 (pt) 2008-12-11 2019-09-24 Bayer Cropscience Ag éteres e hodrazonas de oxima de tiazolila como agentes protetors de culturas.
DE102010000662A1 (de) 2009-03-18 2010-10-21 Bayer Cropscience Ag Aminopropylthiazol-Derivate als Fungizide
EP2272846A1 (de) 2009-06-23 2011-01-12 Bayer CropScience AG Thiazolylpiperidin Derivate als Fungizide
UA107938C2 (en) 2009-08-12 2015-03-10 Syngenta Participations Ag Heterocycles with microbicidal properties
KR20120089644A (ko) 2009-08-12 2012-08-13 신젠타 파티서페이션즈 아게 살미생물성 헤테로사이클
WO2011051243A1 (en) 2009-10-29 2011-05-05 Bayer Cropscience Ag Active compound combinations
EP2493886B1 (de) 2009-10-30 2014-11-26 Bayer CropScience AG Heteroarylpiperidin und -piperazin derivate
JP5785560B2 (ja) * 2009-12-21 2015-09-30 バイエル・クロップサイエンス・アクチェンゲゼルシャフト 殺真菌剤としてのビス(ジフルオロメチル)ピラゾール
EP2516424B1 (en) 2009-12-22 2013-12-18 Syngenta Participations AG Pyrazole derivatives
JP5960683B2 (ja) 2010-04-28 2016-08-02 バイエル・インテレクチュアル・プロパティ・ゲゼルシャフト・ミット・ベシュレンクテル・ハフツングBayer Intellectual Property GmbH 殺真菌剤としてのケトヘテロアリールピペリジンおよび−ピペラジン誘導体
US8815775B2 (en) 2010-05-18 2014-08-26 Bayer Cropscience Ag Bis(difluoromethyl)pyrazoles as fungicides
US8759527B2 (en) * 2010-08-25 2014-06-24 Bayer Cropscience Ag Heteroarylpiperidine and -piperazine derivatives as fungicides
PE20141002A1 (es) * 2010-10-27 2014-08-17 Bayer Ip Gmbh Derivados de heteroarilpiperidina y -piperazina como fungicidas

Also Published As

Publication number Publication date
US20150218152A1 (en) 2015-08-06
US20170044153A1 (en) 2017-02-16
UA112534C2 (uk) 2016-09-26
US9512117B2 (en) 2016-12-06
CN103492379B (zh) 2018-06-15
US20170044154A1 (en) 2017-02-16
IL225766A (en) 2015-09-24
JP2013542212A (ja) 2013-11-21
WO2012055837A1 (de) 2012-05-03
CA2815716C (en) 2019-06-11
BR112013010497B1 (pt) 2018-07-17
CN103492379A (zh) 2014-01-01
US20140005224A1 (en) 2014-01-02
CA2815716A1 (en) 2012-05-03
EP2632922A1 (de) 2013-09-04
US9975889B2 (en) 2018-05-22
CN107033139B (zh) 2019-11-19
CO6731072A2 (es) 2013-08-15
EP2632922B1 (de) 2019-02-27
MX2013004526A (es) 2013-05-30
WO2012055837A9 (de) 2012-09-20
US9914728B2 (en) 2018-03-13
IL225766A0 (en) 2013-06-27
JP5918773B2 (ja) 2016-05-18
JP2016128458A (ja) 2016-07-14
BR112013010497A2 (pt) 2016-07-05
KR101797074B1 (ko) 2017-11-13
MX352731B (es) 2017-12-06
JP6117387B2 (ja) 2017-04-19
CN107033139A (zh) 2017-08-11
KR20130129962A (ko) 2013-11-29

Similar Documents

Publication Publication Date Title
PE20141002A1 (es) Derivados de heteroarilpiperidina y -piperazina como fungicidas
EA201200018A1 (ru) Триазольные соединения, несущие серосодержащий заместитель
PE20140185A1 (es) Derivados de heteroarilpiperidina y piperazina como fungicidas
PE20181288A1 (es) Derivados de dihidroimidazopirazinona usados en el tratamiento del cancer
UY32313A (es) Composiciones herbicidas que contienen compuestos de benzoilpirazol y otro compuesto herbicida
CR11021A (es) Derivados de quinolina como fungicidas
PH12015500119A1 (en) Composition for controlling plant disease and application therefor
AR079342A1 (es) Derivados de azol y metodos para producirlos, compuestos intermediarios para los derivados y metodos para producirlos, asi como tambien agentes agrohorticolas y agentes protectores de materiales industriales que contienen los derivados
MX2013004242A (es) Sulfonamidas nematocidas.
MD4866B1 (ro) Pesticide pe bază de azol biciclic substituit cu heterociclu
UA110657C2 (uk) Сільськогосподарська і садова фунгіцидна композиція
CL2012000310A1 (es) Compuesto derivado de 5-fluoro pirimidinona; composicion fungicida que comprende a dicho compuesto; y un metodo para el control diferencial de ataque fungico en plantas.
MX2010007952A (es) Arilpirrolinas insecticidas.
NI201000054A (es) Compuestos químicos.
AR087119A1 (es) Composiciones plaguicidas y procesos relacionados
MX2012001690A (es) Heterociclos microbicidas.
BRPI0812222A2 (pt) Compostos ciclobutenodiona substituídos anti-inflamatórios.
PE20121047A1 (es) Derivados de tiazolilpiperidina como fungicidas
UY31750A (es) Compuestos y composiciones como inhibidores de quinasa
MX380421B (es) Compuestos herbicidas de pirimidiniloxi benceno sustituido.
EA201270256A1 (ru) Производные т1-замещенного 5-фтор-2-оксопиримидинон-1 (2h) -карбоксамида
PE20141169A1 (es) Derivados de etinilo
AR075763A1 (es) N-alcoxicarboxamidas sustituidas con heterociclos, composiciones microbiocidas que las contienen y metodo para el control y/o prevencion de infestaciones fungicas en plantas.
AR079316A1 (es) Derivado de azol, compuestos intermedios para obtenerlo, metodos para producirlos y agente agro- horticola o agente de proteccion de material industrial que lo comprende
PE20141168A1 (es) Derivados de pirazolidin-3-ona

Legal Events

Date Code Title Description
FG Grant, registration